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Browsing by Author Balzarini, Jan

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RightsPreviewIssue DateTitleAuthor(s)Type
closedAccessaccesoRestringido.pdf.jpg2015Anti-HIV-1 activity of a tripodal receptor that recognizes mannose oligomersRivero-Buceta, Eva ; Carrero, Paula ; Casanova, Elena ; Doyagüez, Elisa G.; Madrona, Andrés; Quesada, Ernesto; Peréz-Pérez, María-Jesús ; Mateos, Raquel  ; Bravo, Laura ; Mathys, Leen; Noppen, Sam; Kiselev, Evgency; Marchand, Christophe; Pommier, Yves; Liekens, Sandra; Balzarini, Jan; Camarasa Rius, María José ; San-Félix, Ana Artículo
closedAccessArtículo.pdf.jpg2001Anti-HIV-1 activity of benzothiadiazine dioxideMartínez, Ana ; Gil, Carmen  ; Castro, Ana ; Pérez, Concepción; Witvrouw, M.; Pannecouque, C.; Balzarini, Jan; De Clercq, ErikArtículo
openAccessCarbohydrate_Binding_Plos_Pathogens_2016.pdf.jpg23-Sep-2016Carbohydrate-Binding Non-Peptidic Pradimicins for the Treatment of Acute Sleeping Sickness in Murine ModelsCastillo Acosta, Víctor M.; Ruiz-Pérez, Luis Miguel; Etxebarria, Juan; Reichardt, Niels Christian; Navarro, M.; Igarashi, Yasuhiro; Liekens, Sandra; Balzarini, Jan; González-Pacanowska, D.Artículo
closedAccess2015Conservation of antiviral activity and improved selectivity in PMEO-DAPym upon pyrimidine to triazine scaffold hoppingCastro, Sonia de ; Fernández-Cureses, Gloria ; Andrei, G; Snoeck, R.; Sánchez-Murcia, Pedro A. ; Korban, B.; Gago, Federico ; Balzarini, Jan; Camarasa Rius, María José Artículo
closedAccess2011Crystal structure of tert -butyldimethylsilyl-spiroaminooxathioledioxide- thymine (TSAO-T) in complex with HIV-1 reverse transcriptase (RT) redefines the elastic limits of the non-nucleoside inhibitor-binding pocketDas, Krishna; Bauman, J. D.; Rim, A. S.; Dharia, C.; Clark, A. D.; Camarasa Rius, María José ; Balzarini, Jan; Arnold, E.Artículo
closedAccess2015Design, synthesis, and biological evaluation of unconventional aminopyrimidine, aminopurine, and amino-1,3,5-triazine methyloxynucleosidesFernández-Cureses, Gloria ; Castro, Sonia de ; Jimeno, M. Luisa ; Balzarini, Jan; Camarasa Rius, María José Artículo
closedAccess2011Dipeptidyl peptidase IV dependent water-soluble prodrugs of highly lipophilic bicyclic nucleoside analoguesDiez-Torrubia, Alberto ; Balzarini, Jan; Andrei, G; Snoeck, R.; De Meester, Ingrid; Camarasa Rius, María José ; Velázquez, Sonsoles Artículo
closedAccess2012Dipeptidyl Peptidase IV-Activated Prodrugs of Anti- Varicella Zoster Virus Bicyclic Nucleoside Analogues Containing Different Self-Cleavage Spacer SystemsDiez-Torrubia, Alberto ; Cabrera, Silvia ; De Meester, Ingrid; Camarasa Rius, María José ; Balzarini, Jan; Velázquez, Sonsoles Artículo
closedAccess2015Dipeptidyl-peptidase IV (DPP IV/CD26)-activated prodrugs: A successful strategy for improving water solubility and oral bioavailabilityVelázquez, Sonsoles ; Castro, Sonia de ; Diez-Torrubia, Alberto ; Balzarini, Jan; Camarasa Rius, María José Artículo
closedAccess3-Feb-2012Dipeptidyl-peptidase IV (DPPIV/CD26)-based prodrugs of hydroxy-containing drugsDiez-Torrubia, Alberto ; Cabrera, Silvia ; Lambeir, Anne-Marie; Balzarini, Jan; Camarasa Rius, María José ; Velázquez, Sonsoles Artículo
