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Derechos | Preview | Fecha Public. | Título | Autor(es) | Tipo |
openAccess | | 13-jun-2019 | Peptides Linked to Vpg1 of Foot-and-Mouth Disease Virus (FMDV): Design, Synthesis and X-Ray Crystallography of the Complexes with FMDV RNA-dependent RNA polymerase | Castro, Sonia de CSIC ORCID; Ferrer-Ortra, C.; Fernández-Cureses, Gloria CSIC; Verdaguer, Núria CSIC ORCID ; Camarasa Rius, María José CSIC ORCID | comunicación de congreso |
openAccess | | 2020 | Peptides mimicking the β7/β8 loop of HIV'1 reverse transcriptase p51 as “hotspot-targeted” dimerization inhibitors | Sánchez-Murcia, Pedro A. CSIC ORCID; Castro, Sonia de CSIC ORCID; García-Aparicio, Carlos CSIC; Jiménez, M. Angeles CSIC ORCID ; Corona, A.; Tramontano, Enzo; Sluis-Cremer, N.; Menéndez-Arias, Luis CSIC ORCID ; Velázquez, Sonsoles CSIC ORCID CVN; Gago, Federico CSIC ORCID; Camarasa Rius, María José CSIC ORCID | artículo |
openAccess | | 2018 | Polypharmacology in HIV inhibition: can a drug with simultaneous action against two relevant targets be an alternative to combination therapy? | Castro, Sonia de CSIC ORCID; Camarasa Rius, María José CSIC ORCID | artículo |
closedAccess | | 6-jun-2013 | Probing the Dimerization Interface of Leishmania infantum Trypanothione Reductase with Site-Directed Mutagenesis and Short Peptides | Toro, Miguel Ángel; Sánchez-Murcia, Pedro A. CSIC ORCID; Moreno, David; Ruiz-Santaquiteria, Marta CSIC ORCID; Alzate, Juan Fernando; Negri, Ana; Camarasa Rius, María José CSIC ORCID; Gago, Federico CSIC ORCID; Velázquez, Sonsoles CSIC ORCID CVN; Jiménez-Ruiz, Antonio | artículo |
openAccess | | 2018 | Prodrugs of Nucleoside Triphosphates as a Sound and Challenging Approach: A Pioneering Work That Opens a New Era in the Direct Intracellular Delivery of Nucleoside Triphosphates | Camarasa Rius, María José CSIC ORCID | artículo; preprint |
openAccess | | 18-nov-2004 | Produgs cleavable by CD26. | Balzarini, Jan; Camarasa Rius, María José CSIC ORCID; Velázquez, Sonsoles CSIC ORCID CVN | patente |
openAccess | | 23-ene-2018 | Protein-ligand complex for structure-based design: impact on the affinity and antitumor activity of new tubulin ligands | Bueno, Oskia CSIC; Estévez-Gallego, Juan CSIC ORCID ; Martins, S.; Prota, Andrea E.; Gago, Federico CSIC ORCID; Gómez-SanJuan, Asier CSIC; Camarasa Rius, María José CSIC ORCID; Barasoain, Isabel CSIC ; Steinmetz, Michel O.; Díaz, José Fernando CSIC ORCID ; Liekens, Sandra; Peréz-Pérez, María-Jesús CSIC ORCID ; Priego, Eva María CSIC ORCID | comunicación de congreso |
openAccess | | 2020 | Pseudoirreversible slow-binding inhibition of trypanothione reductase by a protein–protein interaction disruptor | Lucio, Héctor de; Toro, Miguel Ángel; Camarasa Rius, María José CSIC ORCID; Velázquez, Sonsoles CSIC ORCID CVN; Gago, Federico CSIC ORCID; Jimenez-Ruiz, Antonio | artículo |
openAccess | | 2019 | Pyrrolopyrimidine vs imidazole-phenyl-thiazole scaffolds in nonpeptidic dimerization inhibitors of leishmania infantum trypanothione reductase | Revuelto, Alejandro CSIC ORCID; Ruiz-Santaquiteria, Marta CSIC ORCID; Lucio, Héctor de; Gamo, Ana; Carriles, Alejandra A. CSIC ORCID; Gutiérrez, Kilian Jesús; Sánchez-Murcia, Pedro A. CSIC ORCID; Gago, Federico CSIC ORCID; Camarasa Rius, María José CSIC ORCID; Jiménez-Ruiz, Antonio; Velázquez, Sonsoles CSIC ORCID CVN | artículo |
closedAccess | | 2008 | Reactivity of the 4-amino-5H-1,2-oxathiole-2,2-dioxide heterocyclic system: A combined experimental and theoretical study | Castro, Sonia de CSIC ORCID ; Peromingo, M. T.; Lozano, Ángel E. ; Camarasa Rius, María José CSIC ORCID; Velázquez, Sonsoles CSIC ORCID CVN | artículo |
