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| Rights | Preview | Issue Date | Title | Author(s) | Type |
| openAccess |  | 15-May-2019 | 4,4-Disubstituted N-benzylpiperidines: a novel class of fusion inhibitors of influenza virus H1N1 targeting a new binding site in hemagglutinin | Castro, Sonia de CSIC ORCID; Vanderlinden, E.; Ginex, Tiziana CSIC ORCID ; Laporte, M.; Stevaert, L.; Naesens, L.; Luque, F. Javier; Camarasa Rius, María José CSIC ORCID; Velázquez, Sonsoles CSIC ORCID CVN | comunicación de congreso |
| openAccess | | 26-Sep-2022 | A Novel and Versatile Class of Coronavirus non-covalent Mpro Inhibitors based on 1,4,4-Trisubstituted Piperidines | Maldonado, Miguel CSIC ORCID; De Castro, Sonia; Stevaert, Annelies; Delpal, Adrien; Vandeput, Julie; Van Loy, Benjamin; Eydoux, Cecilia; Guillemot, Jean-Claude; Decroly, Etienne; Canard, Bruno; Naesens, Lieve; Gago, Federico CSIC ORCID; Camarasa, María José; Velázquez, Sonsoles CSIC ORCID CVN | comunicación de congreso |
| openAccess |  | 2022 | A Versatile Class of 1,4,4-Trisubstituted Piperidines Block Coronavirus Replication In Vitro | Castro, Sonia de CSIC ORCID; Stevaert, Annelies; Maldonado, Miguel CSIC ORCID; Delpal, Adrien; Vandeput, Julie; Van Loy, Benjamin; Eydoux, Cecilia; Guillemot, Jean-Claude; Decroly, Etienne; Gago, Federico CSIC ORCID; Canard, Bruno; Camarasa Rius, María José CSIC ORCID; Velázquez, Sonsoles CSIC ORCID CVN; Naesens, Lieve | artículo |
| closedAccess | | 1998 | Abasic analogues of TSAO-T as the first sugar derivatives that specifically inhibit HIV-1 reverse transcriptase | Velázquez, Sonsoles CSIC ORCID CVN; Chamorro, Cristina CSIC; Peréz-Pérez, María-Jesús CSIC ORCID ; Álvarez, Rosa; Jimeno, M. Luisa CSIC ORCID; Martín Domenech, Angel; Pérez, Carlos; Gago, Federico CSIC ORCID; De Clercq, Erik; Balzarini, Jan; San-Félix, Ana CSIC ORCID CVN ; Camarasa Rius, María José CSIC ORCID | artículo |
| openAccess |  | 20-May-2016 | Antivascular and antitumor properties of the tubulin-binding chalcone TUB091 | Canela, María-Dolores CSIC; Noppen, Sam; Bueno, Oskia CSIC; Prota, Andrea E.; Bargsten, Katja; Sáez-Calvo, Gonzalo CSIC; Jimeno, M. Luisa CSIC ORCID; Benkhei, Mohammed; Ribatti, Domenico; Velázquez, Sonsoles CSIC ORCID CVN; Camarasa Rius, María José CSIC ORCID; Díaz, José Fernando CSIC ORCID ; Steinmetz, Michel O.; Priego, Eva María CSIC ORCID; Peréz-Pérez, María-Jesús CSIC ORCID ; Liekens, Sandra | artículo |
| openAccess |  | 2015 | Comparison of hydrocarbon-and lactam-bridged cyclic peptides as dimerization inhibitors of Leishmania infantum trypanothione reductase | Sánchez-Murcia, Pedro A. CSIC ORCID; Ruiz-Santaquiteria, Marta CSIC ORCID; Toro, Miguel Ángel; Lucio, H. de; Jiménez, M. Angeles CSIC ORCID ; Gago, Federico CSIC ORCID; Jiménez-Ruiz, Antonio; Camarasa Rius, María José CSIC ORCID; Velázquez, Sonsoles CSIC ORCID CVN | artículo |
| closedAccess | | 2011 | Dipeptidyl peptidase IV dependent water-soluble prodrugs of highly lipophilic bicyclic nucleoside analogues | Diez-Torrubia, Alberto CSIC; Balzarini, Jan; Andrei, G; Snoeck, R.; De Meester, Ingrid; Camarasa Rius, María José CSIC ORCID; Velázquez, Sonsoles CSIC ORCID CVN | artículo |
| closedAccess | | 2012 | Dipeptidyl Peptidase IV-Activated Prodrugs of Anti- Varicella Zoster Virus Bicyclic Nucleoside Analogues Containing Different Self-Cleavage Spacer Systems | Diez-Torrubia, Alberto CSIC; Cabrera, Silvia CSIC ORCID; De Meester, Ingrid; Camarasa Rius, María José CSIC ORCID; Balzarini, Jan; Velázquez, Sonsoles CSIC ORCID CVN | artículo |
| openAccess |  | 2015 | Dipeptidyl-peptidase IV (DPP IV/CD26)-activated prodrugs: A successful strategy for improving water solubility and oral bioavailability | Velázquez, Sonsoles CSIC ORCID CVN; Castro, Sonia de CSIC ORCID; Diez-Torrubia, Alberto CSIC; Balzarini, Jan; Camarasa Rius, María José CSIC ORCID | artículo |
| closedAccess | | 3-Feb-2012 | Dipeptidyl-peptidase IV (DPPIV/CD26)-based prodrugs of hydroxy-containing drugs | Diez-Torrubia, Alberto CSIC; Cabrera, Silvia CSIC ORCID; Lambeir, Anne-Marie; Balzarini, Jan; Camarasa Rius, María José CSIC ORCID; Velázquez, Sonsoles CSIC ORCID CVN | artículo |
