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Derechos | Preview | Fecha Public. | Título | Autor(es) | Tipo |
openAccess | | 15-may-2019 | 4,4-Disubstituted N-benzylpiperidines: a novel class of fusion inhibitors of influenza virus H1N1 targeting a new binding site in hemagglutinin | Castro, Sonia de CSIC ORCID; Vanderlinden, E.; Ginex, Tiziana CSIC ORCID ; Laporte, M.; Stevaert, L.; Naesens, L.; Luque, F. Javier; Camarasa Rius, María José CSIC ORCID; Velázquez, Sonsoles CSIC ORCID CVN | comunicación de congreso |
closedAccess | | 2009 | 4-Benzyloxy-γ-sultone derivatives: Discovery of a novel family of non-nucleoside inhibitors of human cytomegalovirus and varicella zoster virus | Castro, Sonia de CSIC ORCID; García-Aparicio, C.; Andrei, G.; Snoeck, R.; Balzarini, J.; Camarasa Rius, María José CSIC ORCID; Velázquez, Sonsoles CSIC ORCID CVN | artículo |
closedAccess | | 2022 | 5-Nitroindazole-based compounds: further studies for activity optimization as anti-Trypanosoma cruzi agents | Fonseca-Berzal, Cristina; Ibáñez-Escribano, Alexandra; Castro, Sonia de CSIC ORCID; Escario, José A.; Gómez-Barrio, Alicia; Arán, Vicente J. CSIC ORCID | artículo |
openAccess | | 28-oct-2020 | A genome-scale metabolic reconstruction of Haemophilus influenzae reveals FabH as a potential target for antimicrobial therapeutic development | López-López, Nahikari CSIC ORCID; San León, D.; Castro, Sonia de CSIC ORCID; Díez-Martínez, Roberto CSIC ORCID; Camarasa Rius, María José CSIC ORCID; Menéndez, Margarita CSIC ORCID; Nogales, Juan CSIC ORCID ; Garmendia, Juncal CSIC ORCID | comunicación de congreso |
openAccess | | 2022 | A Versatile Class of 1,4,4-Trisubstituted Piperidines Block Coronavirus Replication In Vitro | Castro, Sonia de CSIC ORCID; Stevaert, Annelies; Maldonado, Miguel CSIC ORCID; Delpal, Adrien; Vandeput, Julie; Van Loy, Benjamin; Eydoux, Cecilia; Guillemot, Jean-Claude; Decroly, Etienne; Gago, Federico CSIC ORCID; Canard, Bruno; Camarasa Rius, María José CSIC ORCID; Velázquez, Sonsoles CSIC ORCID CVN; Naesens, Lieve | artículo |
openAccess | | 2015 | Conservation of antiviral activity and improved selectivity in PMEO-DAPym upon pyrimidine to triazine scaffold hopping | Castro, Sonia de CSIC ORCID; Fernández-Cureses, Gloria CSIC; Andrei, G; Snoeck, R.; Sánchez-Murcia, Pedro A. CSIC ORCID; Korban, B.; Gago, Federico CSIC ORCID; Balzarini, Jan; Camarasa Rius, María José CSIC ORCID | artículo |
closedAccess | | 10-mar-2020 | Design, synthesis and X-Ray crystallography of the complexes of (F)uridylated peptides linked to Vpg1 of Foot-and-Mouth Disease Virus (FMDV) with FMDV RNA-dependent RNA polymerase | Castro, Sonia de CSIC ORCID | comunicación de congreso |
closedAccess | | 14-oct-2014 | Design, synthesis and X-Ray of Foot-and-mouth disease virus (Fluoro)uridylylated peptides linked to the genome (VPgpU and VPgpFU) | Castro, Sonia de CSIC ORCID; Ferrer-Orta, Cristina CSIC ORCID ; Fernández-Cureses, Gloria CSIC; Verdaguer, Núria CSIC ORCID ; Domingo, Esteban CSIC ORCID; Camarasa Rius, María José CSIC ORCID | póster de congreso |
openAccess | | 2015 | Design, synthesis, and biological evaluation of unconventional aminopyrimidine, aminopurine, and amino-1,3,5-triazine methyloxynucleosides | Fernández-Cureses, Gloria CSIC; Castro, Sonia de CSIC ORCID; Jimeno, M. Luisa CSIC ORCID; Balzarini, Jan; Camarasa Rius, María José CSIC ORCID | artículo |
openAccess | | 2015 | Dipeptidyl-peptidase IV (DPP IV/CD26)-activated prodrugs: A successful strategy for improving water solubility and oral bioavailability | Velázquez, Sonsoles CSIC ORCID CVN; Castro, Sonia de CSIC ORCID; Diez-Torrubia, Alberto CSIC; Balzarini, Jan; Camarasa Rius, María José CSIC ORCID | artículo |
closedAccess | | 2014 | Discovery and SAR studies of a novel class of cytotoxic 1,4-disubstituted piperidines via Ugi reaction | Castro, Sonia de CSIC ORCID; Camarasa Rius, María José CSIC ORCID; Balzarini, Jan; Velázquez, Sonsoles CSIC ORCID CVN | artículo |
