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DerechosPreviewFecha Public.TítuloAutor(es)Tipo
openAccessaccesoRestringido.pdf.jpg27-jun-2016Blocking Blood Flow to Solid Tumors by Destabilizing Tubulin : An Approach to Targeting Tumor Growth (Perspective)Peréz-Pérez, María-Jesús CSIC ORCID ; Priego, Eva María CSIC ORCID; Bueno, Oskia CSIC; Martins, Maria Solange; Canela, María-Dolores CSIC; Liekens, Sandraartículo
closedAccessaccesoRestringido.pdf.jpg2019Chalcones and Chalcone-mimetic Derivatives as Notch Inhibitors in a Model of T-cell Acute Lymphoblastic LeukemiaQuaglio, D.; Zhdanovskaya, N.; Tobajas, Gloria; Cuartas, V.; Balducci, S.; Christodoulou, M. S.; Fabrizi, G.; Gargantilla, Marta CSIC ORCID; Priego, Eva María CSIC ORCID; Carmona Pestania, Á.; Passarella, D.; Screpanti, I.; Botta, B.; Palermo, R.; Mori, M.; Ghirga, F.; Peréz-Pérez, María-Jesús CSIC ORCID artículo
openAccessExpert Opinion_Perez-Perez et al_2019.pdf.jpg14-jun-2019Chikungunya virus drug discovery: still a long way to go?Peréz-Pérez, María-Jesús CSIC ORCID ; Delang, Leen; Ng, Lisa; Priego, Eva María CSIC ORCIDartículo
openAccessaccesoRestringido.pdf.jpg2018Conformational mimetics of the α-methyl chalcone TUB091 binding tubulin: Design, synthesis and antiproliferative activityBueno, Oskia CSIC; Tobajas, Gloria; Quesada, Ernesto CSIC ORCID ; Estévez-Gallego, Juan CSIC ORCID ; Noppen, Sam; Camarasa Rius, María José CSIC ORCID; Díaz, José Fernando CSIC ORCID ; Liekens, Sandra; Priego, Eva María CSIC ORCID; Peréz-Pérez, María-Jesús CSIC ORCID artículo
closedAccessaccesoRestringido.pdf.jpg2012CRDOCK: An ultrafast multipurpose protein-ligand docking toolCortés Cabrera, Álvaro CSIC ORCID; Klett, Javier CSIC ORCID; Dos Santos, Helena G.; Perona, Almudena CSIC ORCID CVN; Gil Redondo, Rubén; Francis, Sandrea M. CSIC; Priego, Eva María CSIC ORCID; Gago, Federico CSIC ORCID; Morreale, Antonioartículo
openAccessmolecules-pirazolinas_2019.pdf.jpg2019Design and Synthesis of New 6-Nitro and 6-Amino- 3,3a,4,5-Tetrahydro-2H-Benzo[g]indazole Derivatives: Antiproliferative and Antibacterial ActivityCuartas, Viviana; Crespo, María del Pilar; Priego, Eva María CSIC ORCID; Persoons, Leentje; Daelemans, Dirk; Camarasa Rius, María José CSIC ORCID; Insuasty, Braulio; Peréz-Pérez, María-Jesús CSIC ORCID artículo
openAccessmolecules-24-04236-v2.pdf.jpg2019Design and synthesis of new 6-nitro and 6-Amino-3,3a,4,5-Tetrahydro-2H-Benzo[g]indazole derivatives: Antiproliferative and antibacterial activityCuartas, V.; Crespo, M. D. P.; Priego, Eva María CSIC ORCID; Persoons, L.; Daelemans, D.; Camarasa Rius, María José CSIC ORCID; Insuasty, Braulio; Peréz-Pérez, María-Jesús CSIC ORCID artículo
closedAccessEJMC_Diphenyl_ether_derivatives_2019.pdf.jpgjun-2019Diphenyl ether derivatives occupy the expanded binding site of cyclohexanedione compounds at the colchicine site in tubulin by movement of the aT5 loopBueno, Oskia CSIC; Gargantilla, Marta CSIC ORCID; Estévez-Gallego, Juan CSIC ORCID ; Martins, Solange; Díaz, José Fernando CSIC ORCID ; Camarasa Rius, María José CSIC ORCID; Liekens, Sandra; Peréz-Pérez, María-Jesús CSIC ORCID ; Priego, Eva María CSIC ORCIDartículo
closedAccess2012Efficient synthesis and anti-enteroviral activity of 9-arylpurinesAguado, Leire CSIC; Canela, María-Dolores CSIC; Thibaut, Hendrik Jan; Priego, Eva María CSIC ORCID; Camarasa Rius, María José CSIC ORCID; Leyssen, Pieter; Neyts, Johan; Peréz-Pérez, María-Jesús CSIC ORCID artículo
openAccessScientific reports(2018)4242.pdf.jpg2018High-affinity ligands of the colchicine domain in tubulin based on a structure-guided designBueno, Oskia CSIC; Estévez-Gallego, Juan CSIC ORCID ; Martins, S.; Prota, Andrea E.; Gago, Federico CSIC ORCID; Gómez-SanJuan, Asier CSIC; Camarasa Rius, María José CSIC ORCID; Barasoain, Isabel CSIC ; Steinmetz, Michel O.; Díaz, José Fernando CSIC ORCID ; Peréz-Pérez, María-Jesús CSIC ORCID ; Liekens, Sandra; Priego, Eva María CSIC ORCIDartículo
