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Rights | Preview | Issue Date | Title | Author(s) | Type |
openAccess |  | 14-Mar-2018 | 1-(Benzo[d]thiazol-2-yl)-3-phenylureas as dual inhibitors of casein kinase 1 and ABAD enzymes for treatment of neurodegenerative disorders | Benek, O.; Pérez, Daniel I.; Pérez, Concepción; Martínez, Ana ; Musilek, Kamil | artículo |
openAccess |  | 14-Jul-2015 | 3,4-Dihydro-1,3,5-triazin-2(1H)-ones as the first dual BACE-1/GSK-3β fragment hits against Alzheimer’s disease | Prati, Federica; Pérez, Daniel I.; Pérez Castillo, Ana ; Martínez, Ana ; Bolognesi, Maria Laura | artículo |
closedAccess |  | 2012 | 5-imino-1,2,4-thiadiazoles: first small molecules as substrate competitive inhibitors of glycogen synthase kinase 3 | Palomo, Valle ; Pérez, Daniel I.; Pérez, Concepción; Morales-García, José A. ; Soteras, Ignacio ; Alonso-Gil, Sandra ; Encinas, Arantxa; Castro, Ana ; Campillo, Nuria E. ; Pérez Castillo, Ana ; Gil, Carmen ; Martínez, Ana | artículo |
closedAccess |  | 2013 | A fluorescent styrylquinoline with combined therapeutic and diagnostic activities against Alzheimer's and prion diseases | Staderini, Matteo; Aulic, Suzana; Bartolini, Manuela; Tran, H. N. A.; González-Ruiz, Victor; Pérez, Daniel I.; Cabezas, Nieves; Martínez, Ana ; Martín, M. Antonia; Andrisano, Vincenza; Legname, Giuseppe; Menéndez, J. Carlos; Bolognesi, Maria Laura | artículo |
openAccess |  | Mar-2016 | Application of BACE1 immobilized enzyme reactor for the characterization of multifunctional alkaloids from Corydalis cava (Fumariaceae) as Alzheimer's disease targets | Chlebek, Jakub; De Simone, Angela; Hošťálková, Anna; Opletal, Lubomír; Pérez, Concepción; Pérez, Daniel I.; Havlíková, Lucie; Cahlíková, Lucie; Andrisano, Vincenza | artículo |
openAccess |  | 30-Aug-2017 | Biological and pharmacological characterization of benzothiazole-based CK-1δ inhibitors in models of Parkinson’s disease | Morales-García, José A. ; Salado, Irene G. ; Sanz-SanCristóbal, Marina ; Gil, Carmen ; Pérez Castillo, Ana ; Martínez, Ana ; Pérez, Daniel I. | artículo |
openAccess |  | 27-Sep-2018 | CDC-7-inhibitors compounds and use thereof for the treatment of neurological conditions | Martinez Gil, Ana ; Pérez, Daniel I.; Gil, Carmen ; Martín-Requero, Ángeles ; Rojas-Prats, Elisa; Martínez-González, Loreto ; Pérez, Concepción | solicitud de patente |
closedAccess |  | 2018 | Chameleon-like behavior of indolylpiperidines in complex with cholinesterases targets: Potent butyrylcholinesterase inhibitors | Chierrito, Talita P. C.; Pedersoli-Mantoani, S.; Roca, Carlos; Sebastián-Pérez, Víctor; Martínez-González, Loreto ; Pérez, Daniel I.; Pérez, Concepción; Canales, A.; Cañada, F. Javier ; Campillo, Nuria E. ; Carvalho, Ivone; Martínez, Ana | artículo |
openAccess |  | 22-Oct-2018 | Compuestos inhibidores de CDC-7 y su uso para el tratamiento de patologías neurológicas | Martinez Gil, Ana ; Pérez, Daniel I.; Gil, Carmen ; Martín-Requero, Ángeles ; Rojas-Prats, Elisa; Martínez-González, Loreto ; Pérez, Concepción | solicitud de patente |
openAccess |  | 29-Nov-2012 | Derivados heterocíclicos inhibidores de fosfodiesterasa 7 | Gil, Carmen ; Martínez, Ana ; Redondo, Miriam ; Campillo, Nuria E. ; Pérez, Daniel I.; Loza, María Isabel; Cadavid, María Isabel; Brea, José; Pérez Castillo, Ana  | solicitud de patente |
