Derechos | Preview | Fecha Public. | Título | Autor(es) | Tipo |
openAccess | | 2015 | Anti-HIV-1 activity of a tripodal receptor that recognizes mannose oligomers | Rivero-Buceta, Eva CSIC ORCID; Carrero, Paula CSIC; Casanova, Elena CSIC; Doyagüez, Elisa G. CSIC; Madrona, Andrés CSIC ORCID; Quesada, Ernesto CSIC ORCID ; Peréz-Pérez, María-Jesús CSIC ORCID ; Mateos, Raquel CSIC ORCID ; Bravo, Laura CSIC ORCID; Mathys, Leen; Noppen, Sam; Kiselev, Evgency; Marchand, Christophe; Pommier, Yves; Liekens, Sandra; Balzarini, Jan; Camarasa Rius, María José CSIC ORCID; San-Félix, Ana CSIC ORCID | artículo |
openAccess | | 20-may-2016 | Antivascular and antitumor properties of the tubulin-binding chalcone TUB091 | Canela, María-Dolores CSIC; Noppen, Sam; Bueno, Oskia CSIC; Prota, Andrea E.; Bargsten, Katja; Sáez-Calvo, Gonzalo CSIC; Jimeno, M. Luisa CSIC ORCID; Benkhei, Mohammed; Ribatti, Domenico; Velázquez, Sonsoles CSIC ORCID CVN; Camarasa Rius, María José CSIC ORCID; Díaz, José Fernando CSIC ORCID ; Steinmetz, Michel O.; Priego, Eva María CSIC ORCID; Peréz-Pérez, María-Jesús CSIC ORCID ; Liekens, Sandra | artículo |
openAccess | | 27-jun-2016 | Blocking Blood Flow to Solid Tumors by Destabilizing Tubulin : An Approach to Targeting Tumor Growth (Perspective) | Peréz-Pérez, María-Jesús CSIC ORCID ; Priego, Eva María CSIC ORCID; Bueno, Oskia CSIC; Martins, Maria Solange; Canela, María-Dolores CSIC; Liekens, Sandra | artículo |
openAccess | | 23-sep-2016 | Carbohydrate-Binding Non-Peptidic Pradimicins for the Treatment of Acute Sleeping Sickness in Murine Models | Castillo Acosta, Víctor M.; Ruiz-Pérez, Luis Miguel; Etxebarria, Juan; Reichardt, Niels Christian; Navarro, M.; Igarashi, Yasuhiro; Liekens, Sandra; Balzarini, Jan; González-Pacanowska, Dolores | artículo |
openAccess | | 2018 | Conformational mimetics of the α-methyl chalcone TUB091 binding tubulin: Design, synthesis and antiproliferative activity | Bueno, Oskia CSIC; Tobajas, Gloria; Quesada, Ernesto CSIC ORCID ; Estévez-Gallego, Juan CSIC ORCID ; Noppen, Sam; Camarasa Rius, María José CSIC ORCID; Díaz, José Fernando CSIC ORCID ; Liekens, Sandra; Priego, Eva María CSIC ORCID; Peréz-Pérez, María-Jesús CSIC ORCID | artículo |
closedAccess | | jun-2019 | Diphenyl ether derivatives occupy the expanded binding site of cyclohexanedione compounds at the colchicine site in tubulin by movement of the aT5 loop | Bueno, Oskia CSIC; Gargantilla, Marta CSIC ORCID; Estévez-Gallego, Juan CSIC ORCID ; Martins, Solange; Díaz, José Fernando CSIC ORCID ; Camarasa Rius, María José CSIC ORCID; Liekens, Sandra; Peréz-Pérez, María-Jesús CSIC ORCID ; Priego, Eva María CSIC ORCID | artículo |
openAccess | | 2018 | High-affinity ligands of the colchicine domain in tubulin based on a structure-guided design | Bueno, Oskia CSIC; Estévez-Gallego, Juan CSIC ORCID ; Martins, S.; Prota, Andrea E.; Gago, Federico CSIC ORCID; Gómez-SanJuan, Asier CSIC; Camarasa Rius, María José CSIC ORCID; Barasoain, Isabel CSIC ; Steinmetz, Michel O.; Díaz, José Fernando CSIC ORCID ; Peréz-Pérez, María-Jesús CSIC ORCID ; Liekens, Sandra; Priego, Eva María CSIC ORCID | artículo |
openAccess | | 2014 | Novel colchicine-site binders with a cyclohexanedione scaffold identified through a ligand-based virtual screening approach | Canela, María-Dolores CSIC; Peréz-Pérez, María-Jesús CSIC ORCID ; Noppen, Sam; Sáez-Calvo, Gonzalo CSIC; Díaz, José Fernando CSIC ORCID ; Camarasa Rius, María José CSIC ORCID; Liekens, Sandra; Priego, Eva María CSIC ORCID | artículo |
openAccess | | 23-ene-2018 | Protein-ligand complex for structure-based design: impact on the affinity and antitumor activity of new tubulin ligands | Bueno, Oskia CSIC; Estévez-Gallego, Juan CSIC ORCID ; Martins, S.; Prota, Andrea E.; Gago, Federico CSIC ORCID; Gómez-SanJuan, Asier CSIC; Camarasa Rius, María José CSIC ORCID; Barasoain, Isabel CSIC ; Steinmetz, Michel O.; Díaz, José Fernando CSIC ORCID ; Liekens, Sandra; Peréz-Pérez, María-Jesús CSIC ORCID ; Priego, Eva María CSIC ORCID | comunicación de congreso |
openAccess | | 2017 | Structure-activity relationship studies on a Trp dendrimer with dual activities against HIV and enterovirus A71. Modifications on the amino acid | Martínez-Gualda, Belén CSIC; Sun, L.; Rivero-Buceta, Eva CSIC ORCID; Flores, Aida CSIC; Quesada, Ernesto CSIC ORCID ; Balzarini, Jan; Noppen, Sam; Liekens, Sandra; Schols, Dominique; Neyts, Johan; Leyssen, Pieter; Mirabelli, C.; Camarasa Rius, María José CSIC ORCID; San-Félix, Ana CSIC ORCID | artículo |
closedAccess | | 2016 | Targeting the colchicine site in tubulin through cyclohexanedione derivatives | Canela, María-Dolores CSIC; Bueno, Oskia CSIC; Noppen, Sam; Sáez-Calvo, Gonzalo CSIC; Estévez-Gallego, Juan CSIC ORCID ; Díaz, José Fernando CSIC ORCID ; Camarasa Rius, María José CSIC ORCID; Liekens, Sandra; Peréz-Pérez, María-Jesús CSIC ORCID ; Priego, Eva María CSIC ORCID | artículo |
openAccess | | 2015 | Tryptophan dendrimers that inhibit HIV replication, prevent virus entry and bind to the HIV envelope glycoproteins gp120 and gp41 | Rivero-Buceta, Eva CSIC ORCID; Doyagüez, Elisa G. CSIC; Colomer, Ignacio CSIC ORCID ; Quesada, Ernesto CSIC ORCID ; Mathys, Leen; Noppen, Sam; Liekens, Sandra; Camarasa Rius, María José CSIC ORCID; Peréz-Pérez, María-Jesús CSIC ORCID ; Balzarini, Jan; San-Félix, Ana CSIC ORCID | artículo |