Derechos | Preview | Fecha Public. | Título | Autor(es) | Tipo |
closedAccess | | 30-abr-2002 | 2-Oxopiperazine-based γ-turn conformationally constrained peptides: Synthesis of CCK-4 analogues | Herrero, Susana; García-López, M. Teresa CSIC ; Latorre, Julio; Cenarruzabeitia, Edurne CSIC; Río, Joaquín del CSIC; Herranz, Rosario CSIC ORCID | artículo |
closedAccess | | 15-may-1998 | 2-Oxopyrrolidines and 6-oxoperhydropyrrolo[1,2-a]pyrazines as templates in the search for nonpeptide cholecystokinin ligands | Martín-Martínez, Mercedes CSIC ORCID; Ballaz García, Santiago; Latorre, Miriam; Herranz, Rosario CSIC ORCID; García-López, M. Teresa CSIC ; Cenarruzabeitia, Edurne CSIC; Río, Joaquín del CSIC; González-Muñiz, Rosario CSIC ORCID | artículo |
closedAccess | | 7-oct-1999 | 5-(Tryptophyl)amino-1,3-dioxoperhydropyrido[1,2-c]pyrimidine-based potent and selective CCK1 receptor antagonists: Structural modifications at the tryptophan domain | Bartolomé-Nebreda, José M.; Gómez-Monterrey, Isabel CSIC; García-López, M. Teresa CSIC ; González-Muñiz, Rosario CSIC ORCID; Martín-Martínez, Mercedes CSIC ORCID; Ballaz García, Santiago; Cenarruzabeitia, Edurne CSIC; Latorre, Miriam; Río, Joaquín del CSIC; Herranz, Rosario CSIC ORCID | artículo |
closedAccess | | 18-oct-2001 | 5-(Tryptophyl)amino-1,3-dioxoperhydropyrido[1,2-c]pyrimidine-based potent and selective CCK1 receptor antagonists: Structure-activity relationship studies on the central 1,3-dioxoperhydropyrido[1,2-c]pyrimidine scaffold | Bartolomé-Nebreda, José M.; García-López, M. Teresa CSIC ; González-Muñiz, Rosario CSIC ORCID; Cenarruzabeitia, Edurne CSIC; Latorre, Miriam; Río, Joaquín del CSIC; Herranz, Rosario CSIC ORCID | artículo |
closedAccess | | 25-may-2001 | 5-(Tryptophyl)amino-1,3-dioxoperhydropyrido[1,2-c]pyrimidine-based potent and selective CCK1 receptor antagonists: Structure-activity relationship studies on the substituent at N2-position | Bartolomé-Nebreda, José M.; Patiño-Molina, Rosario; Martín-Martínez, Mercedes CSIC ORCID; Gómez-Monterrey, Isabel CSIC; García-López, M. Teresa CSIC ; González-Muñiz, Rosario CSIC ORCID; Cenarruzabeitia, Edurne CSIC; Latorre, Miriam; Río, Joaquín del CSIC; Herranz, Rosario CSIC ORCID | artículo |
closedAccess | | 4-sep-2004 | 5-(tryptophylamino)-1,3-dioxoperhydropyrido[1,2-c]pyrimidine-based cholecystokinin receptor antagonists: Reversal of CCK1 receptor subtype selectivity toward CCK2 receptors | Muñoz, Pilar; García-López, M. Teresa CSIC ; Cenarruzabeitia, Edurne CSIC; Río, Joaquín del CSIC; Dufresne, Marlene; Foucaud, Magali; Fourmy, Daniel; Herranz, Rosario CSIC ORCID | artículo |
closedAccess | | 3-mar-2005 | Analogues of the neuroprotective tripeptide Gly-Pro-Glu (GPE): synthesis and structure–activity relationships | Alonso De Diego, Sergio A. CSIC; Muñoz, Pilar; González-Muñiz, Rosario CSIC ORCID; Cenarruzabeitia, Edurne CSIC; Frechilla, Diana; Río, Joaquín del CSIC; Jimeno, M. Luisa CSIC ORCID; García-López, M. Teresa CSIC | artículo |
closedAccess | | 2-nov-2005 | Conformationally constrained CCK4 analogues incorporating IBTM and BTD β-turn mimetics | Martín-Martínez, Mercedes CSIC ORCID; Figuera, Natalia De la CSIC; Latorre, Miriam; García-López, M. Teresa CSIC ; Cenarruzabeitia, Edurne CSIC; Río, Joaquín del CSIC; González-Muñiz, Rosario CSIC ORCID | artículo |
