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DerechosPreviewFecha Public.TítuloAutor(es)Tipo
closedAccessaccesoRestringido.pdf.jpg18-jun-20185-Hydroxypyrido[2,3-b]pyrazin-6(5H)-one derivatives as novel dual inhibitors of HIV-1 reverse transcriptase-associated ribonuclease H and integraseSun, Lin; Gao, Ping; Dong, Guanyu; Zhang, Xujie; Ding, Xiao; Wang, Xueshun; Daelemans, Dirk; De Clercq, Erik; Pannecouque, Christophe; Menéndez-Arias, Luis CSIC ORCID ; Zhang, Peng; Liu, Xinyongartículo
closedAccessaccesoRestringido.pdf.jpg2023Chapter 2 - Chalcones: Diverse biological activities and structure–activity relationshipsZhang, Ying; Liu, Chuanfeng; Ju, Han; Jia, Ruifang; Gao, Shenghua; Liu, Xinyong; Menéndez-Arias, Luis CSIC ORCID ; Zhan, Pengcapítulo de libro
embargoedAccessRNase-H-inhibitors.pdf.jpg5-dic-2022Current medicinal chemistry strategies in the discovery of novel HIV-1 ribonuclease H inhibitorsZhang, Lina; Wei, Fenju; Zhang, Jiwei; Liu, Chuanfeng; López-Carrobles, Nerea; Liu, Xinyong; Menéndez-Arias, Luis CSIC ORCID ; Zhan, Pengartículo
openAccess340989_Manuscript-revised_LMA_Gao0702_LMA.pdf.jpg1-sep-2019Design, synthesis and biological evaluation of 3-hydroxyquinazoline-2,4(1H,3H)-diones as dual inhibitors of HIV-1 reverse transcriptase-associated RNase H and integraseGao, Ping; Cheng, Xiqiang; Sun, Lin; Song, Shu; Álvarez, Mar CSIC ORCID; Luczkowiak, Joanna; Pannecouque, Christophe; De Clercq, Erik; Menéndez-Arias, Luis CSIC ORCID ; Zhan, Peng; Liu, Xinyongartículo
openAccessMenéndez-AriasL_DesignSynthesisandBiologic.pdf.jpg24-nov-2018Design, synthesis, and biologic evaluation of novel galloyl derivatives as HIV-1 RNase H inhibitorsGao, Ping; Sun, Lin; Cheng, Xiqiang; Poongavanam, Vasanthanathan; Kongsted, Jacob; Álvarez, Mar CSIC ORCID; Luczkowiak, Joanna; Pannecouque, Christophe; De Clercq, Erik; Lee, Kuo-Hsiung; Chen, Chin-Ho; Liu, Huiqing; Menéndez-Arias, Luis CSIC ORCID ; Liu, Xinyong; Zhang, Pengartículo
embargoedAccessRNase-H-inhibitors.pdf.jpg5-oct-2022Design, synthesis, and biological evaluation of novel double-winged galloyl derivatives as HIV-1 RNase H inhibitorsZhang, Lina; Wei, Fenju; Borrego, David; Zhao, Fabao; Martínez Del Río, Javier; Frutos-Beltrán, Estrella CSIC ORCID; Zhang, Jiwei; Xu, Shujing; López-Carrobles, Nerea; Gao, Shenghua; Kang, Dongwei; Pannecouque, Christophe; Clercq, Erik De; Liu, Xinyong; Menéndez-Arias, Luis CSIC ORCID ; Zhan, Pengartículo
openAccessMenéndez-AriasL_DiscoveryOptimizationAndTarget.pdf.jpg2021Discovery, optimization, and target identification of novel coumarin derivatives as HIV-1 reverse transcriptase-associated ribonuclease H inhibitorsKang, Dongwei; Urhan, Çagil; Wei, Fenju; Frutos-Beltrán, Estrella CSIC ORCID; Sun, Lin; Álvarez, Mar CSIC ORCID; Feng, Da; Tao, Yucen; Pannecouque, Christophe; De Clercq, Erik; Menéndez-Arias, Luis CSIC ORCID ; Liu, Xinyong; Zhan, Pengartículo
1-s2.0-S2211383523003064-main.pdf.jpg3-ago-2023Emerging drug design strategies in anti-influenza drug discoveryLiu, Chuanfeng; Hu, Lide; Dong, Guanyu; Zhang, Ying; Ferreira da Silva-Júnior, Edeildo; Liu, Xinyong; Menéndez-Arias, Luis CSIC ORCID artículo de revisión
openAccessinfluenza-drug-discovery.pdf.jpgdic-2023Emerging drug design strategies in anti-influenza drug discoveryLiu, Chuanfeng; Hu, Lide; Dong, Guanyu; Zhang, Ying; Ferreira da Silva-Júnior, Edeildo; Liu, Xinyong; Menéndez-Arias, Luis CSIC ORCID ; Zhan, Pengartículo
