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Derechos | Preview | Fecha Public. | Título | Autor(es) | Tipo |
closedAccess | | 2010 | 9-Arylpurines as a Novel Class of Enterovirus Inhibitors | Aguado, Leire CSIC; Thibaut, Hendrik Jan; Priego, Eva María CSIC ORCID; Jimeno, M. Luisa CSIC ORCID; Camarasa Rius, María José CSIC ORCID; Neyts, Johan; Peréz-Pérez, María-Jesús CSIC ORCID | artículo |
closedAccess | | 2002 | A new and efficient one-pot synthesis of pyrido[2,1-f]purine-2,4-diones starting from 6-aminouracil derivatives | Peréz-Pérez, María-Jesús CSIC ORCID ; Priego, Eva María CSIC ORCID; Jimeno, M. Luisa CSIC ORCID; Camarasa Rius, María José CSIC ORCID | artículo |
openAccess | | 2022 | Allosteric Inhibition of Neutral Sphingomyelinase 2 (nSMase2) by DPTIP: From Antiflaviviral Activity to Deciphering Its Binding Site through In Silico Studies and Experimental Validation | Álvarez-Fernández, Hadrián CSIC; Mingo-Casas, Patricia; Blázquez, Ana B.; Caridi, Flavia CSIC ORCID; Saiz Calahorra, Juan Carlos; Peréz-Pérez, María-Jesús CSIC ORCID ; Martín-Acebes, M. A.; Priego, Eva María CSIC ORCID | artículo |
openAccess | | 20-may-2016 | Antivascular and antitumor properties of the tubulin-binding chalcone TUB091 | Canela, María-Dolores CSIC; Noppen, Sam; Bueno, Oskia CSIC; Prota, Andrea E.; Bargsten, Katja; Sáez-Calvo, Gonzalo CSIC; Jimeno, M. Luisa CSIC ORCID; Benkhei, Mohammed; Ribatti, Domenico; Velázquez, Sonsoles CSIC ORCID CVN; Camarasa Rius, María José CSIC ORCID; Díaz, José Fernando CSIC ORCID ; Steinmetz, Michel O.; Priego, Eva María CSIC ORCID; Peréz-Pérez, María-Jesús CSIC ORCID ; Liekens, Sandra | artículo |
closedAccess | | 2017 | Antiviral activity of [1,2,3]triazolo[4,5-d]pyrimidin-7(6H)-ones against chikungunya virus targeting the viral capping nsP1 | Gigante, Alba CSIC ORCID; Gómez-SanJuan, Asier CSIC; Delang, Leen; Li, C.; Bueno, Oskia CSIC; Gamo, Ana María CSIC; Priego, Eva María CSIC ORCID; Camarasa Rius, María José CSIC ORCID; Jochmans, D.; Leyssen, Pieter; Decroly, E.; Coutard, Bruno; Querat, Guilles; Neyts, Johan; Peréz-Pérez, María-Jesús CSIC ORCID | artículo |
openAccess | | 8-dic-2021 | Antivirals against (Re)emerging Flaviviruses: Should We Target the Virus or the Host? | Peréz-Pérez, María-Jesús CSIC ORCID ; Saiz Calahorra, Juan Carlos; Priego, Eva María CSIC ORCID; Martín-Acebes, M. A. | artículo |
openAccess | | 27-jun-2016 | Blocking Blood Flow to Solid Tumors by Destabilizing Tubulin : An Approach to Targeting Tumor Growth (Perspective) | Peréz-Pérez, María-Jesús CSIC ORCID ; Priego, Eva María CSIC ORCID; Bueno, Oskia CSIC; Martins, Maria Solange; Canela, María-Dolores CSIC; Liekens, Sandra | artículo |
closedAccess | | 2019 | Chalcones and Chalcone-mimetic Derivatives as Notch Inhibitors in a Model of T-cell Acute Lymphoblastic Leukemia | Quaglio, D.; Zhdanovskaya, N.; Tobajas, Gloria; Cuartas, V.; Balducci, S.; Christodoulou, M. S.; Fabrizi, G.; Gargantilla, Marta CSIC ORCID; Priego, Eva María CSIC ORCID; Carmona Pestania, Á.; Passarella, D.; Screpanti, I.; Botta, B.; Palermo, R.; Mori, M.; Ghirga, F.; Peréz-Pérez, María-Jesús CSIC ORCID | artículo |
openAccess | | 14-jun-2019 | Chikungunya virus drug discovery: still a long way to go? | Peréz-Pérez, María-Jesús CSIC ORCID ; Delang, Leen; Ng, Lisa; Priego, Eva María CSIC ORCID | artículo |
openAccess | | 2018 | Conformational mimetics of the α-methyl chalcone TUB091 binding tubulin: Design, synthesis and antiproliferative activity | Bueno, Oskia CSIC; Tobajas, Gloria; Quesada, Ernesto CSIC ORCID ; Estévez-Gallego, Juan CSIC ORCID ; Noppen, Sam; Camarasa Rius, María José CSIC ORCID; Díaz, José Fernando CSIC ORCID ; Liekens, Sandra; Priego, Eva María CSIC ORCID; Peréz-Pérez, María-Jesús CSIC ORCID | artículo |
