Derechos | Preview | Fecha Public. | Título | Autor(es) | Tipo |
closedAccess | | 19-feb-2019 | A new class of dual HIV and EV71 entry inhibitors: tri and tetrapodal tryptophan derivatives | Martí-Marí, Olaia CSIC ORCID; Martínez-Gualda, Belén CSIC; Puente-Secades, Sofía de la CSIC; Mirabelli, Carmen; Sun, Liang; Delang, Leen; Schols, Dominique; Neyts, Johan; Camarasa Rius, María José CSIC ORCID; San-Félix, Ana CSIC ORCID | comunicación de congreso |
openAccess | | 3-abr-2019 | A second-generation of tryptophan-containing small molecules extremely potent against HIV and EV-A71 clinical isolates | Martí-Marí, Olaia CSIC ORCID; Martínez-Gualda, Belén CSIC; Puente-Secades, Sofía de la CSIC; Quesada, Ernesto CSIC ORCID ; Sun, Liang; Delang, Leen; Mirabelli, Carmen; Noppen, Sam; Schols, Dominique; Neyts, Johan; Gago, Federico CSIC ORCID; Camarasa Rius, María José CSIC ORCID; San-Félix, Ana CSIC ORCID | actas de congreso |
closedAccess | | 2023 | Un ataque combinado químico, virológico, biofísico y estructural hace posible la obtención de nuevos inhibidores de entrada celular de SARS-CoV-2 y la caracterización de su mecanismo de inhibición | Gargantilla, Marta CSIC ORCID; Francés-Gómez, Clara CSIC ORCID; Adhav, Anmol CSIC ORCID; Forcada-Nadal, Alicia CSIC ORCID; Martínez-Gualda, Belén CSIC; Martí-Marí, Olaia CSIC ORCID; López-Redondo, Marisa CSIC; Melero, Roberto CSIC ORCID; Marco-Marín, Clara CSIC ORCID; IBV-Covid 19-Pipeline; Bravo, Jerónimo CSIC ORCID ; Llácer, José Luis CSIC ORCID ; Marina, Alberto CSIC ORCID ; Rubio, Vicente CSIC ORCID ; Geller, Ron CSIC ORCID | comunicación de congreso |
openAccess | | 10-ago-2023 | C-2 Thiophenyl Tryptophan Trimers Inhibit Cellular Entry of SARS-CoV-2 through Interaction with the Viral Spike (S) Protein | Gargantilla, Marta CSIC ORCID; Francés-Gómez, Clara CSIC ORCID; Adhav, Anmol CSIC ORCID; Forcada-Nadal, Alicia CSIC ORCID; Martínez-Gualda, Belén CSIC; Martí-Marí, Olaia CSIC ORCID; López-Redondo, Marisa CSIC; Melero, Roberto CSIC ORCID; Marco-Marín, Clara CSIC ORCID; Gougeard, Nadine CSIC ORCID; Espinosa, Carolina; Rubio-Del-Campo, Antonio; Ruiz-Partida, Rafael; Hernández-Sierra, María del Pilar; Villamayor-Belinchón, Laura; Bravo, Jerónimo CSIC ORCID ; Llácer, José Luis CSIC ORCID ; Marina, Alberto CSIC ORCID ; Rubio, Vicente CSIC ORCID ; San-Félix, Ana CSIC ORCID ; Geller, Ron CSIC ORCID ; Peréz-Pérez, María-Jesús CSIC ORCID | artículo |
openAccess | | 25-ene-2023 | C2-thioether tryptophan trimers and tetramers and use thereof | San-Félix, Ana CSIC ORCID ; Peréz-Pérez, María-Jesús CSIC ORCID ; Quesada, Ernesto CSIC ORCID ; Gargantilla, Marta CSIC ORCID; Martínez-Gualda, Belén CSIC; Geller, Ron CSIC ORCID ; Francés-Gómez, Clara CSIC ORCID | solicitud de patente |
openAccess | | 26-ene-2023 | C2-thioether tryptophan trimers and tetramers for the treatment of betacoronoavirus infections | San-Félix, Ana CSIC ORCID ; Peréz-Pérez, María-Jesús CSIC ORCID ; Quesada, Ernesto CSIC ORCID ; Gargantilla, Marta CSIC ORCID; Martínez-Gualda, Belén CSIC; Geller, Ron CSIC ORCID ; Francés-Gómez, Clara CSIC ORCID | solicitud de patente |
openAccess | | 7-jul-2021 | Double Arylation of the Indole Side Chain of Tri- and Tetrapodal Tryptophan Derivatives Renders Highly Potent HIV‑1 and EV-A71 Entry Inhibitors | Martí-Marí, Olaia CSIC ORCID; Martínez-Gualda, Belén CSIC; Puente-Secades, Sofía de la CSIC; Mills, Alberto; Quesada, Ernesto CSIC ORCID ; Abdelnabi, Rana; Sun, Liang; Boonen, Arnaud; Noppen, Sam; Neyts, Johan; Schols, Dominique; Camarasa Rius, María José CSIC ORCID; Gago, Federico CSIC ORCID; San-Félix, Ana CSIC ORCID | artículo |
openAccess | | 6-jun-2019 | Exploring nanoparticle approaches for in vivo delivery of a potent class of EV-A71 inhibitors | Martí-Marí, Olaia CSIC ORCID; Fernández-Barahona, Irene; Martínez-Gualda, Belén CSIC; Camarasa Rius, María José CSIC ORCID; Herranz, Fernando CSIC ORCID CVN; San-Félix, Ana CSIC ORCID | comunicación de congreso |
