| | Derechos | Preview | Fecha Public. | Título | Autor(es) | Tipo |
| 1 | closedAccess | | 4-sep-2004 | 5-(tryptophylamino)-1,3-dioxoperhydropyrido[1,2-c]pyrimidine-based cholecystokinin receptor antagonists: Reversal of CCK1 receptor subtype selectivity toward CCK2 receptors | Muñoz, Pilar; García-López, M. Teresa CSIC ; Cenarruzabeitia, Edurne CSIC; Río, Joaquín del CSIC; Dufresne, Marlene; Foucaud, Magali; Fourmy, Daniel; Herranz, Rosario CSIC ORCID | artículo |
| 2 | closedAccess | | 1997 | 2,5-Diketopiperidine derivatives as non-peptide ligands for cholecystokinin receptors | González-Muñiz, Rosario CSIC ORCID; Domínguez, María José; Herranz, Rosario CSIC ORCID; García-López, M. Teresa CSIC ; Ballaz García, Santiago; Fortuño Gil, Alejandrona; Río, Joaquín del CSIC | artículo |
| 3 | closedAccess | | 2000 | New conformationally constrained tryptophans by N(α)-C(α)-cyclization to an azetidin-2-one core | Gerona-Navarro, Guillermo CSIC; Bonache de Marcos, María Ángeles CSIC ORCID; Herranz, Rosario CSIC ORCID; García-López, M. Teresa CSIC ; González-Muñiz, Rosario CSIC ORCID | artículo |
| 4 | closedAccess | | ene-1980 | Alkylating nucleosides. 3. The reaction of 3,5-dimethylpyrazole nucleosides with N-bromosuccinimide | García-López, M. Teresa CSIC ; Herranz, Rosario CSIC ORCID; Alonso, Gregorio | artículo |
| 5 | closedAccess | | ago-1991 | Synthesis of 5'-N-(α-amino-β-mercaptoacyl)amino-5'-deoxynucleosides as potential antiviral compounds | Herranz, Rosario CSIC ORCID; Castro-Pichel, J.; García-López, M. Teresa CSIC ; Pérez, Concepción CSIC ORCID; Balzarini, Jan; Clercq, Erik De | artículo |
| 6 | closedAccess | | 23-abr-1996 | CCK-4 restricted analogues containing a 3-oxoindolizidine skeleton | González-Muñiz, Rosario CSIC ORCID; Domínguez, María José; Martín-Martínez, Mercedes CSIC ORCID; Herranz, Rosario CSIC ORCID; García-López, M. Teresa CSIC ; Barber Cárcamo, Ana María; Ballaz García, Santiago; Río, Joaquín del CSIC | artículo |
| 7 | openAccess | | 1-jul-1998 | Derivados de 1,3-dioxoperhidropirido[1,2-c]pirimidinas como antagonistas de colecistoquinina | González-Muñiz, Rosario CSIC ORCID; García-López, M. Teresa CSIC ; Gómez-Monterrey, Isabel CSIC; Herranz, Rosario CSIC ORCID; Martín-Martínez, Mercedes CSIC ORCID; Barber Cárcamo, Ana María; Berjón San Juan, Angel; Fortuño Gil, Alejandrona; Ballaz García, Santiago; Río, Joaquín del CSIC | patente |
| 8 | openAccess | | 26-jul-2016 | Compuestos moduladores del sensor neuronal de calcio dream y sus usos terapéuticos | Gutiérrez-Rodríguez, Marta CSIC ORCID ; Cercós, Pilar CSIC; Martín-Martínez, Mercedes CSIC ORCID; Herranz, Rosario CSIC ORCID; García-López, M. Teresa CSIC ; Valenzuela, Carmen CSIC ORCID CVN; Naranjo, José Ramón CSIC ORCID; Mellström, Britt CSIC; Dopazo, Xose M.; González Pérez, Paz | patente |
| 9 | closedAccess | | 28-may-1993 | Stereospecific synthesis of (2R,3S)-3-amino-2-piperidineacetic acid derivatives for use as conformational constraint in peptides | Gómez-Monterrey, Isabel CSIC; González-Muñiz, Rosario CSIC ORCID; Herranz, Rosario CSIC ORCID; García-López, M. Teresa CSIC | artículo |
| 10 | openAccess | | 8-feb-2018 | Dream neuronal calcium sensor-modulating compounds, and therapeutic uses thereof | Gutiérrez-Rodríguez, Marta CSIC ORCID ; Cercós, Pilar CSIC; Martín-Martínez, Mercedes CSIC ORCID; Herranz, Rosario CSIC ORCID; García-López, M. Teresa CSIC ; Valenzuela, Carmen CSIC ORCID CVN; Naranjo, José Ramón CSIC ORCID; Mellström, Britt CSIC; Dopazo, Xose M.; González Pérez, Paz | solicitud de patente |
