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Derechos | Preview | Fecha Public. | Título | Autor(es) | Tipo |
openAccess | | 3-oct-2021 | Design of inhibitors of the intrinsically disordered protein NUPR1: balance between drug affinity and target function | Rizzuti, Bruno; Lan, Wenjun; Santofimia-Castaño, Patricia; Zhou, Zhengwei; Velázquez-Campoy, Adrián; Abian, Olga CSIC ORCID; Peng, Ling; Neira, José L. CSIC ORCID; Xia, Yi; Iovanna, Juan Lucio | artículo |
openAccess | | 16-may-2019 | Designing and repurposing drugs to target intrinsically disordered proteins for cancer treatment: using NUPR1 as a paradigm | Santofimia-Castaño, Patricia; Rizzuti, Bruno; Xia, Yi; Abian, Olga CSIC ORCID; Peng, Ling; Velázquez-Campoy, Adrián; Iovanna, Juan Lucio; Neira, José L. CSIC ORCID | artículo |
openAccess | | 2020 | Dynamics of the intrinsically disordered inhibitor IF7 of glutamine synthetase in isolation and in complex with its partner | Neira, José L. CSIC ORCID; Ortore, M.G.; Florencio, Francisco J.; Muro-Pastor, M. Isabel CSIC ORCID ; Rizzuti, Bruno | artículo |
closedAccess | | 17-jul-2019 | Dynamics of the intrinsically disordered protein NUPR1 in isolation and in its fuzzy complexes with DNA and prothymosin α | Neira, José L. CSIC ORCID; Palomino-Schätzlein, M.; Ricci, C.; Ortore, M.G.; Rizzuti, Bruno; Iovanna, Juan Lucio | artículo |
closedAccess | | 2020 | Human importin α3 and its N-terminal truncated form, without the importin-β-binding domain, are oligomeric species with a low conformational stability in solution | Díaz-García, Clara; Hornos, Felipe; Giudici, A. Marcela; Cámara-Artigas, Ana; Luque-Ortega, Juan Román CSIC ORCID ; Arbe, Arantxa CSIC ORCID; Rizzuti, Bruno; Alfonso, Carlos CSIC ORCID ; Forwood, Jade K.; Iovanna, Juan Lucio; Gómez, Javier; Prieto, Manuel CSIC; Coutinho, Ana; Neira, José L. CSIC ORCID | artículo |
openAccess | | 2017 | Identification of a Drug Targeting an Intrinsically Disordered Protein Involved in Pancreatic Adenocarcinoma | Neira, J.L.; Bintz, J.; Arruebo, María; Rizzuti, Bruno; Bonacci, T.; Vega, Sonia CSIC ORCID; Lanas, A.; Velázquez-Campoy, Adrián; Iovanna, Juan Lucio; Abian, Olga CSIC ORCID | artículo |
openAccess | | 18-jul-2017 | Intrinsically disordered chromatin protein NUPR1 binds to the C-terminal region of Polycomb RING1B | Santofimia-Castaño, Patricia; Rizzuti, Bruno; Pey, Ángel L.; Soubeyran, Philippe; Vidal, Miguel CSIC ORCID ; Urrutia, Raúl; Iovanna, Juan Lucio; Neira, José L. CSIC ORCID | artículo |
closedAccess | | jun-2017 | Intrinsically disordered inhibitor of glutamine synthetase is a functional protein with random-coil-like pKa values | Cozza, Concetta; Neira, José L. CSIC ORCID; Florencio, Francisco J.; Muro-Pastor, M. Isabel CSIC ORCID ; Rizzuti, Bruno | artículo |
openAccess | | 28-mar-2019 | Ligand-based design identifies a potent NUPR1 inhibitor exerting anticancer activity via necroptosis | Santofimia-Castaño, Patricia; Xia, Yi; Lan, Wenjun; Zhou, Zhengwei; Huang, Can; Peng, Ling; Soubeyran, Philippe; Velázquez-Campoy, Adrián; Abian, Olga CSIC ORCID; Rizzuti, Bruno; Neira, José L. CSIC ORCID; Iovanna, Juan Lucio | artículo |
openAccess | | ago-2023 | New insights into cancer: MDM2 binds to the citrullinating enzyme PADI4 | Araujo-Abad, Salomé; Rizzuti, Bruno; Villamarin-Ortiz, Adrián; Pantoja-Uceda, D.; Moreno-Gonzalez, Celia M; Abian, Olga CSIC ORCID; Velazquez-Campoy, Adrián; Neira, José L. CSIC ORCID; de Juan Romero, Camino | artículo |
