Derechos | Preview | Fecha Public. | Título | Autor(es) | Tipo |
embargoedAccess | | 4-abr-2023 | A Potential Boron Neutron Capture Therapy Agent Selectively Suppresses High-Grade Glioma: In Vitro and in Vivo Exploration | Alamón, Catalina; Dávila, Belén; García, María Fernanda; Nievas, Susana; Dagrosa, María Alejandra; Thorp, Silvia; Kovacs, Mariángeles; Trias, Emiliano; Faccio, Ricardo; Gabay, Martín; Zeineh, Nidal; Weizman, Abraham; Teixidor, Francesc CSIC ORCID; Viñas, Clara CSIC ORCID; Gavish, Moshe; Cerecetto, Hugo; Couto, Marcos | artículo |
closedAccess | | 2012 | Amidines bearing benzofuroxan or benzimidazole 1,3-dioxide core scaffolds as Trypanosoma cruzi-inhibitors: Structural basis for their interactions with cruzipain | Merlino, A.; Benítez, Domingo; Campillo, Nuria E. CSIC ORCID ; Páez, Juan A. CSIC ORCID; Tinoco, L. T.; González, Mercedes; Cerecetto, Hugo | artículo |
closedAccess | | 2009 | Anti-trypanosomatid benzofuroxans and deoxygenated analogues: Synthesis using polymer-supported triphenylphosphine, biological evaluation and mechanism of action studies | Castro, Diego; Boiani, Lucía; Benitez, Diego; Hernández, Paola; Merlino, Alicia; Gil, Carmen CSIC ORCID ; Olea-Azar, Claudio; González, Mercedes; Cerecetto, Hugo; Porcal, Williams | artículo |
closedAccess | | 2013 | Artificial neural networks based on CODES descriptors in pharmacology: Identification of novel trypanocidal drugs against chagas disease | Guerra, Ángela CSIC; González-Naranjo, Pedro CSIC ORCID; Campillo, Nuria E. CSIC ORCID ; Cerecetto, Hugo; González, Mercedes; Páez, Juan A. CSIC ORCID | artículo |
closedAccess | | 11-nov-2020 | Bimodal Therapeutic Agents Against Glioblastoma, One of the Most Lethal Forms of Cancer | Couto, Marcos; Alamón, Catalina; Nievas, Susana; Perona, Marina; Dagrosa, María Alejandra; Teixidor, Francesc CSIC ORCID; Cabral, Pablo; Viñas, Clara CSIC ORCID; Cerecetto, Hugo | artículo |
openAccess | | sep-2019 | Carboranylanilinoquinazoline EGFR-inhibitors: toward ‘lead-to-candidate’ stage in the drug-development pipeline | Couto, Marcos; Alamón, Catalina; Sánchez, Carina; Dávila, Belén; Fernández, Marcelo; Lecot, Nicole; Cabral, Pablo; Teixidor, Francesc CSIC ORCID; Viñas, Clara CSIC ORCID; Cerecetto, Hugo | artículo |
openAccess | | 2020 | Closo-Carboranyl- and Metallacarboranyl [1,2,3]triazolyl-Decorated Lapatinib-Scaffold for Cancer Therapy Combining Tyrosine Kinase Inhibition and Boron Neutron Capture Therapy | Couto, Marcos; Alamón, Catalina; García, María Fernanda; Kovacs, Mariángeles; Trias, Emiliano; Nievas, Susana; Pozzi, Emiliano; Curotto, Paula; Thorp, Silvia; Dagrosa, María Alejandra; Teixidor, Francesc CSIC ORCID; Viñas, Clara CSIC ORCID; Cerecetto, Hugo | artículo |
closedAccess | | 2010 | Development of second generation amidinohydrazones, thio- and semicarbazones as Trypanosoma cruzi-inhibitors bearing benzofuroxan and benzimidazole 1,3-dioxide core scaffolds | Merlino, Alicia; Benitez, Diego; Chavez, Santiago; Hernández, Paola; Tinoco, Luzineide W.; Campillo, Nuria E. CSIC ORCID ; Páez, Juan A. CSIC ORCID; Cerecetto, Hugo; González, Mercedes | artículo |
closedAccess | | 2006 | ESR and electrochemical study of 5-nitroindazole derivatives with antiprotozoal activity | Olea-Azar, Claudio; Cerecetto, Hugo; Gerpe, Alejandra; González, Mercedes; Arán, Vicente J. CSIC ORCID; Rigol, C.; Opazo, L. | artículo |
