Mostrando resultados 8 a 24 de 24
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Derechos | Preview | Fecha Public. | Título | Autor(es) | Tipo |
closedAccess | | 2010 | Design, synthesis and inhibitory activity against Mycobacterium tuberculosis thymidine monophosphate kinase of acyclic nucleoside analogues with a distal imidazoquinolinone | Familiar, Olga CSIC; Munier-Lehmann, Hélène; Aínsa, José A.; Camarasa Rius, María José CSIC ORCID; Peréz-Pérez, María-Jesús CSIC ORCID | artículo |
closedAccess | | 11-jul-2019 | Design, Synthesis, and Efficacy Testing of Nitroethylene- and 7-Nitrobenzoxadiazol-Based Flavodoxin Inhibitors against Helicobacter pylori Drug-Resistant Clinical Strains and in Helicobacter pylori-Infected Mice | Salillas, Sandra; Alías, Miriam CSIC; Michel, V.; Mahía Moros, Alejandro CSIC; Lucía Quintana, Ainhoa; Rodrigues, L.; Bueno, J.; Galano-Frutos, Juan J.; Reuse, Hilde de; Velázquez-Campoy, Adrián; Carrodeguas, José A. CSIC ORCID; Sostres, Carlos; Castillo, Javier; Aínsa, José A.; Díaz de Villegas, María D. CSIC ORCID; Lanas, Ángel; Touati, Eliette; Sancho, Javier CSIC ORCID | artículo |
openAccess | | 2022 | Development of functionalized nanocarriers for drug targeting in tuberculosis | Baranyai, Zsuzsa CSIC ORCID; Alleva, María CSIC ORCID; Martínez-Vicente, Pablo CSIC ORCID; Moros, María CSIC ORCID; Millán-Placer, Ana C.; Picó, Ana; Aínsa, José A.; Fuente, Jesús M. de la CSIC ORCID | comunicación de congreso |
openAccess | | 15-mar-2022 | Discovery of 3H-pyrrolo[2,3-c]quinolines with activity against Mycobacterium tuberculosis by allosteric inhibition of the glutamate-5-kinase enzyme | Panciera, Michele; Lence, Emilio; Rodríguez, Ángela; Gracia, Begoña; Aínsa, José A.; Marco-Marín, Clara CSIC ORCID; Rubio, Vicente CSIC ORCID ; Duarte Correia, Carlos Roque; González-Bello, Concepción | artículo |
openAccess | | 2018 | Discovery of antimicrobial compounds targeting bacterial type FAD synthetases | Sebastián, María; Anoz-Carbonell, E.; Gracia, B.; Cossio, P.; Aínsa, José A.; Lans, Isaias CSIC; Medina, Milagros CSIC ORCID | artículo |
openAccess | | 2018 | Fighting superbugs: new promising compounds against Helicobacter pylori | Salillas, Sandra; Alías, Miriam CSIC; Michel, V.; Mahía Moros, Alejandro CSIC; Lucía Quintana, Ainhoa; Rodrigues, L.; Bueno, J.; Galano-Frutos, Juan J.; Velázquez-Campoy, Adrián; Carrodeguas, José A. CSIC ORCID; Sostres, Carlos; Castillo, Javier; Aínsa, José A.; Díaz de Villegas, María D. CSIC ORCID; Lanas, Ángel; Touati, E.; Sancho, Javier CSIC ORCID | comunicación de congreso |
openAccess | | 14-ago-2020 | In silico discovery and biological validation of ligands of FAD synthase, a promising new antimicrobial target | Lans, Isaias CSIC; Anoz-Carbonell, E.; Palacio-Rodríguez, K.; Aínsa, José A.; Medina, Milagros CSIC ORCID; Cossio, P. | artículo |
closedAccess | | 2018 | Micelas polipetídicas recubiertas con alginato para encapsulación de bedaquilina | Soria-Carrera, Héctor CSIC ORCID; Lucía, Ainhoa; Matteis, Laura de; Aínsa, José A.; Fuente, Jesús M. de la CSIC ORCID; Martín-Rapún, Rafael CSIC ORCID | póster de congreso |