openAccess | | 6-jun-2019 | Exploring nanoparticle approaches for in vivo delivery of a potent class of EV-71 inhibitors | Martí-Marí, Olaia CSIC ORCID; Fernández-Barahona, Irene; Martínez-Gualda, Belén CSIC; Camarasa Rius, María José CSIC ORCID; Herranz, Fernando CSIC ORCID CVN; San-Félix, Ana CSIC ORCID | comunicación de congreso |
openAccess | | 2019 | Galloyl Carbohydrates with Antiangiogenic Activity Mediated by Capillary Morphogenesis Gene 2 (CMG2) Protein Binding | Doyagüez, Elisa G. CSIC; Carrero, Paula CSIC; Madrona, Andrés CSIC ORCID; Rodríguez-Salamanca, Patricia CSIC ORCID; Martínez-Gualda, Belén CSIC; Camarasa Rius, María José CSIC ORCID; Jimeno, M. Luisa CSIC ORCID; Bennallack, P. R.; Finnell, J. G; Tsang, T. M.; Christensen, K. A.; San-Félix, Ana CSIC ORCID ; Rogers, M. S. | artículo |
openAccess | | 2019 | Modifications in the branched arms of a class of dual inhibitors of HIV and EV71 replication expand their antiviral spectrum | Martínez-Gualda, Belén CSIC; Sun, L.; Martí-Marí, Olaia CSIC ORCID; Mirabelli, C.; Delang, Leen; Neyts, Johan; Schols, Dominique; Camarasa Rius, María José CSIC ORCID; San-Félix, Ana CSIC ORCID | artículo |
openAccess | | 2016 | Optimization of a class of tryptophan dendrimers that inhibit HIV replication leads to a selective, specific, and low-nanomolar inhibitor of clinical isolates of enterovirus A71 | Rivero-Buceta, Eva CSIC ORCID; Sun, L.; Martínez-Gualda, Belén CSIC; Doyagüez, Elisa G. CSIC; Donckers, K.; Quesada, Ernesto CSIC ORCID ; Camarasa Rius, María José CSIC ORCID; Delang, Leen; San-Félix, Ana CSIC ORCID ; Neyts, Johan; Leyssen, Pieter | artículo |
openAccess | | abr-2022 | Organotropic dendrons with high potency as HIV-1, HIV-2 and EV-A71 cell entry inhibitors | Martí-Marí, Olaia CSIC ORCID; Martínez-Gualda, Belén CSIC; Fernández-Barahona, Irene; Mills, Alberto; Abdelnabi, Rana; Noppen, Sam; Neyts, Johan; Schols, Dominique; Camarasa Rius, María José CSIC ORCID; Herranz, Fernando CSIC ORCID CVN; Gago, Federico CSIC ORCID; San-Félix, Ana CSIC ORCID | artículo |
openAccess | | ene-2020 | Scaffold Simplification Strategy Leads to a Novel Generation of Dual Human Immunodeficiency Virus and Enterovirus-A71 Entry Inhibitors | Martínez-Gualda, Belén CSIC; Sun, Liang; Martí-Marí, Olaia CSIC ORCID; Abdelnabi, Rana; Noppen, Sam; Bator, Carol M.; Quesada, Ernesto CSIC ORCID ; Delang, Leen; Mirabelli, Carmen; Lee, Hyunwook; Schols, Dominique; Neyts, Johan; Hafenstein, Susan; Camarasa Rius, María José CSIC ORCID; Gago, Federico CSIC ORCID; San-Félix, Ana CSIC ORCID | artículo |
openAccess | | 2017 | Structure-activity relationship studies on a Trp dendrimer with dual activities against HIV and enterovirus A71. Modifications on the amino acid | Martínez-Gualda, Belén CSIC; Sun, L.; Rivero-Buceta, Eva CSIC ORCID; Flores, Aida CSIC; Quesada, Ernesto CSIC ORCID ; Balzarini, Jan; Noppen, Sam; Liekens, Sandra; Schols, Dominique; Neyts, Johan; Leyssen, Pieter; Mirabelli, C.; Camarasa Rius, María José CSIC ORCID; San-Félix, Ana CSIC ORCID | artículo |
openAccess | | 2020 | Tryptophan trimers and tetramers inhibit dengue and Zika virus replication by interfering with viral attachment processes | Fikatas, A.; Vervaeke, P.; Martínez-Gualda, Belén CSIC; Martí-Marí, Olaia CSIC ORCID; Noppen, S.; Meyen, E.; Camarasa Rius, María José CSIC ORCID; San-Félix, Ana CSIC ORCID ; Pannecouque, C.; Schols, Dominique | artículo |
openAccess | | 5-oct-2022 | Tryptophan trimers efficiently inhibit SARS-CoV-2 entry into the host cells | Gargantilla, Marta CSIC ORCID; Francés-Gómez, Clara CSIC ORCID; Adhav, Anmol CSIC ORCID; Martínez-Gualda, Belén CSIC; Marina, Alberto CSIC ORCID ; Rubio, Vicente CSIC ORCID ; Geller, Ron CSIC ORCID ; San-Félix, Ana CSIC ORCID ; Peréz-Pérez, María-Jesús CSIC ORCID | póster de congreso |
openAccess | | 2019 | Viral engagement with host receptors blocked by a novel class of tryptophan dendrimers that targets the 5-fold-axis of the enterovirus-A71 capsid | Sun, L.; Lee, H.; Thibaut, H. J.; Lanko, K.; Rivero-Buceta, E.; Bator, C.; Martínez-Gualda, Belén CSIC; Dallmeier, K.; Delang, L.; Leyssen, P.; Gago, Federico CSIC ORCID; San-Félix, Ana CSIC ORCID ; Hafenstein, S.; Mirabelli, C.; Neyts, Johan | artículo |