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Rights | Preview | Issue Date | Title | Author(s) | Type |
openAccess |  | 15-May-2019 | 4,4-Disubstituted N-benzylpiperidines: a novel class of fusion inhibitors of influenza virus H1N1 targeting a new binding site in hemagglutinin | Castro, Sonia de; Vanderlinden, E.; Ginex, Tiziana CSIC ORCID ; Laporte, M.; Stevaert, L.; Naesens, L.; Luque, F. Javier; Camarasa Rius, María José CSIC ORCID; Velázquez, Sonsoles CSIC ORCID CVN | comunicación de congreso |
closedAccess | | 2013 | 5'-Trityl-substituted thymidine derivatives as a novel class of antileishmanial agents: Leishmania infantum EndoG as a potential target | Casanova, Elena CSIC; Moreno, David; Gigante, Alba CSIC ORCID; Genes, Carlos Mario; Rico, Eva; Oliva, Cristina; Camarasa Rius, María José CSIC ORCID; Gago, Federico CSIC ORCID; Jiménez-Ruiz, Antonio; Peréz-Pérez, María-Jesús CSIC ORCID | artículo |
closedAccess | | 2010 | 9-Arylpurines as a Novel Class of Enterovirus Inhibitors | Aguado, Leire CSIC; Thibaut, Hendrik Jan; Priego, Eva María CSIC ORCID; Jimeno, M. Luisa CSIC ORCID; Camarasa Rius, María José CSIC ORCID; Neyts, Johan; Peréz-Pérez, María-Jesús CSIC ORCID | artículo |
openAccess | | 28-Oct-2020 | A genome-scale metabolic reconstruction of Haemophilus influenzae reveals FabH as a potential target for antimicrobial therapeutic development | López-López, Nahikari CSIC ORCID; San León, D.; Castro, Sonia de; Díez-Martínez, Roberto CSIC ORCID; Camarasa Rius, María José CSIC ORCID; Menéndez, Margarita CSIC ORCID; Nogales, Juan CSIC ORCID ; Garmendia, Juncal CSIC ORCID | comunicación de congreso |
closedAccess | | 2002 | A new and efficient one-pot synthesis of pyrido[2,1-f]purine-2,4-diones starting from 6-aminouracil derivatives | Pérez Pérez, María Jesús; Priego, Eva María CSIC ORCID; Jimeno, M. Luisa CSIC ORCID; Camarasa Rius, María José CSIC ORCID | artículo |
closedAccess |  | 19-Feb-2019 | A new class of dual HIV and EV71 entry inhibitors: tri and tetrapodal tryptophan derivatives | Martí-Marí, Olaia; Martínez-Gualda, Belén; Puente, Sofia de la; Mirabelli, Carmen; Sun, Liang; Delang, Leen; Schols, Dominique; Neyts, Johan; Camarasa Rius, María José CSIC ORCID; San-Félix, Ana CSIC ORCID CVN | comunicación de congreso |
openAccess |  | 22-Jun-2018 | A Novel Class of Cationic and Non-Peptidic Small Molecules as Hits for the Development of Antimicrobial Agents | Jiménez, A.; García, Pablo; Puente, Sofia de la; Madrona, Andrés; Camarasa Rius, María José CSIC ORCID; Peréz-Pérez, María-Jesús CSIC ORCID ; Quintela Fernández, José Carlos; García del Portillo, Francisco CSIC ORCID ; San-Félix, Ana CSIC ORCID CVN | artículo |
openAccess |  | 3-Apr-2019 | A second-generation of tryptophan-containing small molecules extremely potent against HIV and EV-A71 clinical isolates | Martí-Marí, Olaia; Martínez-Gualda, Belén; Puente-Secades, Sofía de la; Quesada, Ernesto CSIC ORCID ; Sun, Liang; Delang, Leen; Mirabelli, Carmen; Noppen, Sam; Schols, Dominique; Neyts, Johan; Gago, Federico CSIC ORCID; Camarasa Rius, María José CSIC ORCID; San-Félix, Ana CSIC ORCID CVN | actas de congreso |
openAccess |  | 2022 | A Versatile Class of 1,4,4-Trisubstituted Piperidines Block Coronavirus Replication In Vitro | Castro, Sonia de; Stevaert, Annelies; Maldonado, Miguel; Delpal, Adrien; Vandeput, Julie; Van Loy, Benjamin; Eydoux, Cecilia; Guillemot, Jean-Claude; Decroly, Etienne; Gago, Federico CSIC ORCID; Canard, Bruno; Camarasa Rius, María José CSIC ORCID; Velázquez, Sonsoles CSIC ORCID CVN; Naesens, Lieve | artículo |
closedAccess | | 1998 | Abasic analogues of TSAO-T as the first sugar derivatives that specifically inhibit HIV-1 reverse transcriptase | Velázquez, Sonsoles CSIC ORCID CVN; Chamorro, Cristina; Pérez Pérez, María Jesús; Alvarez, Rosa; Jimeno, M. Luisa; Martín Domenech, Angel; Pérez, Carlos; Gago, Federico; De Clercq, Erik; Balzarini, Jan; San-Félix, Ana CSIC ORCID CVN; Camarasa Rius, María José CSIC ORCID | artículo |
