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Derechos | Preview | Fecha Public. | Título | Autor(es) | Tipo |
openAccess | | 4-may-2017 | 5-NITROINDAZOLE derivatives and use thereof as antiprotozoal agents | Escario, José Antonio; Gómez-Barrio, Alicia; Nogal-Ruiz, Juan José; Ibanez Escribano, Alexandra; Fonseca-Berzal, Cristina; Arán, Vicente J. CSIC ORCID; Reviriego, Felipe CSIC ORCID; Cumella Montánchez, José María CSIC | solicitud de patente |
openAccess | | ago-2022 | 5-Nitroindazole derivatives as potential therapeutic alternatives against Acanthamoeba castellanii | Martín-Escolano, Rubén; Pérez-Cordón, Gregorio; Arán, Vicente J. CSIC ORCID; Marín, Clotilde; Sánchez-Moreno, Manuel; Rosales, María José | artículo |
closedAccess | | 2022 | 5-Nitroindazole-based compounds: further studies for activity optimization as anti-Trypanosoma cruzi agents | Fonseca-Berzal, Cristina; Ibáñez-Escribano, Alexandra; Castro, Sonia de CSIC ORCID; Escario, José A.; Gómez-Barrio, Alicia; Arán, Vicente J. CSIC ORCID | artículo |
closedAccess | | 2005 | A computer-based approach to the rational discovery of new trichomonacidal drugs by atom-type linear indices | Marrero-Ponce, Yovani; Machado-Tugores, Yanesty; Pereira, David M.; Escario, José Antonio; Barrio, Alicia G.; Nogal-Ruiz, Juan José; Ochoa, Carmen; Arán, Vicente J. CSIC ORCID; Martínez-Fernández, Antonio R.; García Sánchez, Roy N.; Montero-Torres, Alina; Torrens, Francisco; Meneses-Marcel, Alfredo | artículo |
closedAccess | | 2005 | A linear discrimination analysis based virtual screening of trichomonacidal lead-like compounds: Outcomes of in silico studies supported by experimental results | Meneses-Marcel, Alfredo; Marrero-Ponce, Yovani; Machado-Tugores, Yanesty; Montero-Torres, Alina; Montero Pereira, David; Escario, José Antonio; Nogal-Ruiz, Juan José; Ochoa, Carmen; Arán, Vicente J. CSIC ORCID; Martínez-Fernández, Antonio R.; García Sánchez, Roy N. | artículo |
closedAccess | | 2005 | A novel non-stochastic quadratic fingerprints-based approach for the 'in silico' discovery of new antitrypanosomal compounds | Montero-Torres, Alina; Vega, María Celeste; Marrero-Ponce, Yovani; Rolón, Miriam; Gómez-Barrio, Alicia; Escario, José Antonio; Arán, Vicente J. CSIC ORCID; Martínez-Fernández, Antonio R.; Meneses-Marcel, Alfredo | artículo |
closedAccess | | 2014 | A sequential procedure for rapid and accurate identification of putative trichomonacidal agents | Ibáñez-Escribano, Alexandra; Meneses-Marcel, Alfredo; Marrero-Ponce, Yovani; Nogal-Ruiz, Juan José; Arán, Vicente J. CSIC ORCID; Gómez-Barrio, Alicia; Escario, José Antonio | artículo |
closedAccess | | 2020 | Activity profile of two 5-nitroindazole derivatives over the moderately drug-resistant Trypanosoma cruzi Y strain (DTU TcII): in vitro and in vivo studies | Fonseca-Berzal, Cristina; da Silva, C. F.; Batista, D. d. G. J.; de Oliveira, G. M.; Cumella, José; Batista, M. M.; Peres, R. B.; Silva da Gama Nefertiti, A.; Escario, José Antonio; Gómez-Barrio, A.; Arán, Vicente J. CSIC ORCID; Soeiro, M. d. N. C. | artículo |
openAccess | | 8-feb-2018 | Aminas derivadas de 5- Nitroindazol con propiedades antiprotozoarias | Escario, José Antonio; Gómez-Barrio, Alicia; Nogal Ruíz, Juan José; Fonseca-Berzal, Cristina; Arán, Vicente J. CSIC ORCID; Dardonville, Christophe CSIC ORCID ; Vela, Nerea CSIC; Sifontes-Rodríguez, S.; Meneses-Marcel, Alfredo | patente |
openAccess | | 8-feb-2018 | Aminas derivadas de 5-Nitroindazol con propiedades antiprotozoarias | Escario, José Antonio; Gómez-Barrio, Alicia; Nogal Ruíz, Juan José; Fonseca-Berzal, Cristina; javascript:void(0);; Arán, Vicente J. CSIC ORCID; Dardonville, Christophe CSIC ORCID ; Vela, Nerea CSIC; Sifontes-Rodríguez, S; Meneses-Marcel, Alfredo | solicitud de patente |
