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| Rights | Preview | Issue Date | Title | Author(s) | Type |
| openAccess |  | 29-May-2018 | A fluorescence anisotropy assay to discover and characterize ligands targeting the maytansine site of tubulin | Menchon, Grégory; Lucena-Agell, Daniel CSIC ORCID ; Díaz, José Fernando CSIC ORCID ; Steinmetz, Michel O. | artículo |
| closedAccess |  | 12-Oct-2020 | A method for the stereoselective construction of the hemiaminal center in zampanolides | Brütsch, Tobias M.; Berardozzi, Simone; Rothe, Marlene L.; Redondo-Horcajo, Mariano CSIC ORCID; Díaz, José Fernando CSIC ORCID ; Altmann, Karl-Heinz | artículo |
| openAccess |  | Mar-2013 | A structure-based design of new C2- and C13-substituted taxanes: Tubulin binding affinities and extended quantitative structure-activity relationships using comparative binding energy (COMBINE) analysis | Coderch, Claire; Tang, Yong; Klett, Javier CSIC ORCID; Zhang, Shu-En; Ma, Yung-Tao; Shaorong, Wang; Matesanz, Ruth CSIC ; Pera, Benet CSIC; Canales, Ángeles CSIC ORCID; Jiménez-Barbero, Jesús CSIC ORCID; Morreale, Antonio; Díaz, José Fernando CSIC ORCID ; Fang, Wei-shuo S.; Gago, Federico CSIC ORCID | artículo |
| openAccess |  | 18-May-2001 | Activation of cell division protein FtsZ. Control of switch loop T3 conformation by the nucleotide gamma-phosphate | Díaz, José Fernando CSIC ORCID ; Kralicek, Andrew; Mingorance, Jesús; Palacios, Juan Manuel; Vicente, Miguel; Andreu, José Manuel CSIC ORCID | artículo |
| closedAccess |  | 26-Aug-2016 | Aggregated compound biological signatures facilitate phenotypic drug discovery and target elucidation | Cortés Cabrera, Álvaro CSIC ORCID; Lucena-Agell, Daniel CSIC ORCID ; Redondo-Horcajo, Mariano CSIC ORCID ; Barasoain, Isabel CSIC ; Díaz, José Fernando CSIC ORCID ; Fasching, Bernhard; Petrone, Paula M. | artículo |
| openAccess |  | 20-May-2016 | Antivascular and antitumor properties of the tubulin-binding chalcone TUB091 | Canela, María-Dolores CSIC; Noppen, Sam; Bueno, Oskía; Prota, Andrea E.; Bargsten, Katja; Sáez-Calvo, Gonzalo; Jimeno, M. Luisa CSIC ORCID; Benkhei, Mohammed; Ribatti, Domenico; Velázquez, Sonsoles CSIC ORCID CVN; Camarasa Rius, María José CSIC ORCID; Díaz, José Fernando CSIC ORCID ; Steinmetz, Michel O.; Priego, Eva María CSIC ORCID; Peréz-Pérez, María-Jesús CSIC ORCID ; Liekens, Sandra | artículo |
| closedAccess |  | Jul-2008 | Apo-Hsp90 coexists in two open conformational states in solution | Bron, P.; Giudice, E.; Rolland, J.P.; Martínez Buey, Rubén CSIC ORCID CVN; Barbier, Pascale; Díaz, José Fernando CSIC ORCID ; Peyrot, Vincent; Thomas, D.; Garnier, C. | artículo |
| closedAccess | | 2007 | Arylthioindole inhibitors of tubulin polymerization. 3. Biological evaluation, structure-activity relationships and molecular modeling studies | La Regina, Giuseppe; Edler, Michael C.; Brancale, Andrea; Kandil, Sahar; Coluccia, Antonio; Piscitelli, Francesco; Hamel, Ernest; De Martino, Gabriella; Matesanz, Ruth CSIC ; Díaz, José Fernando CSIC ORCID ; Scovassi, Anna Ivana; Prosperi, Ennio; Lavecchia, Antonio; Novellino, Ettore; Artico, Marino; Silvestri, Romano | artículo |
| openAccess |  | 11-Dec-1998 | Changes in microtubule protofilament number induced by Taxol binding to an easily accessible site. Internal microtubule dynamics | Díaz, José Fernando CSIC ORCID ; Valpuesta, José M. CSIC ORCID ; Chacón, Pablo CSIC ORCID; Diakun, Gregory P.; Andreu, José Manuel CSIC ORCID | artículo |
| closedAccess | | 2007 | Characterizing Ligand-Microtubule binding by competition methods | Díaz, José Fernando CSIC ORCID ; Martínez Buey, Rubén CSIC ORCID CVN | artículo |