| closedAccess |  | 2014 | Discovery and SAR studies of a novel class of cytotoxic 1,4-disubstituted piperidines via Ugi reaction | Castro, Sonia de CSIC ORCID; Camarasa Rius, María José CSIC ORCID; Balzarini, Jan; Velázquez, Sonsoles CSIC ORCID CVN | artículo |
| openAccess |  | 2014 | Diseño y desarrollo de una novedosa estrategia profármaco basada en la enzima DPPIV/CD26 | Camarasa Rius, María José CSIC ORCID; Castro, Sonia de CSIC ORCID; Velázquez, Sonsoles CSIC ORCID CVN | artículo |
| openAccess |  | 2021 | Efficient Dimerization Disruption of Leishmania infantum Trypanothione Reductase by Triazole-phenyl-thiazoles | Revuelto, Alejandro CSIC ORCID; Lucio, Héctor de; García-Soriano, Juan Carlos; Sánchez-Murcia, Pedro A. CSIC ORCID; Gago, Federico CSIC ORCID; Jiménez-Ruiz, Antonio; Camarasa Rius, María José CSIC ORCID; Velázquez, Sonsoles CSIC ORCID CVN | artículo |
| openAccess |  | 2017 | First example of peptides targeting the dimer interface of Leishmania infantum trypanothione reductase with potent in vitro antileishmanial activity# | Ruiz-Santaquiteria, Marta CSIC ORCID; Sánchez-Murcia, Pedro A. CSIC ORCID; Toro, Miguel Ángel; Lucio, H. de; Gutiérrez, Kilian Jesús; Castro, Sonia de CSIC ORCID; Carneiro, Filipa A. C.; Gago, Federico CSIC ORCID; Jiménez-Ruiz, Antonio; Camarasa Rius, María José CSIC ORCID; Velázquez, Sonsoles CSIC ORCID CVN | artículo |
| closedAccess | | 2011 | From β-Amino-γ-sultone to Unusual Bicyclic Pyridine and Pyrazine Heterocyclic Systems: Synthesis and Cytostatic and Antiviral Activities | Castro, Sonia de CSIC ORCID; Familiar, Olga CSIC; Andrei, G; Snoeck, R.; Balzarini, Jan; Camarasa Rius, María José CSIC ORCID; Velázquez, Sonsoles CSIC ORCID CVN | artículo |
| closedAccess | | 2000 | HIV-1 specific reverse transcriptase inhibitors: Why are TSAO-nucleosides so unique? | Camarasa Rius, María José CSIC ORCID; San-Felix, Alejandra; Peréz-Pérez, María-Jesús CSIC ORCID ; Velázquez, Sonsoles CSIC ORCID CVN; Álvarez, Rosa; Chamorro, Cristina CSIC; Jimeno, M. Luisa CSIC ORCID; Perez, Carlos; Gago, Federico CSIC ORCID; De Clercq, Erik; Balzarini, Jan | artículo |
| openAccess |  | 2022 | Identification of 1,2,3-triazolium salt-based inhibitors of Leishmania infantum trypanothione disulfide reductase with enhanced antileishmanial potency in cellulo and increased selectivity | Lucio, Héctor de; Revuelto, Alejandro CSIC ORCID; Carriles, Alejandra A. CSIC ORCID; Castro, Sonia de CSIC ORCID; García-González, Sonia; García-Soriano, Juan Carlos; Alcón-Calderón, Mercedes; Sánchez-Murcia, Pedro A. CSIC ORCID; Hermoso, Juan A. CSIC ORCID; Gago, Federico CSIC ORCID; Camarasa Rius, María José CSIC ORCID; Jiménez-Ruiz, Antonio; Velázquez, Sonsoles CSIC ORCID CVN | artículo |
| openAccess |  | 2022 | Identification of L. infantum trypanothione synthetase inhibitors with leishmanicidal activity from a (non-biased) in-house chemical library | Alcón-Calderón, Mercedes; Lucio, Héctor de; García-Soriano, Juan Carlos; Revuelto, Alejandro CSIC ORCID; Castro, Sonia de CSIC ORCID; López-Gutiérrez, Celia; San-Félix, Ana CSIC ORCID CVN ; Quesada, Ernesto CSIC ORCID ; Gago, Federico CSIC ORCID; Camarasa Rius, María José CSIC ORCID; Jiménez-Ruiz, Antonio; Velázquez, Sonsoles CSIC ORCID CVN | artículo |
| openAccess |  | 21-Sep-2017 | Improved proteolytic stability and potent activity against Leishmania infantum trypanothione reductase of α/β-peptide foldamers conjugated to cell-penetrating peptides | Lucio, Héctor de; Gamo, Ana María CSIC; Ruiz-Santaquiteria, Marta CSIC ORCID; Castro, Sonia de CSIC ORCID; Sánchez-Murcia, Pedro A. CSIC ORCID; Toro, Miguel Ángel; Gutiérrez, Kilian Jesús; Gago, Federico CSIC ORCID; Jiménez- Ruiz, Antonio; Camarasa Rius, María José CSIC ORCID; Velázquez, Sonsoles CSIC ORCID CVN | artículo |
| openAccess |  | 12-Mar-2009 | Improvements in or relating to compositions for the treatment or prophylaxis of viral infections | Balzarini, Jan; Camarasa Rius, María José CSIC ORCID; Velázquez, Sonsoles CSIC ORCID CVN | patente |
