Derechos | Preview | Fecha Public. | Título | Autor(es) | Tipo |
openAccess | | 20-may-2016 | Antivascular and antitumor properties of the tubulin-binding chalcone TUB091 | Canela, María-Dolores CSIC; Noppen, Sam; Bueno, Oskia CSIC; Prota, Andrea E.; Bargsten, Katja; Sáez-Calvo, Gonzalo CSIC; Jimeno, M. Luisa CSIC ORCID; Benkhei, Mohammed; Ribatti, Domenico; Velázquez, Sonsoles CSIC ORCID CVN; Camarasa Rius, María José CSIC ORCID; Díaz, José Fernando CSIC ORCID ; Steinmetz, Michel O.; Priego, Eva María CSIC ORCID; Peréz-Pérez, María-Jesús CSIC ORCID ; Liekens, Sandra | artículo |
openAccess | | 2015 | Evaluación de un nuevo quimiotipo de moduladores de tubulina del dominio de vinca | Sáez-Calvo, Gonzalo CSIC | tesis doctoral |
openAccess | | 2014 | Novel colchicine-site binders with a cyclohexanedione scaffold identified through a ligand-based virtual screening approach | Canela, María-Dolores CSIC; Peréz-Pérez, María-Jesús CSIC ORCID ; Noppen, Sam; Sáez-Calvo, Gonzalo CSIC; Díaz, José Fernando CSIC ORCID ; Camarasa Rius, María José CSIC ORCID; Liekens, Sandra; Priego, Eva María CSIC ORCID | artículo |
openAccess | | 22-jun-2017 | Quinolin-6-yloxyacetamides are microtubule destabilizing agents that bind to the colchicine site of tubulin | Sharma, Ashwani; Sáez-Calvo, Gonzalo CSIC; Olieric, Natacha; Balaguer, Francisco de Asís CSIC ORCID; Barasoain, Isabel CSIC ; Lamberth, Clemens; Díaz, José Fernando CSIC ORCID ; Steinmetz, Michel O. | artículo |
closedAccess | | 18-dic-2015 | Restoration of microtubule interaction and cytotoxicity in D-seco taxanes upon incorporation of 20-hydroxymethyl-4-allyloxy groups | Wang, Shao-Rong; Yang, Chun-Gang; Sánchez-Murcia, Pedro A. CSIC ORCID; Snyder, James P.; Yan, Ning; Sáez-Calvo, Gonzalo CSIC; Díaz, José Fernando CSIC ORCID ; Gago, Federico CSIC ORCID; Fang, Wei-Shuo | artículo |
closedAccess | | 2016 | Targeting the colchicine site in tubulin through cyclohexanedione derivatives | Canela, María-Dolores CSIC; Bueno, Oskia CSIC; Noppen, Sam; Sáez-Calvo, Gonzalo CSIC; Estévez-Gallego, Juan CSIC ORCID ; Díaz, José Fernando CSIC ORCID ; Camarasa Rius, María José CSIC ORCID; Liekens, Sandra; Peréz-Pérez, María-Jesús CSIC ORCID ; Priego, Eva María CSIC ORCID | artículo |
openAccess | | 22-jun-2017 | Triazolopyrimidines Are Microtubule-Stabilizing Agents that Bind the Vinca Inhibitor Site of Tubulin | Sáez-Calvo, Gonzalo CSIC; Balaguer, Francisco de Asís CSIC ORCID; Barasoain, Isabel CSIC ; Rodríguez-Salarichs, Javier CSIC; Muñoz-Hernández, Hugo CSIC ORCID; Berbís, Manuel Álvaro CSIC; Peñalva, Miguel Ángel CSIC ORCID ; Matesanz, Ruth CSIC ; Canales, Ángeles CSIC ORCID; Jiménez-Barbero, Jesús CSIC ORCID; Andreu, José Manuel CSIC ORCID ; Díaz, José Fernando CSIC ORCID | artículo |
openAccess | | 12-oct-2017 | Zampanolide binding to tubulin indicates crosstalk of taxane site with colchicine and nucleotide sites | Field, Jessica J.; Pera, Benet CSIC; Estévez-Gallego, Juan CSIC ORCID ; Rodríguez-Salarichs, Javier CSIC; Sáez-Calvo, Gonzalo CSIC; Andreu, José Manuel CSIC ORCID ; Díaz, José Fernando CSIC ORCID | artículo |