Derechos | Preview | Fecha Public. | Título | Autor(es) | Tipo |
closedAccess | | 14-jun-2011 | Corrigendum: Mechanism of Action of the Cytotoxic Macrolides Amphidinolide X and J | Trigili, Chiara CSIC; Pera, Benet CSIC; Barbazanges, Marion; Cossy, Janine; Meyer, Christophe; Pineda, Oriol; Rodríguez-Escrich, Carles; Urpí, Félix; Vilarrasa, Jaume; Díaz, José Fernando CSIC ORCID ; Barasoain, Isabel CSIC | corrigenda |
closedAccess | | may-2011 | Design and Synthesis of Pironetin Analogues with Simplified Structure and Study of Their Interactions with Microtubules | Marco, J. Alberto; García-Pla, Jorge; Carda, Miguel; Murga, Juan; Falomir, Eva; Trigili, Chiara CSIC; Notararigo, Sara CSIC ORCID; Díaz, José Fernando CSIC ORCID ; Barasoain, Isabel CSIC | artículo |
closedAccess | | 15-ago-2011 | Effects of C7 Substitutions in a High Affinity Microtubule-Binding Taxane on Antitumor Activity and Drug Transport | Xiao, Xi; Wu, Ju; Trigili, Chiara CSIC; Chen, Hui; Chu, Joseph W.K.; Zhao, Ying; Lu, Peihua; Sheng, Li; Li, Yan; Sharom, Frances J.; Barasoain, Isabel CSIC ; Díaz, José Fernando CSIC ORCID ; Fang, Wei-Shuo | artículo |
openAccess | | 2013 | Estudio y caracterización del mecanismo de acción bioquímico y celular de compuestos antitumorales dirigidos contra el citoesqueleto | Trigili, Chiara CSIC | tesis doctoral |
closedAccess | | may-2011 | Highly Stereoselective Total Synthesis of (+)-9-epi-Dictyostatin and (–)-12,13-bis-epi-Dictyostatin Eur. J | Zanato, Chiara; Pignataro, Luca; Ambrosi, Andrea; Hao, Zhongyan; Trigili, Chiara CSIC; Díaz, José Fernando CSIC ORCID ; Barasoain, Isabel CSIC ; Gennari, Cesare | artículo |
openAccess | | 19-ago-2011 | Insights into the interaction of discodermolide and docetaxel with tubulin. Mapping the binding sites of microtubule-stabilizing agents by using an integrated NMR and computational approach | Canales, Ángeles CSIC ORCID; Rodríguez-Salarichs, Javier CSIC; Trigili, Chiara CSIC; Nieto, Lidia CSIC; Coderch, Claire; Andreu, José Manuel CSIC ORCID ; Paterson, Ian; Jiménez-Barbero, Jesús CSIC ORCID; Díaz, José Fernando CSIC ORCID | artículo |
closedAccess | | 1-jun-2011 | Mecanismo de accion de los macrolidos citotoxicos amphinolidas X y J | Trigili, Chiara CSIC; Pera, Benet CSIC; Barbazanges, Marion; Cossy, Janine; Meyer, Christophe; Pineda, Oriol; Rodríguez-Escrich, Carles; Urpí, Félix; Vilarrasa, Jaume; Díaz, José Fernando CSIC ORCID ; Barasoain, Isabel CSIC | póster de congreso |
closedAccess | | 2-may-2011 | Mechanism of Action of Cytotoxic Macrolides Amphidinolide X and J. | Trigili, Chiara CSIC; Pera, Benet CSIC; Barbazanges, Marion; Cossy, Janine; Meyer, Christophe; Pineda, Oriol; Rodríguez-Escrich, Carles; Urpí, Félix; Vilarrasa, Jaume; Díaz, José Fernando CSIC ORCID ; Barasoain, Isabel CSIC | artículo |
closedAccess | | 16-ago-2010 | Molecular recognition of peloruside A by microtubules. The C24 primary alcohol is essential for biological activity. | Pera, Benet CSIC; Razzak, Mina; Trigili, Chiara CSIC; Pineda, Oriol; Canales, Ángeles CSIC ORCID; Martínez Buey, Rubén CSIC ORCID; Jiménez-Barbero, Jesús CSIC ORCID; Northcote, Peter; Paterson, Ian; Barasoain, Isabel CSIC ; Díaz, José Fernando CSIC ORCID | artículo |
closedAccess | | 26-mar-2010 | Probing the Pore Drug Binding Site of Microtubules with Fluorescent Taxanes: Evidence of Two Binding Poses | Barasoain, Isabel CSIC ; García-Carril, Ana M.; Matesanz, Ruth CSIC ; Maccari, Giorgio; Trigili, Chiara CSIC; Mori, Mattia; Shi, Jing-Zhe; Fang, Wei-Shuo; Andreu, José Manuel CSIC ORCID ; Botta, Maurizio; Díaz, José Fernando CSIC ORCID | artículo |
