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DerechosPreviewFecha Public.TítuloAutor(es)Tipo
openAccessASF7 revised manuscript 20190326.pdf.jpg2019Galloyl Carbohydrates with Antiangiogenic Activity Mediated by Capillary Morphogenesis Gene 2 (CMG2) Protein BindingDoyagüez, Elisa G. CSIC; Carrero, Paula CSIC; Madrona, Andrés CSIC ORCID; Rodríguez-Salamanca, Patricia CSIC ORCID; Martínez-Gualda, Belén CSIC; Camarasa Rius, María José CSIC ORCID; Jimeno, M. Luisa CSIC ORCID; Bennallack, P. R.; Finnell, J. G; Tsang, T. M.; Christensen, K. A.; San-Félix, Ana CSIC ORCID ; Rogers, M. S.artículo
closedAccess2014Heterocyclic Chemistry in Drug Discovery (Book review)Camarasa Rius, María José CSIC ORCIDartículo
openAccessScientific reports(2018)4242.pdf.jpg2018High-affinity ligands of the colchicine domain in tubulin based on a structure-guided designBueno, Oskia CSIC; Estévez-Gallego, Juan CSIC ORCID ; Martins, S.; Prota, Andrea E.; Gago, Federico CSIC ORCID; Gómez-SanJuan, Asier CSIC; Camarasa Rius, María José CSIC ORCID; Barasoain, Isabel CSIC ; Steinmetz, Michel O.; Díaz, José Fernando CSIC ORCID ; Peréz-Pérez, María-Jesús CSIC ORCID ; Liekens, Sandra; Priego, Eva María CSIC ORCIDartículo
openAccessene-2021HIV-1 Envelope Spike MPER: From a Vaccine Target to a New Druggable Pocket for Novel and Effective Fusion InhibitorsLuque, F. Javier; Camarasa Rius, María José CSIC ORCIDartículo
closedAccess2000HIV-1 specific reverse transcriptase inhibitors: Why are TSAO-nucleosides so unique?Camarasa Rius, María José CSIC ORCID; San-Felix, Alejandra; Peréz-Pérez, María-Jesús CSIC ORCID ; Velázquez, Sonsoles CSIC ORCID CVN; Álvarez, Rosa; Chamorro, Cristina CSIC; Jimeno, M. Luisa CSIC ORCID; Perez, Carlos; Gago, Federico CSIC ORCID; De Clercq, Erik; Balzarini, Janartículo
openAccessEuropean Journal of Medicinal Chemistry 244 (2022).pdf.jpg2022Identification of 1,2,3-triazolium salt-based inhibitors of Leishmania infantum trypanothione disulfide reductase with enhanced antileishmanial potency in cellulo and increased selectivityLucio, Héctor de; Revuelto, Alejandro CSIC ORCID; Carriles, Alejandra A. CSIC ORCID; Castro, Sonia de CSIC ORCID; García-González, Sonia; García-Soriano, Juan Carlos; Alcón-Calderón, Mercedes; Sánchez-Murcia, Pedro A. CSIC ORCID; Hermoso, Juan A. CSIC ORCID; Gago, Federico CSIC ORCID; Camarasa Rius, María José CSIC ORCID; Jiménez-Ruiz, Antonio; Velázquez, Sonsoles CSIC ORCID CVNartículo
closedAccess2014Identification of [1,2,3]triazolo[4,5-d ]pyrimidin-7(6H)-ones as novel inhibitors of chikungunya virus replicationGigante, Alba CSIC ORCID; Canela, María-Dolores CSIC; Delang, Leen; Priego, Eva María CSIC ORCID; Camarasa Rius, María José CSIC ORCID; Querat, Guilles; Neyts, Johan; Leyssen, Pieter; Peréz-Pérez, María-Jesús CSIC ORCID artículo
closedAccessaccesoRestringido.pdf.jpg2009Identification of aspartic acid-203 in human thymidine phosphorylase as an important residue for both catalysis and non-competitive inhibition by the small molecule >crystallization chaperone> 5′-O-tritylinosine (KIN59)Bronckaers, A.; Aguado, Leire CSIC; Negri, Ana; Camarasa Rius, María José CSIC ORCID; Balzarini, Jan; Peréz-Pérez, María-Jesús CSIC ORCID ; Gago, Federico CSIC ORCID; Liekens, S.artículo
openAccessEuropean Journal of Medicinal Chemistry 243 (2022).pdf.jpg2022Identification of L. infantum trypanothione synthetase inhibitors with leishmanicidal activity from a (non-biased) in-house chemical libraryAlcón-Calderón, Mercedes; Lucio, Héctor de; García-Soriano, Juan Carlos; Revuelto, Alejandro CSIC ORCID; Castro, Sonia de CSIC ORCID; López-Gutiérrez, Celia; San-Félix, Ana CSIC ORCID ; Quesada, Ernesto CSIC ORCID ; Gago, Federico CSIC ORCID; Camarasa Rius, María José CSIC ORCID; Jiménez-Ruiz, Antonio; Velázquez, Sonsoles CSIC ORCID CVNartículo
openAccessSV-EJMC 2017- preprint.pdf.jpg21-sep-2017Improved proteolytic stability and potent activity against Leishmania infantum trypanothione reductase of α/β-peptide foldamers conjugated to cell-penetrating peptidesLucio, Héctor de; Gamo, Ana María CSIC; Ruiz-Santaquiteria, Marta CSIC ORCID; Castro, Sonia de CSIC ORCID; Sánchez-Murcia, Pedro A. CSIC ORCID; Toro, Miguel Ángel; Gutiérrez, Kilian Jesús; Gago, Federico CSIC ORCID; Jiménez- Ruiz, Antonio; Camarasa Rius, María José CSIC ORCID; Velázquez, Sonsoles CSIC ORCID CVNartículo