| 11 | openAccess | | 1-jun-1985 | Synthesis and antiviral evaluation of nucleosides of S-methylimidazole-4-carboxamide | Alonso, R.; Andrés, J. Ignacio; García-López, M. Teresa CSIC ; Heras, F. G. de las; Herranz, Rosario CSIC ORCID; Alarcón, Balbino CSIC ORCID; Carrasco, Luis | artículo |
| 12 | closedAccess | | 1-jun-1980 | Alkylating nucleosides. 4. Synthesis and cytostatic activity of chloro- and iodomethylpyrazole nucleosides | García-López, M. Teresa CSIC ; Domínguez, María José; Herranz, Rosario CSIC ORCID; Sanchez-Perez, Rosa M.; Contreras, Antonio; Alonso, Gregorio | artículo |
| 13 | closedAccess | | 1989 | Synthesis and antiviral activity of 5'-O-(substituted) sulfamoyl pyrimidine nucleosides | Castro-Pichel, J.; García-López, M. Teresa CSIC ; Herranz, Rosario CSIC ORCID; Pérez, Concepción CSIC ORCID; Vilas, Pilar | artículo |
| 14 | closedAccess | | 1991 | Synthesis of penicillamine- and cysteine-containing nucleoamino acids as potential antivirals and aminopeptidase B inhibitors | Herranz, Rosario CSIC ORCID; Castro-Pichel, J.; García-López, M. Teresa CSIC ; Pérez, Concepción CSIC ORCID; Balzarini, Jan; Clercq, Erik De | artículo |
| 15 | closedAccess | | 1983 | Studies on the synthesis of 2-bromomethylimidazole nucleosides related to AICA-riboside [5-amino-1-(β-D-ribofuranosyl)imidazole-4-carboxamide] | García-López, M. Teresa CSIC ; Herranz, Rosario CSIC ORCID; Andrés, J. Ignacio | artículo |
| 16 | openAccess | | 26-jul-2016 | Compuestos moduladores del sensor neuronal de calcio dream y sus usos terapéuticos | Gutiérrez-Rodríguez, Marta CSIC ORCID ; Cercós, Pilar CSIC; Martín-Martínez, Mercedes CSIC ORCID; Herranz, Rosario CSIC ORCID; García-López, M. Teresa CSIC ; Valenzuela, Carmen CSIC ORCID CVN; Naranjo, José Ramón CSIC ORCID; Mellström, Britt CSIC; Dopazo, Xose M.; González Pérez, Paz | solicitud de patente |
| 17 | closedAccess | | 16-dic-1991 | Synthesis of Ψ[CH(CN)NH] pseudopeptides. A new peptide bond surrogate | Herranz, Rosario CSIC ORCID; Suárez-Gea, M. Luisa CSIC; Vinuesa, Soledad CSIC; García-López, M. Teresa CSIC ; Martínez Gil, Ana CSIC ORCID | artículo |
| 18 | closedAccess | | 14-jul-2004 | Unprecedented stereospecific synthesis of a novel tetracyclic ring system, a hybrid of tetrahydropyrrolo[2,3-b]indole and tetrahydroimidazo[1,2-a]indole, via a domino reaction upon a tryptophan-derived amino nitrile | González-Vera, Juan A. CSIC ORCID; García-López, M. Teresa CSIC ; Herranz, Rosario CSIC ORCID | artículo |
| 19 | openAccess | | 1-jun-1985 | Un procedimiento para la preparación de derivados N-glicosídicos de alquilimidazoles | Herranz, Rosario CSIC ORCID; Andrés Gil, José Ignacio; García-López, M. Teresa CSIC ; Gómez de las Heras Martín-Maestro, Federico | patente |
| 20 | openAccess | | 2013 | Solvent-free synthesis of α-amino nitrile-derived ureas | Ventosa-Andrés, Pilar CSIC; González-Vera, Juan A. CSIC ORCID; García-López, M. Teresa CSIC ; Herranz, Rosario CSIC ORCID | artículo |
| 21 | closedAccess | | 2-may-2003 | Expedient one-pot synthesis of novel chiral 2-substituted 5-phenyl-1,4-benzodiazepine scaffolds from amino acid-derived amino nitriles | Herrero, Susana; García-López, M. Teresa CSIC ; Herranz, Rosario CSIC ORCID | artículo |