openAccess | | 2019 | Mycobacterial aminoglycoside acetyltransferases: A little of drug resistance, and a lot of other roles | Sanz-García, Fernando; Anoz-Carbonell, Ernesto; Pérez-Herrán, Esther; Martín, Carlos; Lucía, Ainhoa; Rodrigues, Liliana; Aínsa, José A. | artículo de revisión |
closedAccess | | 2018 | Nanoemulsion-based chitosan nanocapsules as efficient delivery system for bedaquiline antibiotic | García-Embid, Sonia; Serrano-Sevilla, Inés; Matteis, Laura de; Lucía, Ainhoa; Aínsa, José A.; Fuente, Jesús M. de la CSIC ORCID | póster de congreso |
openAccess | | 2021 | Nanotechnology-based targeted drug delivery: An emerging tool to overcome tuberculosis | Baranyai, Zsuzsa CSIC ORCID; Soria-Carrera, Héctor CSIC ORCID; Alleva, María CSIC ORCID; Millán-Placer, Ana C.; Lucía, Ainhoa; Martín-Rapún, Rafael CSIC ORCID; Aínsa, José A.; Fuente, Jesús M. de la CSIC ORCID | artículo |
closedAccess | | 2018 | New active formulations against M. tuberculosis: Bedaquiline encapsulation in lipid nanoparticles and chitosan nanocapsules | Matteis, Laura de; Jary, Dorothée; Lucía, Ainhoa; García-Embid, Sonia; Serrano-Sevilla, Inés; Pérez, Daniel; Aínsa, José A.; Navarro, Fabrice; Fuente, Jesús M. de la CSIC ORCID | artículo |
openAccess | | 2019 | Polypeptidic micelles stabilized with sodium alginate enhance the activity of encapsulated bedaquiline | Soria-Carrera, Héctor CSIC ORCID; Lucía, Ainhoa; Matteis, Laura de; Aínsa, José A.; Fuente, Jesús M. de la CSIC ORCID; Martín-Rapún, Rafael CSIC ORCID | artículo |
closedAccess | | 2018 | Polysaccharide-coated polypeptidic micelles for drug delivery | Soria-Carrera, Héctor CSIC ORCID; Matteis, Laura de; Lucía, Ainhoa; Aínsa, José A.; Martín-Rapún, Rafael CSIC ORCID; Fuente, Jesús M. de la CSIC ORCID | comunicación de congreso |
openAccess | | 2020 | Resisting antimicrobial resistance: Flavodoxin inhibitors to combat Helicobacter pylori infection | Salillas, Sandra; Alías, Miriam CSIC; Michel, V.; Mahía Moros, Alejandro CSIC; Conde-Giménez, María; Anoz-Carbonell, Ernesto; Lucía Quintana, Ainhoa; Rodrigues, L.; Bueno, J.; Galano-Frutos, Juan J.; Velázquez-Campoy, Adrián; Carrodeguas, José A. CSIC ORCID; Sostres, Carlos; Castillo, Javier; Gálvez, José A. CSIC ORCID; Aínsa, José A.; Díaz de Villegas, María D. CSIC ORCID; Lanas, Ángel; Touati, Eliette; Sancho, Javier CSIC ORCID | póster de congreso |
openAccess | | 20-sep-2021 | Selective targeting of human and animal pathogens of the Helicobacter genus by flavodoxin inhibitors: Efficacy, synergy, resistance and mechanistic studies | Salillas, Sandra; Galano-Frutos, Juan J.; Mahía Moros, Alejandro CSIC; Maity, Ritwik; Conde-Giménez, María; Anoz-Carbonell, E.; Berlamont, Helena; Velázquez-Campoy, Adrián; Touati, Eliette; Mamat, Uwe; Schaible, Ulrich E.; Gálvez, José A. CSIC ORCID; Díaz de Villegas, María D. CSIC ORCID; Haesebrouck, Freddy; Aínsa, José A.; Sancho, Javier CSIC ORCID | artículo |
closedAccess | | 2019 | Synthesis and biological activity of dehydrophos derivatives | Jiménez-Andreu, M. Mercedes CSIC; Lucía Quintana, Ainhoa; Aínsa, José A.; Sayago, Francisco J. CSIC ORCID; Cativiela, Carlos CSIC ORCID | artículo |