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Browsing by Author Pérez, Daniel I.

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openAccess2360783_A1.pdf.jpg6-Sep-20111,2,4-tiadiazoles-5-imino sustituidos útiles en el tratamiento de enfermedades neurodegenerativasLoza García, María Isabel; Martínez, Ana CSIC ORCID ; Pérez, Daniel I. CSIC ORCID; Brea Floriani, José; Cadavid Torres, María Isabel; Palomo, Valle CSIC ORCID ; Gil, Carmen CSIC ORCID ; Pérez Castillo, Ana CSIC ORCID; Pérez, Concepción CSIC ORCIDsolicitud de patente
openAccess1 Benzo d thiazol 2 yl 3 phenylureas as dual inhibitors of casein kinase 1 and ABAD enzymes for treatment of neurodegenerative disorders.pdf.jpg14-Mar-20181-(Benzo[d]thiazol-2-yl)-3-phenylureas as dual inhibitors of casein kinase 1 and ABAD enzymes for treatment of neurodegenerative disordersBenek, O.; Pérez, Daniel I. CSIC ORCID; Pérez, Concepción CSIC ORCID; Martínez, Ana CSIC ORCID ; Musilek, Kamilartículo
openAccessacs chem. neur._Martínez, Ana_2015(post).pdf.jpg14-Jul-20153,4-Dihydro-1,3,5-triazin-2(1H)-ones as the first dual BACE-1/GSK-3β fragment hits against Alzheimer’s diseasePrati, Federica; Pérez, Daniel I. CSIC ORCID; Pérez Castillo, Ana CSIC ORCID; Martínez, Ana CSIC ORCID ; Bolognesi, Maria Lauraartículo
closedAccessaccesoRestringido.pdf.jpg20125-imino-1,2,4-thiadiazoles: first small molecules as substrate competitive inhibitors of glycogen synthase kinase 3Palomo, Valle CSIC ORCID ; Pérez, Daniel I. CSIC ORCID; Pérez, Concepción CSIC ORCID; Morales-García, José A. CSIC ORCID; Soteras, Ignacio CSIC ORCID; Alonso-Gil, Sandra CSIC; Encinas, Arantxa; Castro, Ana CSIC ORCID; Campillo, Nuria E. CSIC ORCID ; Pérez Castillo, Ana CSIC ORCID; Gil, Carmen CSIC ORCID ; Martínez, Ana CSIC ORCID artículo
closedAccessaccesoRestringido.pdf.jpg20125-Imino-1,2-4-thiadiazoles and quinazolines derivatives as glycogen synthase kinase 3β (GSK-3β) and phosphodiesterase 7 (PDE7) inhibitors: Determination of blood-brain barrier penetration and binding to human serum albuminPérez, Daniel I. CSIC ORCID; Pistolozzi, Marco; Redondo, Miriam CSIC; Fortugno, Cecilia; Gil, Carmen CSIC ORCID ; Felix, Guy; Martínez, Ana CSIC ORCID ; Bertucci, Carloartículo
closedAccessaccesoRestringido.pdf.jpg2013A fluorescent styrylquinoline with combined therapeutic and diagnostic activities against Alzheimer's and prion diseasesStaderini, Matteo; Aulic, Suzana; Bartolini, Manuela; Tran, H. N. A.; González-Ruiz, Victor; Pérez, Daniel I. CSIC ORCID; Cabezas, Nieves; Martínez, Ana CSIC ORCID ; Martín, M. Antonia; Andrisano, Vincenza; Legname, Giuseppe; Menéndez, José Carlos; Bolognesi, Maria Lauraartículo
closedAccessaccesoRestringido.pdf.jpg2012A small chemical library of 2-aminoimidazole derivatives as BACE-1 inhibitors: Structure-based design, synthesis, and biological evaluationChiriano, G.; De Simone, A.; Mancini, Francesca; Pérez, Daniel I. CSIC ORCID; Cavalli, A.; Bolognesi, Maria Laura; Legname, G.; Martínez, A.; Andrisano, Vincenza; Carloni, Paolo; Roberti, M.artículo
openAccessFitoterapia postprint-1.pdf.jpgMar-2016Application of BACE1 immobilized enzyme reactor for the characterization of multifunctional alkaloids from Corydalis cava (Fumariaceae) as Alzheimer's disease targetsChlebek, Jakub; De Simone, Angela; Hošťálková, Anna; Opletal, Lubomír; Pérez, Concepción CSIC ORCID; Pérez, Daniel I. CSIC ORCID; Havlíková, Lucie; Cahlíková, Lucie; Andrisano, Vincenzaartículo
openAccessES2489297_B1.pdf.jpg1-Sep-2014Benzotiazoles sustituidos y sus aplicaciones terapéuticas para el tratamiento de enfermedades humanasMartínez, Ana CSIC ORCID ; Pérez, Daniel I. CSIC ORCID; Gil, Carmen CSIC ORCID ; García Salado, Irene; Redondo, Miriam CSIC; Pérez, Concepción CSIC ORCIDpatente
openAccessES2489297_A1.pdf.jpg1-Sep-2014Benzotiazoles sustituidos y sus aplicaciones terapéuticas para el tratamiento de enfermedades humanasMartínez, Ana CSIC ORCID ; Pérez, Daniel I. CSIC ORCID; Gil, Carmen CSIC ORCID ; García Salado, Irene; Redondo, Miriam CSIC; Pérez, Concepción CSIC ORCIDsolicitud de patente
