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Derechos | Preview | Fecha Public. | Título | Autor(es) | Tipo |
closedAccess | | 2017 | Facile one-pot synthesis of new [1,2,4]triazolo[1,5-a]pyridine derivatives by ultrasonic irradiation | Zribi, L.; Zribi, F.; Marco-Contelles, José CSIC ORCID; Chabchoub, Fakher; Ismaili, L. | artículo |
openAccess | | 24-mar-2016 | Imidazopyranotacrines as Non-Hepatotoxic, Selective Acetylcholinesterase Inhibitors, and Antioxidant Agents for Alzheimer's Disease Therapy | Boulebd, Houssem; Ismaili, L.; Bartolini, Manuela; Bouraiou, Abdelmalek; Andrisano, Vincenza; Martin, Hélène; Bonet, Alexandre; Moraleda, Ignacio; Iriepa, Isabel; Chioua, Mourad CSIC ORCID ; Belfaitah, Ali; Marco-Contelles, José CSIC ORCID | artículo |
closedAccess | | 2019 | Multi-target 1,4-dihydropyridines showing calcium channel blockade and antioxidant capacity for Alzheimer's disease therapy | Malek, R.; Maj, M.; Wnorowski, A.; Józwiak, K.; Martin, Helene; Iriepa, Isabel; Moraleda, I.; Chabchoub, Fakher; Marco-Contelles, José CSIC ORCID; Ismaili, L. | artículo |
closedAccess | | 2017 | Multitarget-Directed Ligands Combining Cholinesterase and Monoamine Oxidase Inhibition with Histamine H3R Antagonism for Neurodegenerative Diseases | Bautista-Aguilera, Óscar M. CSIC ORCID; Hagenow, S.; Palomino-Antolín, Alejandra; Farré-Alins, V.; Ismaili, L.; Joffrin, P. L.; Jimeno, M. Luisa CSIC ORCID; Soukup, Ondrej; Janockova, Jana; Kalinowski, A.; Proschak, E.; Iriepa, Isabel; Moraleda, I.; Schwed, J. S.; Romero Jódar, Alejandro CSIC ORCID; López-Muñoz, Francisco; Chioua, Mourad CSIC ORCID ; Egea, Javier; Ramsay, R. R.; Marco-Contelles, José CSIC ORCID; Stark, H. | artículo |
closedAccess | | 2017 | New (benz)imidazolopyridino tacrines as nonhepatotoxic, cholinesterase inhibitors for Alzheimer disease | Boulebd, Houssem; Ismaili, L.; Martin, Helene; Bonet, A.; Chioua, Mourad CSIC ORCID ; Marco-Contelles, José CSIC ORCID; Belfaitah, A. | artículo |
closedAccess | | 2019 | New method for the synthesis of 4-aryl-3,4-dihydro-2H-benzo[g]chromene-2,5,10-triones | Choura, E.; Ncir, M.; Maalej, E.; Marco-Contelles, José CSIC ORCID; Ismaili, L.; Chabchoub, Fakher | artículo |
openAccess | | 2015 | Novel tacrine-grafted ugi adducts as multipotent anti-alzheimer drugs: A synthetic renewal in tacrine-ferulic acid hybrids | Benchekroun, Mohamed; Bartolini, Manuela; Egea, Javier; Romero Jódar, Alejandro CSIC ORCID; Soriano, Elena CSIC; Pudlo, M.; Luzet, Vincenza; Andrisano, V.; Jimeno, M. Luisa CSIC ORCID; López, M. G.; Wehle, S.; Gharbi, T.; Refouvelet, B.; Andrés, Lucía de CSIC; Herrera-Arozamena, Clara CSIC ORCID CVN; Monti, B.; Bolognesi, Maria Laura; Rodríguez-Franco, María Isabel CSIC ORCID ; Decker, Michael; Marco-Contelles, José CSIC ORCID; Ismaili, L. | artículo |
closedAccess | | 2020 | Propargylamine-derived multi-target directed ligands for Alzheimer's disease therapy | do Carmo Carreiras, María; Ismaili, L.; Marco-Contelles, José CSIC ORCID | artículo |
closedAccess | | 2021 | Regioselective Synthesis of Novel [1,2,4]Triazolo[1,5-a]pyridine Derivatives | Hassen, M. B.; Masmoudi, F.; Zribi, L.; Trigui, M.; Ismaili, L.; Marco-Contelles, José CSIC ORCID; Chabchoub, Fakher | artículo |
closedAccess | | 2021 | Synthesis and Biological Assessment of PyrimidoTacrines as Promising Agents for Alzheimer's Disease Therapy | Dakhlaoui, I.; Maalej, E.; Martin, Helene; Lucht, A.; Iriepa, I.; Moraleda, I.; Marco-Contelles, José CSIC ORCID; Chabchoub, Fakher; Ismaili, L. | artículo |
