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Derechos | Preview | Fecha Public. | Título | Autor(es) | Tipo |
openAccess | | 2020 | N-benzyl 4,4-disubstituted piperidines as a potent class of influenza H1N1 virus inhibitors showing a novel mechanism of hemagglutinin fusion peptide interaction | Castro, Sonia de CSIC ORCID; Ginex, Tiziana CSIC ORCID ; Vanderlinden, E.; Laporte, M.; Stevaert, A.; Cumella, José; Gago, Federico CSIC ORCID; Camarasa Rius, María José CSIC ORCID; Luque, F. Javier; Naesens, L.; Velázquez, Sonsoles CSIC ORCID CVN | artículo |
openAccess | | 2005 | Novel [2′,5′-Bis-O-(tert-butyldimethylsily)-β-D- ribofuranosyl]-3′-spiro-5″-(4″-amino-1″, 2″-oxathiole-2″,2″-diozide) derivatives with anti-HIV-1 and anti-human-cytomegalovirus activity | Castro, Sonia de CSIC ORCID ; Lobatón, E.; Peréz-Pérez, María-Jesús CSIC ORCID ; San-Félix, Ana CSIC ORCID ; Cordeiro, A.; Andrei, G.; Snoeck, R.; De Clercq, E.; Balzarini, J.; Camarasa Rius, María José CSIC ORCID; Velázquez, Sonsoles CSIC ORCID CVN | artículo |
closedAccess | | 2007 | NOVEL NON-NUCLEOSIDE HUMAN CYTOMEGALOVIRUS INHIBITORS BASED UPON TSAO NUCLEOSIDE DERIVATIVES:STRUCTURE-ACTIVITY RELATIONSHIPS | Castro, Sonia de CSIC ORCID ; Andrei, Graziela; Snoeck, Robert; Balzarini, Jan; Camarasa Rius, María José CSIC ORCID; Velázquez, Sonsoles CSIC ORCID CVN | artículo |
closedAccess | | 2013 | Novel water-soluble prodrugs of acyclovir cleavable by the dipeptidyl-peptidase IV (DPP IV/CD26) enzyme | Diez-Torrubia, Alberto CSIC; Cabrera, Silvia CSIC ORCID; Castro, Sonia de CSIC ORCID; García-Aparicio, Carlos CSIC; Mulder, Gwenn; De Meester, Ingrid; Camarasa Rius, María José CSIC ORCID; Balzarini, Jan; Velázquez, Sonsoles CSIC ORCID CVN; Diez-Torrubia, Alberto CSIC | artículo |
openAccess | | 27-may-2021 | Peptides containing -Dalanine (D-ala) or related amino alcohols | García del Portillo, Francisco CSIC ORCID ; Rico Pérez, Gadea; Ramos Marquès, Estel; San-Félix, Ana CSIC ORCID ; Velázquez, Sonsoles CSIC ORCID CVN; Puente-Secades, Sofía de la CSIC; Doyagüez, Elisa G. CSIC | solicitud de patente |
openAccess | | 2020 | Peptides mimicking the β7/β8 loop of HIV'1 reverse transcriptase p51 as “hotspot-targeted” dimerization inhibitors | Sánchez-Murcia, Pedro A. CSIC ORCID; Castro, Sonia de CSIC ORCID; García-Aparicio, Carlos CSIC; Jiménez, M. Angeles CSIC ORCID ; Corona, A.; Tramontano, Enzo; Sluis-Cremer, N.; Menéndez-Arias, Luis CSIC ORCID ; Velázquez, Sonsoles CSIC ORCID CVN; Gago, Federico CSIC ORCID; Camarasa Rius, María José CSIC ORCID | artículo |
openAccess | | ene-2022 | Peptidoglycan editing in non-proliferating intracellular Salmonella as source of interference with immune signaling | Hernández, Sara B.; Castanheira, Sonia; Pucciarelli,M. Graciela; Cestero, Juan J.; Rico-Pérez, Gadea; Paradela, Alberto; Ayala, Juan A.; Velázquez, Sonsoles CSIC ORCID CVN; San-Félix, Ana CSIC ORCID ; Cava, Felipe CSIC ORCID; García del Portillo, Francisco CSIC ORCID | artículo |
openAccess | | 25-ene-2022 | Peptidoglycan editing in non-proliferating intracellular Salmonella as source of interference with immune signaling | Hernández, Sara B.; Castanheira, Sónia CSIC ORCID; Pucciarelli, María Graciela CSIC ORCID; Cestero, Juan J; Rico-Pérez, Gadea; Paradela, Alberto; Ayala, Juan A; Velázquez, Sonsoles CSIC ORCID CVN; San-Félix, Ana CSIC ORCID ; Cava, Felipe CSIC ORCID; García del Portillo, Francisco CSIC ORCID | artículo |
openAccess | | 19-may-2021 | Péptidos que contienen D-Alanina (D-Ala) o aminoalcoholes relacionados | García del Portillo, Francisco CSIC ORCID ; Rico Pérez, Gadea; Ramos Marquès, Estel; San-Félix, Ana CSIC ORCID ; Velázquez, Sonsoles CSIC ORCID CVN; Puente-Secades, Sofía de la CSIC; Doyagüez, Elisa G. CSIC | solicitud de patente |
