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Derechos | Preview | Fecha Public. | Título | Autor(es) | Tipo |
openAccess | | 2015 | Deciphering the Non-Equivalence of Serine and Threonine O-Glycosylation Points: Implications for Molecular Recognition of the Tn Antigen by an anti-MUC1 Antibody | Martínez-Sáez, N.; Castro-López, Jorge; Valero-González, Jessika; Madariaga, David; Compañón, Ismael; Somovilla, Víctor J.; Salvadó, M.; Asensio, Juan Luis CSIC ORCID; Jiménez-Barbero, Jesús CSIC ORCID; Avenoza, A.; Busto, J.H.; Bernardes, G.J.L.; Peregrina, Jesús M.; Hurtado-Guerrero, Ramón CSIC ORCID; Corzana, Francisco | artículo |
closedAccess | | 2013 | Design and synthesis of fungical transglycosidase inhibitors | Gomollón-Bel, Fernando CSIC ORCID; Marca, Eduardo CSIC; Hurtado-Guerrero, Ramón CSIC ORCID; Delso, J. Ignacio CSIC ORCID; Tejero, Tomás CSIC ORCID; Merino, Pedro CSIC ORCID | comunicación de congreso |
closedAccess | | 2016 | Design of α-S-Neoglycopeptides Derived from MUC1 with a Flexible and Solvent-Exposed Sugar Moiety | Rojas-Ocáriz, V.; Compañón, Ismael; Aydillo, C.; Castro-López, Jorge; Jiménez-Barbero, Jesús CSIC ORCID; Hurtado-Guerrero, Ramón CSIC ORCID; Avenoza, A.; Zurbano, M.M.; Peregrina, Jesús M.; Busto, J.H.; Corzana, Francisco | artículo |
openAccess | | 31-mar-2016 | Design, synthesis, crystallization and biological evaluation of new symmetrical biscationic compounds as selective inhibitors of human Choline Kinase α1 (ChoKα1) | Schiaffino-Ortega, Santiago; Baglioni, Eleonora; Mariotto, Elena; Bortolozzi, Roberta; Serran Aguilera, Lucia; Ríos Marco, Pablo; Carrasco-Jiménez, Maria Paz; Gallo, Miguel A.; Hurtado-Guerrero, Ramón CSIC ORCID; Marco, Carmen; Basso, Giuseppe; Viola, Giampietro; Entrena, Antonio; López-Cara, Luisa C. | artículo |
closedAccess | | 2013 | Determination of potential scaffolds for human choline kinase α1 by chemical deconvolution studies | Sahún-Roncero, M.; Rubio-Ruiz, B.; Conejo-García, A.; Velázquez-Campoy, Adrián; Entrena, Antonio; Hurtado-Guerrero, Ramón CSIC ORCID | artículo |
closedAccess | | 2014 | Discovery of a new binding site on human choline kinase α1: Design, synthesis, crystallographic studies, and biological evaluation of asymmetrical bispyridinium derivatives | Rubio-Ruiz, B.; Figuerola-Conchas, A.; Ramos-Torrecillas, J.; Capitán-Cañadas, F.; Ríos-Marco, P.; Carrasco, M.P.; Gallo, M.A.; Espinosa, A. CSIC ORCID; Marco, C.; Ruiz, C.; Entrena, Antonio; Hurtado-Guerrero, Ramón CSIC ORCID; Conejo-García, A. | artículo |
openAccess | | 6-nov-2018 | Dynamic acetylation of phosphoenolpyruvate carboxykinase toggles enzyme activity between gluconeogenic and anaplerotic reactions | Latorre-Muro, Pedro; Baeza, Josue; Armstrong, Eric A.; Hurtado-Guerrero, Ramón CSIC ORCID; Corzana, Francisco; Wu, Lindsay E.; Sinclair, David A.; Lopez-Buesa, P.; Carrodeguas, José A. CSIC ORCID; Denu, John M. | artículo |
openAccess | | 2015 | Dynamic interplay between catalytic and lectin domains of GalNAc-transferases modulates protein O-glycosylation | Lira-Navarrete, Erandi; de las Rivas, Matilde; Compañón, Ismael; Pallarés, M.C.; Kong, Y.; Iglesias-Fernández, J.; Bernardes, G. J. L.; Peregrina, Jesús M.; Rovira, C.; Bernadó, P.; Bruscolini, P.; Clausen, H.; Lostao, Anabel CSIC ORCID; Corzana, Francisco; Hurtado-Guerrero, Ramón CSIC ORCID | artículo |
openAccess | | 16-ago-2018 | Evidence for substrate-assisted catalysis in N-acetylphosphoglucosamine mutase | Raimi, Olawale G.; Hurtado-Guerrero, Ramón CSIC ORCID; van Aalten, D.M.F. | artículo |
openAccess | | 2021 | Fucosyltransferase-specific inhibitionvianext generation of fucose mimetics | Martin, Kyle C.; Tricomi, Jacopo; Corzana, Francisco; García-García, Ana; Ceballos-Laita, Laura CSIC ORCID; Hicks,Thomas; Monaco, Serena; Angulo, Jesús CSIC ORCID ; Hurtado-Guerrero, Ramón CSIC ORCID; Richichi, Barbara; Sakstein, Robert | artículo |