| 22 | closedAccess | | may-2000 | Studies on the synthesis of β-keto esters derived from dipeptides: Search for a low-epimerizing method | Patiño-Molina, Rosario; Martín-Martínez, Mercedes CSIC ORCID; Herranz, Rosario CSIC ORCID; García-López, M. Teresa CSIC ; González-Muñiz, Rosario CSIC ORCID | artículo |
| 23 | closedAccess | | 1992 | Aminopeptidase inhibitory properties and analgesic activity of (2S,3R)-3,7-diamino-2-hydroxy-heptanoic acid containing tripeptide analogues of the N-terminal tripeptide of probestin | Herranz, Rosario CSIC ORCID; Vinuesa, Soledad CSIC; Pérez, Concepción CSIC ORCID; García-López, M. Teresa CSIC ; Ceballos, María L. de CSIC ORCID; Murillo, Francisco M.; Río, Joaquín del CSIC | artículo |
| 24 | openAccess | | 11-dic-2020 | Compuestos moduladores del sensor neuronal de calcio DREAM y sus usos terapéuticos | Gutiérrez-Rodríguez, Marta CSIC ORCID ; Cercós, Pilar CSIC; Martín-Martínez, Mercedes CSIC ORCID; Herranz, Rosario CSIC ORCID; García-López, M. Teresa CSIC ; Valenzuela, Carmen CSIC ORCID CVN; Naranjo, José Ramón CSIC ORCID; Dopazo Santos, José Manuel; González Pérez, Paz | traducción de patente |
| 25 | closedAccess | | may-1987 | Analgesic dipeptide derivatives. II. Synthetic dipeptides containing a C-terminal 2-(2-nitrophenylsulfenyl) tryptophan residue | García-López, M. Teresa CSIC ; González-Muñiz, Rosario CSIC ORCID; Herranz, Rosario CSIC ORCID; Molinero, M. Teresa; Río, Joaquín del CSIC | artículo |
| 26 | closedAccess | | 2013 | Targeting the dream protein: new avenues for the search of drugs for neurodegenerative diseases | Cercós, Pilar CSIC; García-López, M. Teresa CSIC ; Herranz, Rosario CSIC ORCID; Martín-Martínez, Mercedes CSIC ORCID; Prieto, Ángela CSIC; Valenzuela, Carmen CSIC ORCID CVN; Naranjo, José Ramón CSIC ORCID; Gutiérrez-Rodríguez, Marta CSIC ORCID | póster de congreso |
| 27 | closedAccess | | 1995 | 2-Amino-3-oxohexahydroindolizino[8,7-b]indole-5-carboxylate derivatives as new scaffolds for mimicking β-turn secondary structures. Molecular dynamics and stereoselective synthesis | Figuera, Natalia De la CSIC; Alkorta, Ibon CSIC ORCID ; García-López, M. Teresa CSIC ; Herranz, Rosario CSIC ORCID; González-Muñiz, Rosario CSIC ORCID | artículo |
| 28 | closedAccess | | 18-oct-2001 | 5-(Tryptophyl)amino-1,3-dioxoperhydropyrido[1,2-c]pyrimidine-based potent and selective CCK1 receptor antagonists: Structure-activity relationship studies on the central 1,3-dioxoperhydropyrido[1,2-c]pyrimidine scaffold | Bartolomé-Nebreda, José M.; García-López, M. Teresa CSIC ; González-Muñiz, Rosario CSIC ORCID; Cenarruzabeitia, Edurne CSIC; Latorre, Miriam; Río, Joaquín del CSIC; Herranz, Rosario CSIC ORCID | artículo |
| 29 | openAccess | | 2012 | Design, synthesis and biological evaluation of new peptide-based ureas and thioureas as potential antagonists of the thrombin receptor PAR1 | Ventosa-Andrés, Pilar CSIC; Valdivielso, Ángel M. CSIC; Pappos, Ioannis; García-López, M. Teresa CSIC ; Tsopanoglou, Nikos E.; Herranz, Rosario CSIC ORCID | artículo |
| 30 | openAccess | | 2014 | Chameleonic reactivity of α-amino nitrile-derived ureas. Synthesis of highly functionalized imidazolidin-2-one and imidazolidine-2,4-dione derivatives | Ventosa-Andrés, Pilar CSIC; González-Verdejo, Juan A.; García-López, M. Teresa CSIC ; Herranz, Rosario CSIC ORCID | artículo |
| 31 | closedAccess | | 2007 | Strategies for design of non peptide CCK1R agonist/antagonist ligands | García-López, M. Teresa CSIC ; González-Muñiz, Rosario CSIC ORCID; Martín-Martínez, Mercedes CSIC ORCID; Herranz, Rosario CSIC ORCID | artículo de revisión |