openAccess |  | Apr-2017 | Drugs on clinical development for the treatment of amyotrophic lateral sclerosis | Martínez, Ana ; Palomo, Valle ; Pérez, Daniel I.; Gil, Carmen | artículo |
openAccess |  | 2012 | Effect of phosphodiesterase 7 (PDE7) inhibitors in experimental autoimmune encephalomyelitis mice. Discovery of a new chemically diverse family of compounds | Redondo, Miriam ; Brea, José; Pérez, Daniel I.; Soteras, Ignacio ; Val, Cristina; Pérez, Concepción; Morales-García, José A. ; Alonso-Gil, Sandra ; Paul-Fernández, Nuria ; Martín-Álvarez, Rocío ; Cadavid, María Isabel; Loza, María Isabel; Pérez Castillo, Ana ; Mengod Los Arcos, Guadalupe ; Campillo, Nuria E. ; Martínez, Ana ; Gil, Carmen | artículo |
openAccess | | 2015 | From bitopic inhibitors to multitarget drugs for Alzheimer’s disease future treatment | Pérez, Daniel I.; Martínez, Ana ; Gil, Carmen ; Campillo, Nuria E. | artículo |
closedAccess |  | 2013 | Glycogen synthase kinase-3 inhibitors as potent therapeutic agents for the treatment of Parkinson disease | Morales-García, José A. ; Susín, Cristina ; Alonso-Gil, Sandra ; Pérez, Daniel I.; Palomo, Valle ; Pérez, Concepción; Conde, Santiago ; Santos, Ángel; Gil, Carmen ; Martínez, Ana ; Pérez Castillo, Ana  | artículo |
openAccess |  | 5-Apr-2019 | In Vitro and In Silico Acetylcholinesterase Inhibitory Activity of Thalictricavine and Canadine and Their Predicted Penetration across the Blood-Brain Barrier | Chlebek, Jakub; Korábečný, Jan; Doležal, Rafael; Štěpánková, Šárka; Pérez, Daniel I.; Hošťálková, Anna; Opletal, Lubomír; Cahlíková, Lucie; Macáková, Kateřina; Kučera, Tomáš; Hrabinová, Martina; Jun, Daniel | artículo |
openAccess |  | 29-Sep-2017 | Leucine rich repeat kinase 2 (LRRK2) inhibitors based on indolinone scaffold: Potential pro-neurogenic agents | Salado, Irene G. ; Zaldívar-Díez, Josefa; Sebastián-Pérez, Víctor; Li, Lingling; Geiger, Larissa; González, Silvia; Campillo, Nuria E. ; Gil, Carmen ; Morales, Aixa V. ; Pérez, Daniel I.; Martínez, Ana | artículo |
closedAccess |  | 2012 | Microwave-assisted synthesis of hydroxyphenyl nitrones with protective action against oxidative stress | Chavarría, Cecilia; Pérez, Daniel I.; Pérez, Concepción; Morales-García, José A. ; Alonso-Gil, Sandra ; Pérez Castillo, Ana ; Gil, Carmen ; Souza, José M.; Porcal, Williams | artículo |
closedAccess |  | 2014 | Modulation of cAMP-specific PDE without emetogenic activity: New sulfide-like PDE7 inhibitors | García, Ana M. ; Brea, José; Morales-García, José A. ; Pérez, Daniel I.; González, A. ; Alonso-Gil, Sandra ; Conde, Santiago ; Cadavid, María Isabel; Loza, María Isabel; Pérez Castillo, Ana ; Martínez, Ana ; Gil, Carmen | artículo |
closedAccess |  | 2015 | Multitarget drug discovery for Alzheimer's disease: Triazinones as BACE-1 and GSK-3ß inhibitors | Pérez, Daniel I.; Pérez Castillo, Ana ; Martínez, Ana ; Bolognesi, Maria Laura; Cavalli, Andrea | artículo |
closedAccess |  | 2015 | Neuroprotection of CK-1 inhibitors against TDP-43 and LPS toxicity | Martínez, Ana ; Pérez, Daniel I.; Salado, Irene G. ; Gil, Carmen ; Morales-García, José A. ; Pérez Castillo, Ana  | comunicación de congreso |