openAccess | | 25-abr-2019 | Amines derived from 2-benzyl-5-nitroindazole with antiprotozoal properties against trypanosoma, leishmania and trichomonas | Escario, José Antonio; Gómez-Barrio, Alicia; Nogal Ruíz, Juan José; Fonseca-Berzal, Cristina; Arán, Vicente J. CSIC ORCID; Dardonville, Christophe CSIC ORCID ; Vela, Nerea CSIC; Sifontes-Rodríguez, S; Meneses-Marcel, Alfredo | solicitud de patente |
closedAccess | | 2018 | Antichagasic, Leishmanicidal, and Trichomonacidal Activity of 2-Benzyl-5-nitroindazole-Derived Amines | Fonseca-Berzal, Cristina; Ibáñez-Escribano, Alexandra; Vela, Nerea CSIC; Cumella, José; Nogal-Ruiz, Juan José; Escario, José Antonio; da Silva, P. B.; Soeiro, M. N. C.; Sifontes-Rodríguez, S; Meneses-Marcel, Alfredo; Gómez-Barrio, Alicia; Arán, Vicente J. CSIC ORCID | artículo |
openAccess | | 2012 | Antileishmanial, antitrypanosomal and cytotoxic screening of ethnopharmacologically selected Peruvian plants | González-Coloma, Azucena CSIC ORCID; Reina, Matías CSIC; Sáenz, Claudia; Lacret, Rodney; Ruiz Mesia, Lastenia; Arán, Vicente J. CSIC ORCID; Sanz Perucha, Jesús CSIC; Martínez Díaz, Rafael | artículo |
openAccess | | 2019 | Antimalarial quinoline drugs inhibit β-hematin and increase free hemin catalyzing peroxidative reactions and inhibition of cysteine proteases | Herraiz Tomico, Tomás CSIC ORCID ; Guillén Fuerte, Hugo CSIC; González Peña, Diana CSIC; Arán, Vicente J. CSIC ORCID | artículo |
closedAccess | | 2014 | Antiprotozoan lead discovery by aligning dry and wet screening: Prediction, synthesis, and biological assay of novel quinoxalinones | Martins Alho, Miriam A.; Marrero-Ponce, Yovani; Barigye, S. J.; Meneses-Marcel, Alfredo; Machado Tugores, Y.; Montero-Torres, Alina; Gómez-Barrio, Alicia; Nogal, Juan José; García-Sánchez, R. N.; Vega, María Celeste; Rolón, M.; Martínez-Fernández, Antonio R.; Escario, José Antonio; Pérez-Giménez, F.; Garcia-Domenech, Ramon; Rivera, N.; Mondragón, R.; Mondragón, M.; Ibarra-Velarde, Froylán; López-Arencibia, A.; Martín-Navarro, C.; Lorenzo-Morales, J.; Cabrera-Serra, M. G.; Piñero, J.; Tytgat, J.; Chicharro, Roberto CSIC; Arán, Vicente J. CSIC ORCID | artículo |
closedAccess | | 2012 | Biological and chemical study of fused tri- and tetracyclic indazoles and analogues with important antiparasitic activity | Díaz-Urrua, Christian A.; Olea-Azar, Claudio; Zapata, Gerald A.; Lapier, Michael; Mura, Francisco; Aguilera-Venegas, Benjamín; Arán, Vicente J. CSIC ORCID; López-Múñoz, Rodrigo A.; Maya, Juan D. | artículo |
closedAccess | | 2013 | Biological assay of a novel quinoxalinone with antimalarial efficacy on Plasmodium yoelii yoelii | Rivera, Nrma; Marrero Ponce, Yovani; Arán, Vicente J. CSIC ORCID; Martínez, Cecilia; Malagón, Filiberto | artículo |
closedAccess | | 2014 | Cannabinoid agonists showing BuChE inhibition as potential therapeutic agents for Alzheimer's disease | González-Naranjo, Pedro CSIC ORCID; Pérez-Macías, Natalia CSIC ORCID; Campillo, Nuria E. CSIC ORCID ; Pérez, Concepción CSIC ORCID; Arán, Vicente J. CSIC ORCID; Girón, Rocío CSIC ORCID; Sánchez-Robles, E.; Martín, M. Isabel CSIC; Gómez-Cañas, María; García-Arencibia, Moisés; Fernández-Ruiz, Javier; Páez, Juan A. CSIC ORCID | artículo |
closedAccess | | 2008 | Characterization, phase-solubility, and molecular modeling of inclusion complex of 5-nitroindazole derivative with cyclodextrins | Jullian, Carolina; Morales-Montecinos, J.; Zapata-Torres, G.; Aguilera, Benjamín; Rodríguez, J.; Arán, Vicente J. CSIC ORCID; Olea-Azar, Claudio | artículo |
closedAccess | | 2006 | Comparative aromatic hydroxylation and N-demethylation of MPTP neurotoxin and its analogs, N-methylated β-carboline and isoquinoline alkaloids, by human cytochrome P450 2D6 | Herraiz, Tomás; Guillén, Hugo; Arán, Vicente J. CSIC ORCID; Idle, Jeffrey R.; González, Frank J. | artículo |