openAccessWO2009030410A1.pdf.jpg12-mar-2009Improvements in or relating to compositions for the treatment or prophylaxis of viral infectionsBalzarini, Jan; Camarasa Rius, María José CSIC ORCID; Velázquez, Sonsoles CSIC ORCID CVNpatente
openAccessACS Infect Dis 2018.pdf.jpg2018Inhibition of the Replication of Different Strains of Chikungunya Virus by 3-Aryl-[1,2,3]triazolo[4,5- d] pyrimidin-7(6 H)-onesGómez-SanJuan, Asier CSIC; Gamo, Ana María CSIC; Delang, Leen; Pérez-Sánchez, Alfonso; Amrun, S. N.; Abdelnabi, Rana; Jacobs, S.; Priego, Eva María CSIC ORCID; Camarasa Rius, María José CSIC ORCID; Jochmans, D.; Leyssen, Pieter; Ng, L. F. P.; Querat, Guilles; Neyts, Johan; Peréz-Pérez, María-Jesús CSIC ORCID artículo
openAccesspharmaceuticals-14-01131-1.pdf.jpg6-nov-2021Inhibition of XPO-1 Mediated Nuclear Export through the Michael-Acceptor Character of ChalconesGargantilla, Marta CSIC ORCID; López-Fernández, José; Camarasa Rius, María José CSIC ORCID; Persoons, Leentje; Daelemans, Dirk; Priego, Eva María CSIC ORCID; Peréz-Pérez, María-Jesús CSIC ORCID artículo
openAccessijms-24-03539-v2.pdf.jpg10-feb-2023Insertion of an Amphipathic Linker in a Tetrapodal Tryptophan Derivative Leads to a Novel and Highly Potent Entry Inhibitor of Enterovirus A71 Clinical IsolatesMartí-Marí, Olaia CSIC ORCID; Abdelnabi, Rana; Schols, Dominique; Neyts, Johan; Camarasa Rius, María José CSIC ORCID; Gago, Federico CSIC ORCID; San-Félix, Ana CSIC ORCID artículo
openAccessmsystems.01459-21.pdf.jpg16-mar-2022Interrogation of Essentiality in the Reconstructed Haemophilus influenzae Metabolic Network Identifies Lipid Metabolism Antimicrobial Targets: Preclinical Evaluation of a FabH β-Ketoacyl-ACP Synthase InhibitorLópez-López, Nahikari CSIC ORCID; San León, David ; Castro, Sonia de CSIC ORCID; Díez-Martínez, Roberto CSIC ORCID; Iglesias-Bexiga, Manuel CSIC; Camarasa Rius, María José CSIC ORCID; Menéndez, Margarita CSIC ORCID; Nogales, Juan CSIC ORCID ; Garmendia, Juncal CSIC ORCID artículo
closedAccess2009Intramolecular Cation-π Interactions As the Driving Force To Restrict the Conformation of Certain NucleosidesCasanova, Elena; Priego, Eva María CSIC ORCID; Jimeno, M. Luisa CSIC ORCID; Aguado, Leire CSIC; Negri, Ana; Gago, Federico CSIC ORCID; Camarasa Rius, María José CSIC ORCID; Peréz-Pérez, María-Jesús CSIC ORCID artículo
openAccessPLoS ONE 9 (2014).pdf.jpg2014Leishmania infantum EndoG is an endo/exo-nuclease essential for parasite survivalRico, Eva; Oliva, Cristina; Gutiérrez, Kilian Jesús; Alzate, Juan Fernando; Genes, Carlos Mario; Moreno, David; Casanova, Elena CSIC; Gigante, Alba CSIC ORCID; Peréz-Pérez, María-Jesús CSIC ORCID ; Camarasa Rius, María José CSIC ORCID; Clos, Joachim; Gago, Federico CSIC ORCID; Jiménez-Ruiz, Antonioartículo
openAccessASF2Manuscript EJMECH-D-14-01438R2.pdf.jpg2015Linear and branched alkyl-esters and amides of gallic acid and other (mono-, di- and tri-) hydroxy benzoyl derivatives as promising anti-HCV inhibitorsRivero-Buceta, Eva CSIC ORCID; Carrero, Paloma CSIC; Doyagüez, Elisa G. CSIC; Madrona, Andrés CSIC ORCID; Quesada, Ernesto CSIC ORCID ; Camarasa Rius, María José CSIC ORCID; Peréz-Pérez, María-Jesús CSIC ORCID ; Leyssen, Pieter; Paeshuyse, Jan; Balzarini, Jan; Neyts, Johan; San-Félix, Ana CSIC ORCID artículo
closedAccessaccesoRestringido.pdf.jpg3-nov-2012Mechanism for VPg inhibition by FUTP in foot-and-mouth disease virusCastro, Sonia de CSIC ORCID; Ferrer-Orta, Cristina CSIC ORCID ; Fernández-Cureses, Gloria CSIC; Verdaguer, Núria CSIC ORCID ; Domingo, Esteban CSIC ORCID; Camarasa Rius, María José CSIC ORCIDpóster de congreso
closedAccessaccesoRestringido.pdf.jpg25-jun-2013Mechanism for VPg inhibition by FUTP in foot-and-mouth disease virusCastro, Sonia de CSIC ORCID; Ferrer-Orta, Cristina CSIC ORCID ; Fernández-Cureses, Gloria CSIC; Verdaguer, Núria CSIC ORCID ; Domingo, Esteban CSIC ORCID; Camarasa Rius, María José CSIC ORCIDpóster de congreso