Derechos | Preview | Fecha Public. | Título | Autor(es) | Tipo |
openAccess | | 8-feb-2019 | Evaluation of a class of isatinoids identified from a high-throughput screen of human kinase inhibitors as anti-Sleeping Sickness agents | Klug, Dana M.; Díaz-González, Rosario; Pérez-Moreno, Guiomar; Ceballos-Pérez, Gloria; García-Hernández, Raquel CSIC ORCID; Gómez-Pérez, Veronica; Ruiz-Pérez, Luis Miguel; Rojas-Barros, Domingo I.; Gamarro, Francisco; González-Pacanowska, Dolores; Martínez-Martínez, María S.; Manzano, Pilar; Ferrins, Lori; Caffrey, Conor R.; Navarro, M.; Pollastri, M.P. | artículo |
closedAccess | | 2019 | Hit-to-Lead Optimization of Benzoxazepinoindazoles As Human African Trypanosomiasis Therapeutics | Klug, DM; Tschiegg, L; Díaz, Rosario; Rojas-Barros, D; Pérez-Moreno, Guiomar; Ceballos, G; García-Hernández, Raquel CSIC ORCID; Martinez-Martinez, MS; Manzano, Pilar; Ruiz, LM; Caffrey, CR; Gamarro, Francisco; González-Pacanowska, Dolores; Ferrins, L; Navarro, M.; Pollastri, M.P. | artículo |
openAccess | | 2014 | Identification and Characterization of Hundreds of Potent and Selective Inhibitors of Trypanosoma brucei Growth from a Kinase-Targeted Library Screening Campaign | Diaz, Rosa; Luengo-Arratta, Sandra A.; Seixas, Joao D.; Amata, Emanuele; Devine, William; Cordon-Obras, Carlos; Rojas-Barros, Domingo I.; Jiménez, Elena; Ortega, F.; Crouch, Sabrinia; Colmenarejo, Gonzalo; Fiandor, José M.; Martin, José Julio; Berlanga, M.; Gonzalez, S.; Manzano, Pilar; Navarro, M.; Pollastri, M.P. | artículo |
closedAccess | | mar-2016 | Identification of "Preferred" Human Kinase Inhibitors for Sleeping Sickness Lead Discovery. Are Some Kinases Better than Others for Inhibitor Repurposing? | Amata, Emanuele; Xi, Hualin; Colmenarejo, Gonzalo; Díaz-González, Rosario; Cordon-Obras, Carlos; Berlanga, M.; Manzano, Pilar; Erath, Jessey; Roncal, Norma E.; Lee, Patricia J.; Leed, Susan E.; Rodríguez López, Ana CSIC ORCID; Sciotti, Richard J.; Navarro, M.; Pollastri, M.P. | artículo |
closedAccess | | 2020 | Medicinal Chemistry Optimization of a Diaminopurine Chemotype: Toward a Lead for Trypanosoma brucei Inhibitors | Singh, Baljinder; Díaz-González, Rosario; Ceballos-Pérez, Gloria; Rojas-Barros, Domingo I.; Gunaganti, Naresh; Gillingwater, Kirsten; Santos Martinez-Martinez, María; Manzano, Pilar; Navarro, M.; Pollastri, M.P. | artículo |
openAccess | | 2020 | Selectivity and Physicochemical Optimization of Repurposed Pyrazolo[1,5-b]pyridazines for the Treatment of Human African Trypanosomiasis | Tear, WF; Bag S; Díaz-González, Rosario; Ceballos-Pérez, G.; Rojas-Barros, Domingo I.; Cordon-Obras, Carlos; Pérez-Moreno, Guiomar; García-Hernández, Raquel CSIC ORCID; Martinez-Martinez, MS; Ruiz-Pérez, Luis Miguel; Gamarro, Francisco; González- Pacanowska, D.; Caffrey, CR; Ferrins, L; Manzano, Pilar; Navarro, M.; Pollastri, M.P. | artículo |
closedAccess | | 2020 | Structure-property studies of an imidazoquinoline chemotype with antitrypanosomal activity | Klug, Dana M.; Díaz-González, Rosario; DeLano, Travis J.; Mavrogiannaki, Eftychia M.; Buske, Melissa J.; Dalton, Raeann M.; Fisher, John K.; Schneider, Katherine M.; Hilborne, Vivian; Fritsche, Melanie G.; Simpson, Quillon J.; Tear, Westley F.; Devine, William G.; Pérez-Moreno, Guiomar; Ceballos-Pérez, Gloria; García-Hernández, Raquel CSIC ORCID; Bosch-Navarrete, Cristina; Ruiz-Pérez, Luis Miguel; Gamarro, Francisco; González-Pacanowska, Dolores; Martínez-Martínez, María S.; Manzano-Chinchón, Pilar; Navarro, M.; Pollastri, M.P.; Ferrins, L | artículo |
openAccess | | 2011 | The susceptibility of trypanosomatid pathogens to PI3/mTOR kinase inhibitors affords a new opportunity for drug repurposing | Díaz-González, Rosario; Kuhlmann, F.M.; Galan-Rodriguez, C.; Madeira da Silva, L.; Saldivia, M.; Karver, C.E.; Rodríguez, A.; Beverley, S. M.; Navarro, M.; Pollastri, M.P. | artículo |