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openAccessangewandtechemie_Nozal_2021.pdf.jpg24-jun-2021From kinase inhibitors to multitarget ligands as powerful drug leads for Alzheimer’s disease using protein-templated synthesisMartínez Gil, Ana CSIC ORCID ; Nozal, Vanesa CSIC ORCID; García-Rubia, Alfonso CSIC; Cuevas, Eva P. CSIC ORCID ; Pérez, Concepción CSIC ORCID; Palomo, Valle CSIC ORCID ; Tosat-Bitrian, Carlota CSIC ORCID ; Bartolomé Robledo, Fernando CSIC ORCID; Carro, Eva CSIC ORCID; Ramírez, Davidartículo
openAccesspharmaceuticals-14-00332-v3.pdf.jpg6-abr-2021Host-Directed FDA-Approved Drugs with Antiviral Activity against SARS-CoV-2 Identified by Hierarchical In Silico/In Vitro Screening MethodsGinex, Tiziana CSIC ORCID ; Garaigorta, Urtzi ; Ramírez, David; Castro, Victoria; Nozal, Vanesa CSIC ORCID; Maestro, Inés CSIC ORCID; Garcia-Carceles, Javier CSIC ORCID; Campillo, Nuria E. CSIC ORCID ; Martínez Gil, Ana CSIC ORCID ; Gastaminza, Pablo CSIC ORCID; Gil, Carmen CSIC ORCID artículo
openAccessHost-directed_Ginex.pdf.jpg26-nov-2020Host-directed FDA-approved drugs with antiviral activity against SARS-CoV-2 identified by hierarchical in silico/in vitro screening methodsGinex, Tiziana CSIC ORCID ; Garaigorta, Urtzi ; Ramírez, David; Castro, Victoria; Nozal, Vanesa CSIC ORCID; Maestro, Inés CSIC ORCID; Garcia-Carceles, Javier CSIC ORCID; Campillo, Nuria E. CSIC ORCID ; Martínez Gil, Ana CSIC ORCID ; Gastaminza, Pablo CSIC ORCID; Gil, Carmen CSIC ORCID preprint
openAccessijms_nozal_2021.pdf.jpg22-mar-2021Improved controlled release and brain penetration of the small molecule S14 using PLGA nanoparticlesNozal, Vanesa CSIC ORCID; Rojas-Prats, Elisa CSIC ORCID; Maestro, Inés CSIC ORCID; Gil, Carmen CSIC ORCID ; Pérez, Daniel I. CSIC ORCID; Martínez Gil, Ana CSIC ORCID artículo
openAccessAnal. Real Acad. Nal. Farm._Nozal_ 2019.pdf.jpg2019Improved linkage design for the discovery of multitarget ligands as powerful drugs for Alzheimer’s diseaseNozal, Vanesa CSIC ORCID; García-Rubia, Alfonso CSIC; Pérez, Concepción CSIC ORCID; Martínez Gil, Ana CSIC ORCID ; Palomo, Valle CSIC ORCID artículo
openAccesspharmaceutics_rojas-prats_2021.pdf.jpg28-ene-2021Increasing brain permeability of PHA-767491, a cell division cycle 7 kinase inhibitor, with biodegradable polymeric nanoparticlesRojas-Prats, Elisa CSIC ORCID; Tosat-Bitrian, Carlota CSIC ORCID ; Martínez-González, Loreto CSIC ORCID ; Nozal, Vanesa CSIC ORCID; Pérez, Daniel I. CSIC ORCID; Martínez Gil, Ana CSIC ORCID artículo
openAccessTesis_Vanesa_Nozal_Garcia_UCM.pdf.jpg7-abr-2022Modulación de la neurodegeneración con nuevas aproximaciones multidiana: diseño y síntesis de compuestos innovadoresNozal, Vanesa CSIC ORCIDtesis doctoral
openAccessCongreso Atenas p.110.pdf.jpgsep-2019Multitarget triazoles: an innovative approach for the treatment of Alzheimer’s diseaseNozal, Vanesa CSIC ORCID; García-Rubia, Alfonso CSIC; Roca, Carlos CSIC ORCID; Pérez, Concepción CSIC ORCID; Palomo, Valle CSIC ORCID ; Martínez Gil, Ana CSIC ORCID comunicación de congreso
