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DerechosPreviewFecha Public.TítuloAutor(es)Tipo
openAccess1-s2.0-S2451945624000436-main.pdf.jpg6-feb-2024Identification of differential biological activity and synergy between the PARP inhibitor rucaparib and its major metaboliteHu, Huabin; Serra, Carme; Zhang, Wenjie; Scrivo, Aurora; Fernández-Carasa, Irene; Consiglio, Antonella; Aytes, Alvaro; Pujana, Miguel Angel; Llebaria, Amadeu CSIC ORCID; Antolin, Albert A.artículo
openAccessIlluminating Phenylazopyridines to Photoswitch Metabotropic Glutamate Receptors. From the Flask to the Animals.pdf.jpg25-ene-2017Illuminating Phenylazopyridines to Photoswitch Metabotropic Glutamate Receptors: From the Flask to the AnimalsGómez-Santacana, Xavier CSIC ORCID; Pittolo, Silvia; Rovira, Xavier CSIC ORCID; Llebaria, Amadeu CSIC ORCIDartículo
openAccessIn the search for photocages cleavable with visible light.pdf.jpg4-dic-2020In the Search for Photocages Cleavable with Visible Light: An Overview of Recent Advances and Chemical StrategiesJosa-Culleré, Laia CSIC ORCID; Llebaria, Amadeu CSIC ORCIDartículo
openAccess2170030_B1.pdf.jpg16-nov-2003Inhibidores de la dihidroceramida desaturasaFabriàs, Gemma CSIC ORCID ; Llebaria, Amadeu CSIC ORCID; Triola Guillem, Gemma CSIC ORCIDpatente
closedAccess1-sep-2006Inhibitors of sphingolipid metabolism enzymesDelgado Cirilo, Antonio CSIC ORCID; Casas, Josefina CSIC ORCID ; Llebaria, Amadeu CSIC ORCID; Abad, José Luis CSIC ORCID ; Fabriàs, Gemma CSIC ORCID artículo
closedAccess2011Integrated Synthetic, Pharmacological, and Computational Investigation of cis-2-(3,5-Dichlorophenylcarbamoyl)cyclohexanecarboxylic Acid Enantiomers As Positive Allosteric Modulators of Metabotropic Glutamate Receptor Subtype 4Christov, Christo; González-Bulnes, Patricia CSIC; Malhaire, Fanny; Karabencheva, Tatyana; Goudet, Cyril; Pin, Jean Philippe; Llebaria, Amadeu CSIC ORCID; Giraldo, Jesúsartículo
openAccessijms-23-08018-v2.pdf.jpg20-jul-2022Light-Induced Activation of a Specific Type-5 Metabotropic Glutamate Receptor Antagonist in the Ventrobasal Thalamus Causes Analgesia in a Mouse Model of Breakthrough Cancer PainNotartomaso, Serena; Antenucci, Nico; Liberatore, Francesca; Mascio, Giada; Boccadamo Pompili, Stefano Vito; Font, Joan CSIC ORCID; Scioli, Mariarosaria; Luongo, Livio; Arcella, Antonietta; Gradini, Roberto; Llebaria, Amadeu CSIC ORCID; Nicoletti, Ferdinandoartículo
openAccess5fa12230b334c5000712c26a.pdf.jpg9-nov-2020Mimetics of extra virgin olive oil phenols with anti-cancer stem cell activityCuyàs, Elisabet; Gumuzio, Juan; Lozano-Sánchez, Jesús; Segura-Carretero, Antonio; Verdura, Sara; Bosch-Barrera, Joaquim; Martín-Castillo, Begoña; Nonell-Canals, Alfons; Llebaria, Amadeu CSIC ORCID; Cabello, Silvia CSIC; Serra, Carmen CSIC ORCID; Sánchez-Martinez, Melchor; Martín, Ángel G.; Menéndez, Javier A.artículo
embargoedAccess1-s2.0-S2451945623002374-main.pdf.jpg17-ago-2023Mitochondria-targeted melatonin photorelease supports the presence of melatonin MT1 receptors in mitochondria inhibiting respirationSomalo-Barranco, Gloria; Pagano Zottola, Antonio C.; Abdulrahman, Abdulrasheed O.; El Zein, Rami M; Cannich, Astrid; Muñoz, Lourdes CSIC ORCID; Serra, Carmen CSIC ORCID; Oishi, Atsuro; Marsicano, Giovanni; Masri, Bernard; Bellocchio, Luigi; Llebaria, Amadeu CSIC ORCID; Jockers, Ralfartículo
closedAccess2-oct-2008Molecular Basis for β-Glucosidase Inhibition by Ring-Modified Calystegine AnaloguesAguilar Moncayo, Matilde; Gloster, Tracey M.; García Moreno, María Isabel; Ortiz-Mellet, Carmen; Davies, Gideon J.; Llebaria, Amadeu CSIC ORCID; Casas, Josefina CSIC ORCID ; Egido-Gabás, Meritxell CSIC; García Fernández, José Manuel CSIC ORCIDartículo
