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Rights | Preview | Issue Date | Title | Author(s) | Type |
openAccess |  | 28-Jun-2016 | ASS234, As a New Multi-Target Directed Propargylamine for Alzheimer's Disease Therapy | Marco-Contelles, José CSIC ORCID; Unzeta, Mercedes; Bolea, Irene; Esteban, Gerard; Ramsay, Rona R.; Romero, Alejandro CSIC ORCID; Martínez-Murillo, Ricardo CSIC ORCID; Carreiras, M. Carmo; Ismaili, L. | artículo |
closedAccess |  | 2020 | Automated Synthesis of New Quinoxalinetacrines | Bautista-Aguilera, Óscar M.; Ismaili, L.; Chioua, Mourad CSIC ORCID ; Iriepa, Isabel; Martínez-Grau, Angeles; Beadle, C. D.; Vetman, T.; López-Muñoz, Francisco; Marco-Contelles, José CSIC ORCID | artículo |
openAccess |  | 2022 | Benzochromenopyrimidines: Synthesis, Antiproliferative Activity against Colorectal Cancer and Physicochemical Properties | Choura, E.; Elghali, F.; Bernard, P. J.; Msalbi, D.; Marco-Contelles, José CSIC ORCID; Aifa, Sami; Ismaili, L.; Chabchoub, Fakher | artículo |
closedAccess |  | 2021 | (±)- BIGI-3h: Pentatarget-Directed Ligand combining Cholinesterase, Monoamine Oxidase, and Glycogen Synthase Kinase 3β Inhibition with Calcium Channel Antagonism and Antiaggregating Properties for Alzheimer's Disease | Ismaili, L.; Monnin, J.; Etievant, A.; Arribas, R. L.; Viejo, L.; Refouvelet, B.; Soukup, O.; Janockova, J.; Hepnarova, V.; Korábečný, Jan; Kucera, T.; Jun, D.; Andrys, R.; Musilek, K.; Baguet, A.; García-Frutos, Eva M. CSIC ORCID; De Simone, A.; Andrisano, V.; Bartolini, M.; De Los Ríos, C.; Marco-Contelles, José CSIC ORCID; Haffen, E. | artículo |
closedAccess |  | 2021 | (±)- BIGI-3h: Pentatarget-Directed Ligand combining Cholinesterase, Monoamine Oxidase, and Glycogen Synthase Kinase 3β Inhibition with Calcium Channel Antagonism and Antiaggregating Properties for Alzheimer's Disease | Ismaili, L.; Monnin, J.; Etievant, A.; Arribas, R. L.; Viejo, L.; Refouvelet, B.; Soukup, O.; Janockova, J.; Hepnarova, V.; Korábečný, Jan; Kucera, T.; Jun, D.; Andrys, R.; Musilek, K.; Baguet, A.; García-Frutos, Eva M. CSIC ORCID; De Simone, A.; Andrisano, V.; Bartolini, M.; De Los Ríos, C.; Marco-Contelles, José CSIC ORCID; Haffen, E. | artículo |
openAccess |  | 2019 | Donepezil + chromone + melatonin hybrids as promising agents for Alzheimer’s disease therapy | Pachón-Angona, I.; Refouvelet, B.; Andrýs, R.; Martin, Hélène; Luzet, V.; Iriepa, Isabel; Moraleda, I.; Diez-Iriepa, Daniel; Oset-Gasque, María Jesús; Marco-Contelles, José CSIC ORCID; Musilek, K.; Ismaili, L. | artículo |
closedAccess |  | 2015 | Donepezil-ferulic acid hybrids as anti-Alzheimer drugs | Benchekroun, M.; Ismaili, L.; Pudlo, M.; Luzet, V.; Gharbi, T.; Refouvelet, B.; Marco-Contelles, José CSIC ORCID | artículo |
closedAccess |  | 2017 | Facile one-pot synthesis of new [1,2,4]triazolo[1,5-a]pyridine derivatives by ultrasonic irradiation | Zribi, L.; Zribi, F.; Marco-Contelles, José CSIC ORCID; Chabchoub, Fakher; Ismaili, L. | artículo |
openAccess |  | 24-Mar-2016 | Imidazopyranotacrines as Non-Hepatotoxic, Selective Acetylcholinesterase Inhibitors, and Antioxidant Agents for Alzheimer's Disease Therapy | Boulebd, Houssem; Ismaili, L.; Bartolini, Manuela; Bouraiou, Abdelmalek; Andrisano, Vincenza; Martin, Hélène; Bonet, Alexandre; Moraleda, Ignacio; Iriepa, Isabel; Chioua, Mourad CSIC ORCID ; Belfaitah, Ali; Marco-Contelles, José CSIC ORCID | artículo |
