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Showing results 1 to 14 of 14
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openAccessproceedings-22-00108 (1).pdf.jpg15-May-20194,4-Disubstituted N-benzylpiperidines: a novel class of fusion inhibitors of influenza virus H1N1 targeting a new binding site in hemagglutininCastro, Sonia de; Vanderlinden, E.; Ginex, Tiziana CSIC ORCID ; Laporte, M.; Stevaert, L.; Naesens, L.; Luque, F. Javier; Camarasa Rius, María José CSIC ORCID; Velázquez, Sonsoles CSIC ORCID CVNcomunicación de congreso
openAccessJMC2020.pdf.jpg24-Jul-2020Centrally Active Multitarget Anti-Alzheimer Agents Derived from the Antioxidant Lead CR-6Pérez-Areales, F. Javier; Garrido, María; Aso, Ester; Bartolini, Manuela; De Simone, Angela; Espargaró, Alba; Ginex, Tiziana CSIC ORCID ; Sabate, Raimon; Pérez, Belén; Andrisano, Vincenza; Puigoriol-Illamola, Dolors; Pallàs, Mercè; Luque, F. Javier; Loza, María Isabel; Brea, José; Ferrer, Isidro; Ciruela, Francisco; Messeguer Peypoch, Ángel CSIC ORCID; Muñoz-Torrero, Diegoartículo
openAccessacs.jmedchem-Gil, C._2020.pdf.jpg8-Jun-2020COVID-19: Drug targets and potential treatmentsGil, Carmen CSIC ORCID ; Ginex, Tiziana CSIC ORCID ; Maestro, Inés; Nozal, Vanesa; Barrado-Gil, Lucía; Cuesta-Geijo, Miguel Ángel; Urquiza, Jesús; Ramírez, David; Alonso, Covadonga; Campillo, Nuria E. CSIC ORCID ; Martínez, Ana CSIC ORCID artículo
openAccesspharmaceuticals-14-00332-v3.pdf.jpg6-Apr-2021Host-Directed FDA-Approved Drugs with Antiviral Activity against SARS-CoV-2 Identified by Hierarchical In Silico/In Vitro Screening MethodsGinex, Tiziana CSIC ORCID ; Garaigorta, Urtzi ; Ramírez, David; Castro, Victoria; Nozal, Vanesa; Maestro, Inés; Garcia-Carceles, Javier; Campillo, Nuria E. CSIC ORCID ; Martínez, Ana CSIC ORCID ; Gastaminza, Pablo; Gil, Carmen CSIC ORCID artículo
openAccessHost-directed_Ginex.pdf.jpg26-Nov-2020Host-directed FDA-approved drugs with antiviral activity against SARS-CoV-2 identified by hierarchical in silico/in vitro screening methodsGinex, Tiziana CSIC ORCID ; Garaigorta, Urtzi ; Ramírez, David; Castro, Victoria; Nozal, Vanesa; Maestro, Inés; Garcia-Carceles, Javier; Campillo, Nuria E. CSIC ORCID ; Martínez, Ana CSIC ORCID ; Gastaminza, Pablo; Gil, Carmen CSIC ORCID preprint
openAccessSVelazquez_manuscript-ACSID 2020_compressed.pdf.jpg2020N-benzyl 4,4-disubstituted piperidines as a potent class of influenza H1N1 virus inhibitors showing a novel mechanism of hemagglutinin fusion peptide interactionCastro, Sonia de; Ginex, Tiziana CSIC ORCID ; Vanderlinden, E.; Laporte, M.; Stevaert, A.; Cumella, José; Gago, Federico CSIC ORCID; Camarasa Rius, María José CSIC ORCID; Luque, F. Javier; Naesens, L.; Velázquez, Sonsoles CSIC ORCID CVNartículo
openAccessAbstract_YRS_A. Martínez_2021.pdf.jpg18-Jun-2021P25 Ligand and structure-based virtual screening toward identifying new potent inhibitors against SGK 1Madruga, Enrique; Maestro, Inés; Ginex, Tiziana CSIC ORCID ; Martínez, Ana CSIC ORCID comunicación de congreso
closedAccessaccesoRestringido.pdf.jpg2020Pharmacology and preclinical validation of a novel anticancer compound targeting PEPCK-MAragó, M.; Moreno-Felici, J.; Abás, S.; Rodríguez-Arévalo, S.; Hyroššová, P.; Figueras, A.; Viñals, F.; Pérez, B.; Loza, María Isabel; Brea, J.; Latorre, P.; Carrodeguas, José A. CSIC ORCID; García-Rovés, Pablo M.; Galdeano, Carles; Ginex, Tiziana CSIC ORCID ; Luque, F. Javier; Escolano, Carmen; Perales, J.Cartículo