| openAccess |  | 2009 | Chloroacetylation of cyclostreptin influences its interaction with tubulin | Calvo, Enrique; Barasoain, Isabel CSIC ; Camafeita, Emilio; Andreu, José Manuel CSIC ORCID ; López, Juan Antonio; Díaz, José Fernando CSIC ORCID | comunicación de congreso |
| closedAccess |  | 2012 | Comparative Binding Energy (COMBINE) Analysis Supports a Proposal for the Binding Mode of Epothilones to β-Tubulin | Coderch, Claire; Klett, Javier CSIC ORCID; Morreale, Antonio; Díaz, José Fernando CSIC ORCID ; Gago, Federico CSIC ORCID | artículo |
| openAccess |  | 2018 | Conformational mimetics of the α-methyl chalcone TUB091 binding tubulin: Design, synthesis and antiproliferative activity | Bueno, Oskía; Tobajas, Gloria; Quesada, Ernesto; Estévez-Gallego, Juan CSIC ORCID ; Noppen, Sam; Camarasa Rius, María José CSIC ORCID; Díaz, José Fernando CSIC ORCID ; Liekens, Sandra; Priego, Eva María CSIC ORCID; Peréz-Pérez, María-Jesús CSIC ORCID | artículo |
| openAccess |  | 2-Jan-1998 | Control of the structural stability of the tubulin dimer by one high affinity bound magnesium ion at nucleotide N-site | Menéndez, Margarita CSIC ORCID; Rivas, Germán CSIC ORCID ; Díaz, José Fernando CSIC ORCID ; Andreu, José Manuel CSIC ORCID | artículo |
| closedAccess |  | 14-Jun-2011 | Corrigendum: Mechanism of Action of the Cytotoxic Macrolides Amphidinolide X and J | Trigili, Chiara CSIC; Pera, Benet CSIC; Barbazanges, Marion; Cossy, Janine; Meyer, Christophe; Pineda, Oriol; Rodríguez-Escrich, Carles; Urpí, Félix; Vilarrasa, Jaume; Díaz, José Fernando CSIC ORCID ; Barasoain, Isabel CSIC | corrigenda |
| openAccess |  | 22-Oct-2010 | Cpl-7, a Lysozyme Encoded by a Pneumococcal Bacteriophage with a Novel Cell Wall-Binding Motif | Bustamante, Noemí CSIC; Campillo, Nuria E. CSIC ORCID ; García, Ernesto CSIC ORCID ; Gallego, Cristina; Pera, Benet CSIC; Diakun, Gregory P.; Saiz, José L.; García, Pedro CSIC ORCID ; Díaz, José Fernando CSIC ORCID ; Menéndez, Margarita CSIC ORCID | artículo |
| openAccess |  | 20-Mar-2019 | Crystal Structure of the Cyclostreptin-Tubulin Adduct: Implications for Tubulin Activation by Taxane-Site Ligands | Balaguer, Francisco de Asís; Mühlethaler, Tobias; Estévez-Gallego, Juan CSIC ORCID ; Calvo, Enrique; Giménez-Abián, Juan F. CSIC ; Risinger, April L.; Sorensen, Erik J.; Vanderwal, Christopher D.; Altmann, Karl-Heinz; Mooberry, Susan; Steinmetz, Michel O.; Oliva, María A. CSIC ORCID ; Prota, Andrea E.; Díaz, José Fernando CSIC ORCID | artículo |
| closedAccess |  | 30-Aug-2005 | Cyclostreptin (FR182877), an Antitumour Tubulin-Polymerizing Agent Deficient in Enhancing Tubulin Assembly Despite Its High Affinity for the Taxoid Site | Edler, Michael C.; Martínez Buey, Rubén CSIC ORCID CVN; Gussio, Rick; Marcus, Adam I.; Vanderwal, Christopher D.; Sorensen, Erik J.; Díaz, José Fernando CSIC ORCID ; Giannakakou, Paraskevi; Hamel, Ernest | artículo |
| openAccess |  | Jan-2007 | Cyclostreptin binds covalently to microtubule pores and lumenal taxoid binding sites | Martínez Buey, Rubén CSIC ORCID CVN; Calvo, Enrique; Barasoain, Isabel CSIC ; Pineda, Oriol; Edler, Michael C.; Matesanz, Ruth CSIC ; Cerezo, Gemma; Vanderwal, Christopher D.; Day, Billy W.; Sorensen, Erik J.; López, Juan Antonio; Andreu, José Manuel CSIC ORCID ; Hamel, Ernest; Díaz, José Fernando CSIC ORCID | artículo |
| closedAccess |  | Jan-2012 | Cyclostreptin Derivatives Specifically Target Cellular Tubulin and Further Map the Paclitaxel Site | Calvo, Enrique; Barasoain, Isabel CSIC ; Matesanz, Ruth CSIC ; Pera, Benet CSIC; Camafeita, Emilio; Pineda, Oriol; Hamel, Ernest; Vanderwal, Christopher D.; Andreu, José Manuel CSIC ORCID ; López, Juan Antonio; Díaz, José Fernando CSIC ORCID | artículo |
