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Browsing by Author Brea, José

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Showing results 1 to 16 of 16
RightsPreviewIssue DateTitleAuthor(s)Type
openAccesspharmaceuticals-14-01323-v3.pdf.jpg17-Dec-20212-(Piperidin-4-yl)acetamides as Potent Inhibitors of Soluble Epoxide Hydrolase with Anti-Inflammatory ActivityMartín-López, Juan; Codony, Sandra; Bartra Cabré, Clara CSIC ORCID; Morisseau, Christophe; Loza, María Isabel; Sanfeliu, Coral CSIC ORCID; Hammock, Bruce D.; Brea, José; Vázquez, Santiagoartículo
openAccess1-s2.0-S0223523423000065-main.pdf.jpg20238-Amide and 8-carbamate substitution patterns as modulators of 7-hydroxy-4-methylcoumarin's antidepressant profile: Synthesis, biological evaluation and docking studiesMatos, María de Jesús; Novo, Paula; Mayán, Lucía; Torres, I.; Uriarte, Eugenio; Yáñez, Matilde; Fontenla, José Ángel; Ortuso, F.; Alcaro, Stefano; Procopio, Francesca; Rodríguez-Franco, María Isabel CSIC ORCID ; Val, Cristina; Loza, María Isabel; Brea, José; Borges, Fernanda; Viña, Doloresartículo
openAccessA new family of subnanomolar inhibitors of soluble epoxide hydrolase.pdf.jpg3-Apr-2022A new family of subnanomolar inhibitors of soluble epoxide hydrolaseEscolano, Carmen; Bagán, Andrea; Turcu, Andreea L.; Morisseau, Christophe; Loza, María Isabel; Brea, José; Bartra Cabré, Clara CSIC ORCID; Sanfeliu, Coral CSIC ORCID; Hammock, Bruce D.; Vázquez, Santiagopóster de congreso
openAccessRodriguez_EurJMedChem_2021_editorial.pdf.jpg15-Oct-2021Benzofuranyl-2-imidazoles as imidazoline I2 receptor ligands for Alzheimer's diseaseRodriguez Arévalo, Sergio; Bagán, Andrea; Griñán Ferré, Christian; Vasilopoulou, Foteini; Pallàs, Mercè; Brocos Mosquera, Iria; Callado, Luis F.; Loza, M Isabel; Martínez, Antón L.; Brea, José; Pérez, Belén; Molins, Elies CSIC ORCID ; De Jonghe, Steven; Daelemans, Dirk; Radan, Milica; Djikic, Teodora; Nikolic, Katarina; Hernández Hernández, Elena; García-Fuster, M. Julia; García Sevilla, Jesús A.; Escolano, Carmenartículo
openAccessAbas_JMedChem_2020_postprint.pdf.jpg9-Apr-2020Bicyclic alfa-iminophosphonates as highly affinity imidazoline I2 receptor ligands for Alzheimer’s DiseaseAbás, Sònia; Rodríguez Arévalo, Sergio; Bagán, Andrea; Griñán Ferré, Christian; Vasilopoulou, Foteini; Brocos Mosquera, Iria; Muguruza, Carolina; Pérez, Belén; Molins, Elies CSIC ORCID ; Luque, F. Javier; Pérez Lozano, Pilar; Jonghe, Steven de; Daelemans, Dirk; Naesens, Lieve; Brea, José; Loza, María Isabel; Hernández Hernández, Elena; García-Sevilla, Jesús Andrés; García Fuster, M. Julia; Radan, Milica; Djikic, Teodora; Nikolic, Katarina; Pallàs, Mercè; Callado, Luis F.; Escolano, Carmenartículo
openAccessJMC2020.pdf.jpg24-Jul-2020Centrally Active Multitarget Anti-Alzheimer Agents Derived from the Antioxidant Lead CR-6Pérez-Areales, F. Javier; Garrido, María; Aso, Ester; Bartolini, Manuela; De Simone, Angela; Espargaró, Alba; Ginex, Tiziana CSIC ORCID ; Sabate, Raimon; Pérez, Belén; Andrisano, Vincenza; Puigoriol-Illamola, Dolors; Pallàs, Mercè; Luque, F. Javier; Loza, María Isabel; Brea, José; Ferrer, Isidro; Ciruela, Francisco; Messeguer Peypoch, Ángel CSIC ORCID; Muñoz-Torrero, Diegoartículo
openAccessES2391732A1.pdf.jpg29-Nov-2012Derivados heterocíclicos inhibidores de fosfodiesterasa 7Gil, Carmen CSIC ORCID ; Martínez, Ana CSIC ORCID ; Redondo, Miriam CSIC; Campillo, Nuria E. CSIC ORCID ; Pérez, Daniel I.; Loza, María Isabel; Cadavid, María Isabel; Brea, José; Pérez Castillo, Ana CSIC ORCIDsolicitud de patente
openAccessEffect of phosphodiesterase.pdf.jpg2012Effect of phosphodiesterase 7 (PDE7) inhibitors in experimental autoimmune encephalomyelitis mice. Discovery of a new chemically diverse family of compoundsRedondo, Miriam CSIC; Brea, José; Pérez, Daniel I.; Soteras, Ignacio CSIC ORCID; Val, Cristina; Pérez, Concepción; Morales-García, José A. CSIC ORCID; Alonso-Gil, Sandra CSIC; Paul-Fernández, Nuria CSIC; Martín-Álvarez, Rocío CSIC; Cadavid, María Isabel; Loza, María Isabel; Pérez Castillo, Ana CSIC ORCID; Mengod Los Arcos, Guadalupe CSIC ORCID; Campillo, Nuria E. CSIC ORCID ; Martínez, Ana CSIC ORCID ; Gil, Carmen CSIC ORCID artículo
