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Browsing by Author Noppen, Sam

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Showing results 1 to 12 of 12
RightsPreviewIssue DateTitleAuthor(s)Type
openAccessA second-generation of tryptophan.pdf.jpg3-Apr-2019A second-generation of tryptophan-containing small molecules extremely potent against HIV and EV-A71 clinical isolatesMartí-Marí, Olaia; Martínez-Gualda, Belén; Puente-Secades, Sofía de la; Quesada, Ernesto CSIC ORCID ; Sun, Liang; Delang, Leen; Mirabelli, Carmen; Noppen, Sam; Schols, Dominique; Neyts, Johan; Gago, Federico CSIC ORCID; Camarasa Rius, María José CSIC ORCID; San-Félix, Ana CSIC ORCID CVN actas de congreso
openAccessaccesoRestringido.pdf.jpg2015Anti-HIV-1 activity of a tripodal receptor that recognizes mannose oligomersRivero-Buceta, Eva CSIC; Carrero, Paula CSIC; Casanova, Elena CSIC; García-Doyagüez, Elisa CSIC ORCID; Madrona, Andrés; Quesada, Ernesto; Peréz-Pérez, María-Jesús CSIC ORCID ; Mateos, Raquel CSIC ORCID ; Bravo, Laura CSIC ORCID; Mathys, Leen; Noppen, Sam; Kiselev, Evgency; Marchand, Christophe; Pommier, Yves; Liekens, Sandra; Balzarini, Jan; Camarasa Rius, María José CSIC ORCID; San-Félix, Ana CSIC ORCID CVN artículo
openAccessOncotarget.pdf.jpg20-May-2016Antivascular and antitumor properties of the tubulin-binding chalcone TUB091Canela, María-Dolores CSIC; Noppen, Sam; Bueno, Oskía; Prota, Andrea E.; Bargsten, Katja; Sáez-Calvo, Gonzalo; Jimeno, M. Luisa CSIC ORCID; Benkhei, Mohammed; Ribatti, Domenico; Velázquez, Sonsoles CSIC ORCID CVN; Camarasa Rius, María José CSIC ORCID; Díaz, José Fernando CSIC ORCID ; Steinmetz, Michel O.; Priego, Eva María CSIC ORCID; Peréz-Pérez, María-Jesús CSIC ORCID ; Liekens, Sandraartículo
openAccessaccesoRestringido.pdf.jpg2018Conformational mimetics of the α-methyl chalcone TUB091 binding tubulin: Design, synthesis and antiproliferative activityBueno, Oskía; Tobajas, Gloria; Quesada, Ernesto; Estévez-Gallego, Juan CSIC ORCID ; Noppen, Sam; Camarasa Rius, María José CSIC ORCID; Díaz, José Fernando CSIC ORCID ; Liekens, Sandra; Priego, Eva María CSIC ORCID; Peréz-Pérez, María-Jesús CSIC ORCID artículo
openAccessacs.jmedchem.1c00315-1.pdf.jpg7-Jul-2021Double Arylation of the Indole Side Chain of Tri- and Tetrapodal Tryptophan Derivatives Renders Highly Potent HIV‑1 and EV-A71 Entry InhibitorsMartí-Marí, Olaia; Martínez-Gualda, Belén; Puente-Secades, Sofía de la; Mills, Alberto; Quesada, Ernesto CSIC ORCID ; Abdelnabi, Rana; Sun, Liang; Boonen, Arnaud; Noppen, Sam; Neyts, Johan; Schols, Dominique; Camarasa Rius, María José CSIC ORCID; Gago, Federico CSIC ORCID; San-Félix, Ana CSIC ORCID CVN artículo