openAccess | | 14-may-2016 | Synthesis and Biological Evaluation of Benzochromenopyrimidinones as Cholinesterase Inhibitors and Potent Antioxidant, Non-Hepatotoxic Agents for Alzheimer’s Disease | Dgachi, Youssef; Bautista-Aguilera, Óscar M. CSIC ORCID; Benchekroun, Mohamed; Martin, Hélène; Bonet, Alexandre; Knez, Damijan; Godyń, Justyna; Malawska, Bárbara; Gobec, Stanislav; Chioua, Mourad CSIC ORCID ; Janockova, Jana; Soukup, O.; Chabchoub, Fakher; Marco-Contelles, José CSIC ORCID; Ismaili, L. | artículo |
closedAccess | | 2019 | Synthesis and Biological Evaluation of Novel Chromone+Donepezil Hybrids for Alzheimer's Disease Therapy | Malek, R.; Refouvelet, B.; Benchekroun, Mohamed; Iriepa, Isabel; Moraleda, I.; Andrys, R.; Musilek, K.; Marco-Contelles, José CSIC ORCID; Ismaili, L. | artículo |
closedAccess | | 2021 | Synthesis and Fluorescence of (E)-3-Aryl-2-(5-aryl-4H-1,2,4-triazol-3-yl) Acrylonitriles | Zribi, L.; Ismaili, L.; Vieira-Ferreira, L. F.; Ferreira-Machado, I. L.; Marco-Contelles, José CSIC ORCID; Chabchoub, Fakher | artículo |
closedAccess | | 2019 | Synthesis of (±)-cis-1-Aryl-3-oxo-2,3-dihydro-1H-benzo[f]chromene-2-carbonitriles and (±)-trans-4-Aryl-2-oxo-3,4-dihydro-2H-benzo[h]chromene-3-carbonitriles | Mkaouar, K.; Iriepa, Isabel; Diez-Iriepa, Daniel CSIC; Marco-Contelles, José CSIC ORCID; Ismaili, L.; Chabchoub, Fakher | artículo |
closedAccess | | 2019 | Synthesis of new ferulic/lipoic/comenic acid-melatonin hybrids as antioxidants and Nrf2 activators via Ugi reaction | Pachón-Angona, I.; Martin, Helene; Chhor, S.; Oset-Gasque, María Jesús; Refouvelet, B.; Marco-Contelles, José CSIC ORCID; Ismaili, L. | artículo |
closedAccess | | 2019 | Synthesis, antioxidant and Aβ anti-aggregation properties of new ferulic, caffeic and lipoic acid derivatives obtained by the Ugi four-component reaction | Benchekroun, Mohamed; Pachón-Angona, I.; Luzet, V.; Martin, Helene; Oset-Gasque, María Jesús; Marco-Contelles, José CSIC ORCID; Ismaili, L. | artículo |
closedAccess | | 2016 | Synthesis, regioselectivity, and DFT analysis of new antioxidant pyrazolo[4,3-c]quinoline-3,4-diones | Tomassoli, I.; Herlem, G.; Picaud, F.; Benchekroun, Mohamed; Bautista-Aguilera, Óscar M. CSIC ORCID; Luzet, Vincenza; Jimeno, M. Luisa CSIC ORCID; Gharbi, T.; Refouvelet, B.; Ismaili, L. | artículo |
openAccess | | 2021 | Tacrines as Therapeutic Agents for Alzheimer's Disease. V. Recent Developments | Bautista-Aguilera, Óscar M. CSIC ORCID; Ismaili, L.; Iriepa, Isabel; Diez-Iriepa, Daniel CSIC; Chabchoub, Fakher; Marco-Contelles, José CSIC ORCID; Pérez-García, Marta CSIC ORCID | artículo |
closedAccess | | 2017 | Tetrahydropyranodiquinolin-8-amines as new, non hepatotoxic, antioxidant, and acetylcholinesterase inhibitors for Alzheimer's disease therapy | Dgachi, Youssef; Sokolov, O.; Luzet, V.; Godyn, J.; Panek, D.; Bonet, A.; Martin, Helene; Iriepa, Isabel; Moraleda, I.; García-Iriepa, C.; Janockova, J.; Richert, L.; Soukup, O.; Malawska, B.; Chabchoub, Fakher; Marco-Contelles, José CSIC ORCID; Ismaili, L. | artículo |
closedAccess | | 2016 | The Antioxidant Additive Approach for Alzheimer's Disease Therapy: New Ferulic (Lipoic) Acid Plus Melatonin Modified Tacrines as Cholinesterases Inhibitors, Direct Antioxidants, and Nuclear Factor (Erythroid-Derived 2)-Like 2 Activators | Benchekroun, Mohamed; Romero Jódar, Alejandro CSIC ORCID; Egea, Javier; León, Rafael CSIC ORCID ; Michalska, P.; Buendía, I.; Jimeno, M. Luisa CSIC ORCID; Jun, Daniel; Janockova, Jana; Sepsova, V.; Soukup, Ondrej; Bautista-Aguilera, Óscar M. CSIC ORCID; Refouvelet, B.; Ouari, O.; Marco-Contelles, José CSIC ORCID; Ismaili, L. | artículo |