Derechos | Preview | Fecha Public. | Título | Autor(es) | Tipo |
closedAccess | | 2008 | 4″-benzoylureido-TSAO derivatives as potent and selective non-nucleoside HCMV inhibitors. Structure-activity relationship and mechanism of antiviral action | Castro, Sonia de CSIC ORCID ; Peromingo, M. T.; Naesens, L.; Andrei, G.; Snoeck, R.; Balzarini, J.; Velázquez, Sonsoles CSIC ORCID CVN; Camarasa Rius, María José CSIC ORCID | artículo |
openAccess | | 2006 | Discovery of TSAO derivatives with an unusual HIV-1 activity/resistance profile | Castro, Sonia de CSIC ORCID ; García-Aparicio, Carlos CSIC; Van Laethem, K.; Gago, Federico CSIC ORCID; Lobatón, E.; De Clercq, E.; Balzarini, J.; Camarasa Rius, María José CSIC ORCID; Velázquez, Sonsoles CSIC ORCID CVN | artículo |
openAccess | | 2005 | Novel [2′,5′-Bis-O-(tert-butyldimethylsily)-β-D- ribofuranosyl]-3′-spiro-5″-(4″-amino-1″, 2″-oxathiole-2″,2″-diozide) derivatives with anti-HIV-1 and anti-human-cytomegalovirus activity | Castro, Sonia de CSIC ORCID ; Lobatón, E.; Peréz-Pérez, María-Jesús CSIC ORCID ; San-Félix, Ana CSIC ORCID ; Cordeiro, A.; Andrei, G.; Snoeck, R.; De Clercq, E.; Balzarini, J.; Camarasa Rius, María José CSIC ORCID; Velázquez, Sonsoles CSIC ORCID CVN | artículo |
closedAccess | | 2007 | NOVEL NON-NUCLEOSIDE HUMAN CYTOMEGALOVIRUS INHIBITORS BASED UPON TSAO NUCLEOSIDE DERIVATIVES:STRUCTURE-ACTIVITY RELATIONSHIPS | Castro, Sonia de CSIC ORCID ; Andrei, Graziela; Snoeck, Robert; Balzarini, Jan; Camarasa Rius, María José CSIC ORCID; Velázquez, Sonsoles CSIC ORCID CVN | artículo |
closedAccess | | 2008 | Reactivity of the 4-amino-5H-1,2-oxathiole-2,2-dioxide heterocyclic system: A combined experimental and theoretical study | Castro, Sonia de CSIC ORCID ; Peromingo, M. T.; Lozano, Ángel E. ; Camarasa Rius, María José CSIC ORCID; Velázquez, Sonsoles CSIC ORCID CVN | artículo |
closedAccess | | 2005 | The N137 and P140 amino acids in the p51 and the P95 amino acid in the p66 subunit of human immunodeficiency virus type 1 (HIV-1) reverse transcriptase are instrumental to maintain catalytic activity and to design new classes of anti-HIV-1 drugs | Auwerx, J.; Van Nieuwenhove, J.; Rodríguez-Barrios, F.; Castro, Sonia de CSIC ORCID ; Velázquez, Sonsoles CSIC ORCID CVN; Ceccherini-Silberstein, F.; De Clercq, E.; Camarasa Rius, María José CSIC ORCID; Perno, C.-F.; Gago, Federico CSIC ORCID; Balzarini, J. | artículo |
closedAccess | | 2006 | TSAO derivatives, inhibitors of HIV-1 reverse transcriptase dimerization: Recent progress | Camarasa Rius, María José CSIC ORCID; Velázquez, Sonsoles CSIC ORCID CVN; San-Félix, Ana CSIC ORCID ; Peréz-Pérez, María-Jesús CSIC ORCID ; Bonache, María-Cruz CSIC; Castro, Sonia de CSIC ORCID | artículo de revisión |
openAccess | | 2006 | Unprecedented lability of the 5′-O-tert-butyldimethylsilyl group from 3′-spiro-5″-(4″-acylamino-1″,2″-oxathiole- 2″,2″-dioxide) nucleoside derivatives via neighboring group participation of the 4″-acylamino residue | Castro, Sonia de CSIC ORCID ; Lozano López, Ángel Emilio CSIC ORCID ; Jimeno, M. Luisa CSIC ORCID; Peréz-Pérez, María-Jesús CSIC ORCID ; San-Félix, Ana CSIC ORCID ; Camarasa Rius, María José CSIC ORCID; Velázquez, Sonsoles CSIC ORCID CVN | artículo |