Rights | Preview | Issue Date | Title | Author(s) | Type |
embargoedAccess |  | 2020 | 2-Oxaadamant-1-yl Ureas as Soluble Epoxide Hydrolase Inhibitors: In Vivo Evaluation in a Murine Model of Acute Pancreatitis | Codony, Sandra; Pujol, E.; Pizarro, J.; Feixas, Ferran; Valverde,E.; Loza, María Isabel; Brea, José Manuel; Saez, Elena; Oyarzabal, Julen; Pineda-Lucena, Antonio; Pérez, Belén ; Pérez, Concepción; Rodríguez-Franco, María Isabel ; Leiva, Rosana; Osuna, Sílvia; Morissea, Christophe; Hammock, Bruce D.; Vázquez-Carrera, Manuel; Vázquez, Santiago | artículo |
openAccess |  | Feb-2020 | A comprehensive tyrosine phosphoproteomic analysis reveals novel components of the platelet CLEC-2 signaling cascade | Izquierdo, Irene; Barrachina, Maria N.; Hermida-Nogueira, Lidia; Casas, Vanessa ; Morán, Luis A.; Lacerenza, Serena; Pinto-Llorente, Roberto; Eble, Johannes A.; Ríos, Vivian de los ; Domínguez, Eduardo; Loza, María Isabel; Casal, J. Ignacio ; Carrascal, Montserrat ; Abián, Joaquín ; García, Ángel | artículo |
openAccess |  | 9-Apr-2020 | Bicyclic alfa-iminophosphonates as highly affinity imidazoline I2 receptor ligands for Alzheimer’s Disease | Abás, Sònia; Rodríguez Arévalo, Sergio; Bagán, Andrea; Griñán Ferré, Christian; Vasilopoulou, Foteini; Brocos Mosquera, Iria; Muguruza, Carolina; Pérez, Belén ; Molins, Elies ; Luque, F. Javier; Pérez Lozano, Pilar; Jonghe, Steven de; Daelemans, Dirk; Naesens, Lieve; Brea, José; Loza, María Isabel; Hernández Hernández, Elena; García-Sevilla, Jesús A.; García Fuster, M. Julia; Radan, Milica; Djikic, Teodora; Nikolic, Katarina; Pallàs, Mercè; Callado, Luis F.; Escolano, Carmen | artículo |
openAccess |  | 29-Nov-2012 | Derivados heterocíclicos inhibidores de fosfodiesterasa 7 | Gil, Carmen ; Martínez, Ana ; Redondo, Miriam ; Campillo, Nuria E. ; Pérez, Daniel I.; Loza, María Isabel; Cadavid, María Isabel; Brea, José; Pérez Castillo, Ana  | solicitud de patente |
openAccess |  | 2012 | Effect of phosphodiesterase 7 (PDE7) inhibitors in experimental autoimmune encephalomyelitis mice. Discovery of a new chemically diverse family of compounds | Redondo, Miriam ; Brea, José; Pérez, Daniel I.; Soteras, Ignacio ; Val, Cristina; Pérez, Concepción; Morales-García, José A. ; Alonso-Gil, Sandra ; Paul-Fernández, Nuria ; Martín-Álvarez, Rocío ; Cadavid, María Isabel; Loza, María Isabel; Pérez Castillo, Ana ; Mengod Los Arcos, Guadalupe ; Campillo, Nuria E. ; Martínez, Ana ; Gil, Carmen | artículo |
closedAccess |  | 2020 | Essential role of the C148–C227 disulphide bridge in the human 5-HT2A homodimeric receptor | Cimadevila, M.; Gómez-García, L.; Martínez, A.L.; Iglesias, A.; López-Giménez, Juan F. ; Castro, M.; Cadavid, M.I.; Loza, María Isabel; Brea, J. | artículo |
closedAccess |  | 11-Mar-2009 | Evidence for distinct antagonist-revealed functional states of 5-hydroxytryptamine(2A) receptor homodimers | Vilaró, Maria Teresa ; Mengod Los Arcos, Guadalupe ; Loza, María Isabel | artículo |
closedAccess |  | 2014 | Modulation of cAMP-specific PDE without emetogenic activity: New sulfide-like PDE7 inhibitors | García, Ana M. ; Brea, José; Morales-García, José A. ; Pérez, Daniel I.; González, A. ; Alonso-Gil, Sandra ; Conde, Santiago ; Cadavid, María Isabel; Loza, María Isabel; Pérez Castillo, Ana ; Martínez, Ana ; Gil, Carmen | artículo |