openAccessJ Med Chemistry_Morales-Tenorio_2021.pdf.jpg5-Nov-2021Potential pharmacological strategies targeting the Niemann-Pick C1receptor and Ebola virus glycoprotein interactionMorales-Tenorio, Marcos; Ginex, Tiziana CSIC ORCID ; Cuesta-Geijo, Miguel Ángel; Campillo, Nuria E. CSIC ORCID ; Muñoz-Fontela, César; Alonso, Covadonga; Delgado, Rafael; Gil, Carmen CSIC ORCID artículo
openAccesseotp_ginex_2020.pdf.jpg5-Oct-2020Searching for effective antiviral small molecules against influenza A virus: A patent reviewGinex, Tiziana CSIC ORCID ; Luque, F. Javierartículo
openAccessproceedings-22-00071.pdf.jpg14-Aug-2019Synthesis, in vitro profiling, and in vivo efficacy studies of a new family of multitarget anti-alzheimer compoundsPérez-Areales, Francisco Javier; Garrido, María; Aso, Ester; Bartolini, Manuela; Simone, Angela; Espargaró, Alba; Ginex, Tiziana CSIC ORCID ; Sabate, Raimon; Pérez, Belén; Andrisano, Vincenza; Luque, F. Javier; Ferrer, Isidro; Ciruela, Francisco; Messeguer Peypoch, Ángel CSIC ORCID; Muñoz-Torrero, Diegoartículo
openAccessrolemuta.pdf.jpg2022The role of SARS-CoV-2 genetic background in the emergence and success of spike mutations: the case of the spike A222V mutationGinex, Tiziana CSIC ORCID ; Marco-Marín, Clara CSIC ORCID; Wieczor, Milosz; Mata, Carlos P.; Krieger, James; Ruiz-Rodríguez, Paula CSIC ORCID ; López-Redondo, Marisa CSIC; Francés-Gómez, Clara CSIC; Melero, Roberto CSIC ORCID; Sorzano, Carlos Óscar S.; Martínez, Marta; Gougeard, Nadine CSIC; Forcada-Nadal, Alicia CSIC ORCID; Zamora-Caballero, Sara; Gozalbo-Rovira, Roberto CSIC ORCID ; Sanz-Frasquet, Carla; Arranz, Rocío; Bravo, Jerónimo CSIC ORCID ; Rubio, Vicente CSIC ORCID ; Marina, Alberto CSIC ORCID; The IBV-Covid19-Pipeline; Geller, Ron CSIC ORCID ; Comas, Iñaki CSIC ORCID ; Gil, Carmen CSIC ORCID ; Coscollá, Mireia CSIC ORCID; Orozco, Modesto; Llácer, José Luis CSIC ORCID ; Carazo, José M.comunicación de congreso
closedAccessaccesoRestringido.pdf.jpg8-Dec-2021The structural role of SARS-CoV-2 genetic background in the emergence and success of spike mutations: the case of the spike A222V mutationGinex, Tiziana CSIC ORCID ; Marco-Marín, Clara CSIC ORCID; Wieczor, Milosz; Mata, Carlos P.; Krieger, James; López-Redondo, Marisa CSIC; Francés-Gómez, Clara CSIC; Ruiz-Rodríguez, Paula CSIC ORCID ; Melero, Roberto CSIC ORCID; Sorzano, Carlos Óscar S.; Martínez, Marta; Gougeard, Nadine CSIC; Forcada-Nadal, Alicia CSIC ORCID; Zamora-Caballero, Sara; Gozalbo-Rovira, Roberto CSIC ORCID ; Sanz-Frasquet, Carla; Bravo, Jerónimo CSIC ORCID ; Rubio, Vicente CSIC ORCID ; Marina, Alberto CSIC ORCID ; Geller, Ron CSIC ORCID ; Comas, Iñaki CSIC ORCID ; Gil, Carmen CSIC ORCID ; Coscollá, Mireia CSIC ORCID; Orozco, Modesto; Llácer, José Luis CSIC ORCID ; Carazo, José M.preprint
openAccessppat_Ginex_2022.pdf.jpg11-Jul-2022The structural role of SARS-CoV-2 genetic background in the emergence and success of spike mutations: The case of the spike A222V mutationGinex, Tiziana CSIC ORCID ; Marco-Marín, Clara CSIC ORCID; Wieczor, Milosz; Mata, Carlos P.; Krieger, James; Ruiz-Rodríguez, Paula CSIC ORCID ; López-Redondo, Marisa CSIC; Francés-Gómez, Clara CSIC; Melero, Roberto CSIC ORCID; Sorzano, Carlos Óscar S.; Martínez, Marta; Gougeard, Nadine CSIC; Forcada-Nadal, Alicia CSIC ORCID; Zamora-Caballero, Sara; Gozalbo-Rovira, Roberto CSIC ORCID ; Sanz-Frasquet, Carla; Arranz, Rocío; Bravo, Jerónimo CSIC ORCID ; Rubio, Vicente CSIC ORCID ; Marina, Alberto CSIC ORCID ; The IBV-Covid19-Pipeline; Geller, Ron CSIC ORCID ; Comas, Iñaki CSIC ORCID ; Gil, Carmen CSIC ORCID ; Coscollá, Mireia CSIC ORCID; Orozco, Modesto; Llácer, José Luis CSIC ORCID ; Carazo, José M.artículo