| 32 | closedAccess | | 1999 | New scaffolds for peptidomimetics. Synthetic approaches towards 2,4- dioxooctahydropyrimido[1',6':1,2]pyrido[3,4-b]indole-6-carboxylic acid derivatives | Figuera, Natalia De la CSIC; García-López, M. Teresa CSIC ; Herranz, Rosario CSIC ORCID; González-Muñiz, Rosario CSIC ORCID | artículo |
| 33 | closedAccess | | 2015 | Dream-modulators for dreaming of novel drugs for neurodegenerative diseases | Cercós, Pilar CSIC; Peraza, Diego A. CSIC ORCID; Prieto, Ángela CSIC; González, Teresa CSIC ORCID; Mellström, Britt CSIC; García-López, M. Teresa CSIC ; Herranz, Rosario CSIC ORCID; Martín-Martínez, Mercedes CSIC ORCID; Valenzuela, Carmen CSIC ORCID CVN; Naranjo, José Ramón CSIC ORCID; Gutiérrez-Rodríguez, Marta CSIC ORCID | póster de congreso |
| 34 | closedAccess | | may-1995 | Constrained C-terminal hexapeptide neurotensin analogues containing a 3-oxoindolizidine skeleton | García-López, M. Teresa CSIC ; Alkorta, Ibon CSIC ORCID; Domínguez, María José; González-Muñiz, Rosario CSIC ORCID; Herranz, Rosario CSIC ORCID; Johansen, Nils L.; Madsen, Kjeld; Thøgersen, Henning; Suzdak, Peter | artículo |
| 35 | closedAccess | | 1993 | Ketomethylenebestatin: Synthesis and aminopeptidase inhibition | Herranz, Rosario CSIC ORCID; Castro-Pichel, J.; García-López, M. Teresa CSIC ; Gómez-Monterrey, Isabel CSIC; Pérez, Concepción CSIC ORCID; Vinuesa, Soledad CSIC | artículo |
| 36 | openAccess | | 30-jun-2016 | Dream neuronal calcium sensor-modulating compounds, and therapeutic uses thereof | Gutiérrez-Rodríguez, Marta CSIC ORCID ; Cercós, Pilar CSIC; Martín-Martínez, Mercedes CSIC ORCID; Herranz, Rosario CSIC ORCID; García-López, M. Teresa CSIC ; Valenzuela, Carmen CSIC ORCID CVN; Naranjo, José Ramón CSIC ORCID; Mellström, Britt CSIC; Dopazo, Xose M.; González Pérez, Paz | solicitud de patente |
| 37 | openAccess | | 2014 | Exploring the Phe-Gly Dipeptide-derived Piperazinone Scaffold in the search for Antagonists of the Thrombin receptor PAR1 | Valdivielso, Ángel M. CSIC; García-López, M. Teresa CSIC ; Gutiérrez-Rodríguez, Marta CSIC ORCID ; Herranz, Rosario CSIC ORCID | artículo |
| 38 | closedAccess | | 1996 | Synthesis of highly functionalized γ-lactam derivatives for use as conformational constraints in peptides | Martín-Martínez, Mercedes CSIC ORCID; García-López, M. Teresa CSIC ; Herranz, Rosario CSIC ORCID; González-Muñiz, Rosario CSIC ORCID | artículo |
| 39 | closedAccess | | 1995 | Ketomethylene and (Cyanomethy1ene)amino Pseudopeptide Analogues of the C-Terminal Hexapeptide of Neurotensin | González-Muñiz, Rosario CSIC ORCID; García-López, M. Teresa CSIC ; Gómez-Monterrey, Isabel CSIC; Herranz, Rosario CSIC ORCID; Jimeno, M. Luisa CSIC ORCID; Suárez-Gea, M. Luisa CSIC; Johansen, Nils L.; Madsen, Kjeld; Thøgersen, Henning | artículo |
| 40 | closedAccess | | 9-sep-2000 | β-Turned dipeptoids as potent and selective CCK1 receptor antagonists | Martín-Martínez, Mercedes CSIC ORCID; Figuera, Natalia De la CSIC; Latorre, Miriam; Herranz, Rosario CSIC ORCID; García-López, M. Teresa CSIC ; Cenarruzabeitia, Edurne CSIC; Río, Joaquín del CSIC; González-Muñiz, Rosario CSIC ORCID | artículo |
