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openAccess1 Benzo d thiazol 2 yl 3 phenylureas as dual inhibitors of casein kinase 1 and ABAD enzymes for treatment of neurodegenerative disorders.pdf.jpg14-Mar-20181-(Benzo[d]thiazol-2-yl)-3-phenylureas as dual inhibitors of casein kinase 1 and ABAD enzymes for treatment of neurodegenerative disordersBenek, O.; Pérez, Daniel I.; Pérez, Concepción; Martínez, Ana CSIC ORCID ; Musilek, Kamilartículo
closedAccessrestringido.pdf.jpg29-Apr-20191-Aryl-3-(4-methoxybenzyl)ureas as potentially irreversible glycogen synthase kinase 3 inhibitors: Synthesis and biological evaluationVenter, Jana; Pérez, Concepción; van Otterlo, Willem A. L.; Martínez, Ana CSIC ORCID ; Blackie, Margaret A.L.artículo
openAccess20 JMC 9237  (2-Oxaadamant-1-yl ureas).pdf.jpg20202-Oxaadamant-1-yl Ureas as Soluble Epoxide Hydrolase Inhibitors: In Vivo Evaluation in a Murine Model of Acute PancreatitisCodony, Sandra; Pujol, Eugènia; Pizarro, J.; Feixas, Ferran; Valverde,E.; Loza, María Isabel; Brea, José Manuel; Saez, Elena; Oyarzabal, Julen; Pineda-Lucena, Antonio; Pérez, Belén; Pérez, Concepción; Rodríguez-Franco, María Isabel CSIC ORCID ; Leiva, Rosana; Osuna, Sílvia; Morissea, Christophe; Hammock, Bruce D.; Vázquez-Carrera, Manuel; Vázquez, Santiagoartículo
closedAccessaccesoRestringido.pdf.jpg20125-imino-1,2,4-thiadiazoles: first small molecules as substrate competitive inhibitors of glycogen synthase kinase 3Palomo, Valle CSIC ORCID ; Pérez, Daniel I.; Pérez, Concepción; Morales-García, José A. CSIC ORCID; Soteras, Ignacio CSIC ORCID; Alonso-Gil, Sandra CSIC; Encinas, Arantxa; Castro, Ana CSIC ORCID; Campillo, Nuria E. CSIC ORCID ; Pérez Castillo, Ana CSIC ORCID; Gil, Carmen CSIC ORCID ; Martínez, Ana CSIC ORCID artículo
openAccessCNS postprint 2018.pdf.jpg7-May-2018Activation of the cannabinoid type 2 receptor by a novel indazole derivative normalizes the survival pattern of lymphoblasts from patients with late-onset alzheimer’s diseaseDel Cerro, Patricia; Alquézar, Carolina CSIC ORCID; Bartolomé Robledo, Fernando CSIC ORCID; González-Naranjo, Pedro CSIC ORCID; Pérez, Concepción; Carro, Eva; Páez, Juan A. CSIC ORCID; Campillo, Nuria E. CSIC ORCID ; Martín-Requero, Ángeles CSIC ORCID artículo
closedAccessaccesoRestringido.pdf.jpg1991Analgesic dipeptide derivatives. Part 8. 3-amino-2-hydroxy-4-[2-(o- nitrophenylthio)indol-3-yl]butanoic acid [AH(NPS)IBA]-containing dipeptide analogues of the analgesic compound H-Trp(Nps)-Lys-OMeHerranz, Rosario CSIC ORCID; Vinuesa, Soledad; Pérez, Concepción; García-López, M. T.; Ceballos, María L. de CSIC ORCID; Río, Joaquín delartículo
closedAccessaccesoRestringido.pdf.jpg2014Anthocyanins constituents, antioxidant and anti-Inflammatory activity of strawberries. Comparison with other berry fruitsPérez, Concepción; Ruiz del Castillo, M. Luisa CSIC ORCID ; Gil, Carmen CSIC ORCID ; Blanch, Gracia Patricia CSIC ORCID ; Flores, Gema CSICcapítulo de libro
closedAccessArtículo.pdf.jpg2001Anti-HIV-1 activity of benzothiadiazine dioxideMartínez, Ana CSIC ORCID ; Gil, Carmen CSIC ORCID ; Castro, Ana CSIC ORCID; Pérez, Concepción; Witvrouw, M.; Pannecouque, C.; Balzarini, Jan; De Clercq, Erikartículo
openAccessFitoterapia postprint-1.pdf.jpgMar-2016Application of BACE1 immobilized enzyme reactor for the characterization of multifunctional alkaloids from Corydalis cava (Fumariaceae) as Alzheimer's disease targetsChlebek, Jakub; De Simone, Angela; Hošťálková, Anna; Opletal, Lubomír; Pérez, Concepción; Pérez, Daniel I.; Havlíková, Lucie; Cahlíková, Lucie; Andrisano, Vincenzaartículo