openAccesspharmaceuticals-15-00835.pdf.jpg2022Hybridization Approach to Identify Salicylanilides as Inhibitors of Tubulin Polymerization and Signal Transducers and Activators of Transcription 3 (STAT3)Gargantilla, Marta CSIC ORCID; Persoons, Leentje; Kauerová, Tereza; Río, Natalia del CSIC ORCID; Daelemans, Dirk; Priego, Eva María CSIC ORCID; Kollar, Peter; Peréz-Pérez, María-Jesús CSIC ORCID artículo
closedAccess2014Identification of [1,2,3]triazolo[4,5-d ]pyrimidin-7(6H)-ones as novel inhibitors of chikungunya virus replicationGigante, Alba CSIC ORCID; Canela, María-Dolores CSIC; Delang, Leen; Priego, Eva María CSIC ORCID; Camarasa Rius, María José CSIC ORCID; Querat, Guilles; Neyts, Johan; Leyssen, Pieter; Peréz-Pérez, María-Jesús CSIC ORCID artículo
openAccessScientific reports (2018).pdf.jpg2018Identification of a novel 2-oxindole fluorinated derivative as in vivo antitumor agent for prostate cancer acting via AMPK activationBort Bueno, Alicia; Quesada Sánchez, Sergio CSIC; Ramos-Torres, Ágata; Gargantilla, Marta CSIC ORCID; Priego, Eva María CSIC ORCID; Raynal, S.; Lepifre, F.; Gasalla, José María; Rodriguez-Henche, Nieves; Castro, Ana CSIC ORCID; Díaz-Laviada, Inésartículo
openAccessACS Infect Dis 2018.pdf.jpg2018Inhibition of the Replication of Different Strains of Chikungunya Virus by 3-Aryl-[1,2,3]triazolo[4,5- d] pyrimidin-7(6 H)-onesGómez-SanJuan, Asier CSIC; Gamo, Ana María CSIC; Delang, Leen; Pérez-Sánchez, Alfonso; Amrun, S. N.; Abdelnabi, Rana; Jacobs, S.; Priego, Eva María CSIC ORCID; Camarasa Rius, María José CSIC ORCID; Jochmans, D.; Leyssen, Pieter; Ng, L. F. P.; Querat, Guilles; Neyts, Johan; Peréz-Pérez, María-Jesús CSIC ORCID artículo
openAccesspharmaceuticals-14-01131-1.pdf.jpg6-nov-2021Inhibition of XPO-1 Mediated Nuclear Export through the Michael-Acceptor Character of ChalconesGargantilla, Marta CSIC ORCID; López-Fernández, José; Camarasa Rius, María José CSIC ORCID; Persoons, Leentje; Daelemans, Dirk; Priego, Eva María CSIC ORCID; Peréz-Pérez, María-Jesús CSIC ORCID artículo
closedAccess2009Intramolecular Cation-π Interactions As the Driving Force To Restrict the Conformation of Certain NucleosidesCasanova, Elena; Priego, Eva María CSIC ORCID; Jimeno, M. Luisa CSIC ORCID; Aguado, Leire CSIC; Negri, Ana; Gago, Federico CSIC ORCID; Camarasa Rius, María José CSIC ORCID; Peréz-Pérez, María-Jesús CSIC ORCID artículo
openAccessGigante_full_article.pdf.jpg2014Microwave-assisted synthesis of C-8 aryl and heteroaryl inosines and determination of their inhibitory activities against Plasmodium falciparum purine nucleoside phosphorylaseGigante, Alba CSIC ORCID; Priego, Eva María CSIC ORCID; Sánchez-Carrasco, Paula; Ruiz-Pérez, Luis Miguel; Vande Voorde, Johan; Camarasa Rius, María José CSIC ORCID; Balzarini, Jan; González-Pacanowska, Dolores; Peréz-Pérez, María-Jesús CSIC ORCID artículo
openAccess2022 ACS Chem Neurosci 13-275 postprint.pdf.jpg19-ene-2022Neuroprotective Effect of IND1316, an Indole-Based AMPK Activator, in Animal Models of Huntington DiseaseVela, Marta; García-Gimeno, María Adelaida CSIC ORCID; Sanchis, Ana CSIC; Bono-Yagüe, José; Cumella, José; Lagartera, Laura CSIC ORCID; Pérez, Concepción CSIC ORCID; Priego, Eva María CSIC ORCID; Campos, Ángela CSIC; Sanz, Pascual CSIC ORCID ; Vázquez-Manrique, Rafael P. CSIC ORCID; Castro, Ana CSIC ORCIDartículo
openAccessCanela-et-al_2014_JMedChem_57.pdf.jpg2014Novel colchicine-site binders with a cyclohexanedione scaffold identified through a ligand-based virtual screening approachCanela, María-Dolores CSIC; Peréz-Pérez, María-Jesús CSIC ORCID ; Noppen, Sam; Sáez-Calvo, Gonzalo CSIC; Díaz, José Fernando CSIC ORCID ; Camarasa Rius, María José CSIC ORCID; Liekens, Sandra; Priego, Eva María CSIC ORCIDartículo
openAccessProtein ligand complex.pdf.jpg23-ene-2018Protein-ligand complex for structure-based design: impact on the affinity and antitumor activity of new tubulin ligandsBueno, Oskia CSIC; Estévez-Gallego, Juan CSIC ORCID ; Martins, S.; Prota, Andrea E.; Gago, Federico CSIC ORCID; Gómez-SanJuan, Asier CSIC; Camarasa Rius, María José CSIC ORCID; Barasoain, Isabel CSIC ; Steinmetz, Michel O.; Díaz, José Fernando CSIC ORCID ; Liekens, Sandra; Peréz-Pérez, María-Jesús CSIC ORCID ; Priego, Eva María CSIC ORCIDcomunicación de congreso