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openAccessEuropean Journal of Medicinal Chemistry 244 (2022).pdf.jpg2022Identification of 1,2,3-triazolium salt-based inhibitors of Leishmania infantum trypanothione disulfide reductase with enhanced antileishmanial potency in cellulo and increased selectivityLucio, Héctor de; Revuelto, Alejandro CSIC ORCID; Carriles, Alejandra A. CSIC ORCID; Castro, Sonia de CSIC ORCID; García-González, Sonia; García-Soriano, Juan Carlos; Alcón-Calderón, Mercedes; Sánchez-Murcia, Pedro A. CSIC ORCID; Hermoso, Juan A. CSIC ORCID; Gago, Federico CSIC ORCID; Camarasa Rius, María José CSIC ORCID; Jiménez-Ruiz, Antonio; Velázquez, Sonsoles CSIC ORCID CVNartículo
openAccessEuropean Journal of Medicinal Chemistry 243 (2022).pdf.jpg2022Identification of L. infantum trypanothione synthetase inhibitors with leishmanicidal activity from a (non-biased) in-house chemical libraryAlcón-Calderón, Mercedes; Lucio, Héctor de; García-Soriano, Juan Carlos; Revuelto, Alejandro CSIC ORCID; Castro, Sonia de CSIC ORCID; López-Gutiérrez, Celia; San-Félix, Ana CSIC ORCID ; Quesada, Ernesto CSIC ORCID ; Gago, Federico CSIC ORCID; Camarasa Rius, María José CSIC ORCID; Jiménez-Ruiz, Antonio; Velázquez, Sonsoles CSIC ORCID CVNartículo
openAccessaccesoRestringido.pdf.jpg2019Pyrrolopyrimidine vs imidazole-phenyl-thiazole scaffolds in nonpeptidic dimerization inhibitors of leishmania infantum trypanothione reductaseRevuelto, Alejandro CSIC ORCID; Ruiz-Santaquiteria, Marta CSIC ORCID; Lucio, Héctor de; Gamo, Ana; Carriles, Alejandra A. CSIC ORCID; Gutiérrez, Kilian Jesús; Sánchez-Murcia, Pedro A. CSIC ORCID; Gago, Federico CSIC ORCID; Camarasa Rius, María José CSIC ORCID; Jiménez-Ruiz, Antonio; Velázquez, Sonsoles CSIC ORCID CVNartículo
openAccesspharmaceuticals-14-00689-v2-1.pdf.jpg17-jul-2021Small Molecule–Peptide Conjugates as Dimerization Inhibitors of Leishmania infantum Trypanothione Disulfide ReductaseRevuelto, Alejandro CSIC ORCID; López-Martín, Isabel; Lucio, Héctor de; García-Soriano, Juan Carlos; Zanda, Nicola; Castro, Sonia de CSIC ORCID; Gago, Federico CSIC ORCID; Jiménez-Ruiz, Antonio; Velázquez, Sonsoles CSIC ORCID CVN; Camarasa Rius, María José CSIC ORCIDartículo
openAccessEP3502109A1.pdf.jpg26-jun-2018Triazole-phenyl-thiazole heterocycles as innovative inhibitors of trypanothione reductase and their use as leishmanicidesCamarasa Rius, María José CSIC ORCID; Velázquez, Sonsoles CSIC ORCID CVN; Revuelto, Alejandro CSIC ORCID; Gago, Federico CSIC ORCID; Jiménez- Ruiz, Antonio; Toro, Miguel Ángel; Sánchez-Murcia, Pedro A. CSIC ORCID; Lucio, Héctor desolicitud de patente
openAccessWO2019122113A1.pdf.jpg27-jun-2019Triazole-phenyl-thiazole heterocycles as innovative inhibitors of trypanothione reductase and their use as leishmanicidesCamarasa Rius, María José CSIC ORCID; Velázquez, Sonsoles CSIC ORCID CVN; Revuelto, Alejandro CSIC ORCID; Gago, Federico CSIC ORCID; Jiménez- Ruiz, Antonio; Toro, Miguel Ángel; Sánchez-Murcia, Pedro A. CSIC ORCID; Lucio, Héctor desolicitud de patente