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Browsing by Author Priego, Eva María

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RightsPreviewIssue DateTitleAuthor(s)Type
closedAccess20109-Arylpurines as a Novel Class of Enterovirus InhibitorsAguado, Leire CSIC; Thibaut, Hendrik Jan; Priego, Eva María CSIC ORCID; Jimeno, M. Luisa CSIC ORCID; Camarasa Rius, María José CSIC ORCID; Neyts, Johan; Peréz-Pérez, María-Jesús CSIC ORCID artículo
closedAccess2002A new and efficient one-pot synthesis of pyrido[2,1-f]purine-2,4-diones starting from 6-aminouracil derivativesPérez Pérez, María Jesús; Priego, Eva María CSIC ORCID; Jimeno, M. Luisa CSIC ORCID; Camarasa Rius, María José CSIC ORCIDartículo
openAccessijms-23-13935-v2.pdf.jpg2022Allosteric Inhibition of Neutral Sphingomyelinase 2 (nSMase2) by DPTIP: From Antiflaviviral Activity to Deciphering Its Binding Site through In Silico Studies and Experimental ValidationÁlvarez-Fernández, Hadrián; Mingo-Casas, Patricia; Blázquez, Ana-Belén; Caridi, Flavia CSIC ORCID; Saiz, Juan Carlos; Peréz-Pérez, María-Jesús CSIC ORCID ; Martín-Acebes,Miguel A.; Priego, Eva María CSIC ORCIDartículo
openAccessOncotarget.pdf.jpg20-May-2016Antivascular and antitumor properties of the tubulin-binding chalcone TUB091Canela, María-Dolores CSIC; Noppen, Sam; Bueno, Oskía; Prota, Andrea E.; Bargsten, Katja; Sáez-Calvo, Gonzalo; Jimeno, M. Luisa CSIC ORCID; Benkhei, Mohammed; Ribatti, Domenico; Velázquez, Sonsoles CSIC ORCID CVN; Camarasa Rius, María José CSIC ORCID; Díaz, José Fernando CSIC ORCID ; Steinmetz, Michel O.; Priego, Eva María CSIC ORCID; Peréz-Pérez, María-Jesús CSIC ORCID ; Liekens, Sandraartículo
closedAccessaccesoRestringido.pdf.jpg2017Antiviral activity of [1,2,3]triazolo[4,5-d]pyrimidin-7(6H)-ones against chikungunya virus targeting the viral capping nsP1Gigante, Alba CSIC ORCID; Gómez-SanJuan, Asier CSIC; Delang, Leen; Li, C.; Bueno, Oskía; Gamo, Ana María CSIC; Priego, Eva María CSIC ORCID; Camarasa Rius, María José CSIC ORCID; Jochmans, D.; Leyssen, Pieter; Decroly, E.; Coutard, Bruno; Querat, Guilles; Neyts, Johan; Peréz-Pérez, María-Jesús CSIC ORCID artículo
openAccessacsmedchemlett.1c00617.pdf.jpg8-Dec-2021Antivirals against (Re)emerging Flaviviruses: Should We Target the Virus or the Host?Peréz-Pérez, María-Jesús CSIC ORCID ; Saiz, Juan-Carlos; Priego, Eva María CSIC ORCID; Martín-Acebes, Miguel Ángelartículo
openAccessaccesoRestringido.pdf.jpg27-Jun-2016Blocking Blood Flow to Solid Tumors by Destabilizing Tubulin : An Approach to Targeting Tumor Growth (Perspective)Peréz-Pérez, María-Jesús CSIC ORCID ; Priego, Eva María CSIC ORCID; Bueno, Oskía; Martins, Maria Solange; Canela, María-Dolores CSIC; Liekens, Sandraartículo
closedAccessaccesoRestringido.pdf.jpg2019Chalcones and Chalcone-mimetic Derivatives as Notch Inhibitors in a Model of T-cell Acute Lymphoblastic LeukemiaQuaglio, D.; Zhdanovskaya, N.; Tobajas, Gloria; Cuartas, V.; Balducci, S.; Christodoulou, M. S.; Fabrizi, G.; Gargantilla, Marta; Priego, Eva María CSIC ORCID; Carmona Pestania, Á.; Passarella, D.; Screpanti, I.; Botta, B.; Palermo, R.; Mori, M.; Ghirga, F.; Peréz-Pérez, María-Jesús CSIC ORCID artículo
openAccessExpert Opinion_Perez-Perez et al_2019.pdf.jpg14-Jun-2019Chikungunya virus drug discovery: still a long way to go?Peréz-Pérez, María-Jesús CSIC ORCID ; Delang, Leen; Ng, Lisa; Priego, Eva María CSIC ORCIDartículo
openAccessaccesoRestringido.pdf.jpg2018Conformational mimetics of the α-methyl chalcone TUB091 binding tubulin: Design, synthesis and antiproliferative activityBueno, Oskía; Tobajas, Gloria; Quesada, Ernesto; Estévez-Gallego, Juan CSIC ORCID ; Noppen, Sam; Camarasa Rius, María José CSIC ORCID; Díaz, José Fernando CSIC ORCID ; Liekens, Sandra; Priego, Eva María CSIC ORCID; Peréz-Pérez, María-Jesús CSIC ORCID artículo