openAccess | | 4-sep-2013 | Genetic and structural validation of Aspergillus fumigatus N-acetylphosphoglucosamine mutase as an antifungal target | Fang, Wenxia; Du, Ting; Raimi, Olawale G.; Hurtado-Guerrero, Ramón CSIC ORCID; Mariño, Karina; Albarbarawi, Osama; Ferguson, Michael A. J.; Jin, C.; Aalten, Daan M. F. van | artículo |
openAccess | | 10-jun-2013 | Genetic and structural validation of Aspergillus fumigatusUDP-N-acetylglucosamine pyrophosphorylase as an antifungal target | Fang, Wenxia; Du, Ting; Raimi, Olawale G.; Hurtado-Guerrero, Ramón CSIC ORCID; Urbaniak, Michael D.; Ibrahim, Adel F. M.; Ferguson, Michael A. J.; Jin, Cheng Jun; van Aalten, D.M.F. | artículo |
closedAccess | | 2016 | Glycomimetics targeting glycosyltransferases: Synthetic, computational and structural studies of less-polar conjugates | Ghirardello, Mattia CSIC ORCID; Rivas, Matilde de las; Lacetera, Alessandra CSIC ORCID; Delso, J. Ignacio CSIC ORCID; Lira-Navarrete, Erandi; Tejero, Tomás CSIC ORCID; Martín-Santamaría, Sonsoles CSIC ORCID ; Hurtado-Guerrero, Ramón CSIC ORCID; Merino, Pedro CSIC ORCID | artículo |
closedAccess | | 2018 | Inhibitors against fungal cell wall remodeling enzymes | Delso, J. Ignacio CSIC ORCID; Valero-González, Jessika; Gomollón-Bel, Fernando CSIC ORCID; Castro-López, Jorge; Fang, Wenxia; Navratilova, Iva; Aalten, Daan M. F. van; Tejero, Tomás CSIC ORCID; Merino, Pedro CSIC ORCID ; Hurtado-Guerrero, Ramón CSIC ORCID | artículo |
openAccess | | 2016 | Kinetic and functional properties of human mitochondrial phosphoenolpyruvate carboxykinase | Escós, M.; Latorre, P.; Hidalgo, Jorge; Hurtado-Guerrero, Ramón CSIC ORCID; Carrodeguas, José A. CSIC ORCID; Lopez-Buesa, P. | artículo |
openAccess | | 10-abr-2019 | Mechanisms of redundancy and specificity of the Aspergillus fumigatus Crh transglycosylases | Fang, W.; Sanz, A.B.; Bartual, Sergio G. CSIC ORCID; Wang, B.; Ferenbach, A.T.; Farkaš, V.; Hurtado-Guerrero, Ramón CSIC ORCID; Arroyo, J.; van Aalten, D.M.F. | artículo |
openAccess | | 2020 | Molecular basis for fibroblast growth factor 23 O-glycosylation by GalNAc-T3 | Rivas, Matilde de las; Paul Daniel, Earnest James; Narimatsu, Yoshiki; Compañón, Ismael; Kato, Kentaro; Hermosilla, Pablo CSIC ORCID; Thureau, Aurélien; Ceballos-Laita, Laura CSIC ORCID; Coelho, Helena; Bernardó, Pau; Marcelo, Filipa CSIC ORCID; Hansen, Lars; Maeda, Ryota; Lostao, Anabel CSIC ORCID; Corzana, Francisco; Clausen, Henrik; Gerken, Thomas A.; Hurtado-Guerrero, Ramón CSIC ORCID | artículo |
openAccess | | 2016 | Mucin architecture behind the immune response: Design, evaluation and conformational analysis of an antitumor vaccine derived from an unnatural MUC1 fragment | Martínez-Sáez, N.; Supekar, N.T.; Wolfert, M.A.; Bermejo, I.A.; Hurtado-Guerrero, Ramón CSIC ORCID; Asensio, Juan Luis CSIC ORCID; Jiménez-Barbero, Jesús CSIC ORCID; Busto, J.H.; Avenoza, A.; Boons, G.J.; Peregrina, Jesús M.; Corzana, Francisco | artículo |
closedAccess | | 2016 | New glycomimetics targeting human GalNAc-T2, synthesis, computational and structural studies | Ghirardello, Mattia CSIC ORCID; Delso, J. Ignacio CSIC ORCID; Tejero, Tomás CSIC ORCID; Martín-Santamaría, Sonsoles CSIC ORCID ; Hurtado-Guerrero, Ramón CSIC ORCID; Merino, Pedro CSIC ORCID | póster de congreso |
openAccess | | 2017 | NleB/SseK effectors from Citrobacter rodentium, Escherichia coli, and Salmonella enterica display distinct differences in host substrate specificity | El Qaidi, S.; Chen, K.; Halim, A.; Siukstaite, L.; Rueter, C.; Hurtado-Guerrero, Ramón CSIC ORCID; Clausen, H.; Hardwidge, P.R. | artículo |