Derechos | Preview | Fecha Public. | Título | Autor(es) | Tipo |
closedAccess | | 26-nov-2014 | Design and synthesis of pironetin analogue/colchicine hybrids and study of their cytotoxic activity and mechanisms of interaction with tubulin | Vilanova, Concepción; Díaz-Oltra, Santiago; Murga, Juan; Falomir, Eva; Carda, Miguel; Redondo-Horcajo, Mariano CSIC ORCID ; Díaz, José Fernando CSIC ORCID ; Barasoain, Isabel CSIC ; Marco, J. Alberto | artículo |
closedAccess | | may-2011 | Design and Synthesis of Pironetin Analogues with Simplified Structure and Study of Their Interactions with Microtubules | Marco, J. Alberto; García-Pla, Jorge; Carda, Miguel; Murga, Juan; Falomir, Eva; Trigili, Chiara CSIC; Notararigo, Sara CSIC ORCID; Díaz, José Fernando CSIC ORCID ; Barasoain, Isabel CSIC | artículo |
openAccess | | 31-jul-2016 | Pironetin binds covalently to Cys316 and perturbs a major loop and helix of -tubulin to inhibit microtubule formation | Prota, Andrea E.; Setter, J.; Waight, Andrew B.; Bargsten, Katja; Murga, Juan; Díaz, José Fernando CSIC ORCID ; Steinmetz, Michel O. | artículo |
closedAccess | | 28-feb-2013 | Synthesis and biological evaluation as microtubule-active agents of several tetrahydrofuran and spiroacetal derivatives | Carda, Miguel; Murga, Juan; Paños, Julián; Angulo-Pachón, C.A.; García-Pla, Jorge; Díaz-Oltra, Santiago; Marco, J. Alberto; Trigili, Chiara CSIC; Redondo-Horcajo, Mariano CSIC ORCID ; Díaz, José Fernando CSIC ORCID ; Barasoain, Isabel CSIC | artículo |
closedAccess | | 2013 | Synthesis and biological evaluation of truncated α-tubulin-binding pironetin analogues lacking alkyl pendants in the side chain or the dihydropyrone ring | Paños, Julián; Díaz-Oltra, Santiago; Sánchez-Peris, María; García-Pla, Jorge; Murga, Juan; Falomir, Eva; Carda, Miguel; Redondo-Horcajo, Mariano CSIC ORCID ; Díaz, José Fernando CSIC ORCID ; Barasoain, Isabel CSIC ; Marco, J. Alberto | artículo |
closedAccess | | feb-2013 | Synthesis and Biological Evaluation of α-Tubulin-Binding Pironetin Analogues with Enhanced Lipophilicity | Carda, Miguel; Murga, Juan; Díaz-Oltra, Santiago; García-Pla, Jorge; Paños, Julián; Falomir, Eva; Trigili, Chiara CSIC; Díaz, José Fernando CSIC ORCID ; Barasoain, Isabel CSIC ; Marco, J. Alberto | artículo |
closedAccess | | 2021 | Synthesis of N-acyl Derivatives of Aminocombretastatin A-4 and Study of their Interaction with Tubulin and downregulation of c-Myc | Agut, Raül; Falomir, Eva; Murga, Juan; Martín-Beltrán, Celia; Gil-Edo, Raquel; Pla, Alberto; Carda, Miguel; Díaz, José Fernando CSIC ORCID ; Josa-Prado, Fernando CSIC ORCID; Marco, J. Alberto | artículo |
closedAccess | | ago-2015 | The Mechanism of the Interactions of Pironetin Analog/Combretastatin A-4 Hybrids with Tubulin | Torijano-Gutiérrez, Sandra; Vilanova, Concepción; Díaz-Oltra, Santiago; Murga, Juan; Falomir, Eva; Carda, Miguel; Redondo-Horcajo, Mariano CSIC ORCID ; Díaz, José Fernando CSIC ORCID ; Barasoain, Isabel CSIC ; Marco, J. Alberto | artículo |
closedAccess | | 15-jun-2007 | The Total Synthesis and Biological Properties of the Cytotoxic Macrolide FD-891 and Its Non-Natural (Z)-C12 Isomer | García-Fortanet, Jorge; Murga, Juan; Carda, Miguel; Marco, J. Alberto; Matesanz, Ruth CSIC ; Díaz, José Fernando CSIC ORCID ; Barasoain, Isabel CSIC | artículo |