Mostrando resultados 12 a 31 de 39
< Anterior
Siguiente >
Derechos | Preview | Fecha Public. | Título | Autor(es) | Tipo |
openAccess | | 2018 | Identification of a Tool Compound to Study the Mechanisms of Functional Selectivity between D2 and D3 Dopamine Receptors | Reyes-Resina, I.; Samadi, Abdelouahid CSIC ORCID; Navarro, Gemma; Saadeh, H. A.; Khasawneh, M. A.; Mestres, Jordi; Marco-Contelles, José CSIC ORCID; Franco, Rafael | artículo |
closedAccess | | 2015 | α-aryl-N-alkyl nitrones, as potential agents for stroke treatment: Synthesis, theoretical calculations, antioxidant, anti-inflammatory, neuroprotective, and brain-blood barrier permeability properties | Chioua, Mourad CSIC ORCID ; Sucunza, D.; Soriano, Elena CSIC; Hadjipavlou-Litina, Dimitra; Alcázar González, Alberto; Ayuso, I.; Oset-Gasque, María Jesús; Gonzalez, M. P.; Monjas, Leticia CSIC ORCID; Rodríguez-Franco, María Isabel CSIC ORCID ; Marco-Contelles, José CSIC ORCID; Marco-Contelles, José CSIC ORCID; Samadi, Abdelouahid CSIC ORCID | artículo |
closedAccess | | 2014 | Kinetic and structural analysis of the irreversible inhibition of human monoamine oxidases by ASS234, a multi-target compound designed for use in Alzheimer's disease | Esteban, Gerard; Allan, Jennifer; Samadi, Abdelouahid CSIC ORCID; Mattevi, Andrea; Unzeta, Mercedes; Marco-Contelles, José CSIC ORCID; Binda, Claudia; Ramsay, Rona R. | artículo |
openAccess | | 2014 | Multipotent cholinesterase/monoamine oxidase inhibitors for the treatment of Alzheimer’s disease: Design, synthesis, biochemical evaluation, ADMET, molecular modeling, and QSAR analysis of novel donepezil-pyridyl hybrids | Bautista-Aguilera, Óscar M. CSIC ORCID; Esteban, Gerard; Chioua, Mourad CSIC ORCID ; Nikolic, Katarina; Agbaba, Danica; Moraleda, Ignacio; Iriepa, Isabel; Soriano, Elena CSIC; Samadi, Abdelouahid CSIC ORCID; Unzeta, Mercedes; Marco-Contelles, José CSIC ORCID | artículo |
closedAccess | | 2013 | Multipotent, permeable drug ASS234 inhibits Aβ aggregation, possesses antioxidant properties and protects from Aβ-induced apoptosis in vitro | Bolea, Irene; Gella, Alejandro; Monjas, Leticia CSIC ORCID; Pérez, Concepción CSIC ORCID; Rodríguez-Franco, María Isabel CSIC ORCID ; Marco-Contelles, José CSIC ORCID; Samadi, Abdelouahid CSIC ORCID; Unzeta, Mercedes | artículo |
closedAccess | | 2016 | N-Benzylpiperidine derivatives as α7 nicotinic receptor antagonists | Criado, Manuel CSIC ORCID; Mulet, José CSIC ORCID; Sala, Francisco CSIC ORCID; Sala, Salvador CSIC ORCID; Colmena, Inés CSIC; Gandía, Luis; Bautista-Aguilera, Oscar M.; Samadi, Abdelouahid CSIC ORCID; Chioua, Mourad CSIC ORCID ; Marco-Contelles, José CSIC ORCID | artículo |
closedAccess | | 2014 | N-methyl-N-((1-methyl-5-(3-(1-(2-methylbenzyl)piperidin-4-yl)propoxy)-1H-indol-2-yl)methyl)prop-2-yn-1-amine, a new cholinesterase and monoamine oxidase dual inhibitor | Bautista-Aguilera, Óscar M. CSIC ORCID; Samadi, Abdelouahid CSIC ORCID; Chioua, Mourad CSIC ORCID ; Nikolic, K.; Filipic, S.; Agbaba, Danica; Soriano, Elena CSIC; Andrés, Lucía de CSIC; Rodríguez-Franco, María Isabel CSIC ORCID ; Alcaro, S.; Ramsay, R. R.; Ortuso, F.; Yáñez, Matilde; Marco-Contelles, José CSIC ORCID | artículo |
openAccess | | 22-ago-2011 | New derivatives of propargylamine having neuroprotective capacity for the treatment of alzheimer's and parkinson's diseases | Samadi, Abdelouahid CSIC ORCID; Marco-Contelles, José CSIC ORCID; Bolea Tomás, Irene; Luque, Francisco J.; Unzeta López, Mercedes | solicitud de patente |