closedAccess |  | 2001 | Multiple conformations of native and recombinant human 5-hydroxytryptamine2A receptors are labeled by agonists and discriminated by antagonists | López-Giménez, Juan F. ; Villazón, María; Brea, José Manuel; Loza, María Isabel; Palacios, José M.; Mengod Los Arcos, Guadalupe ; Vilaró, Maria Teresa  | artículo |
closedAccess |  | 2012 | Neuroprotective efficacy of quinazoline type phosphodiesterase 7 inhibitors in cellular cultures and experimental stroke model | Redondo, Miriam ; Zarruk, Juan G.; Ceballos, Placido ; Pérez, Daniel I.; Pérez Martín, María Concepción; Pérez Castillo, Ana ; Moro, María A.; Brea, José; Val, Cristina; Cadavid, María Isabel; Loza, María Isabel; Campillo, Nuria E. ; Martínez, Ana ; Gil, Carmen | artículo |
closedAccess |  | 8-Dec-2001 | New serotonin 5-HT2A, 5-HT2B, and 5-HT2C receptor antagonists: Synthesis, pharmacology, 3D-QSAR, and molecular modeling of (aminoalkyl)benzo and heterocycloalkanones | Brea, José Manuel; Mengod Los Arcos, Guadalupe ; Loza, María Isabel | artículo |
closedAccess |  | 2-Jun-2020 | Pharmacological Inhibition of Soluble Epoxide Hydrolase as a New Therapy for Alzheimer's Disease | Griñán-Ferré, Christian; Codony, Sandra; Pujol, Eugènia; Yang, Jun; Leiva, Rosana; Escolano, Carmen; Puigoriol-Illamola, Dolors; Companys-Alemany, Júlia; Corpas, Rubén ; Sanfeliu, Coral ; Pérez, Belén ; Loza, María Isabel; Brea, José; Morisseau, Christophe; Hammock, Bruce D.; Vázquez, Santiago; Pallàs, Mercè; Galdeano, Carles | artículo |
closedAccess |  | 2017 | Pharmacological tools based on imidazole scaffold proved the utility of PDE10A inhibitors for Parkinson’s disease | García, Ana M. ; Salado, Irene G. ; Pérez, Daniel I.; Brea, José; Morales-García, José A. ; González-García, Alejandro; Cadavid, María Isabel; Loza, María Isabel; Luque, Francisco Javier; Pérez Castillo, Ana ; Martínez, Ana ; Gil, Carmen | artículo |
closedAccess |  | 2020 | Pharmacology and preclinical validation of a novel anticancer compound targeting PEPCK-M | Aragó, M.; Moreno-Felici, J.; Abás, S.; Rodríguez-Arévalo, S.; Hyroššová, P.; Figueras, A.; Viñals, F.; Pérez, B.; Loza, María Isabel; Brea, J.; Latorre, P.; Carrodeguas, J.A.; García-Rovés, P.M.; Galdeano, C.; Ginex, Tiziana ; Luque, F.J.; Escolano, C.; Perales, J.C | artículo |
openAccess |  | 7-Apr-2011 | Substituted 5-IMINO-1,2,4-THIADIAZOLES that can be used to treat neurodegenerative diseases | Martínez, Ana ; Gil, Carmen ; Palomo, Valle ; Pérez, Daniel I.; Pérez Martín, María Concepción; Pérez Castillo, Ana ; Loza, María Isabel; Cadavid, María Isabel; Brea, José | solicitud de patente |
closedAccess | | 2010 | Synthesis, biological activity and molecular docking analysis of new A2A adenosine receptor agonists | Rodríguez, Anna M. ; Rosell, Gloria ; Bujons Vilàs, Jordi ; Gutiérrez-de-Terán, Hugo; Rodríguez, David; Brea, José Manuel; Loza, María Isabel; Guerrero, Ángel ; Bosch, María Pilar  | artículo |
closedAccess |  | 2013 | Unraveling phosphodiesterase surfaces. Identification of phosphodiesterase 7 allosteric modulation cavities | Redondo, Miriam ; Soteras, Ignacio ; Brea, José Manuel; González-García, A.; Cadavid, Maria Isabel; Loza, María Isabel; Martínez, Ana ; Gil, Carmen ; Campillo, Nuria E. | artículo |