openAccessEuropean Journal of Medicinal Chemistry_Staderini_2022.pdf.jpg15-Nov-2022Bifunctional carbazole derivatives for simultaneous therapy and fluorescence imaging in prion disease murine cell modelsStaderini, Matteo; Vanni, Silvia; Colini Baldeschi, Arianna; Giachin, Gabriele; Zattoni, Marco; Celauro, Luigi; Ferracin, Chiara; Bistaffa, Edoardo; Moda, F.; Pérez, Daniel I. CSIC ORCID; Martínez, Ana CSIC ORCID ; Martín, M. Antonia; Martín-Cámara, Olmo; Cores, Ángel; Bianchini, Giulia; Kammerer, Robert; Menéndez, J. Carlos; Legname, G.; Bolognesi, Maria Lauraartículo
openAccessacsomega.7b00869.pdf.jpg30-Aug-2017Biological and pharmacological characterization of benzothiazole-based CK-1δ inhibitors in models of Parkinson’s diseaseMorales-García, José A. CSIC ORCID; Salado, Irene G. CSIC; Sanz-SanCristóbal, Marina CSIC; Gil, Carmen CSIC ORCID ; Pérez Castillo, Ana CSIC ORCID; Martínez, Ana CSIC ORCID ; Pérez, Daniel I. CSIC ORCIDartículo
openAccessEP3604310A1.pdf.jpg5-Feb-2020CDC-7-inhibitors compounds and use thereof for the treatment of neurological conditionsMartínez, Ana CSIC ORCID ; Pérez, Daniel I. CSIC ORCID; Gil, Carmen CSIC ORCID ; Martín-Requero, Ángeles CSIC ORCID ; Rojas-Prats, Elisa; Martínez-González, Loreto CSIC ORCID ; Pérez, Concepción CSIC ORCIDsolicitud de patente
openAccessWO2018172587A1.pdf.jpg27-Sep-2018CDC-7-inhibitors compounds and use thereof for the treatment of neurological conditionsMartínez, Ana CSIC ORCID ; Pérez, Daniel I. CSIC ORCID; Gil, Carmen CSIC ORCID ; Martín-Requero, Ángeles CSIC ORCID ; Rojas-Prats, Elisa; Martínez-González, Loreto CSIC ORCID ; Pérez, Concepción CSIC ORCIDsolicitud de patente
openAccessUS2020093828A1.pdf.jpg26-Mar-2020CDC-7-inhibitors compounds and use thereof for the treatment of neurological conditionsMartínez, Ana CSIC ORCID ; Pérez, Daniel I. CSIC ORCID; Gil, Carmen CSIC ORCID ; Martín-Requero, Ángeles CSIC ORCID ; Rojas-Prats, Elisa; Martínez-González, Loreto CSIC ORCID ; Pérez, Concepción CSIC ORCIDsolicitud de patente
closedAccessaccesoRestringido.pdf.jpg2018Chameleon-like behavior of indolylpiperidines in complex with cholinesterases targets: Potent butyrylcholinesterase inhibitorsChierrito, Talita P. C.; Pedersoli-Mantoani, S.; Roca, Carlos; Sebastián-Pérez, Víctor; Martínez-González, Loreto CSIC ORCID ; Pérez, Daniel I. CSIC ORCID; Pérez, Concepción CSIC ORCID; Canales, A.; Cañada, F. Javier ; Campillo, Nuria E. CSIC ORCID ; Carvalho, Ivone; Martínez, Ana CSIC ORCID artículo
openAccessWO_2003_055479_A1.pdf.jpg10-Jul-2003Compounds and their therapeutic use related to the phophorylating activity of the enzyme GSK-3Conde, Santiago CSIC; Martínez, Ana CSIC ORCID ; Pérez, Daniel I. CSIC ORCID; Pérez, Concepción CSIC ORCID; Moreno Muñoz, Francisco José; Wandosell, Francisco CSIC ORCID patente
openAccessES2686909A1.pdf.jpg22-Oct-2018Compuestos inhibidores de CDC-7 y su uso para el tratamiento de patologías neurológicasMartínez, Ana CSIC ORCID ; Pérez, Daniel I. CSIC ORCID; Gil, Carmen CSIC ORCID ; Martín-Requero, Ángeles CSIC ORCID ; Rojas-Prats, Elisa; Martínez-González, Loreto CSIC ORCID ; Pérez, Concepción CSIC ORCIDsolicitud de patente
openAccessES2686909B1.pdf.jpg22-Oct-2018Compuestos inhibidores de CDC-7 y su uso para el tratamiento de patologías neurológicasMartínez, Ana CSIC ORCID ; Pérez, Daniel I. CSIC ORCID; Gil, Carmen CSIC ORCID ; Martín-Requero, Ángeles CSIC ORCID ; Rojas-Prats, Elisa; Martínez-González, Loreto CSIC ORCID ; Pérez, Concepción CSIC ORCIDpatente
openAccessJEIMC_Sciú_2018.pdf.jpg1-Jan-2019Computer-aided molecular design of pyrazolotriazines targeting glycogen synthase kinase 3Sciú, María Lourdes; Sebastián-Pérez, Víctor; Martínez-González, Loreto CSIC ORCID ; Benítez, Rocio; Pérez, Daniel I. CSIC ORCID; Pérez, Concepción CSIC ORCID; Campillo, Nuria E. CSIC ORCID ; Martínez, Ana CSIC ORCID ; Moyano, Elizabeth Lauraartículo