closedAccess |  | 2019 | Multi-target 1,4-dihydropyridines showing calcium channel blockade and antioxidant capacity for Alzheimer's disease therapy | Malek, R.; Maj, M.; Wnorowski, A.; Józwiak, K.; Martin, Helene; Iriepa, Isabel; Moraleda, I.; Chabchoub, Fakher; Marco-Contelles, José CSIC ORCID; Ismaili, L. | artículo |
closedAccess |  | 2017 | Multitarget-Directed Ligands Combining Cholinesterase and Monoamine Oxidase Inhibition with Histamine H3R Antagonism for Neurodegenerative Diseases | Bautista-Aguilera, Óscar M.; Hagenow, S.; Palomino-Antolín, Alejandra; Farré-Alins, V.; Ismaili, L.; Joffrin, P. L.; Jimeno, M. Luisa; Soukup, O.; Janockova, Jana; Kalinowski, A.; Proschak, E.; Iriepa, Isabel; Moraleda, I.; Schwed, J. S.; Romero Martínez, Alejandro; López-Muñoz, Francisco; Chioua, Mourad CSIC ORCID ; Egea, Javier; Ramsay, R. R.; Marco-Contelles, José CSIC ORCID; Stark, H. | artículo |
closedAccess |  | 2017 | New (benz)imidazolopyridino tacrines as nonhepatotoxic, cholinesterase inhibitors for Alzheimer disease | Boulebd, Houssem; Ismaili, L.; Martin, Helene; Bonet, A.; Chioua, Mourad CSIC ORCID ; Marco-Contelles, José CSIC ORCID; Belfaitah, A. | artículo |
closedAccess |  | 2019 | New method for the synthesis of 4-aryl-3,4-dihydro-2H-benzo[g]chromene-2,5,10-triones | Choura, E.; Ncir, M.; Maalej, E.; Marco-Contelles, José CSIC ORCID; Ismaili, L.; Chabchoub, Fakher | artículo |
openAccess |  | 2015 | Novel tacrine-grafted ugi adducts as multipotent anti-alzheimer drugs: A synthetic renewal in tacrine-ferulic acid hybrids | Benchekroun, M.; Bartolini, Manuela; Egea, Javier; Romero, A.; Soriano, Elena CSIC; Pudlo, M.; Luzet, Vincenza; Andrisano, V.; Jimeno, M. Luisa CSIC ORCID; López, M. G.; Wehle, S.; Gharbi, T.; Refouvelet, B.; Andrés, L. de; Herrera-Arozamena, Clara; Monti, B.; Bolognesi, Maria Laura; Rodríguez-Franco, María Isabel CSIC ORCID ; Decker, Michael; Marco-Contelles, José CSIC ORCID; Ismaili, L. | artículo |
closedAccess |  | 2020 | Propargylamine-derived multi-target directed ligands for Alzheimer's disease therapy | do Carmo Carreiras, María; Ismaili, L.; Marco-Contelles, José CSIC ORCID | artículo |
closedAccess |  | 2021 | Regioselective Synthesis of Novel [1,2,4]Triazolo[1,5-a]pyridine Derivatives | Hassen, M. B.; Masmoudi, F.; Zribi, L.; Trigui, M.; Ismaili, L.; Marco-Contelles, José CSIC ORCID; Chabchoub, Fakher | artículo |
closedAccess |  | 2021 | Synthesis and Biological Assessment of PyrimidoTacrines as Promising Agents for Alzheimer's Disease Therapy | Dakhlaoui, I.; Maalej, E.; Martin, Helene; Lucht, A.; Iriepa, I.; Moraleda, I.; Marco-Contelles, José CSIC ORCID; Chabchoub, Fakher; Ismaili, L. | artículo |
openAccess |  | 14-May-2016 | Synthesis and Biological Evaluation of Benzochromenopyrimidinones as Cholinesterase Inhibitors and Potent Antioxidant, Non-Hepatotoxic Agents for Alzheimer’s Disease | Dgachi, Youssef; Bautista-Aguilera, Óscar M.; Benchekroun, M.; Martin, Hélène; Bonet, Alexandre; Knez, Damijan; Godyń, Justyna; Malawska, Bárbara; Gobec, Stanislav; Chioua, Mourad CSIC ORCID ; Janockova, Jana; Soukup, O.; Chabchoub, Fakher; Marco-Contelles, José CSIC ORCID; Ismaili, L. | artículo |
closedAccess |  | 2019 | Synthesis and Biological Evaluation of Novel Chromone+Donepezil Hybrids for Alzheimer's Disease Therapy | Malek, R.; Refouvelet, B.; Benchekroun, M.; Iriepa, Isabel; Moraleda, I.; Andrys, R.; Musilek, K.; Marco-Contelles, José CSIC ORCID; Ismaili, L. | artículo |
closedAccess |  | 2021 | Synthesis and Fluorescence of (E)-3-Aryl-2-(5-aryl-4H-1,2,4-triazol-3-yl) Acrylonitriles | Zribi, L.; Ismaili, L.; Vieira-Ferreira, L. F.; Ferreira-Machado, I. L.; Marco-Contelles, José CSIC ORCID; Chabchoub, Fakher | artículo |