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Browsing by Author Balzarini, Jan

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RightsPreviewIssue DateTitleAuthor(s)Type
closedAccess1998Abasic analogues of TSAO-T as the first sugar derivatives that specifically inhibit HIV-1 reverse transcriptaseVelázquez, Sonsoles CSIC ORCID CVN; Chamorro, Cristina; Pérez Pérez, María Jesús; Alvarez, Rosa; Jimeno, M. Luisa; Martín Domenech, Angel; Pérez, Carlos; Gago, Federico; De Clercq, Erik; Balzarini, Jan; San-Félix, Ana CSIC ORCID CVN; Camarasa Rius, María José CSIC ORCIDartículo
openAccessaccesoRestringido.pdf.jpg2015Anti-HIV-1 activity of a tripodal receptor that recognizes mannose oligomersRivero-Buceta, Eva CSIC; Carrero, Paula CSIC; Casanova, Elena CSIC; García-Doyagüez, Elisa CSIC ORCID; Madrona, Andrés; Quesada, Ernesto; Peréz-Pérez, María-Jesús CSIC ORCID ; Mateos, Raquel CSIC ORCID ; Bravo, Laura CSIC ORCID; Mathys, Leen; Noppen, Sam; Kiselev, Evgency; Marchand, Christophe; Pommier, Yves; Liekens, Sandra; Balzarini, Jan; Camarasa Rius, María José CSIC ORCID; San-Félix, Ana CSIC ORCID CVNartículo
closedAccessArtículo.pdf.jpg2001Anti-HIV-1 activity of benzothiadiazine dioxideMartínez, Ana CSIC ORCID ; Gil, Carmen ; Castro, Ana CSIC ORCID; Pérez, Concepción; Witvrouw, M.; Pannecouque, C.; Balzarini, Jan; De Clercq, Erikartículo
openAccessCarbohydrate_Binding_Plos_Pathogens_2016.pdf.jpg23-Sep-2016Carbohydrate-Binding Non-Peptidic Pradimicins for the Treatment of Acute Sleeping Sickness in Murine ModelsCastillo Acosta, Víctor M.; Ruiz-Pérez, Luis Miguel; Etxebarria, Juan; Reichardt, Niels Christian; Navarro, M.; Igarashi, Yasuhiro; Liekens, Sandra; Balzarini, Jan; González-Pacanowska, D.artículo
openAccessMJC-1.pdf.jpg2015Conservation of antiviral activity and improved selectivity in PMEO-DAPym upon pyrimidine to triazine scaffold hoppingCastro, Sonia de; Fernández-Cureses, Gloria CSIC; Andrei, G; Snoeck, R.; Sánchez-Murcia, Pedro A. CSIC ORCID; Korban, B.; Gago, Federico CSIC ORCID; Balzarini, Jan; Camarasa Rius, María José CSIC ORCIDartículo
closedAccess2011Crystal structure of tert -butyldimethylsilyl-spiroaminooxathioledioxide- thymine (TSAO-T) in complex with HIV-1 reverse transcriptase (RT) redefines the elastic limits of the non-nucleoside inhibitor-binding pocketDas, Krishna; Bauman, J. D.; Rim, A. S.; Dharia, C.; Clark, A. D.; Camarasa Rius, María José CSIC ORCID; Balzarini, Jan; Arnold, E.artículo
openAccessMJC-3.pdf.jpg2015Design, synthesis, and biological evaluation of unconventional aminopyrimidine, aminopurine, and amino-1,3,5-triazine methyloxynucleosidesFernández-Cureses, Gloria CSIC; Castro, Sonia de; Jimeno, M. Luisa CSIC ORCID; Balzarini, Jan; Camarasa Rius, María José CSIC ORCIDartículo
closedAccess2011Dipeptidyl peptidase IV dependent water-soluble prodrugs of highly lipophilic bicyclic nucleoside analoguesDiez-Torrubia, Alberto CSIC; Balzarini, Jan; Andrei, G; Snoeck, R.; De Meester, Ingrid; Camarasa Rius, María José CSIC ORCID; Velázquez, Sonsoles CSIC ORCID CVNartículo
closedAccess2012Dipeptidyl Peptidase IV-Activated Prodrugs of Anti- Varicella Zoster Virus Bicyclic Nucleoside Analogues Containing Different Self-Cleavage Spacer SystemsDiez-Torrubia, Alberto CSIC; Cabrera, Silvia CSIC ORCID; De Meester, Ingrid; Camarasa Rius, María José CSIC ORCID; Balzarini, Jan; Velázquez, Sonsoles CSIC ORCID CVNartículo
openAccessMJC-2.pdf.jpg2015Dipeptidyl-peptidase IV (DPP IV/CD26)-activated prodrugs: A successful strategy for improving water solubility and oral bioavailabilityVelázquez, Sonsoles CSIC ORCID CVN; Castro, Sonia de; Diez-Torrubia, Alberto CSIC; Balzarini, Jan; Camarasa Rius, María José CSIC ORCIDartículo