closedAccess | | 2012 | Recent Advances in Thymidine Kinase 2 (TK2) Inhibitors and New Perspectives for Potential Applications | Priego, Eva María CSIC ORCID; Karlsson, Anna; Gago, Federico CSIC ORCID; Camarasa Rius, María José CSIC ORCID; Balzarini, Jan; Peréz-Pérez, María-Jesús CSIC ORCID | artículo |
openAccess | | ene-2020 | Scaffold Simplification Strategy Leads to a Novel Generation of Dual Human Immunodeficiency Virus and Enterovirus-A71 Entry Inhibitors | Martínez-Gualda, Belén CSIC; Sun, Liang; Martí-Marí, Olaia CSIC ORCID; Abdelnabi, Rana; Noppen, Sam; Bator, Carol M.; Quesada, Ernesto CSIC ORCID ; Delang, Leen; Mirabelli, Carmen; Lee, Hyunwook; Schols, Dominique; Neyts, Johan; Hafenstein, Susan; Camarasa Rius, María José CSIC ORCID; Gago, Federico CSIC ORCID; San-Félix, Ana CSIC ORCID | artículo |
closedAccess | | 2001 | Second generation of TSAO compounds directed against HIV-1 TSAO-resistant strains | Lobaton, E.; Velázquez, Sonsoles CSIC ORCID CVN; Peréz-Pérez, María-Jesús CSIC ORCID ; Jimeno, M. Luisa CSIC ORCID; San-Felix, S.; De Clercq, Erik; Balzarini, Jan; Camarasa Rius, María José CSIC ORCID | artículo |
closedAccess | | 2008 | Selective human adenosine A3 antagonists based on pyrido[2,1-f]purine-2,4-diones: Novel features of hA3 antagonist binding | Priego, Eva María CSIC ORCID; Peréz-Pérez, María-Jesús CSIC ORCID ; Von Frijtag Drabbe Kuenzel, J. K.; de Vries, H.; Ijzerman, A. P.; Camarasa Rius, María José CSIC ORCID; Martín-Santamaría, Sonsoles CSIC ORCID | artículo |
openAccess | | 2011 | Selective inhibition of Human Immunodeficiency Virus type 1 (HIV-1) by a novel family of tricyclic nucleosides | Bonache, María-Cruz CSIC; Cordeiro, Alessandra CSIC; Quesada, Ernesto CSIC ORCID ; Vanstreels, Els; Daelemans, Dirk; Camarasa Rius, María José CSIC ORCID; Balzarini, Jan; San-Félix, Ana CSIC ORCID | artículo |
closedAccess | | 1982 | Síntesis, actividad citostática y mecanismo de acción de N-glicosil-halometilazoles. Un nuevo tipo de agentes alquilantes | Alonso, Gregorio; Alonso, R.; Camarasa Rius, María José CSIC ORCID; Contreras, Antonio; García-López, M. Teresa CSIC ; Heras, F. G. de las; Herranz, Rosario CSIC ORCID; Sanchez-Perez, Rosa M. | artículo |
openAccess | | 17-jul-2021 | Small Molecule–Peptide Conjugates as Dimerization Inhibitors of Leishmania infantum Trypanothione Disulfide Reductase | Revuelto, Alejandro CSIC ORCID; López-Martín, Isabel; Lucio, Héctor de; García-Soriano, Juan Carlos; Zanda, Nicola; Castro, Sonia de CSIC ORCID; Gago, Federico CSIC ORCID; Jiménez-Ruiz, Antonio; Velázquez, Sonsoles CSIC ORCID CVN; Camarasa Rius, María José CSIC ORCID | artículo |
closedAccess | | 2008 | Structure, physiological role, and specific inhibitors of human thymidine kinase 2 (TK2): Present and future | Peréz-Pérez, María-Jesús CSIC ORCID ; Priego, Eva María CSIC ORCID; Hernández, Ana-Isabel CSIC; Familiar, Olga CSIC; Camarasa Rius, María José CSIC ORCID; Negri, Ana; Gago, Federico CSIC ORCID; Balzarini, Jan | artículo |
openAccess | | 2017 | Structure-activity relationship studies on a Trp dendrimer with dual activities against HIV and enterovirus A71. Modifications on the amino acid | Martínez-Gualda, Belén CSIC; Sun, L.; Rivero-Buceta, Eva CSIC ORCID; Flores, Aida CSIC; Quesada, Ernesto CSIC ORCID ; Balzarini, Jan; Noppen, Sam; Liekens, Sandra; Schols, Dominique; Neyts, Johan; Leyssen, Pieter; Mirabelli, C.; Camarasa Rius, María José CSIC ORCID; San-Félix, Ana CSIC ORCID | artículo |
closedAccess | | 2-sep-2012 | Studies on the molecular basis for VPg inhibition by FUTP in foot-and-mouth disease virus | Castro, Sonia de CSIC ORCID; Ferrer-Orta, Cristina CSIC ORCID ; Fernández-Cureses, Gloria CSIC; Verdaguer, Núria CSIC ORCID ; Domingo, Esteban CSIC ORCID; Camarasa Rius, María José CSIC ORCID | póster de congreso |