openAccessEgido_Meritxell_et_al.pdf.jpg1-mar-2005New aminocyclitols as modulators of glucosylceramide metabolismEgido-Gabás, Meritxell CSIC; Serrano, Pedro; Casas, Josefina CSIC ORCID ; Llebaria, Amadeu CSIC ORCID; Delgado Cirilo, Antonio CSIC ORCIDartículo
closedAccess2011New Glucocerebrosidase Inhibitors by Exploration of Chemical Diversity of N-Substituted Aminocyclitols Using Click Chemistry and in Situ ScreeningDíaz-Bueno, Lucía CSIC ORCID; Casas, Josefina CSIC ORCID ; Bujons, Jordi CSIC ORCID; Llebaria, Amadeu CSIC ORCID; Delgado Huertas, Antonio CSIC ORCID artículo
openAccesscmdc.202000992.pdf.jpg6-abr-2021New Paradigm in NKT Cell Antigens: MCS-0208 (2-(Hydroxymethyl)phenylthio-phytoceramide) – an Aryl-Phytoceramide Compound with a Single Hydroxyl Group Stimulates NKT CellsBorràs-Tudurí, Roser CSIC; Alcaide, Anna CSIC; Aspeslag, Sandrine; Usero, Lorena; Serra, Carmen CSIC ORCID; Roura-Mir, Carme; Elewaut, Dirk; Llebaria, Amadeu CSIC ORCIDartículo
closedAccess2011NKT TCR Recognition of CD1d-α-C-GalactosylceramidePatel, Onisha; Cameron, Garth; Pellicci, Daniel G.; Liu, Zheng; Byun, Hoe-Sup; Beddoe, Travis; McCluskey, James; Franck, Richard W.; Castaño, A. Raúl; Harrak Serifi, Youssef CSIC; Llebaria, Amadeu CSIC ORCID; Bittman, Robert; Porcelli, Steven A.; Godfrey, Dale I.; Rossjohn, Jamieartículo
openAccessES2713775A1.pdf.jpg31-may-2019Non-glycosidic analogues of alpha-galactosylceramide as NKT cell activatorsLlebaria, Amadeu CSIC ORCID; Borràs-Tudurí, Roser CSIC; Serra, Carmen CSIC ORCID; Alcaide, Anna CSICsolicitud de patente
closedAccess13-may-2005On the regio- and stereoselective synthesis of aminocyclitols from cyclitol epoxides: the effect of Li as a chelating agentSerrano, Pedro; Llebaria, Amadeu CSIC ORCID; Vázquez, Jordi; Pablo, Joan de; Anglada Rull, Josep M. CSIC ORCID; Delgado Cirilo, Antonio CSIC ORCIDartículo
embargoedAccessdumazer-et-al-2024-optical-control-of-adenosine-a2a-receptor-using-istradefylline-photosensitivity.pdf.jpg7-feb-2024Optical Control of Adenosine A2A Receptor Using Istradefylline PhotosensitivityDumazer, Anaëlle; Gómez-Santacana, Xavier CSIC ORCID; Malhaire, Fanny; Jopling, Chris; Maurel, Damien; Lebon, Guillaume; Llebaria, Amadeu CSIC ORCID; Goudet, Cyrilartículo
openAccessOptical control of endogenous receptors and cellular excitability using targeted covalent photoswitches.pdf.jpg20-jul-2016Optical control of endogenous receptors and cellular excitability using targeted covalent photoswitchesIzquierdo-Serra, Mercè; Trapero, Ana CSIC ORCID; Llebaria, Amadeu CSIC ORCID; Gorost́iza, Pauartículo
openAccesselife-23545-v1 (2).pdf.jpg11-abr-2017Optical control of pain in vivo with a photoactive mGlu5 receptor negative allosteric modulatorFont, Joan CSIC ORCID; López-Cano, Marc; Notartomaso, Serena; Scarselli, Pamela; Di Pietro, Paola Di; Bresolí-Obach, Roger; Battaglia, Giuseppe; Malhaire, Fanny; Rovira, Xavier CSIC ORCID; Catena, Juan Lorenzo CSIC ORCID; Giraldo, Jesús; Pin, Jean Philippe; Fernández-Dueñas, Víctor; Goudet, Cyril; Nonell, Santi; Nicoletti, Ferdinando; Llebaria, Amadeu CSIC ORCID; Ciruela, Franciscoartículo
openAccessOptoGluNAM4.1, a Photoswitchable Allosteric.pdf.jpg18-ago-2016OptoGluNAM4.1, a Photoswitchable Allosteric Antagonist for Real-Time Control of mGlu4 Receptor ActivityRovira, Xavier CSIC ORCID; Trapero, Ana CSIC ORCID; Llebaria, Amadeu CSIC ORCIDartículo