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openAccessScientific reports(2018)4242.pdf.jpg2018High-affinity ligands of the colchicine domain in tubulin based on a structure-guided designBueno, Oskia CSIC; Estévez-Gallego, Juan CSIC ORCID ; Martins, S.; Prota, Andrea E.; Gago, Federico CSIC ORCID; Gómez-SanJuan, Asier CSIC; Camarasa Rius, María José CSIC ORCID; Barasoain, Isabel CSIC ; Steinmetz, Michel O.; Díaz, José Fernando CSIC ORCID ; Peréz-Pérez, María-Jesús CSIC ORCID ; Liekens, Sandra; Priego, Eva María CSIC ORCIDartículo
openAccesspharmaceuticals-15-00835.pdf.jpg2022Hybridization Approach to Identify Salicylanilides as Inhibitors of Tubulin Polymerization and Signal Transducers and Activators of Transcription 3 (STAT3)Gargantilla, Marta CSIC ORCID; Persoons, Leentje; Kauerová, Tereza; Río, Natalia del CSIC ORCID; Daelemans, Dirk; Priego, Eva María CSIC ORCID; Kollar, Peter; Peréz-Pérez, María-Jesús CSIC ORCID artículo
closedAccess2014Identification of [1,2,3]triazolo[4,5-d ]pyrimidin-7(6H)-ones as novel inhibitors of chikungunya virus replicationGigante, Alba CSIC ORCID; Canela, María-Dolores CSIC; Delang, Leen; Priego, Eva María CSIC ORCID; Camarasa Rius, María José CSIC ORCID; Querat, Guilles; Neyts, Johan; Leyssen, Pieter; Peréz-Pérez, María-Jesús CSIC ORCID artículo
openAccessScientific reports (2018).pdf.jpg2018Identification of a novel 2-oxindole fluorinated derivative as in vivo antitumor agent for prostate cancer acting via AMPK activationBort Bueno, Alicia; Quesada Sánchez, Sergio CSIC; Ramos-Torres, Ágata; Gargantilla, Marta CSIC ORCID; Priego, Eva María CSIC ORCID; Raynal, S.; Lepifre, F.; Gasalla, José María; Rodriguez-Henche, Nieves; Castro, Ana CSIC ORCID; Díaz-Laviada, Inésartículo
openAccessACS Infect Dis 2018.pdf.jpg2018Inhibition of the Replication of Different Strains of Chikungunya Virus by 3-Aryl-[1,2,3]triazolo[4,5- d] pyrimidin-7(6 H)-onesGómez-SanJuan, Asier CSIC; Gamo, Ana María CSIC; Delang, Leen; Pérez-Sánchez, Alfonso; Amrun, S. N.; Abdelnabi, Rana; Jacobs, S.; Priego, Eva María CSIC ORCID; Camarasa Rius, María José CSIC ORCID; Jochmans, D.; Leyssen, Pieter; Ng, L. F. P.; Querat, Guilles; Neyts, Johan; Peréz-Pérez, María-Jesús CSIC ORCID artículo
openAccesspharmaceuticals-14-01131-1.pdf.jpg6-nov-2021Inhibition of XPO-1 Mediated Nuclear Export through the Michael-Acceptor Character of ChalconesGargantilla, Marta CSIC ORCID; López-Fernández, José; Camarasa Rius, María José CSIC ORCID; Persoons, Leentje; Daelemans, Dirk; Priego, Eva María CSIC ORCID; Peréz-Pérez, María-Jesús CSIC ORCID artículo
closedAccess2009Intramolecular Cation-π Interactions As the Driving Force To Restrict the Conformation of Certain NucleosidesCasanova, Elena; Priego, Eva María CSIC ORCID; Jimeno, M. Luisa CSIC ORCID; Aguado, Leire CSIC; Negri, Ana; Gago, Federico CSIC ORCID; Camarasa Rius, María José CSIC ORCID; Peréz-Pérez, María-Jesús CSIC ORCID artículo
openAccessGigante_full_article.pdf.jpg2014Microwave-assisted synthesis of C-8 aryl and heteroaryl inosines and determination of their inhibitory activities against Plasmodium falciparum purine nucleoside phosphorylaseGigante, Alba CSIC ORCID; Priego, Eva María CSIC ORCID; Sánchez-Carrasco, Paula; Ruiz-Pérez, Luis Miguel; Vande Voorde, Johan; Camarasa Rius, María José CSIC ORCID; Balzarini, Jan; González-Pacanowska, Dolores; Peréz-Pérez, María-Jesús CSIC ORCID artículo