| 41 | closedAccess | | oct-2004 | Pharmacological study of IQM-97,423, a potent and selective CCK1 receptor antagonist with protective effect in experimental acute pancreatitis | Latorre, Miriam; Bartolomé-Nebreda, José M.; García-López, M. Teresa CSIC ; González-Muñiz, Rosario CSIC ORCID; Herranz, Rosario CSIC ORCID; Río, Joaquín del CSIC; Cenarruzabeitia, Edurne CSIC | artículo |
| 42 | closedAccess | | dic-2001 | Conformationally restricted PACAP27 analogues incorporating type II/II′ IBTM β-Turn mimetics. Synthesis, NMR structure determination, and binding affinity | González-Muñiz, Rosario CSIC ORCID; Martín-Martínez, Mercedes CSIC ORCID; Granata, Cesare; Oliveira, Eliandre de; Santiveri, Clara M. CSIC ORCID; González, Carlos CSIC; Frechilla, Diana; Herranz, Rosario CSIC ORCID; García-López, M. Teresa CSIC ; Río, Joaquín del CSIC; Jiménez, M. Angeles CSIC ORCID ; Andreu, David | artículo |
| 43 | closedAccess | | 1990 | 5'-O-[N-(aminoacyl)sulfamoyl]nucleosides. Synthesis and antiviral and cytostatic activities | Castro-Pichel, J.; García-López, M. Teresa CSIC ; Herranz, Rosario CSIC ORCID; Pérez, Concepción CSIC ORCID | artículo |
| 44 | closedAccess | | ene-2007 | Regioselective base-promoted nucleophilic ring opening of spirocyclic 2,6-dioxopiperazines: Synthesis of N-(1-carboxycyclohexyl)amino acid derivatives | González-Vera, Juan A. CSIC ORCID; García-López, M. Teresa CSIC ; Herranz, Rosario CSIC ORCID | artículo |
| 45 | closedAccess | | 1-mar-1990 | An improved one-pot method for the stereoselective synthesis of the (2S,3R)-3-amino-2-hydroxy acids: Key intermediates for bestatin and amastatin | Herranz, Rosario CSIC ORCID; Castro-Pichel, J.; Vinuesa, Soledad CSIC; García-López, M. Teresa CSIC | artículo |
| 46 | closedAccess | | 7-oct-1999 | 5-(Tryptophyl)amino-1,3-dioxoperhydropyrido[1,2-c]pyrimidine-based potent and selective CCK1 receptor antagonists: Structural modifications at the tryptophan domain | Bartolomé-Nebreda, José M.; Gómez-Monterrey, Isabel CSIC; García-López, M. Teresa CSIC ; González-Muñiz, Rosario CSIC ORCID; Martín-Martínez, Mercedes CSIC ORCID; Ballaz García, Santiago; Cenarruzabeitia, Edurne CSIC; Latorre, Miriam; Río, Joaquín del CSIC; Herranz, Rosario CSIC ORCID | artículo |
| 47 | closedAccess | | 30-sep-2004 | Synthesis, conformational analysis, and cytotoxicity of conformationally constrained aplidine and tamandarin A analogues incorporating a spirolactam β-turn mimetic | Gutiérrez-Rodríguez, Marta CSIC ORCID ; Martín-Martínez, Mercedes CSIC ORCID; García-López, M. Teresa CSIC ; Herranz, Rosario CSIC ORCID; Cuevas, Félix; Polanco, Concepción; Rodríguez-Campos, Ignacio; Manzanares, Ignacio; Cárdenas, Francisco; Feliz, Miguel; Lloyd-Williams, Paul; Giralt, Ernest | artículo |
| 48 | closedAccess | | 1-jul-1979 | Alkylating nucleosides. 2. Synthesis and cytostatic activity of bromomethylpyrazole and pyrazole nitrogen mustard nucleosides | García-López, M. Teresa CSIC ; Herranz, Rosario CSIC ORCID; Alonso, Gregorio | artículo |
| 49 | closedAccess | | 1986 | Antinociceptive effects in rodents of the dipeptide Lys-Trp (Nps) and related compounds | García-López, M. Teresa CSIC ; Herranz, Rosario CSIC ORCID; González-Muñiz, R.; Naranjo, José Ramón CSIC ORCID; Ceballos, María L. de CSIC ORCID; Río, Joaquín del CSIC | artículo |
| 50 | closedAccess | | 30-abr-2002 | 2-Oxopiperazine-based γ-turn conformationally constrained peptides: Synthesis of CCK-4 analogues | Herrero, Susana; García-López, M. Teresa CSIC ; Latorre, Julio; Cenarruzabeitia, Edurne CSIC; Río, Joaquín del CSIC; Herranz, Rosario CSIC ORCID | artículo |