Rights | Preview | Issue Date | Title | Author(s) | Type |
openAccess |  | 20-May-2016 | Antivascular and antitumor properties of the tubulin-binding chalcone TUB091 | Canela, María-Dolores ; Noppen, Sam; Bueno, Oskía; Prota, Andrea E.; Bargsten, Katja; Sáez-Calvo, Gonzalo; Jimeno, M. Luisa ; Benkhei, Mohammed; Ribatti, Domenico; Velázquez, Sonsoles ; Camarasa Rius, María José ; Díaz, José Fernando ; Steinmetz, Michel O.; Priego, Eva María ; Peréz-Pérez, María-Jesús ; Liekens, Sandra | artículo |
openAccess |  | 20-Mar-2019 | Crystal Structure of the Cyclostreptin-Tubulin Adduct: Implications for Tubulin Activation by Taxane-Site Ligands | Balaguer, Francisco de Asís; Mühlethaler, Tobias; Estévez-Gallego, Juan ; Calvo, Enrique; Giménez-Abián, Juan F. ; Risinger, April L.; Sorensen, Erik J.; Vanderwal, Christopher D.; Altmann, Karl-Heinz; Mooberry, Susan; Steinmetz, Michel O.; Oliva, María A. ; Prota, Andrea E.; Díaz, José Fernando | artículo |
openAccess |  | 2018 | High-affinity ligands of the colchicine domain in tubulin based on a structure-guided design | Bueno, Oskía; Estévez-Gallego, Juan ; Martins, S.; Prota, Andrea E.; Gago, Federico ; Gómez-SanJuan, Asier; Camarasa Rius, María José ; Barasoain, Isabel ; Steinmetz, Michel O.; Díaz, Fernando J.; Peréz-Pérez, María-Jesús ; Liekens, Sandra; Priego, Eva María  | artículo |
closedAccess |  | 1-Feb-2013 | Molecular Mechanism of Action of Microtubule-Stabilizing Anticancer Agents | Prota, Andrea E.; Bargsten, Katja; Zurwerra, Didier; Field, Jessica J.; Díaz, José Fernando ; Altmann, Karl-Heinz; Steinmetz, Michel O. | artículo |
openAccess |  | 31-Jul-2016 | Pironetin binds covalently to Cys316 and perturbs a major loop and helix of -tubulin to inhibit microtubule formation | Prota, Andrea E.; Setter, J.; Waight, Andrew B.; Bargsten, Katja; Murga, Juan; Díaz, José Fernando ; Steinmetz, Michel O. | artículo |
openAccess |  | 22-Nov-2019 | Structural basis of colchicine-site targeting acylhydrazones active against multidrug-resistant acute lymphoblastic leukemia | Cury, Nathália Moreno; Mühlethaler, Tobias; Laranjeira, Angelo Brunelli Albertoni; Canevarolo, Rafael Renatino; Zenatti, Priscila Pini; Lucena-Agell, Daniel ; Barasoain, Isabel ; Song, Chunhua; Sun,Dongxiao; Dovat, Sinisa; Yunes, Rosendo Augusto; Prota, Andrea E.; Steinmetz, Michel O.; Díaz, José Fernando ; Yunes, José Andrés | artículo |
embargoedAccess |  | 13-Jul-2020 | Structural basis of noscapine activation for tubulin binding | Oliva, María A. ; Prota, Andrea E.; Rodríguez-Salarichs, Javier; Wenxin, Gu; Bennani, Y. L.; Jiménez-Barbero, Jesús ; Bargsten, Katja; Canales, Ángeles ; Steinmetz, Michel O.; Díaz, José Fernando | artículo |
openAccess |  | 10-Mar-2020 | Structural model for differential cap maturation at growing microtubule ends | Estévez-Gallego, Juan ; Josa-Prado, Fernando; Ku, Siou; Martínez Buey, Rubén ; Balaguer, Francisco de Asís; Prota, Andrea E.; Lucena-Agell, Daniel ; Kamma-Lorger, C.S.; Yagi, Toshiki; Iwamoto, Hiroyuki; Duchesne, Laurence; Barasoain, Isabel ; Steinmetz, Michel O.; Chrétien, Denis; Kamimura, Shinji; Díaz, José Fernando ; Oliva, María A. | artículo |