openAccessMenéndez-AriasL_MedicinalChemistryStrategies.pdf.jpg17-feb-2021Medicinal chemistry strategies for discovering antivirals effective against drug-resistant virusesMa, Yue; Frutos-Beltrán, Estrella CSIC ORCID; Kang, Dongwei; Pannecouque, Christophe; De Clercq, Erik; Menéndez-Arias, Luis CSIC ORCID ; Liu, Xinyong; Zhan, Pengartículo de revisión
openAccessMenéndez-AriasL_MedicinalChemistryStrategies.pdf.jpg17-feb-2021Medicinal chemistry strategies for discovering antivirals effective against drug-resistant virusesMa, Yue; Frutos-Beltrán, Estrella CSIC ORCID; Kang, Dongwei; Pannecouque, Christophe; De Clercq, Erik; Menéndez-Arias, Luis CSIC ORCID ; Liu, Xinyong; Zhan, Pengartículo de revisión
openAccessMenéndez-AriasL_MedicinalChemistryStrategies.pdf.jpg17-feb-2021Medicinal chemistry strategies for discovering antivirals effective against drug-resistant virusesMa, Yue; Frutos-Beltrán, Estrella CSIC ORCID; Kang, Dongwei; Pannecouque, Christophe; De Clercq, Erik; Menéndez-Arias, Luis CSIC ORCID ; Liu, Xinyong; Zhan, Pengartículo de revisión
openAccessnon-covalent-SARS-CoV-2-Mpro-inhibitors.pdf.jpg9-ago-2023Medicinal chemistry strategies towards the development of non-covalent SARS-CoV-2 Mpro inhibitorsSong, Letian; Gao, Shenghua; Ye, Bing; Yang, Mianling; Yusen, Cheng; Kang, Dongwei; Yi, Fan; Sun, Jin-Peng; Menéndez-Arias, Luis CSIC ORCID ; Neyts, Johan; Liu, Xinyong; Zhan, Pengartículo
openAccessMenéndezAriasL_NovelIndolylarylsulfonederivatives.pdf.jpg12-oct-2020Novel indolylarylsulfone derivatives as covalent HIV-1 reverse transcriptase inhibitors specifically targeting the drug-resistant mutant Y181CGao, Ping; Song, Shu; Frutos-Beltrán, Estrella CSIC ORCID; Li, Wenxin; Sun, Bin; Kang, Dongwei; Zou, Jinmi; Zhang, Jian; Pannecouque, Christophe; De Clercq, Erik; Menéndez-Arias, Luis CSIC ORCID ; Zhan, Peng; Liu, Xinyongartículo
openAccessHIV-1-Reverse-Transcriptase.pdf.jpg15-abr-2022Novel RNase H Inhibitors Blocking RNA-directed Strand Displacement DNA Synthesis by HIV-1 Reverse TranscriptaseMartín-Alonso, Samar; Kang, Dongwei; Martínez Del Río, Javier; Luczkowiak, Joanna; Frutos-Beltrán, Estrella CSIC ORCID; Zhang, Lina; Cheng, Xiqiang; Liu, Xinyong; Zhan, Peng; Menéndez-Arias, Luis CSIC ORCID artículo
closedAccessaccesoRestringido.pdf.jpgmay-2023Rapid discovery and crystallography study of highly potent and selective butylcholinesterase inhibitors based on oxime-containing libraries and conformational restriction strategiesJing, Lanlan; Wei, Wenxiu; Meng, Bairu; Chantegreil, Fabien; Nachon, Florian; Martínez Gil, Ana CSIC ORCID ; Wu, Gaochan; Zhao, Huajun; Song, Yuning; Kang, Dongwei; Brazzolotto, Xavier; Zhan, Peng; Liu, Xinyongartículo
closedAccessaccesoRestringido.pdf.jpg2021Search, Identification, and Design of Effective Antiviral Drugs Against Pandemic Human CoronavirusesHuang, Tianguang; Sun, Lin; Kang, Dongwei; Poongavanam, Vasanthanathan; Liu, Xinyong; Zhan, Peng; Menéndez-Arias, Luis CSIC ORCID capítulo de libro
embargoedAccesscccDNA-DDT-Revised-Manuscript.pdf.jpgjul-2023Targeting hepatitis B virus cccDNA levels: Recent progress in seeking small molecule drug candidatesJin, Yu; Wang, Shuo; Xu, Shujing; Zhao, Shujie; Xu, Xiangrui; Poongavanam, Vasanthanathan; Menéndez-Arias, Luis CSIC ORCID ; Zhan, Peng; Liu, Xinyongartículo