closedAccess | | 2013 | Nontoxic and neuroprotective β-naphthotacrines for alzheimer's disease | Esquivias-Pérez, Mario; Maalej, Enma; Romero Jódar, Alejandro CSIC ORCID; Chabchoub, Fakher; Samadi, Abdelouahid CSIC ORCID; Marco-Contelles, José CSIC ORCID; Oset-Gasque, María Jesús | artículo |
closedAccess | | 2013 | Novel tacrine-related drugs as potential candidates for the treatment of Alzheimer's disease | Romero Jódar, Alejandro CSIC ORCID; Cacabelos, Ramón; Oset-Gasque, María Jesús; Samadi, Abdelouahid CSIC ORCID; Marco-Contelles, José CSIC ORCID | artículo |
openAccess | | 18-ene-2012 | Nuevas 2,2'-azopiridinas a partir de 2-aminopiridinas de interés farmacéutico e industrial | Samadi, Abdelouahid CSIC ORCID; Marco-Contelles, José CSIC ORCID; Botelho da Silva, Daniel | solicitud de patente |
openAccess | | 29-sep-2011 | Nuevos derivados de propargilamina con capacidad neuroprotectora para el tratamiento de las enfermedades de Alzheimer y Parkinson | Samadi, Abdelouahid CSIC ORCID; Marco-Contelles, José CSIC ORCID; Bolea Tomás, Irene; Luque, Francisco J.; Unzeta, Mercedes | solicitud de patente |
closedAccess | | 2013 | PP2A ligand ITH12246 protects against memory impairment and focal cerebral ischemia in mice | Lorrio, Silvia; Romero Jódar, Alejandro CSIC ORCID; González-Lafuente, Laura; Lajarín-Cuesta, Rocío; Martínez-Sanz, Francisco J.; Estrada, Martín CSIC ORCID CVN; Samadi, Abdelouahid CSIC ORCID; Marco-Contelles, José CSIC ORCID; Rodríguez-Franco, María Isabel CSIC ORCID ; Villarroya, Mercedes; López, Manuela G.; Ríos, Cristobal de los | artículo |
openAccess | | 15-feb-2013 | Quinolilnitronas | Chioua, Mourad CSIC ORCID ; Samadi, Abdelouahid CSIC ORCID; Soriano, Elena CSIC; Marco-Contelles, José CSIC ORCID; Oset-Gasque, María Jesús; Alcázar, Alberto | solicitud de patente |
openAccess | | 7-feb-2013 | Quinolyl nitrones | Chioua, Mourad CSIC ORCID ; Samadi, Abdelouahid CSIC ORCID; Soriano, Elena CSIC; Marco-Contelles, José CSIC ORCID; Oset-Gasque, María Jesús; Alcázar, Alberto | patente |
openAccess | | 17-abr-2019 | QuinoxalineTacrine QT78, a Cholinesterase Inhibitor as a Potential Ligand for Alzheimer’s Disease Therapy | Ramos, Eva; Palomino-Antolín, Alejandra; Bartolini, Manuela; Iriepa, Isabel; Moraleda, Ignacio; Diez-Iriepa, Daniel CSIC; Samadi, Abdelouahid CSIC ORCID; Cortina, Carol V.; Chioua, Mourad CSIC ORCID ; Egea, Javier; Romero Jódar, Alejandro CSIC ORCID; Marco-Contelles, José CSIC ORCID | artículo |
closedAccess | | 2014 | Silver triflate-catalyzed cyclization of 2-amino-6-propargyl- amineazines leading to iminoimidazoazines | Chioua, Mourad CSIC ORCID ; Samadi, Abdelouahid CSIC ORCID; Soriano, Elena CSIC; Infantes, L. CSIC ORCID; Marco-Contelles, José CSIC ORCID | artículo |
closedAccess | | 2013 | Silver-catalyzed cyclization of N-(prop-2-yn-1-yl)pyridin-2-amines | Chioua, Mourad CSIC ORCID ; Soriano, Elena CSIC; Infantes, L. CSIC ORCID; Jimeno, M. Luisa CSIC ORCID; Marco-Contelles, José CSIC ORCID; Samadi, Abdelouahid CSIC ORCID | artículo |
openAccess | | 7-may-2012 | Síntesis de piridonas bicíclicas que contienen el sistema heterocíclico de imidazo[1,2-a]piridina, a partir de 2-amino-6-(prop-2-in-1-ilamino)piridinas | Samadi, Abdelouahid CSIC ORCID; Marco-Contelles, José CSIC ORCID; Sucunza Sáez, David CSIC ORCID; Chioua, Mourad CSIC ORCID | solicitud de patente |
closedAccess | | 2011 | Synthesis and pharmacological assessment of diversely substituted pyrazolo[3,4-b]quinoline, and benzo[b]pyrazolo[4,3-g][1,8]naphthyridine derivatives | Silva, Daniel; Chioua, Mourad CSIC ORCID ; Samadi, Abdelouahid CSIC ORCID; Carreiras, M. Carmo; Jimeno, M. Luisa CSIC ORCID; Mendes, Eduarda; Ríos, Cristóbal de los; Romero Jódar, Alejandro CSIC ORCID; Villarroya, Mercedes; Marco-Contelles, José CSIC ORCID | artículo |