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Mostrando resultados 1 a 12 de 12
DerechosPreviewFecha Public.TítuloAutor(es)Tipo
closedAccessaccesoRestringido.pdf.jpg2014Design, synthesis, pharmacological evaluation, QSAR analysis, molecular modeling and ADMET of novel donepezil-indolyl hybrids as multipotent cholinesterase/monoamine oxidase inhibitors for the potential treatment of Alzheimer's diseaseBautista-Aguilera, Óscar M. CSIC ORCID; Esteban, Gerard; Bolea, Irene; Nikolic, Katarina; Agbaba, Danica; Moraleda, Ignacio; Iriepa, Isabel; Samadi, Abdelouahid CSIC ORCID; Soriano, Elena CSIC; Unzeta, Mercedes; Marco-Contelles, José CSIC ORCIDartículo
closedAccessaccesoRestringido.pdf.jpg2014Donepezil + propargylamine + 8-hydroxyquinoline hybrids as new multifunctional metal-chelators, ChE and MAO inhibitors for the potential treatment of Alzheimer's diseaseWang, L.; Esteban, Gerard; Ojima, Masaki; Bautista-Aguilera, Óscar M. CSIC ORCID; Inokuchi, Tsutomu; Moraleda, Ignacio; Iriepa, Isabel; Samadi, Abdelouahid CSIC ORCID; Youdim, Moussa B. H.; Romero Jódar, Alejandro CSIC ORCID; Soriano, Elena CSIC; Herrero-Labrador, Raquel CSIC ORCID; Fernández Fernández, Ana Patricia CSIC; Martínez-Murillo, Ricardo CSIC ORCID; Marco-Contelles, José CSIC ORCID; Unzeta, Mercedesartículo
openAccessmolecules-21-00400.pdf.jpg24-mar-2016Imidazopyranotacrines as Non-Hepatotoxic, Selective Acetylcholinesterase Inhibitors, and Antioxidant Agents for Alzheimer's Disease TherapyBoulebd, Houssem; Ismaili, L.; Bartolini, Manuela; Bouraiou, Abdelmalek; Andrisano, Vincenza; Martin, Hélène; Bonet, Alexandre; Moraleda, Ignacio; Iriepa, Isabel; Chioua, Mourad CSIC ORCID ; Belfaitah, Ali; Marco-Contelles, José CSIC ORCIDartículo
openAccessDrug Design, Development and Therapy.pdf.jpg2014Multipotent cholinesterase/monoamine oxidase inhibitors for the treatment of Alzheimer’s disease: Design, synthesis, biochemical evaluation, ADMET, molecular modeling, and QSAR analysis of novel donepezil-pyridyl hybridsBautista-Aguilera, Óscar M. CSIC ORCID; Esteban, Gerard; Chioua, Mourad CSIC ORCID ; Nikolic, Katarina; Agbaba, Danica; Moraleda, Ignacio; Iriepa, Isabel; Soriano, Elena CSIC; Samadi, Abdelouahid CSIC ORCID; Unzeta, Mercedes; Marco-Contelles, José CSIC ORCIDartículo
closedAccessaccesoRestringido.pdf.jpg2015Pyranopyrazolotacrines as nonneurotoxic, Aβ-anti-aggregating and neuroprotective agents for Alzheimer's diseaseChioua, Mourad CSIC ORCID ; Pérez-Peña, Javier; García-Font, Nuria; Moraleda, Ignacio; Iriepa, Isabel; Soriano, Elena CSIC; Marco-Contelles, José CSIC ORCID; Oset-Gasque, María Jesúsartículo
openAccessmolecules-24-01503.pdf.jpg17-abr-2019QuinoxalineTacrine QT78, a Cholinesterase Inhibitor as a Potential Ligand for Alzheimer’s Disease TherapyRamos, Eva; Palomino-Antolín, Alejandra; Bartolini, Manuela; Iriepa, Isabel; Moraleda, Ignacio; Diez-Iriepa, Daniel CSIC; Samadi, Abdelouahid CSIC ORCID; Cortina, Carol V.; Chioua, Mourad CSIC ORCID ; Egea, Javier; Romero Jódar, Alejandro CSIC ORCID; Marco-Contelles, José CSIC ORCIDartículo
openAccessJOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY.pdf.jpg2019Synthesis and biological assessment of KojoTacrines as new agents for Alzheimer’s disease therapyDgachi, Youssef; Martin, Helene; Martin, Hélène; Malek, R; Jun, D.; Janockova, Jana; Sepsova, Vendula; Soukup, Ondrej; Iriepa, Isabel; Moraleda, Ignacio; Maalej, Enma; Carreiras, M. Carmo; Refouvelet, B.; Chabchoub, Fakher; Marco-Contelles, José CSIC ORCID; Ismaili, Lhassaneartículo
closedAccessaccesoRestringido.pdf.jpg2017Synthesis and biological assessment of racemic benzochromenopyrimidinetriones as promising agents for Alzheimer's disease therapyDgachi, Youssef; Martin, Hélène; Bonet, Alexandre; Chioua, Mourad CSIC ORCID ; Iriepa, Isabel; Moraleda, Ignacio; Chabchoub, Fakher; Marco-Contelles, José CSIC ORCID; Ismaili, Lhassaneartículo
closedAccessaccesoRestringido.pdf.jpg2018Synthesis, Biological Assessment and Molecular Modeling of Racemic QuinoPyranoTacrines for Alzheimer's Disease TherapyChioua, Mourad CSIC ORCID ; Serrano, Estefanía; Dgachi, Youssef; Martin, Hélène; Jun. Daniel Jun; Janockova, Jana; Sepsova, Vendula; Soukup, Ondrej; Moraleda, Ignacio; Chabchoub, Fakher; Ismaili, Lhassan; Iriepa, Isabel; Marco-Contelles, José CSIC ORCIDartículo
closedAccessaccesoRestringido.pdf.jpg2013Synthesis, pharmacological assessment, and molecular modeling of 6-chloro-pyridonepezils: New dual AChE inhibitors as potential drugs for the treatment of Alzheimer's diseaseSamadi, Abdelouahid CSIC ORCID; Fuente Revenga, Mario de la CSIC ORCID; Pérez, Concepción CSIC ORCID; Iriepa, Isabel; Moraleda, Ignacio; Rodríguez-Franco, María Isabel CSIC ORCID ; Marco-Contelles, José CSIC ORCIDartículo
closedAccessaccesoRestringido.pdf.jpg2013Synthesis, pharmacological assessment, and molecular modeling of acetylcholinesterase/butyrylcholinesterase inhibitors: Effect against amyloid-β-induced neurotoxicitySilva, Daniel; Chioua, Mourad CSIC ORCID ; Samadi, Abdelouahid CSIC ORCID; Agostinho, Paula; Garção, Pedro; Lajarín-Cuesta, Rocío; Ríos, Cristobal de los; Iriepa, Isabel; Moraleda, Ignacio; González-Lafuente, Laura; Mendes, Eduarda; Pérez, Concepción CSIC ORCID; Rodríguez-Franco, María Isabel CSIC ORCID ; Marco-Contelles, José CSIC ORCID; Carreiras, M. Carmoartículo
closedAccessaccesoRestringido.pdf.jpg2018Tacripyrimidines, the first tacrine-dihydropyrimidine hybrids, asmulti-target-directed ligands for Alzheimer's diseaseChioua, Mourad CSIC ORCID ; Buzzi, Eleonora; Moraleda, Ignacio; Iriepa, Isabel; Maj, Maciej; Wnorowski, Artur; Giovannini, Catia; Tamarin, Anna; Portali, Federica; Ismaili, Lhassane; López-Alvarado, Pilar; Bolognesi, Maria Laura; Jóźwiak, Krzysztof; Menéndez, J. Carlos; Marco-Contelles, José CSIC ORCID; Bartolini, Manuelaartículo