closedAccess3-Feb-2012Dipeptidyl-peptidase IV (DPPIV/CD26)-based prodrugs of hydroxy-containing drugsDiez-Torrubia, Alberto CSIC; Cabrera, Silvia CSIC ORCID; Lambeir, Anne-Marie; Balzarini, Jan; Camarasa Rius, María José CSIC ORCID; Velázquez, Sonsoles CSIC ORCID CVNartículo
closedAccessaccesoRestringido.pdf.jpg2014Discovery and SAR studies of a novel class of cytotoxic 1,4-disubstituted piperidines via Ugi reactionCastro, Sonia de; Camarasa Rius, María José CSIC ORCID; Balzarini, Jan; Velázquez, Sonsoles CSIC ORCID CVNartículo
openAccessExposure_pntd.PDF.jpg6-Mar-2015Exposure of Trypanosoma brucei to an N-acetylglucosamine-Binding Lectin Induces VSG Switching and Glycosylation Defects Resulting in Reduced InfectivityCastillo Acosta, Víctor M.; Ruiz-Pérez, Luis Miguel; Van Damme, Els J. M.; Balzarini, Jan; González-Pacanowska, D.artículo
closedAccess2011From β-Amino-γ-sultone to Unusual Bicyclic Pyridine and Pyrazine Heterocyclic Systems: Synthesis and Cytostatic and Antiviral ActivitiesCastro, Sonia de; Familiar, Olga CSIC; Andrei, G; Snoeck, R.; Balzarini, Jan; Camarasa Rius, María José CSIC ORCID; Velázquez, Sonsoles CSIC ORCID CVNartículo
openAccessWO2011085454A1.pdf.jpg21-Jul-2011gp120 -binding benzene compounds and saccharide compoundsBalzarini, Jan; Carrero, Paula CSIC; Casanova, Elena; Peréz-Pérez, María-Jesús CSIC ORCID ; San-Félix, Ana CSIC ORCID CVNsolicitud de patente
closedAccess2000HIV-1 specific reverse transcriptase inhibitors: Why are TSAO-nucleosides so unique?Camarasa Rius, María José CSIC ORCID; San-Felix, Alejandra; Pérez Pérez, María Jesús; Velázquez, Sonsoles CSIC ORCID CVN; Álvarez, Rosa; Chamorro, Cristina; Jimeno, M. Luisa CSIC ORCID; Perez, Carlos; Gago, Federico CSIC ORCID; De Clercq, Erik; Balzarini, Janartículo
closedAccessaccesoRestringido.pdf.jpg2009Identification of aspartic acid-203 in human thymidine phosphorylase as an important residue for both catalysis and non-competitive inhibition by the small molecule >crystallization chaperone> 5′-O-tritylinosine (KIN59)Bronckaers, A.; Aguado, Leire CSIC; Negri, Ana; Camarasa Rius, María José CSIC ORCID; Balzarini, Jan; Peréz-Pérez, María-Jesús CSIC ORCID ; Gago, Federico CSIC ORCID; Liekens, S.artículo
openAccessWO2009030410A1.pdf.jpg12-Mar-2009Improvements in or relating to compositions for the treatment or prophylaxis of viral infectionsBalzarini, Jan; Camarasa Rius, María José CSIC ORCID; Velázquez, Sonsoles CSIC ORCID CVNpatente
openAccessASF2Manuscript EJMECH-D-14-01438R2.pdf.jpg2015Linear and branched alkyl-esters and amides of gallic acid and other (mono-, di- and tri-) hydroxy benzoyl derivatives as promising anti-HCV inhibitorsRivero-Buceta, Eva CSIC; Carrero, P.; García-Doyagüez, Elisa CSIC ORCID; Madrona, Andrés; Quesada, Ernesto CSIC ORCID ; Camarasa Rius, María José CSIC ORCID; Peréz-Pérez, María-Jesús CSIC ORCID ; Leyssen, Pieter; Paeshuyse, Jan; Balzarini, Jan; Neyts, Johan; San-Félix, Ana CSIC ORCID CVNartículo
openAccessGigante_full_article.pdf.jpg2014Microwave-assisted synthesis of C-8 aryl and heteroaryl inosines and determination of their inhibitory activities against Plasmodium falciparum purine nucleoside phosphorylaseGigante, Alba CSIC ORCID; Priego, Eva María CSIC ORCID; Sánchez-Carrasco, Paula; Ruiz-Pérez, Luis Miguel; Vande Voorde, Johan; Camarasa Rius, María José CSIC ORCID; Balzarini, Jan; González-Pacanowska, D.; Peréz-Pérez, María-Jesús CSIC ORCID artículo