openAccess | | 21-sep-2021 | Polyphenols from citrus tacle® extract endowed with hmgcr inhibitory activity: An antihypercholesterolemia natural remedy | Grande, Fedora; Occhiuzzi, María Antonietta; Perri, Maria Rosaria; Ioele, Giuseppina; Rizzuti, Bruno; Statti, Giancarlo; Garofalo, Antonio | artículo |
openAccess | | 6-oct-2021 | Residual helicity at the active site of the histidine phosphocarrier, HPr, modulates binding affinity to its natural partners | Neira, José L. CSIC ORCID; Ortega-Alarcón, David; Rizzuti, Bruno; Palomino-Schätzlein, M.; Velázquez-Campoy, Adrián; Falcó, Alberto | artículo |
openAccess | | 2-abr-2021 | Rutin Is a Low Micromolar Inhibitor of SARS-CoV-2 Main Protease 3CLpro: Implications for Drug Design of Quercetin Analogs | Rizzuti, Bruno; Grande, Fedora; Conforti, Filomena; Jiménez-Alesanco, Ana CSIC; Ceballos-Laita, Laura CSIC ORCID; Ortega-Alarcón, David; Vega, Sonia CSIC ORCID; Reyburn, H. T. ; Abian, Olga CSIC ORCID; Velázquez-Campoy, Adrián | artículo |
openAccess | | 30-jun-2021 | Seleno-Functionalization of Quercetin Improves the Non-Covalent Inhibition of Mpro and Its Antiviral Activity in Cells against SARS-CoV-2 | Mangiavacchi, Fancesca; Botwina, Pawel; Menichetti, Elena; Bagnoli, Luana; Rosati, Ornelo; Marini, Francesca; Fonseca, Sergio F.; Abenante, Laura; Alves, Diego; Dabrowska, Agnieszka; Kula-Pacurar, Anna; Ortega-Alarcón, David; Jiménez-Alesanco, Ana CSIC; Ceballos-Laita, Laura CSIC ORCID; Vega, Sonia CSIC ORCID; Rizzuti, Bruno; Abian, Olga CSIC ORCID; Lenardão, Eder J.; Velázquez-Campoy, Adrián; Pyrc, Krzysztof; Sancineto, Luca; Santi, Claudio | artículo |
openAccess | | 1-ago-2020 | Structural stability of SARS-CoV-2 3CLpro and identification of quercetin as an inhibitor by experimental screening | Abian, Olga CSIC ORCID; Ortega-Alarcón, David; Jiménez-Alesanco, Ana CSIC; Ceballos-Laita, Laura CSIC ORCID; Vega, Sonia CSIC ORCID; Reyburn, H. T. ; Rizzuti, Bruno; Velázquez-Campoy, Adrián | artículo |
openAccess | | 1-sep-2021 | Sub-Micromolar Inhibition of SARS-CoV-2 3CLpro by Natural Compounds | Rizzuti, Bruno; Ceballos-Laita, Laura CSIC ORCID; Ortega-Alarcón, David; Jiménez-Alesanco, Ana CSIC; Vega, Sonia CSIC ORCID; Grande, Fedora; Conforti, Filomena; Abian, Olga CSIC ORCID; Velázquez-Campoy, Adrián | artículo |
openAccess | | 30-oct-2019 | Targeting intrinsically disordered proteins involved in cancer | Santofimia-Castaño, P.; Rizzuti, Bruno; Xia, Y.; Abian, Olga CSIC ORCID; Peng, L.; Velázquez-Campoy, Adrián; Neira, José L. CSIC ORCID; Iovanna, Juan Lucio | artículo |
openAccess | | 17-nov-2019 | Targeting the stress-induced protein NUPR1 to treat pancreatic adenocarcinoma | Santofimia-Castaño, Patricia; Xia, Yi; Peng, Ling; Velázquez-Campoy, Adrián; Abian, Olga CSIC ORCID; Lan, Wenjun; Lomberk, Gwen; Urrutia, Raul; Rizzuti, Bruno; Soubeyran, Philippe; Neira, José L. CSIC ORCID; Iovanna, Juan Lucio | artículo |
closedAccess | | 1-jul-2021 | The armadillo-repeat domain of plakophilin 1 binds the C-terminal sterile alpha motif (SAM) of p73 | Neira, José L. CSIC ORCID; Rizzuti, Bruno; Ortega-Alarcón, David; Giudici, A. Marcela; Abian, Olga CSIC ORCID; Fárez-Vidal, María Esther; Velázquez-Campoy, Adrián | artículo |
openAccess | | 2018 | The C terminus of the ribosomal-associated protein LrtA is an intrinsically disordered oligomer | Neira, José L. CSIC ORCID; Giudici, A. Marcela; Hornos, Felipe; Arbe, Arantxa CSIC ORCID; Rizzuti, Bruno | artículo |