Derechos | Preview | Fecha Public. | Título | Autor(es) | Tipo |
closedAccess | | 2015 | 2-Phenoxy-1,4-naphthoquinones: From a Multitarget Antitrypanosomal to a Potential Antitumor Profile | Prati, F.; Bergamini, C.; Molina Orden, María Teresa CSIC; Falchi, F.; Cavalli, A.; Kaiser, M.; Brun, R.; Fato, R.; Bolognesi, Maria Laura | artículo |
openAccess | | 14-jul-2015 | 3,4-Dihydro-1,3,5-triazin-2(1H)-ones as the first dual BACE-1/GSK-3β fragment hits against Alzheimer’s disease | Prati, Federica; Pérez, Daniel I. CSIC ORCID; Pérez Castillo, Ana CSIC ORCID; Martínez Gil, Ana CSIC ORCID ; Bolognesi, Maria Laura | artículo |
closedAccess | | 2013 | A fluorescent styrylquinoline with combined therapeutic and diagnostic activities against Alzheimer's and prion diseases | Staderini, Matteo; Aulic, Suzana; Bartolini, Manuela; Tran, H. N. A.; González-Ruiz, Victor; Pérez, Daniel I. CSIC ORCID; Cabezas, Nieves; Martínez Gil, Ana CSIC ORCID ; Martín, M. Antonia; Andrisano, Vincenza; Legname, Giuseppe; Menéndez, José Carlos; Bolognesi, Maria Laura | artículo |
openAccess | | 9-oct-2018 | A focused library of psychotropic analogs with neuroprotective and neuroregenerative potential | Uliassi, Elisa; Peña-Altamira, Luis Emiliano; Morales, Aixa V. CSIC ORCID; Massenzio, Francesca; Petralla, Sabrina; Rossi, Michele; Roberti, Marinella; Martínez-González, Loreto CSIC ORCID ; Martínez Gil, Ana CSIC ORCID ; Monti, B.; Bolognesi, Maria Laura | artículo |
closedAccess | | 2012 | A small chemical library of 2-aminoimidazole derivatives as BACE-1 inhibitors: Structure-based design, synthesis, and biological evaluation | Chiriano, G.; De Simone, A.; Mancini, Francesca; Pérez, Daniel I. CSIC ORCID; Cavalli, A.; Bolognesi, Maria Laura; Legname, G.; Martínez, A.; Andrisano, Vincenza; Carloni, Paolo; Roberti, M. | artículo |
openAccess | | 15-nov-2022 | Bifunctional carbazole derivatives for simultaneous therapy and fluorescence imaging in prion disease murine cell models | Staderini, Matteo; Vanni, Silvia; Colini Baldeschi, Arianna; Giachin, Gabriele; Zattoni, Marco; Celauro, Luigi; Ferracin, Chiara; Bistaffa, Edoardo; Moda, F.; Pérez, Daniel I. CSIC ORCID; Martínez Gil, Ana CSIC ORCID ; Martín, M. Antonia; Martín-Cámara, Olmo; Cores, Ángel; Bianchini, Giulia; Kammerer, Robert; Menéndez, J. Carlos; Legname, G.; Bolognesi, Maria Laura | artículo |
openAccess | | dic-2006 | Design, synthesis, and biological evaluation of substituted 2,3-dihydro-1H-cyclopenta[b]quinolin-9-ylamine related compounds as fructose-1,6-bisphosphatase inhibitors | Rosini, Michela; Mancini, Francesca; Tarozzi, Andrea; Colizzi, Francesco CSIC ORCID; Andrisano, Vincenza; Bolognesi, Maria Laura; Hrelia, Patrizia; Melchiorre, Carlo | artículo |
openAccess | | 2022 | Discovery of Dual Aβ/Tau Inhibitors and Evaluation of Their Therapeutic Effect on a Drosophila Model of Alzheimer's Disease | Gandini, Annachiara; Gonçalves, Ana Elisa; Strocchi, Silvia; Albertini, Claudia; Janockova, Jana; Tramarin, Anna; Grifoni, Daniela; Poeta, Eleonora; Soukup, Ondrej; Muñoz-Torrero, Diego; Monti, Barbara; Sabate, Raimon; Bartolini, Manuela; Legname, Giuseppe; Bolognesi, Maria Laura | artículo |