openAccess |  | 2015 | Anti-HIV-1 activity of a tripodal receptor that recognizes mannose oligomers | Rivero-Buceta, Eva CSIC; Carrero, Paula CSIC; Casanova, Elena CSIC; García-Doyagüez, Elisa CSIC ORCID; Madrona, Andrés; Quesada, Ernesto; Peréz-Pérez, María-Jesús CSIC ORCID ; Mateos, Raquel CSIC ORCID ; Bravo, Laura CSIC ORCID; Mathys, Leen; Noppen, Sam; Kiselev, Evgency; Marchand, Christophe; Pommier, Yves; Liekens, Sandra; Balzarini, Jan; Camarasa Rius, María José CSIC ORCID; San-Félix, Ana CSIC ORCID CVN | artículo |
openAccess |  | 20-May-2016 | Antivascular and antitumor properties of the tubulin-binding chalcone TUB091 | Canela, María-Dolores CSIC; Noppen, Sam; Bueno, Oskía; Prota, Andrea E.; Bargsten, Katja; Sáez-Calvo, Gonzalo; Jimeno, M. Luisa CSIC ORCID; Benkhei, Mohammed; Ribatti, Domenico; Velázquez, Sonsoles CSIC ORCID CVN; Camarasa Rius, María José CSIC ORCID; Díaz, José Fernando CSIC ORCID ; Steinmetz, Michel O.; Priego, Eva María CSIC ORCID; Peréz-Pérez, María-Jesús CSIC ORCID ; Liekens, Sandra | artículo |
closedAccess |  | 2017 | Antiviral activity of [1,2,3]triazolo[4,5-d]pyrimidin-7(6H)-ones against chikungunya virus targeting the viral capping nsP1 | Gigante, Alba CSIC ORCID; Gómez-SanJuan, Asier CSIC; Delang, Leen; Li, C.; Bueno, Oskía; Gamo, Ana María CSIC; Priego, Eva María CSIC ORCID; Camarasa Rius, María José CSIC ORCID; Jochmans, D.; Leyssen, Pieter; Decroly, E.; Coutard, Bruno; Querat, Guilles; Neyts, Johan; Peréz-Pérez, María-Jesús CSIC ORCID | artículo |
openAccess | | 5-Feb-2020 | Comité Organizador (Congreso Internacional) | Camarasa Rius, María José CSIC ORCID | actas de congreso |
openAccess |  | 2015 | Comparison of hydrocarbon-and lactam-bridged cyclic peptides as dimerization inhibitors of Leishmania infantum trypanothione reductase | Sánchez-Murcia, Pedro A. CSIC ORCID; Ruiz-Santaquiteria, Marta CSIC ORCID; Toro, Miguel A.; Lucio, H. de; Jiménez, M. Angeles CSIC ORCID ; Gago, Federico CSIC ORCID; Jiménez-Ruiz, Antonio; Camarasa Rius, María José CSIC ORCID; Velázquez, Sonsoles CSIC ORCID CVN | artículo |
openAccess |  | 2018 | Conformational mimetics of the α-methyl chalcone TUB091 binding tubulin: Design, synthesis and antiproliferative activity | Bueno, Oskía; Tobajas, Gloria; Quesada, Ernesto; Estévez-Gallego, Juan CSIC ORCID ; Noppen, Sam; Camarasa Rius, María José CSIC ORCID; Díaz, José Fernando CSIC ORCID ; Liekens, Sandra; Priego, Eva María CSIC ORCID; Peréz-Pérez, María-Jesús CSIC ORCID | artículo |
closedAccess | | 1997 | Conformational studies of 3'-spironucleosides (TSAO-T and analogues) by NMR spectroscopy | Álvarez, Rosa; Jimeno, M. Luisa CSIC ORCID; Tomas-Gil, Francisco J.; Pérez Pérez, María Jesús; Camarasa Rius, María José CSIC ORCID | artículo |
openAccess |  | 2015 | Conservation of antiviral activity and improved selectivity in PMEO-DAPym upon pyrimidine to triazine scaffold hopping | Castro, Sonia de; Fernández-Cureses, Gloria CSIC; Andrei, G; Snoeck, R.; Sánchez-Murcia, Pedro A. CSIC ORCID; Korban, B.; Gago, Federico CSIC ORCID; Balzarini, Jan; Camarasa Rius, María José CSIC ORCID | artículo |
closedAccess | | 2011 | Crystal structure of tert -butyldimethylsilyl-spiroaminooxathioledioxide- thymine (TSAO-T) in complex with HIV-1 reverse transcriptase (RT) redefines the elastic limits of the non-nucleoside inhibitor-binding pocket | Das, Krishna; Bauman, J. D.; Rim, A. S.; Dharia, C.; Clark, A. D.; Camarasa Rius, María José CSIC ORCID; Balzarini, Jan; Arnold, E. | artículo |
openAccess |  | 28-Apr-2011 | Derivados de nucleósidos para el tratamiento de infecciones por Leishmania | Gago Badenas, Federico; Rico Galán, Eva; Camarasa Rius, María José CSIC ORCID; Jiménez, A. R.; Casanova Malpica, Elena; Moreno Mateos, David; Peréz-Pérez, María-Jesús CSIC ORCID | patente |