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Derechos | Preview | Fecha Public. | Título | Autor(es) | Tipo |
openAccess | | abr-2015 | Fitness of Leishmania donovani Parasites Resistant to Drug Combinations | García-Hernández, Raquel CSIC ORCID; Gómez-Pérez, Veronica; Castanys, Santiago; Gamarro, Francisco | artículo |
closedAccess | | 2003 | Functional cloning of the miltefosine transporter: A novel p-type phospholipid translocase from leishmania involved in drug resistance | Pérez-Victoria, F. J.; Gamarro, Francisco; Ouellette, M.; Castanys, Santiago | artículo |
openAccess | | 11-abr-2019 | Functional diversity of ABC transporters in Leishmania | Gamarro, Francisco | comunicación de congreso |
closedAccess | | 2005 | Functional expression of a multidrug P-glycoprotein transporter of Leishmania | Cortés-Selva, F.; Muñoz-Martínez, F.; Iliás, A.; Jiménez, I. A.; Váradi, A.; Gamarro, Francisco; Castanys, Santiago | artículo |
openAccess | | 28-abr-2016 | Genomic and Molecular Characterization of Miltefosine Resistance in Leishmania infantum Strains with Either Natural or Acquired Resistance through Experimental Selection of Intracellular Amastigotes | Mondelaers, Annelies; Sánchez-Cañete, María P.; Hendrickx, Sarah; Eberhardt, Eline; García-Hernández, Raquel CSIC ORCID; Lachaud, Laurence; Cotton, James; Sanders, Mandy; Cuypers, Bart; Imamura, Hideo; Dujardin, J. C.; Delputte, Peter; Cos, Paul; Caljon, Guy; Gamarro, Francisco; Castanys, Santiago; Maes, Louis | artículo |
closedAccess | | 2001 | High-affinity binding of silybin derivatives to the nucleotide-binding domain of a Leishmania tropica P-glycoprotein-like transporter and chemosensitization of a multidrug-resistant parasite to daunomycin | Pérez-Victoria, J. M. ; Pérez-Victoria, F. J.; Conseil, G.; Maitrejean, M.; Barron, D.; Castanys, Santiago; Gamarro, Francisco; Di Pietro, A.; Comte, Gilles | artículo |
openAccess | | 8-nov-2020 | Hit-to lead and target identification studies within a novel class of anti-trypanosomal agents | Ferrins, L; Díaz González, R.; Ceballos-Pérez, G.; Saura, A.; Pérez-Moreno, Guiomar; García-Hernández, Raquel CSIC ORCID; Bosch-Navarrete, Cristina; Gamarro, Francisco; Ruiz-Pérez, Luis Miguel; González-Pacanowska, Dolores; Navarro, M.; Pollastri, M. | actas de congreso |
openAccess | | 8-mar-2020 | Hit-to-lead and target identification studies within a novel class of antitrypanosomal agents | Ferrins, L; Díaz-González, Rosario; Ceballos-Pérez, Gloria; Saura, A.; Pérez-Moreno, Guiomar; García-Hernández, Raquel CSIC ORCID; Boch-Navarrete, C; Gamarro, Francisco; Ruiz-Pérez, Luis Miguel; González-Pacanowska, Dolores; Navarro, M.; Pollastri, M. | actas de congreso |
closedAccess | | 2019 | Hit-to-Lead Optimization of Benzoxazepinoindazoles As Human African Trypanosomiasis Therapeutics | Klug, DM; Tschiegg, L; Díaz, Rosario; Rojas-Barros, D; Pérez-Moreno, Guiomar; Ceballos, G; García-Hernández, Raquel CSIC ORCID; Martinez-Martinez, MS; Manzano, Pilar; Ruiz, LM; Caffrey, CR; Gamarro, Francisco; González-Pacanowska, Dolores; Ferrins, L; Navarro, M.; Pollastri, M.P. | artículo |