closedAccessaccesoRestringido.pdf.jpg2014Modulation of cAMP-specific PDE without emetogenic activity: New sulfide-like PDE7 inhibitorsGarcía, Ana M. CSIC ORCID; Brea, José; Morales-García, José A. CSIC ORCID; Pérez, Daniel I.; González, A.; Alonso-Gil, Sandra CSIC; Conde, Santiago CSIC; Cadavid, María Isabel; Loza, María Isabel; Pérez Castillo, Ana CSIC ORCID; Martínez, Ana CSIC ORCID ; Gil, Carmen CSIC ORCID artículo
closedAccessaccesoRestringido.pdf.jpg2012Neuroprotective efficacy of quinazoline type phosphodiesterase 7 inhibitors in cellular cultures and experimental stroke modelRedondo, Miriam CSIC; Zarruk, Juan G.; Ceballos, Placido CSIC; Pérez, Daniel I.; Pérez Martín, María Concepción; Pérez Castillo, Ana CSIC ORCID; Moro, María A.; Brea, José; Val, Cristina; Cadavid, María Isabel; Loza, María Isabel; Campillo, Nuria E. CSIC ORCID ; Martínez, Ana CSIC ORCID ; Gil, Carmen CSIC ORCID artículo
closedAccessaccesoRestringido.pdf.jpg2-Jun-2020Pharmacological Inhibition of Soluble Epoxide Hydrolase as a New Therapy for Alzheimer's DiseaseGriñán-Ferré, Christian; Codony, Sandra; Pujol, Eugènia; Yang, Jun; Leiva, Rosana; Escolano, Carmen; Puigoriol-Illamola, Dolors; Companys-Alemany, Júlia; Corpas, Rubén CSIC ORCID; Sanfeliu, Coral CSIC ORCID; Pérez, Belén; Loza, María Isabel; Brea, José; Morisseau, Christophe; Hammock, Bruce D.; Vázquez, Santiago; Pallàs, Mercè; Galdeano, Carlesartículo
closedAccessaccesoRestringido.pdf.jpg2017Pharmacological tools based on imidazole scaffold proved the utility of PDE10A inhibitors for Parkinson’s diseaseGarcía, Ana M. CSIC ORCID; Salado, Irene G. CSIC; Pérez, Daniel I.; Brea, José; Morales-García, José A. CSIC ORCID; González-García, Alejandro; Cadavid, María Isabel; Loza, María Isabel; Luque, F. Javier; Pérez Castillo, Ana CSIC ORCID; Martínez, Ana CSIC ORCID ; Gil, Carmen CSIC ORCID artículo
openAccessSoluble epoxide hydrolase inhibitors_poster.pdf.jpg3-Apr-2022Soluble epoxide hydrolase inhibitors: design, synthesis, in vitro profiling and in vivo evaluation in murine models of painVázquez, Santiago; Codony, Sandra; Entrena, José M.; Jora, Beatrice; González-Cano, Rafael; Loza, María Isabel; Brea, José; Morisseau, Christophe; Bartra Cabré, Clara CSIC ORCID; Sanfeliu, Coral CSIC ORCID; Hammock, Bruce D.; Cobos, Enrique J.póster de congreso
closedAccessaccesoRestringido.pdf.jpgMay-2022Soluble Epoxide Hydrolase Inhibitors: Design, Synthesis, in vitro Profiling and in vivo Evaluation in Murine Models of PainVázquez, Santiago; Codony, Sandra; Entrena, José M.; Jora, Beatrice; González-Cano, Rafael; Loza, María Isabel; Brea, José; Morisseau, Christophe; Bartra Cabré, Clara CSIC ORCID; Sanfeliu, Coral CSIC ORCID; Hammock, Bruce D.; Cobos, Enrique J.artículo
openAccessWO2011039403A1.pdf.jpg7-Apr-2011Substituted 5-IMINO-1,2,4-THIADIAZOLES that can be used to treat neurodegenerative diseasesMartínez, Ana CSIC ORCID ; Gil, Carmen CSIC ORCID ; Palomo, Valle CSIC ORCID ; Pérez, Daniel I.; Pérez Martín, María Concepción; Pérez Castillo, Ana CSIC ORCID; Loza, María Isabel; Cadavid, María Isabel; Brea, Josésolicitud de patente
openAccessacs.jmedchem.2c00515.pdf.jpg2022Synthesis, in vitro profiling and in vivo evaluation of benzohomoadamantane-based ureas for visceral pain: a new indication for soluble epoxide hydrolase inhibitorsCodony, Sandra; Entrena, José M.; Calvó-Tusell, Carla; Osuna, Sílvia; Jora, Beatrice; González-Cano, Rafael; Corpas, Rubén CSIC ORCID; Morisseau, Christophe; Pérez, Belén; Barniol-Xicota, Marta; Griñán-Ferré, Christian; Pérez, Concepción; Rodríguez-Franco, María Isabel CSIC ORCID ; Martínez, Antón L.; Loza, María Isabel; Pallàs, Mercè; Verhelst, Steven H. L.; Sanfeliu, Coral CSIC ORCID; Feixas, Ferran; Hammock, Bruce D.; Brea, José; Cobos, Enrique J.; Vázquez, Santiagoartículo