Rights | Preview | Issue Date | Title | Author(s) | Type |
closedAccess |  | 2015 | 2-Phenoxy-1,4-naphthoquinones: From a Multitarget Antitrypanosomal to a Potential Antitumor Profile | Prati, F.; Bergamini, C.; Molina, María Teresa ; Falchi, F.; Cavalli, A.; Kaiser, M.; Brun, R.; Fato, R.; Bolognesi, Maria Laura | artículo |
openAccess |  | 14-Jul-2015 | 3,4-Dihydro-1,3,5-triazin-2(1H)-ones as the first dual BACE-1/GSK-3β fragment hits against Alzheimer’s disease | Prati, Federica; Pérez, Daniel I.; Pérez Castillo, Ana ; Martínez, Ana ; Bolognesi, Maria Laura | artículo |
closedAccess |  | 2013 | A fluorescent styrylquinoline with combined therapeutic and diagnostic activities against Alzheimer's and prion diseases | Staderini, Matteo; Aulic, Suzana; Bartolini, Manuela; Tran, H. N. A.; González-Ruiz, Victor; Pérez, Daniel I.; Cabezas, Nieves; Martínez, Ana ; Martín, M. Antonia; Andrisano, Vincenza; Legname, Giuseppe; Menéndez, J. Carlos; Bolognesi, Maria Laura | artículo |
openAccess |  | 9-Oct-2018 | A focused library of psychotropic analogs with neuroprotective and neuroregenerative potential | Uliassi, Elisa; Peña-Altamira, Luis Emiliano; Morales, Aixa V. ; Massenzio, Francesca; Petralla, Sabrina; Rossi, Michele; Roberti, Marinella; Martínez-González, Loreto ; Martínez, Ana ; Monti, B.; Bolognesi, Maria Laura | artículo |
closedAccess |  | 2012 | A small chemical library of 2-aminoimidazole derivatives as BACE-1 inhibitors: Structure-based design, synthesis, and biological evaluation | Chiriano, G.; De Simone, A.; Mancini, F.; Perez, D.I.; Cavalli, A.; Bolognesi, Maria Laura; Legname, G.; Martinez, A. ; Andrisano, Vincenza; Carloni, P.; Roberti, M. | artículo |
closedAccess |  | 2015 | Multitarget drug discovery for Alzheimer's disease: Triazinones as BACE-1 and GSK-3ß inhibitors | Pérez, Daniel I.; Pérez Castillo, Ana ; Martínez, Ana ; Bolognesi, Maria Laura; Cavalli, Andrea | artículo |
closedAccess |  | Jun-2014 | Multitarget ligands and theranostics: Sharpening the medicinal chemistry sword against prion diseases | Bongarzone, Salvatore; Staderini, Matteo; Bolognesi, Maria Laura | artículo |
openAccess |  | 2015 | Novel tacrine-grafted ugi adducts as multipotent anti-alzheimer drugs: A synthetic renewal in tacrine-ferulic acid hybrids | Benchekroun, M.; Bartolini, Manuela; Egea, Javier; Romero, A. ; Soriano, Elena ; Pudlo, M.; Luzet, Vincenza; Andrisano, V.; Jimeno, M. Luisa ; López, M. G.; Wehle, S.; Gharbi, T.; Refouvelet, B.; Andrés, L. de; Herrera-Arozamena, Clara; Monti, B.; Bolognesi, Maria Laura; Rodríguez-Franco, María Isabel ; Decker, M.; Marco-Contelles, José ; Ismaili, L. | artículo |
openAccess |  | 14-Mar-2019 | Structure-activity relationships and mechanistic studies of novel mitochondria-targeted, leishmanicidal derivatives of the 4-aminostyrylquinoline scaffold | Staderini, Matteo; Piquero, Marta; Abengozar, M. A. ; Nácher-Vázquez, Montserrat ; Romanelli, Giulia; López-Alvarado, Pilar; Rivas, Luis ; Bolognesi, Maria Laura; Menéndez, J. Carlos | artículo |
closedAccess |  | 2018 | Tacripyrimidines, the first tacrine-dihydropyrimidine hybrids, asmulti-target-directed ligands for Alzheimer's disease | Chioua, Mourad ; Buzzi, Eleonora; Moraleda, Ignacio; Iriepa, Isabel; Maj, Maciej; Wnorowski, Artur; Giovannini, Catia; Tamarin, Anna; Portali, Federica; Ismaili, Lhassane; López-Alvarado, Pilar; Bolognesi, Maria Laura; Jozwiak, Krzysztof; Menéndez, J. Carlos; Marco-Contelles, José ; Bartolini, Manuela | artículo |
closedAccess |  | 2018 | Tau-Centric Multitarget Approach for Alzheimer's Disease: Development of First-in-Class Dual Glycogen Synthase Kinase 3β and Tau-Aggregation Inhibitors | Gandini, A.; Bartolini, M.; Tedesco, D.; Martínez-González, Loreto ; Roca, Carlos; Campillo, Nuria E. ; Zaldívar-Díez, Josefa; Pérez, Concepción; Zuccheri, G.; Miti, A.; Feoli, A.; Castellano, S.; Petralla, S.; Monti, B.; Rossi, M.; Moda, F.; Legname, G.; Martínez, Ana; Bolognesi, Maria Laura | artículo |
closedAccess |  | 2013 | The bivalent ligand approach as a tool for improving the in vitro anti-alzheimer multitarget profile of dimebon | Rosini, M.; Simoni, E.; Bartolini, Manuela; Soriano, Elena ; Marco-Contelles, José ; Andrisano, V.; Monti, B.; Windisch, M.; Hutter-Paier, B.; McClymont, D. W.; Mellor, I. R.; Bolognesi, Maria Laura | artículo |