closedAccess | | 1999 | Potential multifunctional inhibitors of HIV-1 reverse transcriptase. Novel [AZT]-[TSAO-T] and [d4T]-[TSAO-T] heterodimers modified in the linker and in the dideoxynucleoside region | Velázquez, Sonsoles CSIC ORCID CVN; Tuñón, Victoria; Jimeno, M. Luisa CSIC ORCID; Chamorro, Cristina CSIC; De Clercq, Erik; Balzarini, Jan; Camarasa, María José | artículo |
closedAccess | | 6-jun-2013 | Probing the Dimerization Interface of Leishmania infantum Trypanothione Reductase with Site-Directed Mutagenesis and Short Peptides | Toro, Miguel Ángel; Sánchez-Murcia, Pedro A. CSIC ORCID; Moreno, David; Ruiz-Santaquiteria, Marta CSIC ORCID; Alzate, Juan Fernando; Negri, Ana; Camarasa Rius, María José CSIC ORCID; Gago, Federico CSIC ORCID; Velázquez, Sonsoles CSIC ORCID CVN; Jiménez-Ruiz, Antonio | artículo |
openAccess | | 18-nov-2004 | Produgs cleavable by CD26. | Balzarini, Jan; Camarasa Rius, María José CSIC ORCID; Velázquez, Sonsoles CSIC ORCID CVN | patente |
openAccess | | 2020 | Pseudoirreversible slow-binding inhibition of trypanothione reductase by a protein–protein interaction disruptor | Lucio, Héctor de; Toro, Miguel Ángel; Camarasa Rius, María José CSIC ORCID; Velázquez, Sonsoles CSIC ORCID CVN; Gago, Federico CSIC ORCID; Jimenez-Ruiz, Antonio | artículo |
openAccess | | 2019 | Pyrrolopyrimidine vs imidazole-phenyl-thiazole scaffolds in nonpeptidic dimerization inhibitors of leishmania infantum trypanothione reductase | Revuelto, Alejandro CSIC ORCID; Ruiz-Santaquiteria, Marta CSIC ORCID; Lucio, Héctor de; Gamo, Ana; Carriles, Alejandra A. CSIC ORCID; Gutiérrez, Kilian Jesús; Sánchez-Murcia, Pedro A. CSIC ORCID; Gago, Federico CSIC ORCID; Camarasa Rius, María José CSIC ORCID; Jiménez-Ruiz, Antonio; Velázquez, Sonsoles CSIC ORCID CVN | artículo |
closedAccess | | 2008 | Reactivity of the 4-amino-5H-1,2-oxathiole-2,2-dioxide heterocyclic system: A combined experimental and theoretical study | Castro, Sonia de CSIC ORCID ; Peromingo, M. T.; Lozano, Ángel E. ; Camarasa Rius, María José CSIC ORCID; Velázquez, Sonsoles CSIC ORCID CVN | artículo |
closedAccess | | 2001 | Second generation of TSAO compounds directed against HIV-1 TSAO-resistant strains | Lobaton, E.; Velázquez, Sonsoles CSIC ORCID CVN; Peréz-Pérez, María-Jesús CSIC ORCID ; Jimeno, M. Luisa CSIC ORCID; San-Felix, S.; De Clercq, Erik; Balzarini, Jan; Camarasa Rius, María José CSIC ORCID | artículo |
openAccess | | 17-jul-2021 | Small Molecule–Peptide Conjugates as Dimerization Inhibitors of Leishmania infantum Trypanothione Disulfide Reductase | Revuelto, Alejandro CSIC ORCID; López-Martín, Isabel; Lucio, Héctor de; García-Soriano, Juan Carlos; Zanda, Nicola; Castro, Sonia de CSIC ORCID; Gago, Federico CSIC ORCID; Jiménez-Ruiz, Antonio; Velázquez, Sonsoles CSIC ORCID CVN; Camarasa Rius, María José CSIC ORCID | artículo |
closedAccess | | 1995 | Synthesis and Anti-HIV Activity of [UT]-[TSAO-TI and [UT]-[HEPT] Dimers as Potential Multifunctional Inhibitors of HIV-1 Reverse Transcriptase | Velázquez, Sonsoles CSIC ORCID CVN; Álvarez, Rosa; San-Félix, Ana CSIC ORCID ; Jimeno, M. Luisa CSIC ORCID; De Clercq, Erik; Camarasa Rius, María José CSIC ORCID | artículo |
closedAccess | | 2003 | Synthesis and structural characterization of pyrimidine bi- and tricyclic nucleosides with sugar puckers conformationally locked into the eastern region of the pseudorotational cycle | Chamorro, Cristina CSIC; Luengo, Santos M.; Bonache, María-Cruz CSIC; Velázquez, Sonsoles CSIC ORCID CVN; Peréz-Pérez, María-Jesús CSIC ORCID ; Camarasa Rius, María José CSIC ORCID; Gago, Federico CSIC ORCID; Jimeno, M. Luisa CSIC ORCID; San-Félix, Ana CSIC ORCID | artículo |
closedAccess | | 2013 | Synthesis of 3'-Spiro-substituted Nucleosides: Chemistry of TSAO Nucleoside Derivatives | Camarasa Rius, María José CSIC ORCID; Velázquez, Sonsoles CSIC ORCID CVN; San-Félix, Ana CSIC ORCID ; Peréz-Pérez, María-Jesús CSIC ORCID | capítulo de libro |