closedAccessaccesoRestringido.pdf.jpg2014Discovery and SAR studies of a novel class of cytotoxic 1,4-disubstituted piperidines via Ugi reactionCastro, Sonia de ; Camarasa Rius, María José ; Balzarini, Jan; Velázquez, Sonsoles Artículo
openAccessExposure_pntd.PDF.jpg6-Mar-2015Exposure of Trypanosoma brucei to an N-acetylglucosamine-Binding Lectin Induces VSG Switching and Glycosylation Defects Resulting in Reduced InfectivityCastillo Acosta, Víctor M.; Ruiz-Pérez, Luis Miguel; Van Damme, Els J. M.; Balzarini, Jan; González-Pacanowska, D.Artículo
closedAccess2011From β-Amino-γ-sultone to Unusual Bicyclic Pyridine and Pyrazine Heterocyclic Systems: Synthesis and Cytostatic and Antiviral ActivitiesCastro, Sonia de ; Familiar, Olga ; Andrei, G; Snoeck, R.; Balzarini, Jan; Camarasa Rius, María José ; Velázquez, Sonsoles Artículo
openAccessWO2011085454A1.pdf.jpg21-Jul-2011gp120 -binding benzene compounds and saccharide compoundsBalzarini, Jan; Carrero, Paula ; Casanova, Elena; Peréz-Pérez, María-Jesús ; San-Félix, Ana Solicitud de patente
closedAccess2000HIV-1 specific reverse transcriptase inhibitors: Why are TSAO-nucleosides so unique?Camarasa Rius, María José ; San-Felix, Alejandra; Pérez Pérez, María Jesús; Velázquez, Sonsoles ; Álvarez, Rosa; Chamorro, Cristina; Jimeno, M. Luisa ; Perez, Carlos; Gago, Federico ; De Clercq, Erik; Balzarini, JanArtículo
closedAccessaccesoRestringido.pdf.jpg2009Identification of aspartic acid-203 in human thymidine phosphorylase as an important residue for both catalysis and non-competitive inhibition by the small molecule >crystallization chaperone> 5′-O-tritylinosine (KIN59)Bronckaers, A.; Aguado, Leire ; Negri, Ana; Camarasa Rius, María José ; Balzarini, Jan; Peréz-Pérez, María-Jesús ; Gago, Federico ; Liekens, S.Artículo
openAccessWO2009030410A1.pdf.jpg12-Mar-2009Improvements in or relating to compositions for the treatment or prophylaxis of viral infectionsBalzarini, Jan; Camarasa Rius, María José ; Velázquez, Sonsoles Patente
closedAccess2015Linear and branched alkyl-esters and amides of gallic acid and other (mono-, di- and tri-) hydroxy benzoyl derivatives as promising anti-HCV inhibitorsRivero-Buceta, Eva ; Carrero, P.; Doyagüez, Elisa G.; Madrona, Andrés; Quesada, Ernesto ; Camarasa Rius, María José ; Peréz-Pérez, María-Jesús ; Leyssen, Pieter; Paeshuyse, Jan; Balzarini, Jan; Neyts, Johan; San-Félix, Ana Artículo
openAccessGigante_full_article.pdf.jpg2014Microwave-assisted synthesis of C-8 aryl and heteroaryl inosines and determination of their inhibitory activities against Plasmodium falciparum purine nucleoside phosphorylaseGigante, Alba ; Priego, Eva María ; Sánchez-Carrasco, Paula; Ruiz-Pérez, Luis Miguel; Vande Voorde, Johan; Camarasa Rius, María José ; Balzarini, Jan; González-Pacanowska, D.; Peréz-Pérez, María-Jesús Artículo
openAccessOrg. Biomol. Chem., 2014.pdf.jpg2014Multivalent agents containing 1-substituted 2,3,4-trihydroxyphenyl moieties as novel synthetic polyphenols directed against HIV-1Flores, Aida ; Camarasa Rius, María José ; Peréz-Pérez, María-Jesús ; San-Félix, Ana ; Balzarini, Jan; Quesada, Ernesto Artículo