Derechos | Preview | Fecha Public. | Título | Autor(es) | Tipo |
closedAccess | | 2014 | Choline kinase active site provides features for designing versatile inhibitors | Serrán-Aguilera, L.; Nuti, R.; López-Cara, Luisa C.; Ríos-Marco, Pablo; Carrasco, M.P.; Marco, C.; Entrena, Antonio; Macchiarulo, A.; Hurtado-Guerrero, Ramón CSIC ORCID | artículo |
openAccess | | 31-mar-2016 | Design, synthesis, crystallization and biological evaluation of new symmetrical biscationic compounds as selective inhibitors of human Choline Kinase α1 (ChoKα1) | Schiaffino-Ortega, Santiago; Baglioni, Eleonora; Mariotto, Elena; Bortolozzi, Roberta; Serran Aguilera, Lucia; Ríos Marco, Pablo; Carrasco-Jiménez, Maria Paz; Gallo, Miguel A.; Hurtado-Guerrero, Ramón CSIC ORCID; Marco, Carmen; Basso, Giuseppe; Viola, Giampietro; Entrena, Antonio; López-Cara, Luisa C. | artículo |
closedAccess | | 2013 | Determination of potential scaffolds for human choline kinase α1 by chemical deconvolution studies | Sahún-Roncero, M.; Rubio-Ruiz, B.; Conejo-García, A.; Velázquez-Campoy, Adrián; Entrena, Antonio; Hurtado-Guerrero, Ramón CSIC ORCID | artículo |
closedAccess | | 2014 | Discovery of a new binding site on human choline kinase α1: Design, synthesis, crystallographic studies, and biological evaluation of asymmetrical bispyridinium derivatives | Rubio-Ruiz, B.; Figuerola-Conchas, A.; Ramos-Torrecillas, J.; Capitán-Cañadas, F.; Ríos-Marco, P.; Carrasco, M.P.; Gallo, M.A.; Espinosa, A. CSIC ORCID; Marco, C.; Ruiz, C.; Entrena, Antonio; Hurtado-Guerrero, Ramón CSIC ORCID; Conejo-García, A. | artículo |
openAccess | | 1-jun-2015 | Pharmacophore-Based Virtual Screening to Discover New Active Compounds for Human Choline Kinase α1 | Serran Aguilera, Lucia; Nuti, Roberto; López-Cara, Luisa C.; Gallo Meza, Miguel Angel; Macchiarulo, Antonio; Entrena, Antonio; Hurtado-Guerrero, Ramón CSIC ORCID | artículo |
openAccess | | 2016 | Plasmodium falciparum Choline Kinase Inhibition Leads to a Major Decrease in Phosphatidylethanolamine Causing Parasite Death | Serrán-Aguilera, L.; Denton, H.; Rubio-Ruiz, B.; López-Gutiérrez, B.; Entrena, Antonio; Izquierdo, L.; Smith, T.K.; Conejo-García, A.; Hurtado-Guerrero, Ramón CSIC ORCID | artículo |
openAccess | | 9-abr-2013 | The mechanism of allosteric coupling in choline kinase α1 revealed by the action of a rationally designed inhibitor | Sahún-Roncero, M.; Rubio-Ruiz, B.; Saladino, Giorgio; Conejo-García, A.; Espinosa, Antonio; Velázquez-Campoy, Adrián; Gervasio, Francesco Luigi; Entrena, Antonio; Hurtado-Guerrero, Ramón CSIC ORCID | artículo |