closedAccess | | 2015 | Multitarget drug discovery for Alzheimer's disease: Triazinones as BACE-1 and GSK-3ß inhibitors | Pérez, Daniel I. CSIC ORCID; Pérez Castillo, Ana CSIC ORCID; Martínez Gil, Ana CSIC ORCID ; Bolognesi, Maria Laura; Cavalli, Andrea | artículo |
closedAccess | | jun-2014 | Multitarget ligands and theranostics: Sharpening the medicinal chemistry sword against prion diseases | Bongarzone, Salvatore CSIC ORCID; Staderini, Matteo; Bolognesi, Maria Laura | artículo |
openAccess | | 2015 | Novel tacrine-grafted ugi adducts as multipotent anti-alzheimer drugs: A synthetic renewal in tacrine-ferulic acid hybrids | Benchekroun, Mohamed; Bartolini, Manuela; Egea, Javier; Romero, Alejandro CSIC ORCID; Soriano, Elena CSIC; Pudlo, M.; Luzet, Vincenza; Andrisano, V.; Jimeno, M. Luisa CSIC ORCID; López, M. G.; Wehle, S.; Gharbi, T.; Refouvelet, B.; Andrés, Lucía de CSIC; Herrera-Arozamena, Clara CSIC ORCID CVN; Monti, B.; Bolognesi, Maria Laura; Rodríguez-Franco, María Isabel CSIC ORCID ; Decker, Michael; Marco-Contelles, José CSIC ORCID; Ismaili, L. | artículo |
openAccess | | 14-mar-2019 | Structure-activity relationships and mechanistic studies of novel mitochondria-targeted, leishmanicidal derivatives of the 4-aminostyrylquinoline scaffold | Staderini, Matteo; Piquero, Marta; Abengozar, M. A. CSIC; Nácher-Vázquez, Montserrat CSIC ORCID; Romanelli, Giulia; López-Alvarado, Pilar; Rivas, Luis CSIC ORCID ; Bolognesi, Maria Laura; Menéndez, J. Carlos | artículo |
closedAccess | | 2018 | Tacripyrimidines, the first tacrine-dihydropyrimidine hybrids, asmulti-target-directed ligands for Alzheimer's disease | Chioua, Mourad CSIC ORCID ; Buzzi, Eleonora; Moraleda, Ignacio; Iriepa, Isabel; Maj, Maciej; Wnorowski, Artur; Giovannini, Catia; Tamarin, Anna; Portali, Federica; Ismaili, Lhassane; López-Alvarado, Pilar; Bolognesi, Maria Laura; Jóźwiak, Krzysztof; Menéndez, J. Carlos; Marco-Contelles, José CSIC ORCID; Bartolini, Manuela | artículo |
closedAccess | | 2018 | Tau-Centric Multitarget Approach for Alzheimer's Disease: Development of First-in-Class Dual Glycogen Synthase Kinase 3β and Tau-Aggregation Inhibitors | Gandini, A.; Bartolini, M.; Tedesco, D.; Martínez-González, Loreto CSIC ORCID ; Roca, Carlos CSIC ORCID; Campillo, Nuria E. CSIC ORCID ; Zaldívar-Díez, Josefa CSIC ORCID; Pérez, Concepción CSIC ORCID; Zuccheri, G.; Miti, Andrea; Feoli, A.; Castellano, S.; Petralla, Sabrina; Monti, B.; Rossi, M.; Moda, F.; Legname, G.; Martínez Gil, Ana CSIC ORCID ; Bolognesi, Maria Laura | artículo |
closedAccess | | 2013 | The bivalent ligand approach as a tool for improving the in vitro anti-alzheimer multitarget profile of dimebon | Rosini, M.; Simoni, E.; Bartolini, Manuela; Soriano, Elena CSIC; Marco-Contelles, José CSIC ORCID; Andrisano, V.; Monti, B.; Windisch, M.; Hutter-Paier, B.; McClymont, D. W.; Mellor, I. R.; Bolognesi, Maria Laura | artículo |