closedAccess | | 31-ago-2021 | Glycogen synthase kinase‑3 maleimide inhibitors as potential PET-tracers for imaging Alzheimer’s disease: 11C‑synthesis and in vivo proof of concept | Giglio, Javier; Fernandez, Soledad; Martínez Gil, Ana CSIC ORCID ; Zeni, Maia; Reyes, L.; Rey, A.; Cerecetto, Hugo | artículo |
closedAccess | | 2007 | In vivo anti-chagas vinylthio-, vinylsulfinyl-, and vinylsulfonylbenzofuroxan derivatives | Porcal, Williams; Hernández, Paola; Boiani, Mariana; Aguirre, Gabriela; Boiani, Lucía; Chidichimo, Agustina; Cazzulo, Juan J.; Campillo, Nuria E. CSIC ORCID ; Páez, Juan A. CSIC ORCID; Castro, Ana CSIC ORCID; Krauth-Siegel, R. Luise; Davies, Carolina; Basombrío, Miguel Ángel; González, Mercedes; Cerecetto, Hugo | artículo |
closedAccess | | 2006 | Indazole N-oxide derivatives as antiprotozoal agents: Synthesis, biological evaluation and mechanism of action studies | Gerpe, Alejandra; Aguirre, Gabriela; Boiani, Lucía; Cerecetto, Hugo; González, Mercedes; Olea-Azar, Claudio; Rigol, C.; Maya, Juan D.; Morello, A.; Piro, Óscar E.; Arán, Vicente J. CSIC ORCID; Azqueta, Amaya; Ceráin, A. L. de; Monge, M. Ángeles CSIC ORCID; Yaluff, G. | artículo |
closedAccess | | 2009 | Interaction studies between human α-tocopherol transfer protein and nitric oxide donor tocopherol analogues with LDL-protective activity | López, Gloria V.; Gómez, Luis E.; Campillo, Nuria E. CSIC ORCID ; Páez, Juan A. CSIC ORCID; Giles, Kaleigh; Atkinson, Jeffrey; González, Mercedes; Rubbo, Homero; Cerecetto, Hugo | artículo |
closedAccess | | 2014 | Mutagenicity of N-oxide containing heterocycles and related compounds: Experimental and theoretical studies | Gabay, Martín; Cabrera, M.; Di Maio, R.; Páez, Juan A. CSIC ORCID; Campillo, Nuria E. CSIC ORCID ; Lavaggi, M. L.; Cerecetto, Hugo | artículo |
openAccess | | 5-ago-2010 | New family of antichagasics derived from imidazo[4,5-c][1,2,6]thiadi azine 2,2-dioxide | Páez, Juan A. CSIC ORCID; Campillo, Nuria E. CSIC ORCID ; Guerra, Ángela CSIC; González Hormaizteguy, M. M; Cerecetto, Hugo | solicitud de patente |
closedAccess | | may-2004 | Novel antiprotozoal products: Imidazole and benzimidazole N-oxide derivatives and related compounds | Aguirre, Gabriela; Boiani, Mariana; Cerecetto, Hugo; Gerpe, Alejandra; González, Mercedes; Fernández Sainz, Yolanda; Denicola, Ana; Ochoa de Ocáriz Herrero, Carmen CSIC ; Nogal, Juan José; Montero, David; Escario, José Antonio | artículo |
closedAccess | | 2005 | Pharmacological properties of indazole derivatives: Recent developments | Cerecetto, Hugo; Gerpe, Alejandra; González, Mercedes; Arán, Vicente J. CSIC ORCID; Ochoa de Ocáriz Herrero, Carmen CSIC | artículo |
openAccess | | 18-nov-2020 | Sunitinib-Containing Carborane Pharmacophore with the Ability to Inhibit Tyrosine Kinases Receptors FLT3, KIT and PDGFR-β, Exhibits Powerful In Vivo Anti-Glioblastoma Activity | Alamón, Catalina; Dávila, Belén; García, María Fernanda; Sánchez, Carina; Kovacs, Mariángeles; Trias, Emiliano; Barbeito, Luis; Gabay, Martín; Zeineh, Nidal; Gavish, Moshe; Teixidor, Francesc CSIC ORCID; Viñas, Clara CSIC ORCID; Couto, Marcos; Cerecetto, Hugo | artículo |
closedAccess | | 2005 | Synthesis and biological properties of new 5-nitroindazole derivatives | Arán, Vicente J. CSIC ORCID; Ochoa, Carmen; Boiani, Lucía; Buccino, Pablo; Cerecetto, Hugo; Gerpe, Alejandra; González, Mercedes; Montero, David; Nogal, Juan José; Gómez-Barrio, Alicia; Azqueta, Amaya; López de Cerain, Adela; Piro, Óscar E.; Castellano, Eduardo E. | artículo |