Mostrando resultados 2 a 12 de 12
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Derechos | Preview | Fecha Public. | Título | Autor(es) | Tipo |
openAccess | | 2015 | Comparison of hydrocarbon-and lactam-bridged cyclic peptides as dimerization inhibitors of Leishmania infantum trypanothione reductase | Sánchez-Murcia, Pedro A. CSIC ORCID; Ruiz-Santaquiteria, Marta CSIC ORCID; Toro, Miguel Ángel; Lucio, H. de; Jiménez, M. Angeles CSIC ORCID ; Gago, Federico CSIC ORCID; Jiménez-Ruiz, Antonio; Camarasa Rius, María José CSIC ORCID; Velázquez, Sonsoles CSIC ORCID CVN | artículo |
openAccess | | 2021 | Efficient Dimerization Disruption of Leishmania infantum Trypanothione Reductase by Triazole-phenyl-thiazoles | Revuelto, Alejandro CSIC ORCID; Lucio, Héctor de; García-Soriano, Juan Carlos; Sánchez-Murcia, Pedro A. CSIC ORCID; Gago, Federico CSIC ORCID; Jiménez-Ruiz, Antonio; Camarasa Rius, María José CSIC ORCID; Velázquez, Sonsoles CSIC ORCID CVN | artículo |
openAccess | | 2017 | First example of peptides targeting the dimer interface of Leishmania infantum trypanothione reductase with potent in vitro antileishmanial activity# | Ruiz-Santaquiteria, Marta CSIC ORCID; Sánchez-Murcia, Pedro A. CSIC ORCID; Toro, Miguel Ángel; Lucio, H. de; Gutiérrez, Kilian Jesús; Castro, Sonia de CSIC ORCID; Carneiro, Filipa A. C.; Gago, Federico CSIC ORCID; Jiménez-Ruiz, Antonio; Camarasa Rius, María José CSIC ORCID; Velázquez, Sonsoles CSIC ORCID CVN | artículo |
openAccess | | 2022 | Identification of L. infantum trypanothione synthetase inhibitors with leishmanicidal activity from a (non-biased) in-house chemical library | Alcón-Calderón, Mercedes; Lucio, Héctor de; García-Soriano, Juan Carlos; Revuelto, Alejandro CSIC ORCID; Castro, Sonia de CSIC ORCID; López-Gutiérrez, Celia; San-Félix, Ana CSIC ORCID ; Quesada, Ernesto CSIC ORCID ; Gago, Federico CSIC ORCID; Camarasa Rius, María José CSIC ORCID; Jiménez-Ruiz, Antonio; Velázquez, Sonsoles CSIC ORCID CVN | artículo |
closedAccess | | 2019 | Identification of NEK3 and MOK as novel targets for lithium | Bravo, Ana; de Lucio, H.; Sánchez-Murcia, Pedro A. CSIC ORCID; Jiménez-Ruiz, Antonio; Petrone, Paula M.; Gago, Federico CSIC ORCID; Cortés Cabrera, Álvaro CSIC ORCID | artículo |
openAccess | | 2014 | Leishmania infantum EndoG is an endo/exo-nuclease essential for parasite survival | Rico, Eva; Oliva, Cristina; Gutiérrez, Kilian Jesús; Alzate, Juan Fernando; Genes, Carlos Mario; Moreno, David; Casanova, Elena CSIC; Gigante, Alba CSIC ORCID; Peréz-Pérez, María-Jesús CSIC ORCID ; Camarasa Rius, María José CSIC ORCID; Clos, Joachim; Gago, Federico CSIC ORCID; Jiménez-Ruiz, Antonio | artículo |
closedAccess | | 6-jun-2013 | Probing the Dimerization Interface of Leishmania infantum Trypanothione Reductase with Site-Directed Mutagenesis and Short Peptides | Toro, Miguel Ángel; Sánchez-Murcia, Pedro A. CSIC ORCID; Moreno, David; Ruiz-Santaquiteria, Marta CSIC ORCID; Alzate, Juan Fernando; Negri, Ana; Camarasa Rius, María José CSIC ORCID; Gago, Federico CSIC ORCID; Velázquez, Sonsoles CSIC ORCID CVN; Jiménez-Ruiz, Antonio | artículo |
openAccess | | 2019 | Pyrrolopyrimidine vs imidazole-phenyl-thiazole scaffolds in nonpeptidic dimerization inhibitors of leishmania infantum trypanothione reductase | Revuelto, Alejandro CSIC ORCID; Ruiz-Santaquiteria, Marta CSIC ORCID; Lucio, Héctor de; Gamo, Ana; Carriles, Alejandra A. CSIC ORCID; Gutiérrez, Kilian Jesús; Sánchez-Murcia, Pedro A. CSIC ORCID; Gago, Federico CSIC ORCID; Camarasa Rius, María José CSIC ORCID; Jiménez-Ruiz, Antonio; Velázquez, Sonsoles CSIC ORCID CVN | artículo |
openAccess | | 17-jul-2021 | Small Molecule–Peptide Conjugates as Dimerization Inhibitors of Leishmania infantum Trypanothione Disulfide Reductase | Revuelto, Alejandro CSIC ORCID; López-Martín, Isabel; Lucio, Héctor de; García-Soriano, Juan Carlos; Zanda, Nicola; Castro, Sonia de CSIC ORCID; Gago, Federico CSIC ORCID; Jiménez-Ruiz, Antonio; Velázquez, Sonsoles CSIC ORCID CVN; Camarasa Rius, María José CSIC ORCID | artículo |
openAccess | | 2017 | Structure-based domain assignment in Leishmania infantum EndoG: Characterization of a pH-dependent regulatory switch and a C-Terminal extension that largely dictates DNA substrate preferences | Oliva, C.; Sánchez-Murcia, Pedro A. CSIC ORCID; Rico, E.; Bravo, A.; Menéndez, Margarita CSIC ORCID; Gago, Federico CSIC ORCID; Jiménez-Ruiz, Antonio | artículo |
openAccess | | 2018 | Trypanothione reductase inhibition and anti-leishmanial activity of all-hydrocarbon stapled α-helical peptides with improved proteolytic stability | Ruiz-Santaquiteria, Marta CSIC ORCID; Castro, Sonia de CSIC ORCID; Toro, Miguel Ángel; Lucio, Héctor de; Gutiérrez, Kilian Jesús; Sánchez-Murcia, Pedro A. CSIC ORCID; Jiménez, M. Angeles CSIC ORCID ; Gago, Federico CSIC ORCID; Jiménez-Ruiz, Antonio; Camarasa Rius, María José CSIC ORCID; Velázquez, Sonsoles CSIC ORCID CVN | artículo |