Rights | Preview | Issue Date | Title | Author(s) | Type |
openAccess |  | 17-Dec-2021 | 2-(Piperidin-4-yl)acetamides as Potent Inhibitors of Soluble Epoxide Hydrolase with Anti-Inflammatory Activity | Martín-López, Juan; Codony, Sandra; Bartra Cabré, Clara CSIC ORCID; Morisseau, Christophe; Loza, María Isabel; Sanfeliu, Coral CSIC ORCID; Hammock, Bruce D.; Brea, José; Vázquez, Santiago | artículo |
openAccess |  | 2023 | 8-Amide and 8-carbamate substitution patterns as modulators of 7-hydroxy-4-methylcoumarin's antidepressant profile: Synthesis, biological evaluation and docking studies | Matos, María de Jesús; Novo, Paula; Mayán, Lucía; Torres, I.; Uriarte, Eugenio; Yáñez, Matilde; Fontenla, José Ángel; Ortuso, F.; Alcaro, Stefano; Procopio, Francesca; Rodríguez-Franco, María Isabel CSIC ORCID ; Val, Cristina; Loza, María Isabel; Brea, José; Borges, Fernanda; Viña, Dolores | artículo |
openAccess |  | 3-Apr-2022 | A new family of subnanomolar inhibitors of soluble epoxide hydrolase | Escolano, Carmen; Bagán, Andrea; Turcu, Andreea L.; Morisseau, Christophe; Loza, María Isabel; Brea, José; Bartra Cabré, Clara CSIC ORCID; Sanfeliu, Coral CSIC ORCID; Hammock, Bruce D.; Vázquez, Santiago | póster de congreso |
openAccess |  | 15-Oct-2021 | Benzofuranyl-2-imidazoles as imidazoline I2 receptor ligands for Alzheimer's disease | Rodriguez Arévalo, Sergio; Bagán, Andrea; Griñán Ferré, Christian; Vasilopoulou, Foteini; Pallàs, Mercè; Brocos Mosquera, Iria; Callado, Luis F.; Loza, M Isabel; Martínez, Antón L.; Brea, José; Pérez, Belén; Molins, Elies CSIC ORCID ; De Jonghe, Steven; Daelemans, Dirk; Radan, Milica; Djikic, Teodora; Nikolic, Katarina; Hernández Hernández, Elena; García-Fuster, M. Julia; García Sevilla, Jesús A.; Escolano, Carmen | artículo |
openAccess |  | 9-Apr-2020 | Bicyclic alfa-iminophosphonates as highly affinity imidazoline I2 receptor ligands for Alzheimer’s Disease | Abás, Sònia; Rodríguez Arévalo, Sergio; Bagán, Andrea; Griñán Ferré, Christian; Vasilopoulou, Foteini; Brocos Mosquera, Iria; Muguruza, Carolina; Pérez, Belén; Molins, Elies CSIC ORCID ; Luque, F. Javier; Pérez Lozano, Pilar; Jonghe, Steven de; Daelemans, Dirk; Naesens, Lieve; Brea, José; Loza, María Isabel; Hernández Hernández, Elena; García-Sevilla, Jesús Andrés; García Fuster, M. Julia; Radan, Milica; Djikic, Teodora; Nikolic, Katarina; Pallàs, Mercè; Callado, Luis F.; Escolano, Carmen | artículo |
openAccess |  | 24-Jul-2020 | Centrally Active Multitarget Anti-Alzheimer Agents Derived from the Antioxidant Lead CR-6 | Pérez-Areales, F. Javier; Garrido, María; Aso, Ester; Bartolini, Manuela; De Simone, Angela; Espargaró, Alba; Ginex, Tiziana CSIC ORCID ; Sabate, Raimon; Pérez, Belén; Andrisano, Vincenza; Puigoriol-Illamola, Dolors; Pallàs, Mercè; Luque, F. Javier; Loza, María Isabel; Brea, José; Ferrer, Isidro; Ciruela, Francisco; Messeguer Peypoch, Ángel CSIC ORCID; Muñoz-Torrero, Diego | artículo |
openAccess |  | 29-Nov-2012 | Derivados heterocíclicos inhibidores de fosfodiesterasa 7 | Gil, Carmen CSIC ORCID ; Martínez, Ana CSIC ORCID ; Redondo, Miriam CSIC; Campillo, Nuria E. CSIC ORCID ; Pérez, Daniel I.; Loza, María Isabel; Cadavid, María Isabel; Brea, José; Pérez Castillo, Ana CSIC ORCID | solicitud de patente |
openAccess |  | 2012 | Effect of phosphodiesterase 7 (PDE7) inhibitors in experimental autoimmune encephalomyelitis mice. Discovery of a new chemically diverse family of compounds | Redondo, Miriam CSIC; Brea, José; Pérez, Daniel I.; Soteras, Ignacio CSIC ORCID; Val, Cristina; Pérez, Concepción; Morales-García, José A. CSIC ORCID; Alonso-Gil, Sandra CSIC; Paul-Fernández, Nuria CSIC; Martín-Álvarez, Rocío CSIC; Cadavid, María Isabel; Loza, María Isabel; Pérez Castillo, Ana CSIC ORCID; Mengod Los Arcos, Guadalupe CSIC ORCID; Campillo, Nuria E. CSIC ORCID ; Martínez, Ana CSIC ORCID ; Gil, Carmen CSIC ORCID | artículo |