openAccess | | 16-jul-2019 | Imidazo[2,1-a]isoindole as a new leishmanicidal scaffold. | Rivas, L.; Arsène, S.; Gómez-Pérez, V.; Escarcena, Ricardo; Abengozar, M. A. CSIC; García-Hernández, Raquel CSIC ORCID; Nácher-Vázquez, M.; San Feliciano, A.; Gamarro, Francisco; del Olmo, Esther | comunicación de congreso |
openAccess | | 29-jul-2019 | Imidazo[2,1-a]isoindole scaffold as an uncharted structure active on Leishmania donovani | Arsène, Sobinson; Gómez-Pérez, Veronica; Escarcena, Ricardo; Abengozar, M. A. CSIC; García-Hernández, Raquel CSIC ORCID; Nácher-Vázquez, Montserrat CSIC ORCID; San Feliciano, A.; Gamarro, Francisco; Rivas, Luis CSIC ORCID ; del Olmo, Esther | artículo |
closedAccess | | 2007 | Inactivation of the miltefosine transporter, LdMT, causes miltefosine resistance that is conferred to the amastigote stage of Leishmania donovani and persists in vivo | Seifert, K.; Pérez-Victoria, F. J.; Stettler, M.; Sánchez-Cañete, María P.; Castanys, Santiago; Gamarro, Francisco; Croft, S.L. | artículo |
closedAccess | | 2011 | Increased glycolytic ATP synthesis is associated with tafenoquine resistance in Leishmania major | Manzano, José Ignacio CSIC ORCID; Carvalho, L.; Pérez-Victoria, J. M. ; Castanys, Santiago; Gamarro, Francisco | artículo |
closedAccess | | 2006 | Insights into the molecular mechanism of action of Celastraceae sesquiterpenes as specific, non-transported inhibitors of human P-glycoprotein | Muñoz-Martínez, F.; Reyes, C. P.; Pérez-Lomas, Antonio L.; Jiménez, I. A.; Gamarro, Francisco; Castanys, Santiago | artículo |
closedAccess | | 1998 | Involvement of thiol metabolism in resistance to glucantime in Leishmania tropica | Arana, F. E.; Pérez-Victoria, J. M. ; Repetto, Y.; Morello, A.; Castanys, Santiago; Gamarro, Francisco | artículo |
openAccess | | 2013 | LABCG2, a New ABC Transporter Implicated in Phosphatidylserine Exposure, Is Involved in the Infectivity and Pathogenicity of Leishmania | Campos-Salinas, Jenny; León-Guerrero, D.; González-Rey, Elena CSIC ORCID; Delgado, M.; Castanys, Santiago; Pérez-Victoria, J. M. ; Gamarro, Francisco | artículo |
openAccess | | 10-feb-2023 | Label-Free Mass Spectrometry Proteomics Reveals Different Pathways Modulated in THP-1 Cells Infected with Therapeutic Failure and Drug Resistance Leishmania infantum Clinical Isolates | Tagliazucchi, Lorenzo; Perea-Martínez, Ana; Fiorini, Greta; Manzano, José Ignacio CSIC ORCID; Genovese, Filippo; García-Hernández, Raquel CSIC ORCID; Pinetti, Diego; Gamarro, Francisco; Costi, Maria Paola | artículo |
openAccess | | 2012 | Leishmania donovani Develops Resistance to Drug Combinations | García-Hernández, Raquel CSIC ORCID; Manzano, José Ignacio CSIC ORCID; Castanys, Santiago; Gamarro, Francisco | artículo |
closedAccess | | 2003 | Leishmania donovani resistance to miltefosine involves a defective inward translocation of the drug | Pérez-Victoria, F. J.; Castanys, Santiago; Gamarro, Francisco | artículo |
closedAccess | | 2011 | Leishmanicidal and reversal multidrug resistance constituents from Aeonium lindleyi | Kennedy, M. L.; Cortés, Fernando; Piñero, J. E.; Castanys, Santiago; López-Arencibia, A.; Gamarro, Francisco; Bazzocchi, I. L.; Jiménez, I. A. | artículo |