openAccess | | 2014 | Diseño y desarrollo de una novedosa estrategia profármaco basada en la enzima DPPIV/CD26 | Camarasa Rius, María José CSIC ORCID; Castro, Sonia de CSIC ORCID; Velázquez, Sonsoles CSIC ORCID CVN | artículo |
closedAccess | | 18-sep-2016 | (F)Uridylylated peptides linked to the viral Protein VPg1 of foot-and-mouth disease virus | Camarasa Rius, María José CSIC ORCID; Castro, Sonia de CSIC ORCID; Ferrer-Orta, Cristina CSIC ORCID ; Verdaguer, Núria CSIC ORCID ; Gago, Federico CSIC ORCID | póster de congreso |
openAccess | | 2019 | (F)uridylylated peptides linked to VPg1 of foot-and-mouth disease virus (FMDV): Design, synthesis and X-Ray crystallography of the complexes with FMDV RNA-Dependent RNA Polymerase | Castro, Sonia de CSIC ORCID; Ferrer-Orta, Cristina CSIC ORCID ; Mills, A.; Fernández-Cureses, Gloria CSIC; Gago, Federico CSIC ORCID; Verdaguer, Núria CSIC ORCID ; Camarasa Rius, María José CSIC ORCID | artículo |
openAccess | | 2017 | First example of peptides targeting the dimer interface of Leishmania infantum trypanothione reductase with potent in vitro antileishmanial activity# | Ruiz-Santaquiteria, Marta CSIC ORCID; Sánchez-Murcia, Pedro A. CSIC ORCID; Toro, Miguel Ángel; Lucio, H. de; Gutiérrez, Kilian Jesús; Castro, Sonia de CSIC ORCID; Carneiro, Filipa A. C.; Gago, Federico CSIC ORCID; Jiménez-Ruiz, Antonio; Camarasa Rius, María José CSIC ORCID; Velázquez, Sonsoles CSIC ORCID CVN | artículo |
closedAccess | | 2011 | From β-Amino-γ-sultone to Unusual Bicyclic Pyridine and Pyrazine Heterocyclic Systems: Synthesis and Cytostatic and Antiviral Activities | Castro, Sonia de CSIC ORCID; Familiar, Olga CSIC; Andrei, G; Snoeck, R.; Balzarini, Jan; Camarasa Rius, María José CSIC ORCID; Velázquez, Sonsoles CSIC ORCID CVN | artículo |
openAccess | | 2022 | Identification of 1,2,3-triazolium salt-based inhibitors of Leishmania infantum trypanothione disulfide reductase with enhanced antileishmanial potency in cellulo and increased selectivity | Lucio, Héctor de; Revuelto, Alejandro CSIC ORCID; Carriles, Alejandra A. CSIC ORCID; Castro, Sonia de CSIC ORCID; García-González, Sonia; García-Soriano, Juan Carlos; Alcón-Calderón, Mercedes; Sánchez-Murcia, Pedro A. CSIC ORCID; Hermoso, Juan A. CSIC ORCID; Gago, Federico CSIC ORCID; Camarasa Rius, María José CSIC ORCID; Jiménez-Ruiz, Antonio; Velázquez, Sonsoles CSIC ORCID CVN | artículo |
openAccess | | 2022 | Identification of L. infantum trypanothione synthetase inhibitors with leishmanicidal activity from a (non-biased) in-house chemical library | Alcón-Calderón, Mercedes; Lucio, Héctor de; García-Soriano, Juan Carlos; Revuelto, Alejandro CSIC ORCID; Castro, Sonia de CSIC ORCID; López-Gutiérrez, Celia; San-Félix, Ana CSIC ORCID ; Quesada, Ernesto CSIC ORCID ; Gago, Federico CSIC ORCID; Camarasa Rius, María José CSIC ORCID; Jiménez-Ruiz, Antonio; Velázquez, Sonsoles CSIC ORCID CVN | artículo |
openAccess | | 21-sep-2017 | Improved proteolytic stability and potent activity against Leishmania infantum trypanothione reductase of α/β-peptide foldamers conjugated to cell-penetrating peptides | Lucio, Héctor de; Gamo, Ana María CSIC; Ruiz-Santaquiteria, Marta CSIC ORCID; Castro, Sonia de CSIC ORCID; Sánchez-Murcia, Pedro A. CSIC ORCID; Toro, Miguel Ángel; Gutiérrez, Kilian Jesús; Gago, Federico CSIC ORCID; Jiménez- Ruiz, Antonio; Camarasa Rius, María José CSIC ORCID; Velázquez, Sonsoles CSIC ORCID CVN | artículo |
openAccess | | 16-mar-2022 | Interrogation of Essentiality in the Reconstructed Haemophilus influenzae Metabolic Network Identifies Lipid Metabolism Antimicrobial Targets: Preclinical Evaluation of a FabH β-Ketoacyl-ACP Synthase Inhibitor | López-López, Nahikari CSIC ORCID; San León, David ; Castro, Sonia de CSIC ORCID; Díez-Martínez, Roberto CSIC ORCID; Iglesias-Bexiga, Manuel CSIC; Camarasa Rius, María José CSIC ORCID; Menéndez, Margarita CSIC ORCID; Nogales, Juan CSIC ORCID ; Garmendia, Juncal CSIC ORCID | artículo |