closedAccess | | 21-ene-2002 | Effects of the incorporation of IBTM β-turn mimetics into the dipeptoid CCK1 receptor agonist PD 170292 | Martín-Martínez, Mercedes CSIC ORCID; Latorre, Miriam; García-López, M. Teresa CSIC ; Cenarruzabeitia, Edurne CSIC; Río, Joaquín del CSIC; González-Muñiz, Rosario CSIC ORCID | artículo |
closedAccess | | 4-ene-1999 | Highly constrained dipeptoid analogues containing a type II' β-turn mimic as novel and selective CCK-A receptor ligands | Figuera, Natalia De la CSIC; Martín-Martínez, Mercedes CSIC ORCID; Herranz, Rosario CSIC ORCID; García-López, M. Teresa CSIC ; Latorre, Miriam; Cenarruzabeitia, Edurne CSIC; Río, Joaquín del CSIC; González-Muñiz, Rosario CSIC ORCID | artículo |
closedAccess | | 2006 | New Gly-Pro-Glu (GPE) analogues: Expedite solid-phase synthesis and biological activity | Alonso De Diego, Sergio A. CSIC; Gutiérrez-Rodríguez, Marta CSIC ORCID ; Pérez de Vega, M. Jesús CSIC ORCID; Casabona, Diego; Cativiela, Carlos CSIC ORCID; González-Muñiz, Rosario CSIC ORCID; Herranz, Rosario CSIC ORCID; Cenarruzabeitia, Edurne CSIC; Frechilla, Diana; Río, Joaquín del CSIC; Jimeno, M. Luisa CSIC ORCID; García-López, M. Teresa CSIC | artículo |
closedAccess | | oct-2004 | Pharmacological study of IQM-97,423, a potent and selective CCK1 receptor antagonist with protective effect in experimental acute pancreatitis | Latorre, Miriam; Bartolomé-Nebreda, José M.; García-López, M. Teresa CSIC ; González-Muñiz, Rosario CSIC ORCID; Herranz, Rosario CSIC ORCID; Río, Joaquín del CSIC; Cenarruzabeitia, Edurne CSIC | artículo |
closedAccess | | 2007 | Simple approach to highly functionalized trisubstituted tetrahydropyrimidine-2,4-diones from perhydropyrazino[1,2-f]pyrimidine-3,6,8- trione precursors | Patiño-Molina, Rosario; García-López, M. Teresa CSIC ; Cenarruzabeitia, Edurne CSIC; Río, Joaquín del CSIC; González-Muñiz, Rosario CSIC ORCID | artículo |
closedAccess | | 2005 | Studies on structure-activity relationships of the neuroprotective tripeptide H-Gly-Pro-Glu-OH (GPE) | Alonso De Diego, Sergio A. CSIC; Gutiérrez-Rodríguez, Marta CSIC ORCID ; González-Muñiz, Rosario CSIC ORCID; Herranz, Rosario CSIC ORCID; Jimeno, M. Luisa CSIC ORCID; Cenarruzabeitia, Edurne CSIC; Frechilla, Diana; Río, Joaquín del CSIC; García-López, M. Teresa CSIC | capítulo de libro |
closedAccess | | 1-jul-2006 | The neuroprotective activity of GPE tripeptide analogues does not correlate with glutamate receptor binding affinity | Alonso De Diego, Sergio A. CSIC; Gutiérrez-Rodríguez, Marta CSIC ORCID ; Pérez de Vega, M. Jesús CSIC ORCID; González-Muñiz, Rosario CSIC ORCID; Herranz, Rosario CSIC ORCID; Martín-Martínez, Mercedes CSIC ORCID; Cenarruzabeitia, Edurne CSIC; Frechilla, Diana; Río, Joaquín del CSIC; Jimeno, M. Luisa CSIC ORCID; García-López, M. Teresa CSIC | artículo |
closedAccess | | 16-jun-2003 | Versatile synthesis of chiral 2-substituted-5-oxo-1,2,3,4-tetrahydro-5H-1,4-benzodiazepines as novel scaffolds for peptidomimetic building | Herrero, Susana; García-López, M. Teresa CSIC ; Cenarruzabeitia, Edurne CSIC; Río, Joaquín del CSIC; Herranz, Rosario CSIC ORCID | artículo |
closedAccess | | 9-sep-2000 | β-Turned dipeptoids as potent and selective CCK1 receptor antagonists | Martín-Martínez, Mercedes CSIC ORCID; Figuera, Natalia De la CSIC; Latorre, Miriam; Herranz, Rosario CSIC ORCID; García-López, M. Teresa CSIC ; Cenarruzabeitia, Edurne CSIC; Río, Joaquín del CSIC; González-Muñiz, Rosario CSIC ORCID | artículo |