Derechos | Preview | Fecha Public. | Título | Autor(es) | Tipo |
openAccess | | 20-ago-2021 | A conformation selective mode of inhibiting SRC improves drug efficacy and tolerability | Temps, Caroline; Lietha, Daniel CSIC ORCID ; Webb, Emily R.; Li, Xue-Feng; Dawson, John C.; Muir, Morwenna; Macleod, Kenneth G.; Valero, Teresa; Munro, Alison F.; Contreras-Montoya, Rafael; Luque-Ortega, Juan Román CSIC ORCID ; Fraser, Craig; Beetham, Henry; Schoenherr, Christina; Lopalco, Maria; Arends, Mark J.; Frame, Margaret C.; Qian, Bin-Zhi; Brunton, Valerie G.; Carragher, Neil O.; Unciti-Broceta, Asier | artículo |
openAccess | | 27-jul-2021 | A new layer of phosphoinositide-mediated allosteric regulation uncovered for SHIP2 | Le Coq, Johanne; López-Navajas, Pilar CSIC ; Rodrigo Martín, Bárbara CSIC; Alfonso, Carlos CSIC ORCID ; Lietha, Daniel CSIC ORCID | artículo |
openAccess | | 21-mar-2022 | A tethered ligand assay to probe SARS-CoV-2:ACE2 interactions | Bauer, Magnus Sebastian; Gruber, Sophia; Hausch, Adina; Gomes, Priscila S. F. C.; Milles, Lukas Frederik; Nicolaus, Thomas; Schendel, Leonard C.; López-Navajas, Pilar CSIC ; Procko, Erik; Lietha, Daniel CSIC ORCID ; Melo, Marcelo C. R.; Bernardi, Rafael C.; Gaub, Hermann Eduard; Lipfert, Jan | artículo |
openAccess | | 9-ago-2021 | A Tethered Ligand Assay to Probe SARS-CoV-2:ACE2 Interactions | Bauer, Magnus Sebastian; Gruber, Sophia; Hausch, Adina; Milles, Lukas Frederik; Nicolaus, Thomas; Schendel, Leonard C.; López-Navajas, Pilar CSIC ; Procko, Erik; Lietha, Daniel CSIC ORCID ; Bernardi, Rafael C.; Gaub, Hermann Eduard; Lipfert, Jan | preprint |
openAccess | | 29-oct-2020 | Design, synthesis and biological evaluations of covalent inhibitors of Focal Adhesion Kinase (FAK) against human malignant glioblastoma | Li, Bo; Li, Yongliang; Tomkiewicz-Raulet, Céline; Dao, Pascal; Lietha, Daniel CSIC ORCID ; Yen-Pon, Expédite; Du, Zhiyun; Coumoul, Xavier; Garbay, Christiane; Etheve-Quelquejeu, Mélanie; Chen, Huixiong | artículo |
openAccess | | 24-ene-2020 | FAK structure and regulation by membrane interactions and force in focal adhesions | Tapial Martínez, Paula CSIC; López-Navajas, Pilar CSIC ; Lietha, Daniel CSIC ORCID | artículo |
openAccess | | 15-oct-2022 | New insights into FAK structure and function in focal adhesions | Le Coq, Johanne; Acebrón, Iván CSIC ORCID; Rodrigo Martín, Bárbara CSIC; López-Navajas, Pilar CSIC ; Lietha, Daniel CSIC ORCID | artículo |
openAccess | | jun-2021 | ORP2 couples LDL-cholesterol transport to FAKactivation by endosomal cholesterol/PI(4,5)P2exchange | Takahashi, Kohta; Kanerva, Kristiina; Vanharanta, Lauri; Almeida-Souza, Leonardo; Lietha, Daniel CSIC ORCID ; Olkkonen, Vesa M.; Ikonen, Elina | artículo |
openAccess | | 2-abr-2019 | Structural and mechanistic insights into mechanoactivation of focal adhesion kinase | Bauer, Magnus Sebastian; Baumann, Fabian; Daday, Csaba; Redondo, Pilar; Durner, Ellis; Markus Andreas, Jobst; Milles, Lukas Frederik; Mercadante, Davide; Pippig, Diana Angela; Gaub, Hermann Eduard; Gräter, Frauke; Lietha, Daniel CSIC ORCID | artículo |
openAccess | | 11-ago-2020 | Structural basis of Focal Adhesion Kinase activation on lipid membranes | Acebrón, Iván CSIC ORCID; Righetto, Ricardo D.; Schoenherr, Christina; de Buhr, Svenja; Redondo, Pilar; Culley, Jayne; Rodríguez, Carlos F. CSIC ORCID; Daday, Csaba; Biyani, Nikhil; Llorca, Óscar CSIC ORCID; Byron, Adam; Chami, Mohamed; Gräter, Frauke; Boskovic, Jasminka; Frame, Margaret C.; Stahlberg, Henning; Lietha, Daniel CSIC ORCID | artículo |
openAccess | | 3-ene-2022 | TDP-43 modulation by Tau-Tubulin kinase 1 inhibitors: A new avenue for future amyotrophic lateral sclerosis therapy | Nozal, Vanesa CSIC ORCID; Martínez-González, Loreto CSIC ORCID ; Gómez-Almería, Marta; Gonzalo-Consuegra, Claudia; Santana, Paula; Chaikuad, Apirat; Cuevas, Eva P. CSIC ORCID ; Knapp, Stefan; Lietha, Daniel CSIC ORCID ; Ramírez, David; Petralla, Sabrina; Monti, B.; Gil, Carmen CSIC ORCID ; Martín-Requero, Ángeles CSIC ORCID ; Palomo, Valle CSIC ORCID ; De Lago, E.; Martínez Gil, Ana CSIC ORCID | artículo |