openAccess | | 13-dic-2016 | Structural Determinants of the Dictyostatin Chemotype for Tubulin Binding Affinity and Antitumor Activity Against Taxane- and Epothilone-Resistant Cancer Cells | Trigili, Chiara CSIC; Barasoain, Isabel CSIC ; Sánchez-Murcia, Pedro A. CSIC ORCID; Bargsten, Katja; Redondo-Horcajo, Mariano CSIC ORCID ; Nogales, Aurora CSIC ORCID; Gardner, Nicola M.; Meyer, Arndt; Naylor, Guy J.; Gomez-Rubio, Elena CSIC ORCID; Gago, Federico CSIC ORCID; Steinmetz, Michel O.; Paterson, Ian; Prota, Andrea E.; Díaz, José Fernando CSIC ORCID | artículo |
closedAccess | | nov-2012 | Structure-activity relationships of novel substituted naphthalene diimides as anticancer agents | Milelli, Andrea; Tumiatti, Vicenzo; Micco, Marialuisa; Rosini, Michela; Zuccari, Guendalina; Raffaghello, Lizzia; Bianchi, Giovanna; Pistoia, Vito; Pistoia, Vito; Díaz, José Fernando CSIC ORCID ; Díaz, José Fernando CSIC ORCID ; Pera, Benet CSIC; Trigili, Chiara CSIC; Barasoain, Isabel CSIC ; Musetti, Caterina; Toniolo, Marianna; Sissi. Claudia; Alcaro, Stefano; Moraca, Federica; Zini, Maddalena; Stefanelli, Claudio; Minarini, Anna | artículo |
closedAccess | | 21-may-2012 | Synthesis and Antimitotic and Tubulin Interaction Profiles of Novel Pinacol Derivatives of Podophyllotoxins | Abad, Andrés; López-Pérez, José Luis; Olmo, Esther del; García-Fernández, Luis F. CSIC; Francesch, Andrés; Trigili, Chiara CSIC; Barasoain, Isabel CSIC ; Andreu, José Manuel CSIC ORCID ; Díaz, José Fernando CSIC ORCID ; San Feliciano, Arturo | artículo |
closedAccess | | 28-feb-2013 | Synthesis and biological evaluation as microtubule-active agents of several tetrahydrofuran and spiroacetal derivatives | Carda, Miguel; Murga, Juan; Paños, Julián; Angulo-Pachón, C.A.; García-Pla, Jorge; Díaz-Oltra, Santiago; Marco, J. Alberto; Trigili, Chiara CSIC; Redondo-Horcajo, Mariano CSIC ORCID ; Díaz, José Fernando CSIC ORCID ; Barasoain, Isabel CSIC | artículo |
closedAccess | | feb-2013 | Synthesis and Biological Evaluation of α-Tubulin-Binding Pironetin Analogues with Enhanced Lipophilicity | Carda, Miguel; Murga, Juan; Díaz-Oltra, Santiago; García-Pla, Jorge; Paños, Julián; Falomir, Eva; Trigili, Chiara CSIC; Díaz, José Fernando CSIC ORCID ; Barasoain, Isabel CSIC ; Marco, J. Alberto | artículo |
openAccess | | 19-jun-2014 | Taxanes with high potency inducing tubulin assembly overcome tumoural cell resistances | Matesanz, Ruth CSIC ; Trigili, Chiara CSIC; Rodríguez-Salarichs, Javier CSIC; Pera, Benet CSIC; Jiménez-Barbero, Jesús CSIC ORCID; Canales, Ángeles CSIC ORCID; Barasoain, Isabel CSIC ; Díaz, José Fernando CSIC ORCID | artículo |
closedAccess | | 1-jun-2011 | Zampanolida, un novedoso agente estabilizador de microtubulos quew se une covalentemente al sitio de paclitaxel | Field, Jessica J.; Pera, Benet CSIC; Canales, Ángeles CSIC ORCID; Zuwerra, D.; Trigili, Chiara CSIC; Kanakkanthara, Arun; Wakefield, St. John; Singh, A. Jonathan; Jiménez-Barbero, Jesús CSIC ORCID; Northcote, Peter; Miller, J.; López, Juan Antonio; Hamel, Ernest; Barasoain, Isabel CSIC ; Altmann, Karl-Heinz; Díaz, José Fernando CSIC ORCID | póster de congreso |
openAccess | | 22-jun-2012 | Zampanolide, a potent new microtubule stabilizing agent, covalently reacts with the taxane luminal site in both tubulin alpha-beta-heterodimers and microtubules | Field, Jessica J.; Pera, Benet CSIC; Calvo, Enrique; Canales, Ángeles CSIC ORCID; Zurwerra, Didier; Trigili, Chiara CSIC; Rodríguez-Salarichs, Javier CSIC; Matesanz, Ruth CSIC ; Kanakkanthara, Arun; Wakefield, St. John; Singh, A. Jonathan; Jiménez-Barbero, Jesús CSIC ORCID; Northcote, Peter; Miller, John H.; López, Juan Antonio; Hamel, Ernest; Barasoain, Isabel CSIC ; Altmann, Karl-Heinz; Díaz, José Fernando CSIC ORCID | artículo |