closedAccess |  | 2014 | Modulation of cAMP-specific PDE without emetogenic activity: New sulfide-like PDE7 inhibitors | García, Ana M. CSIC ORCID; Brea, José; Morales-García, José A. CSIC ORCID; Pérez, Daniel I.; González, A.; Alonso-Gil, Sandra CSIC; Conde, Santiago CSIC; Cadavid, María Isabel; Loza, María Isabel; Pérez Castillo, Ana CSIC ORCID; Martínez, Ana CSIC ORCID ; Gil, Carmen CSIC ORCID | artículo |
closedAccess |  | 2012 | Neuroprotective efficacy of quinazoline type phosphodiesterase 7 inhibitors in cellular cultures and experimental stroke model | Redondo, Miriam CSIC; Zarruk, Juan G.; Ceballos, Placido CSIC; Pérez, Daniel I.; Pérez Martín, María Concepción; Pérez Castillo, Ana CSIC ORCID; Moro, María A.; Brea, José; Val, Cristina; Cadavid, María Isabel; Loza, María Isabel; Campillo, Nuria E. CSIC ORCID ; Martínez, Ana CSIC ORCID ; Gil, Carmen CSIC ORCID | artículo |
closedAccess |  | 2-Jun-2020 | Pharmacological Inhibition of Soluble Epoxide Hydrolase as a New Therapy for Alzheimer's Disease | Griñán-Ferré, Christian; Codony, Sandra; Pujol, Eugènia; Yang, Jun; Leiva, Rosana; Escolano, Carmen; Puigoriol-Illamola, Dolors; Companys-Alemany, Júlia; Corpas, Rubén CSIC ORCID; Sanfeliu, Coral CSIC ORCID; Pérez, Belén; Loza, María Isabel; Brea, José; Morisseau, Christophe; Hammock, Bruce D.; Vázquez, Santiago; Pallàs, Mercè; Galdeano, Carles | artículo |
closedAccess |  | 2017 | Pharmacological tools based on imidazole scaffold proved the utility of PDE10A inhibitors for Parkinson’s disease | García, Ana M. CSIC ORCID; Salado, Irene G. CSIC; Pérez, Daniel I.; Brea, José; Morales-García, José A. CSIC ORCID; González-García, Alejandro; Cadavid, María Isabel; Loza, María Isabel; Luque, F. Javier; Pérez Castillo, Ana CSIC ORCID; Martínez, Ana CSIC ORCID ; Gil, Carmen CSIC ORCID | artículo |
openAccess |  | 3-Apr-2022 | Soluble epoxide hydrolase inhibitors: design, synthesis, in vitro profiling and in vivo evaluation in murine models of pain | Vázquez, Santiago; Codony, Sandra; Entrena, José M.; Jora, Beatrice; González-Cano, Rafael; Loza, María Isabel; Brea, José; Morisseau, Christophe; Bartra Cabré, Clara CSIC ORCID; Sanfeliu, Coral CSIC ORCID; Hammock, Bruce D.; Cobos, Enrique J. | póster de congreso |
closedAccess |  | May-2022 | Soluble Epoxide Hydrolase Inhibitors: Design, Synthesis, in vitro Profiling and in vivo Evaluation in Murine Models of Pain | Vázquez, Santiago; Codony, Sandra; Entrena, José M.; Jora, Beatrice; González-Cano, Rafael; Loza, María Isabel; Brea, José; Morisseau, Christophe; Bartra Cabré, Clara CSIC ORCID; Sanfeliu, Coral CSIC ORCID; Hammock, Bruce D.; Cobos, Enrique J. | artículo |
openAccess |  | 7-Apr-2011 | Substituted 5-IMINO-1,2,4-THIADIAZOLES that can be used to treat neurodegenerative diseases | Martínez, Ana CSIC ORCID ; Gil, Carmen CSIC ORCID ; Palomo, Valle CSIC ORCID ; Pérez, Daniel I.; Pérez Martín, María Concepción; Pérez Castillo, Ana CSIC ORCID; Loza, María Isabel; Cadavid, María Isabel; Brea, José | solicitud de patente |
openAccess |  | 2022 | Synthesis, in vitro profiling and in vivo evaluation of benzohomoadamantane-based ureas for visceral pain: a new indication for soluble epoxide hydrolase inhibitors | Codony, Sandra; Entrena, José M.; Calvó-Tusell, Carla; Osuna, Sílvia; Jora, Beatrice; González-Cano, Rafael; Corpas, Rubén CSIC ORCID; Morisseau, Christophe; Pérez, Belén; Barniol-Xicota, Marta; Griñán-Ferré, Christian; Pérez, Concepción; Rodríguez-Franco, María Isabel CSIC ORCID ; Martínez, Antón L.; Loza, María Isabel; Pallàs, Mercè; Verhelst, Steven H. L.; Sanfeliu, Coral CSIC ORCID; Feixas, Ferran; Hammock, Bruce D.; Brea, José; Cobos, Enrique J.; Vázquez, Santiago | artículo |