openAccesschem.202101098.pdf.jpg14-Apr-2021Multivalent Tryptophan- and Tyrosine-Containing [60] Fullerene Hexa-Adducts as Dual HIV and Enterovirus A71 Entry InhibitorsRuiz-Santaquiteria, Marta CSIC ORCID; Illescas, Beatriz M.; Abdelnabi, Rana; Boonen, Arnaud; Mills, Alberto; Martí-Marí, Olaia; Noppen, Sam; Neyts, Johan; Schols, Dominique; Gago, Federico CSIC ORCID; San-Félix, Ana CSIC ORCID CVN ; Camarasa Rius, María José CSIC ORCID; Martín, Nazarioartículo
openAccessCanela-et-al_2014_JMedChem_57.pdf.jpg2014Novel colchicine-site binders with a cyclohexanedione scaffold identified through a ligand-based virtual screening approachCanela, María-Dolores CSIC; Peréz-Pérez, María-Jesús CSIC ORCID ; Noppen, Sam; Sáez-Calvo, Gonzalo; Díaz, José Fernando CSIC ORCID ; Camarasa Rius, María José CSIC ORCID; Liekens, Sandra; Priego, Eva María CSIC ORCIDartículo
openAccessApr-2022Organotropic dendrons with high potency as HIV-1, HIV-2 and EV-A71 cell entry inhibitorsMartí-Marí, Olaia; Martínez-Gualda, Belén; Fernández-Barahona, Irene; Mills, Alberto; Abdelnabi, Rana; Noppen, Sam; Neyts, Johan; Schols, Dominique; Camarasa Rius, María José CSIC ORCID; Herranz, Fernando CSIC ORCID CVN; Gago, Federico CSIC ORCID; San-Félix, Ana CSIC ORCID CVN artículo
openAccessASF9 REVISED jm-2019-01737d.pdf.jpgJan-2020Scaffold Simplification Strategy Leads to a Novel Generation of Dual Human Immunodeficiency Virus and Enterovirus-A71 Entry InhibitorsMartínez-Gualda, Belén; Sun, Liang; Martí-Marí, Olaia; Abdelnabi, Rana; Noppen, Sam; Bator, Carol M.; Quesada, Ernesto CSIC ORCID ; Delang, Leen; Mirabelli, Carmen; Lee, Hyunwook; Schols, Dominique; Neyts, Johan; Hafenstein, Susan; Camarasa Rius, María José CSIC ORCID; Gago, Federico CSIC ORCID; San-Félix, Ana CSIC ORCID CVN artículo
openAccessASF5 Revised EJMECH.pdf.jpg2017Structure-activity relationship studies on a Trp dendrimer with dual activities against HIV and enterovirus A71. Modifications on the amino acidMartínez-Gualda, Belén; Sun, L.; Rivero-Buceta, Eva CSIC; Flores, Aida CSIC; Quesada, Ernesto CSIC ORCID ; Balzarini, Jan; Noppen, Sam; Liekens, Sandra; Schols, Dominique; Neyts, Johan; Leyssen, Pieter; Mirabelli, C.; Camarasa Rius, María José CSIC ORCID; San-Félix, Ana CSIC ORCID CVN artículo
closedAccessaccesoRestringido.pdf.jpg2016Targeting the colchicine site in tubulin through cyclohexanedione derivativesCanela, María-Dolores CSIC; Bueno, O.; Noppen, Sam; Sáez-Calvo, Gonzalo; Estévez-Gallego, Juan CSIC ORCID ; Díaz, José Fernando CSIC ORCID ; Camarasa Rius, María José CSIC ORCID; Liekens, Sandra; Peréz-Pérez, María-Jesús CSIC ORCID ; Priego, Eva María CSIC ORCIDartículo
openAccessASF4 Revised EJMECH-D-15-01517.pdf.jpg2015Tryptophan dendrimers that inhibit HIV replication, prevent virus entry and bind to the HIV envelope glycoproteins gp120 and gp41Rivero-Buceta, Eva CSIC; García-Doyagüez, Elisa CSIC ORCID; Colomer, Ignacio CSIC ORCID ; Quesada, Ernesto; Mathys, Leen; Noppen, Sam; Liekens, Sandra; Camarasa Rius, María José CSIC ORCID; Peréz-Pérez, María-Jesús CSIC ORCID ; Balzarini, Jan; San-Félix, Ana CSIC ORCID CVN artículo