openAccessAbstract_YRS_Nozal_2021.pdf.jpg18-jun-2021O2 Improved controlled release and brain penetration of small molecules with therapeutic potential using PLGA nanoparticlesNozal, Vanesa CSIC ORCID; Rojas-Prats, Elisa CSIC ORCID; Pérez, Daniel I. CSIC ORCID; Gil, Carmen CSIC ORCID ; Martínez Gil, Ana CSIC ORCID comunicación de congreso
openAccess2019Optimización de la estrategia de unión en el diseño de compuestos multidiana prometedores para el tratamiento de la enfermedad de AlzheimerNozal, Vanesa CSIC ORCID; García-Rubia, Alfonso CSIC; Pérez, Concepción CSIC ORCID; Martínez Gil, Ana CSIC ORCID ; Palomo, Valle CSIC ORCID artículo
openAccessAbstract_Pérez de la Lastra_YRS_2021.pdf.jpg18-jun-2021P34 Measuring protein aggregation in lymphoblasts from als patients with a turbidometric assayPérez de la Lastra, C. CSIC; Tosat-Bitrian, Carlota CSIC ORCID ; Nozal, Vanesa CSIC ORCID; Martínez Gil, Ana CSIC ORCID ; Martín-Requero, Ángeles CSIC ORCID ; Palomo, Valle CSIC ORCID comunicación de congreso
openAccess1-ago-2020Protein kinase inhibitors for amyotrophic lateral sclerosis therapyPalomo, Valle CSIC ORCID ; Nozal, Vanesa CSIC ORCID; Rojas-Prats, Elisa CSIC ORCID; Gil, Carmen CSIC ORCID ; Martínez Gil, Ana CSIC ORCID artículo
openAccess15-oct-2018Tau Tubulin Kinase 1 (TTBK1), a new player in the fight against neurodegenerative diseasesNozal, Vanesa CSIC ORCID; Martínez Gil, Ana CSIC ORCID artículo
openAccessWO2023281149A1.pdf.jpg12-ene-2023Tau-tubulin kinase (TTBK) inhibitor compoundsMartínez Gil, Ana CSIC ORCID ; Gil, Carmen CSIC ORCID ; Nozal, Vanesa CSIC ORCID; Palomo, Valle CSIC ORCID ; Martín-Requero, Ángeles CSIC ORCID ; Martínez-González, Loreto CSIC ORCID solicitud de patente
openAccess3-ene-2022TDP-43 modulation by Tau-Tubulin kinase 1 inhibitors: A new avenue for future amyotrophic lateral sclerosis therapyNozal, Vanesa CSIC ORCID; Martínez-González, Loreto CSIC ORCID ; Gómez-Almería, Marta; Gonzalo-Consuegra, Claudia; Santana, Paula; Chaikuad, Apirat; Cuevas, Eva P. CSIC ORCID ; Knapp, Stefan; Lietha, Daniel CSIC ORCID ; Ramírez, David; Petralla, Sabrina; Monti, B.; Gil, Carmen CSIC ORCID ; Martín-Requero, Ángeles CSIC ORCID ; Palomo, Valle CSIC ORCID ; De Lago, E.; Martínez Gil, Ana CSIC ORCID artículo
openAccessacs-cn_revised_2019.pdf.jpg20-mar-2019TDP-43: a key therapeutic target beyond amyotrophic lateral sclerosisPalomo, Valle CSIC ORCID ; Tosat-Bitrian, Carlota CSIC ORCID ; Nozal, Vanesa CSIC ORCID; Nagaraj, Siranjeevi; Martín-Requero, Ángeles CSIC ORCID ; Martínez Gil, Ana CSIC ORCID artículo
openAccessFrontiers in Molecular Neuroscience_Martinez-Gonzalez_2023.pdf.jpg9-ago-2023TTBK1 and CK1 inhibitors restore TDP-43 pathology and avoid disease propagation in lymphoblast from Alzheimer’s disease patientsMartínez-González, Loreto CSIC ORCID ; Cuevas, Eva P. CSIC ORCID ; Tosat-Bitrian, Carlota CSIC ORCID ; Nozal, Vanesa CSIC ORCID; Gil, Carmen CSIC ORCID ; Palomo, Valle CSIC ORCID ; Martín-Requero, Ángeles CSIC ORCID ; Martínez Gil, Ana CSIC ORCID artículo