closedAccessaccesoRestringido.pdf.jpg2000Benzothiadiazine dioxide dibenzyl derivatives as potent human cytomegalovirus inhibitors: Synthesis and comparative molecular field analysisMartínez, Ana CSIC ORCID ; Gil, Carmen CSIC ORCID ; Abasolo, M. Inés; Castro, Ana CSIC ORCID; Bruno, Ana M.; Pérez, Concepción; Prieto, Columbiana; Otero, J.artículo
openAccess2003Benzothiadiazine dioxide human cytomegalovirus inhibitors: Synthesis and antiviral evaluation of main heterocycle modified derivativesMartínez, Ana CSIC ORCID ; Gil, Carmen CSIC ORCID ; Castro, Ana CSIC ORCID; Bruno, Ana M.; Pérez, Concepción; Prieto, Columbiana; Otero, Joaquínartículo
closedAccessaccesoRestringido.pdf.jpg2003Benzothiadiazine dioxides (BTD) derivatives as non-nucleoside human cytomegalovirus (HCMV) inhibitors. Study of structural requirements for biological activityMartínez, Ana CSIC ORCID ; Gil, Carmen CSIC ORCID ; Castro, Ana CSIC ORCID; Pérez, Concepción; Prieto, Carlos CSIC ORCID ; Otero, Joaquínartículo
closedAccessaccesoRestringido.pdf.jpg2012Benzothiazepine CGP37157 and its isosteric 2′-ethyl analogue provide neuroprotection and block cell calcium entryGonzález-Lafuente, Laura; Egea, Javier; León, Rafael CSIC ORCID ; Martínez-Sanz, Francisco J.; Monjas, Leticia CSIC ORCID; Pérez, Concepción; Merino, Cristina; García-De Diego. Antonio M.; Rodríguez-Franco, María Isabel CSIC ORCID ; García, Antonio G.; Villarroya, Mercedes; López, Manuela G.; Ríos, Cristóbal de losartículo
openAccessES2489297_B1.pdf.jpg1-Sep-2014Benzotiazoles sustituidos y sus aplicaciones terapéuticas para el tratamiento de enfermedades humanasMartínez, Ana CSIC ORCID ; Pérez Fernández, Daniel Ignacio; Gil, Carmen CSIC ORCID ; García Salado, Irene; Redondo, Miriam CSIC; Pérez, Concepciónpatente
openAccessES2735807T3.pdf.jpg20-Dec-2019Benzotiazoles sustituidos y sus aplicaciones terapéuticas para el tratamiento de enfermedades humanasMartínez, Ana CSIC ORCID ; Pérez Fernández, Daniel Ignacio; Gil, Carmen CSIC ORCID ; García Salado, Irene; Redondo, Miriam CSIC; Pérez, Concepcióntraducción de patente
openAccessES2489297_A1.pdf.jpg1-Sep-2014Benzotiazoles sustituidos y sus aplicaciones terapéuticas para el tratamiento de enfermedades humanasMartínez, Ana CSIC ORCID ; Pérez Fernández, Daniel Ignacio; Gil, Carmen CSIC ORCID ; García Salado, Irene; Redondo, Miriam CSIC; Pérez, Concepciónsolicitud de patente
openAccessUS2020093828A1.pdf.jpg26-Mar-2020CDC-7-inhibitors compounds and use thereof for the treatment of neurological conditionsMartínez, Ana CSIC ORCID ; Pérez, Daniel I.; Gil, Carmen CSIC ORCID ; Martín-Requero, Ángeles CSIC ORCID ; Rojas-Prats, Elisa; Martínez-González, Loreto CSIC ORCID ; Pérez, Concepciónsolicitud de patente
openAccessEP3604310A1.pdf.jpg5-Feb-2020CDC-7-inhibitors compounds and use thereof for the treatment of neurological conditionsMartínez, Ana CSIC ORCID ; Pérez, Daniel I.; Gil, Carmen CSIC ORCID ; Martín-Requero, Ángeles CSIC ORCID ; Rojas-Prats, Elisa; Martínez-González, Loreto CSIC ORCID ; Pérez, Concepciónsolicitud de patente
openAccessWO2018172587A1.pdf.jpg27-Sep-2018CDC-7-inhibitors compounds and use thereof for the treatment of neurological conditionsMartínez, Ana CSIC ORCID ; Pérez, Daniel I.; Gil, Carmen CSIC ORCID ; Martín-Requero, Ángeles CSIC ORCID ; Rojas-Prats, Elisa; Martínez-González, Loreto CSIC ORCID ; Pérez, Concepciónsolicitud de patente
closedAccessaccesoRestringido.pdf.jpg2018Chameleon-like behavior of indolylpiperidines in complex with cholinesterases targets: Potent butyrylcholinesterase inhibitorsChierrito, Talita P. C.; Pedersoli-Mantoani, S.; Roca, Carlos; Sebastián-Pérez, Víctor; Martínez-González, Loreto CSIC ORCID ; Pérez, Daniel I.; Pérez, Concepción; Canales, A.; Cañada, F. Javier ; Campillo, Nuria E. CSIC ORCID ; Carvalho, Ivone; Martínez, Ana CSIC ORCID artículo