Mostrando resultados 7 a 17 de 17
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Derechos | Preview | Fecha Public. | Título | Autor(es) | Tipo |
openAccess | | 2014 | Multipotent cholinesterase/monoamine oxidase inhibitors for the treatment of Alzheimer’s disease: Design, synthesis, biochemical evaluation, ADMET, molecular modeling, and QSAR analysis of novel donepezil-pyridyl hybrids | Bautista-Aguilera, Óscar M. CSIC ORCID; Esteban, Gerard; Chioua, Mourad CSIC ORCID ; Nikolic, Katarina; Agbaba, Danica; Moraleda, Ignacio; Iriepa, Isabel; Soriano, Elena CSIC; Samadi, Abdelouahid CSIC ORCID; Unzeta, Mercedes; Marco-Contelles, José CSIC ORCID | artículo |
closedAccess | | 2017 | Multitarget-Directed Ligands Combining Cholinesterase and Monoamine Oxidase Inhibition with Histamine H3R Antagonism for Neurodegenerative Diseases | Bautista-Aguilera, Óscar M. CSIC ORCID; Hagenow, S.; Palomino-Antolín, Alejandra; Farré-Alins, V.; Ismaili, L.; Joffrin, P. L.; Jimeno, M. Luisa CSIC ORCID; Soukup, Ondrej; Janockova, Jana; Kalinowski, A.; Proschak, E.; Iriepa, Isabel; Moraleda, I.; Schwed, J. S.; Romero Jódar, Alejandro CSIC ORCID; López-Muñoz, Francisco; Chioua, Mourad CSIC ORCID ; Egea, Javier; Ramsay, R. R.; Marco-Contelles, José CSIC ORCID; Stark, H. | artículo |
closedAccess | | 2014 | N-methyl-N-((1-methyl-5-(3-(1-(2-methylbenzyl)piperidin-4-yl)propoxy)-1H-indol-2-yl)methyl)prop-2-yn-1-amine, a new cholinesterase and monoamine oxidase dual inhibitor | Bautista-Aguilera, Óscar M. CSIC ORCID; Samadi, Abdelouahid CSIC ORCID; Chioua, Mourad CSIC ORCID ; Nikolic, K.; Filipic, S.; Agbaba, Danica; Soriano, Elena CSIC; Andrés, Lucía de CSIC; Rodríguez-Franco, María Isabel CSIC ORCID ; Alcaro, S.; Ramsay, R. R.; Ortuso, F.; Yáñez, Matilde; Marco-Contelles, José CSIC ORCID | artículo |
closedAccess | | 2015 | Predicting targets of compounds against neurological diseases using cheminformatic methodology | Nikolic, Katarina; Mavridis, L.; Bautista-Aguilera, Óscar M. CSIC ORCID; Marco-Contelles, José CSIC ORCID; Stark, H.; do Carmo Carreiras, María; Rossi, I.; Massarelli, P.; Agbaba, Danica; Ramsay, Rona R.; Mitchell, J. B. O. | artículo |
openAccess | | 2023 | Straightforward Synthesis of Bis[(trifluoromethyl)sulfonyl]ethylated Isocoumarins from 2-Ethynylbenzoates | Petcu, Sonia A. CSIC; Lázaro-Milla, Carlos; Rodríguez, Francisco Javier; Iriepa, Isabel; Bautista-Aguilera, Óscar M. CSIC ORCID; Aragoncillo, Cristina CSIC ORCID; Alonso, José M. CSIC; Almendros, Pedro CSIC ORCID | artículo |
openAccess | | 14-may-2016 | Synthesis and Biological Evaluation of Benzochromenopyrimidinones as Cholinesterase Inhibitors and Potent Antioxidant, Non-Hepatotoxic Agents for Alzheimer’s Disease | Dgachi, Youssef; Bautista-Aguilera, Óscar M. CSIC ORCID; Benchekroun, Mohamed; Martin, Hélène; Bonet, Alexandre; Knez, Damijan; Godyń, Justyna; Malawska, Bárbara; Gobec, Stanislav; Chioua, Mourad CSIC ORCID ; Janockova, Jana; Soukup, O.; Chabchoub, Fakher; Marco-Contelles, José CSIC ORCID; Ismaili, L. | artículo |
closedAccess | | 2016 | Synthesis, regioselectivity, and DFT analysis of new antioxidant pyrazolo[4,3-c]quinoline-3,4-diones | Tomassoli, I.; Herlem, G.; Picaud, F.; Benchekroun, Mohamed; Bautista-Aguilera, Óscar M. CSIC ORCID; Luzet, Vincenza; Jimeno, M. Luisa CSIC ORCID; Gharbi, T.; Refouvelet, B.; Ismaili, L. | artículo |
openAccess | | 2021 | Tacrines as Therapeutic Agents for Alzheimer's Disease. V. Recent Developments | Bautista-Aguilera, Óscar M. CSIC ORCID; Ismaili, L.; Iriepa, Isabel; Diez-Iriepa, Daniel CSIC; Chabchoub, Fakher; Marco-Contelles, José CSIC ORCID; Pérez-García, Marta CSIC ORCID | artículo |
closedAccess | | 2016 | The Antioxidant Additive Approach for Alzheimer's Disease Therapy: New Ferulic (Lipoic) Acid Plus Melatonin Modified Tacrines as Cholinesterases Inhibitors, Direct Antioxidants, and Nuclear Factor (Erythroid-Derived 2)-Like 2 Activators | Benchekroun, Mohamed; Romero Jódar, Alejandro CSIC ORCID; Egea, Javier; León, Rafael CSIC ORCID ; Michalska, P.; Buendía, I.; Jimeno, M. Luisa CSIC ORCID; Jun, Daniel; Janockova, Jana; Sepsova, V.; Soukup, Ondrej; Bautista-Aguilera, Óscar M. CSIC ORCID; Refouvelet, B.; Ouari, O.; Marco-Contelles, José CSIC ORCID; Ismaili, L. | artículo |
openAccess | | 2020 | Triazolopyridopyrimidine: A New Scaffold for Dual-Target Small Molecules for Alzheimer's Disease Therapy | Zribi, L.; Pachón-Angona, I.; Bautista-Aguilera, Óscar M. CSIC ORCID; Diez-Iriepa, Daniel CSIC; Marco-Contelles, José CSIC ORCID; Ismaili, L.; Iriepa, Isabel; Chabchoub, Fakher | artículo |
closedAccess | | 2014 | Wnt signaling pathway, a potential target for Alzheimer's disease treatment, is activated by a novel multitarget compound ASS234 | Pino, Javier del; Ramos, Eva; Bautista-Aguilera, Óscar M. CSIC ORCID; Marco-Contelles, José CSIC ORCID; Romero Jódar, Alejandro CSIC ORCID | artículo |