openAccess2022 ACS Chem Neurosci 13-275 postprint.pdf.jpg19-ene-2022Neuroprotective Effect of IND1316, an Indole-Based AMPK Activator, in Animal Models of Huntington DiseaseVela, Marta; García-Gimeno, María Adelaida CSIC ORCID; Sanchis, Ana CSIC; Bono-Yagüe, José; Cumella, José; Lagartera, Laura CSIC ORCID; Pérez, Concepción CSIC ORCID; Priego, Eva María CSIC ORCID; Campos, Ángela CSIC; Sanz, Pascual CSIC ORCID ; Vázquez-Manrique, Rafael P. CSIC ORCID; Castro, Ana CSIC ORCIDartículo
openAccessCanela-et-al_2014_JMedChem_57.pdf.jpg2014Novel colchicine-site binders with a cyclohexanedione scaffold identified through a ligand-based virtual screening approachCanela, María-Dolores CSIC; Peréz-Pérez, María-Jesús CSIC ORCID ; Noppen, Sam; Sáez-Calvo, Gonzalo CSIC; Díaz, José Fernando CSIC ORCID ; Camarasa Rius, María José CSIC ORCID; Liekens, Sandra; Priego, Eva María CSIC ORCIDartículo
openAccessProtein ligand complex.pdf.jpg23-ene-2018Protein-ligand complex for structure-based design: impact on the affinity and antitumor activity of new tubulin ligandsBueno, Oskia CSIC; Estévez-Gallego, Juan CSIC ORCID ; Martins, S.; Prota, Andrea E.; Gago, Federico CSIC ORCID; Gómez-SanJuan, Asier CSIC; Camarasa Rius, María José CSIC ORCID; Barasoain, Isabel CSIC ; Steinmetz, Michel O.; Díaz, José Fernando CSIC ORCID ; Liekens, Sandra; Peréz-Pérez, María-Jesús CSIC ORCID ; Priego, Eva María CSIC ORCIDcomunicación de congreso
closedAccess2012Recent Advances in Thymidine Kinase 2 (TK2) Inhibitors and New Perspectives for Potential ApplicationsPriego, Eva María CSIC ORCID; Karlsson, Anna; Gago, Federico CSIC ORCID; Camarasa Rius, María José CSIC ORCID; Balzarini, Jan; Peréz-Pérez, María-Jesús CSIC ORCID artículo
closedAccessaccesoRestringido.pdf.jpg2008Selective human adenosine A3 antagonists based on pyrido[2,1-f]purine-2,4-diones: Novel features of hA3 antagonist bindingPriego, Eva María CSIC ORCID; Peréz-Pérez, María-Jesús CSIC ORCID ; Von Frijtag Drabbe Kuenzel, J. K.; de Vries, H.; Ijzerman, A. P.; Camarasa Rius, María José CSIC ORCID; Martín-Santamaría, Sonsoles CSIC ORCID artículo
closedAccessaccesoRestringido.pdf.jpg2008Structure, physiological role, and specific inhibitors of human thymidine kinase 2 (TK2): Present and futurePeréz-Pérez, María-Jesús CSIC ORCID ; Priego, Eva María CSIC ORCID; Hernández, Ana-Isabel CSIC; Familiar, Olga CSIC; Camarasa Rius, María José CSIC ORCID; Negri, Ana; Gago, Federico CSIC ORCID; Balzarini, Janartículo
closedAccess2014Synthesis and antiproliferative activity of 6-phenylaminopurinesCanela, María-Dolores CSIC; Liekens, S.; Camarasa Rius, María José CSIC ORCID; Priego, Eva María CSIC ORCID; Peréz-Pérez, María-Jesús CSIC ORCID artículo
closedAccessaccesoRestringido.pdf.jpg2016Targeting the colchicine site in tubulin through cyclohexanedione derivativesCanela, María-Dolores CSIC; Bueno, Oskia CSIC; Noppen, Sam; Sáez-Calvo, Gonzalo CSIC; Estévez-Gallego, Juan CSIC ORCID ; Díaz, José Fernando CSIC ORCID ; Camarasa Rius, María José CSIC ORCID; Liekens, Sandra; Peréz-Pérez, María-Jesús CSIC ORCID ; Priego, Eva María CSIC ORCIDartículo