closedAccess | | 2012 | CRDOCK: An ultrafast multipurpose protein-ligand docking tool | Cortés Cabrera, Álvaro CSIC ORCID; Klett, Javier CSIC ORCID; Dos Santos, Helena G.; Perona, Almudena CSIC ORCID CVN; Gil Redondo, Rubén; Francis, Sandrea M. CSIC; Priego, Eva María CSIC ORCID; Gago, Federico CSIC ORCID; Morreale, Antonio | artículo |
openAccess | | 2019 | Design and Synthesis of New 6-Nitro and 6-Amino- 3,3a,4,5-Tetrahydro-2H-Benzo[g]indazole Derivatives: Antiproliferative and Antibacterial Activity | Cuartas, Viviana; Crespo, María del Pilar; Priego, Eva María CSIC ORCID; Persoons, Leentje; Daelemans, Dirk; Camarasa Rius, María José CSIC ORCID; Insuasty, Braulio; Peréz-Pérez, María-Jesús CSIC ORCID | artículo |
openAccess | | 2019 | Design and synthesis of new 6-nitro and 6-Amino-3,3a,4,5-Tetrahydro-2H-Benzo[g]indazole derivatives: Antiproliferative and antibacterial activity | Cuartas, V.; Crespo, M. D. P.; Priego, Eva María CSIC ORCID; Persoons, L.; Daelemans, D.; Camarasa Rius, María José CSIC ORCID; Insuasty, Braulio; Peréz-Pérez, María-Jesús CSIC ORCID | artículo |
closedAccess | | jun-2019 | Diphenyl ether derivatives occupy the expanded binding site of cyclohexanedione compounds at the colchicine site in tubulin by movement of the aT5 loop | Bueno, Oskia CSIC; Gargantilla, Marta CSIC ORCID; Estévez-Gallego, Juan CSIC ORCID ; Martins, Solange; Díaz, José Fernando CSIC ORCID ; Camarasa Rius, María José CSIC ORCID; Liekens, Sandra; Peréz-Pérez, María-Jesús CSIC ORCID ; Priego, Eva María CSIC ORCID | artículo |
closedAccess | | 2012 | Efficient synthesis and anti-enteroviral activity of 9-arylpurines | Aguado, Leire CSIC; Canela, María-Dolores CSIC; Thibaut, Hendrik Jan; Priego, Eva María CSIC ORCID; Camarasa Rius, María José CSIC ORCID; Leyssen, Pieter; Neyts, Johan; Peréz-Pérez, María-Jesús CSIC ORCID | artículo |
openAccess | | 2018 | High-affinity ligands of the colchicine domain in tubulin based on a structure-guided design | Bueno, Oskia CSIC; Estévez-Gallego, Juan CSIC ORCID ; Martins, S.; Prota, Andrea E.; Gago, Federico CSIC ORCID; Gómez-SanJuan, Asier CSIC; Camarasa Rius, María José CSIC ORCID; Barasoain, Isabel CSIC ; Steinmetz, Michel O.; Díaz, José Fernando CSIC ORCID ; Peréz-Pérez, María-Jesús CSIC ORCID ; Liekens, Sandra; Priego, Eva María CSIC ORCID | artículo |
openAccess | | 2022 | Hybridization Approach to Identify Salicylanilides as Inhibitors of Tubulin Polymerization and Signal Transducers and Activators of Transcription 3 (STAT3) | Gargantilla, Marta CSIC ORCID; Persoons, Leentje; Kauerová, Tereza; Río, Natalia del CSIC ORCID; Daelemans, Dirk; Priego, Eva María CSIC ORCID; Kollar, Peter; Peréz-Pérez, María-Jesús CSIC ORCID | artículo |
closedAccess | | 2014 | Identification of [1,2,3]triazolo[4,5-d ]pyrimidin-7(6H)-ones as novel inhibitors of chikungunya virus replication | Gigante, Alba CSIC ORCID; Canela, María-Dolores CSIC; Delang, Leen; Priego, Eva María CSIC ORCID; Camarasa Rius, María José CSIC ORCID; Querat, Guilles; Neyts, Johan; Leyssen, Pieter; Peréz-Pérez, María-Jesús CSIC ORCID | artículo |
openAccess | | 2018 | Identification of a novel 2-oxindole fluorinated derivative as in vivo antitumor agent for prostate cancer acting via AMPK activation | Bort Bueno, Alicia; Quesada Sánchez, Sergio CSIC; Ramos-Torres, Ágata; Gargantilla, Marta CSIC ORCID; Priego, Eva María CSIC ORCID; Raynal, S.; Lepifre, F.; Gasalla, José María; Rodriguez-Henche, Nieves; Castro, Ana CSIC ORCID; Díaz-Laviada, Inés | artículo |
openAccess | | 2018 | Inhibition of the Replication of Different Strains of Chikungunya Virus by 3-Aryl-[1,2,3]triazolo[4,5- d] pyrimidin-7(6 H)-ones | Gómez-SanJuan, Asier CSIC; Gamo, Ana María CSIC; Delang, Leen; Pérez-Sánchez, Alfonso; Amrun, S. N.; Abdelnabi, Rana; Jacobs, S.; Priego, Eva María CSIC ORCID; Camarasa Rius, María José CSIC ORCID; Jochmans, D.; Leyssen, Pieter; Ng, L. F. P.; Querat, Guilles; Neyts, Johan; Peréz-Pérez, María-Jesús CSIC ORCID | artículo |