closedAccessaccesoRestringido.pdf.jpg2012CRDOCK: An ultrafast multipurpose protein-ligand docking toolCortés Cabrera, Álvaro CSIC ORCID; Klett, Javier CSIC ORCID; Dos Santos, Helena G.; Perona, Almudena CSIC ORCID CVN; Gil Redondo, Rubén; Francis, Sandrea M. CSIC; Priego, Eva María CSIC ORCID; Gago, Federico CSIC ORCID; Morreale, Antonioartículo
openAccessmolecules-pirazolinas_2019.pdf.jpg2019Design and Synthesis of New 6-Nitro and 6-Amino- 3,3a,4,5-Tetrahydro-2H-Benzo[g]indazole Derivatives: Antiproliferative and Antibacterial ActivityCuartas, Viviana; Crespo, María del Pilar; Priego, Eva María CSIC ORCID; Persoons, Leentje; Daelemans, Dirk; Camarasa Rius, María José CSIC ORCID; Insuasty, Braulio; Peréz-Pérez, María-Jesús CSIC ORCID artículo
openAccessmolecules-24-04236-v2.pdf.jpg2019Design and synthesis of new 6-nitro and 6-Amino-3,3a,4,5-Tetrahydro-2H-Benzo[g]indazole derivatives: Antiproliferative and antibacterial activityCuartas, V.; Crespo, M. D. P.; Priego, Eva María CSIC ORCID; Persoons, L.; Daelemans, D.; Camarasa Rius, María José CSIC ORCID; Insuasty, Braulio; Peréz-Pérez, María-Jesús CSIC ORCID artículo
closedAccessEJMC_Diphenyl_ether_derivatives_2019.pdf.jpgJun-2019Diphenyl ether derivatives occupy the expanded binding site of cyclohexanedione compounds at the colchicine site in tubulin by movement of the aT5 loopBueno, Oskia; Gargantilla, Marta; Estévez-Gallego, Juan CSIC ORCID ; Martins, Solange; Díaz, José Fernando CSIC ORCID ; Camarasa Rius, María José CSIC ORCID; Liekens, Sandra; Peréz-Pérez, María-Jesús CSIC ORCID ; Priego, Eva María CSIC ORCIDartículo
closedAccess2012Efficient synthesis and anti-enteroviral activity of 9-arylpurinesAguado, Leire CSIC; Canela, María-Dolores CSIC; Thibaut, Hendrik Jan; Priego, Eva María CSIC ORCID; Camarasa Rius, María José CSIC ORCID; Leyssen, Pieter; Neyts, Johan; Peréz-Pérez, María-Jesús CSIC ORCID artículo
openAccessScientific reports(2018)4242.pdf.jpg2018High-affinity ligands of the colchicine domain in tubulin based on a structure-guided designBueno, Oskía; Estévez-Gallego, Juan CSIC ORCID ; Martins, S.; Prota, Andrea E.; Gago, Federico CSIC ORCID; Gómez-SanJuan, Asier CSIC; Camarasa Rius, María José CSIC ORCID; Barasoain, Isabel CSIC ; Steinmetz, Michel O.; Díaz, José Fernando CSIC ORCID ; Peréz-Pérez, María-Jesús CSIC ORCID ; Liekens, Sandra; Priego, Eva María CSIC ORCIDartículo
openAccesspharmaceuticals-15-00835.pdf.jpg2022Hybridization Approach to Identify Salicylanilides as Inhibitors of Tubulin Polymerization and Signal Transducers and Activators of Transcription 3 (STAT3)Gargantilla, Marta; Persoons, Leentje; Kauerová, Tereza; Río, Natalia del; Daelemans, Dirk; Priego, Eva María CSIC ORCID; Kollar, Peter; Peréz-Pérez, María-Jesús CSIC ORCID artículo
closedAccess2014Identification of [1,2,3]triazolo[4,5-d ]pyrimidin-7(6H)-ones as novel inhibitors of chikungunya virus replicationGigante, Alba CSIC ORCID; Canela, María-Dolores CSIC; Delang, Leen; Priego, Eva María CSIC ORCID; Camarasa Rius, María José CSIC ORCID; Querat, Guilles; Neyts, Johan; Leyssen, Pieter; Peréz-Pérez, María-Jesús CSIC ORCID artículo
openAccessScientific reports (2018).pdf.jpg2018Identification of a novel 2-oxindole fluorinated derivative as in vivo antitumor agent for prostate cancer acting via AMPK activationBort Bueno, Alicia; Quesada Sánchez, Sergio; Ramos-Torres, Ágata; Gargantilla, Marta; Priego, Eva María CSIC ORCID; Raynal, S.; Lepifre, F.; Gasalla, José María; Rodriguez-Henche, Nieves; Castro, Ana CSIC ORCID; Díaz-Laviada, Inésartículo
openAccessACS Infect Dis 2018.pdf.jpg2018Inhibition of the Replication of Different Strains of Chikungunya Virus by 3-Aryl-[1,2,3]triazolo[4,5- d] pyrimidin-7(6 H)-onesGómez-SanJuan, Asier CSIC; Gamo, Ana María CSIC; Delang, Leen; Pérez-Sánchez, Alfonso; Amrun, S. N.; Abdelnabi, Rana; Jacobs, S.; Priego, Eva María CSIC ORCID; Camarasa Rius, María José CSIC ORCID; Jochmans, D.; Leyssen, Pieter; Ng, L. F. P.; Querat, Guilles; Neyts, Johan; Peréz-Pérez, María-Jesús CSIC ORCID artículo