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DerechosPreviewFecha Public.TítuloAutor(es)Tipo
openAccessSVelazquez_manuscript-ACSID 2020_compressed.pdf.jpg2020N-benzyl 4,4-disubstituted piperidines as a potent class of influenza H1N1 virus inhibitors showing a novel mechanism of hemagglutinin fusion peptide interactionCastro, Sonia de CSIC ORCID; Ginex, Tiziana CSIC ORCID ; Vanderlinden, E.; Laporte, M.; Stevaert, A.; Cumella, José; Gago, Federico CSIC ORCID; Camarasa Rius, María José CSIC ORCID; Luque, F. Javier; Naesens, L.; Velázquez, Sonsoles CSIC ORCID CVNartículo
openAccessfbioe-08-00593.pdf.jpg2020N-Ribosyltransferase From Archaeoglobus veneficus: A Novel Halotolerant and Thermostable Biocatalyst for the Synthesis of Purine Ribonucleoside AnalogsAcosta, Javier; Arco, J. del; Pisabarro, V.; Gago, Federico CSIC ORCID; Fernández-Lucas, J.artículo
openAccess2341215_A1.pdf.jpg16-jun-2010Nucleósidos modificados para el tratamiento de infecciones por LeishmaniaPeréz-Pérez, María-Jesús CSIC ORCID ; Casanova Malpica, Elena; Camarasa Rius, María José CSIC ORCID; Jiménez Ruiz, Antonio; Moreno Mateos, David; Rico Galán, Eva; Gago, Federico CSIC ORCIDsolicitud de patente
openAccess2341215_B1.pdf.jpg26-abr-2011Nucleósidos modificados para el tratamiento de infecciones por LeishmaniaGago, Federico CSIC ORCID; Rico Galán, Eva; Camarasa Rius, María José CSIC ORCID; Jiménez, A. R.; Casanova Malpica, Elena; Moreno Mateos, David; Peréz-Pérez, María-Jesús CSIC ORCID patente
openAccessijms-22-06973-v2.pdf.jpg2021On the need to tell apart fraternal twins eef1a1 and eef1a2, and their respective outfitsMills, Alberto; Gago, Federico CSIC ORCIDartículo
closedAccessMatesanz et al-2008_Chemistry and Biology.pdf.jpg23-jun-2008Optimization of Taxane Binding to Microtubules: Binding Affinity Dissection and Incremental Construction of a High-Affinity Analog of PaclitaxelMatesanz, Ruth CSIC ; Barasoain, Isabel CSIC ; Yang, Chun-Gang; Wan, L.; Li, Xuan; Inés, Concepción de CSIC; Coderch, Claire; Gago, Federico CSIC ORCID; Jiménez-Barbero, Jesús CSIC ORCID; Andreu, José Manuel CSIC ORCID ; Fang, Wei-Shuo; Díaz, José Fernando CSIC ORCID artículo
openAccessEuropean Journal of Medicinal Chemistry 237.pdf.jpgabr-2022Organotropic dendrons with high potency as HIV-1, HIV-2 and EV-A71 cell entry inhibitorsMartí-Marí, Olaia CSIC ORCID; Martínez-Gualda, Belén CSIC; Fernández-Barahona, Irene; Mills, Alberto; Abdelnabi, Rana; Noppen, Sam; Neyts, Johan; Schols, Dominique; Camarasa Rius, María José CSIC ORCID; Herranz, Fernando CSIC ORCID CVN; Gago, Federico CSIC ORCID; San-Félix, Ana CSIC ORCID artículo
openAccessACSMCL2020_RT-dimeriz-inhibs-3(revised-for publication).pdf.jpg2020Peptides mimicking the β7/β8 loop of HIV'1 reverse transcriptase p51 as “hotspot-targeted” dimerization inhibitorsSánchez-Murcia, Pedro A. CSIC ORCID; Castro, Sonia de CSIC ORCID; García-Aparicio, Carlos CSIC; Jiménez, M. Angeles CSIC ORCID ; Corona, A.; Tramontano, Enzo; Sluis-Cremer, N.; Menéndez-Arias, Luis CSIC ORCID ; Velázquez, Sonsoles CSIC ORCID CVN; Gago, Federico CSIC ORCID; Camarasa Rius, María José CSIC ORCIDartículo
closedAccess6-jun-2013Probing the Dimerization Interface of Leishmania infantum Trypanothione Reductase with Site-Directed Mutagenesis and Short PeptidesToro, Miguel Ángel; Sánchez-Murcia, Pedro A. CSIC ORCID; Moreno, David; Ruiz-Santaquiteria, Marta CSIC ORCID; Alzate, Juan Fernando; Negri, Ana; Camarasa Rius, María José CSIC ORCID; Gago, Federico CSIC ORCID; Velázquez, Sonsoles CSIC ORCID CVN; Jiménez-Ruiz, Antonioartículo
openAccessProtein ligand complex.pdf.jpg23-ene-2018Protein-ligand complex for structure-based design: impact on the affinity and antitumor activity of new tubulin ligandsBueno, Oskia CSIC; Estévez-Gallego, Juan CSIC ORCID ; Martins, S.; Prota, Andrea E.; Gago, Federico CSIC ORCID; Gómez-SanJuan, Asier CSIC; Camarasa Rius, María José CSIC ORCID; Barasoain, Isabel CSIC ; Steinmetz, Michel O.; Díaz, José Fernando CSIC ORCID ; Liekens, Sandra; Peréz-Pérez, María-Jesús CSIC ORCID ; Priego, Eva María CSIC ORCIDcomunicación de congreso
openAccessBrit. J. Pharmacol..pdf.jpg2020Pseudoirreversible slow-binding inhibition of trypanothione reductase by a protein–protein interaction disruptorLucio, Héctor de; Toro, Miguel Ángel; Camarasa Rius, María José CSIC ORCID; Velázquez, Sonsoles CSIC ORCID CVN; Gago, Federico CSIC ORCID; Jimenez-Ruiz, Antonioartículo
openAccessEuropean Journal of Medical Chemistry.pdf.jpg2022Pyridazino-pyrrolo-quinoxalinium salts as highly potent and selective leishmanicidal agents targeting trypanothione reductasede Lucio, H.; García-Marín, Javier CSIC ORCID; Sánchez-Alonso, Patricio; García-Soriano, Juan Carlos; Toro, Miguel Ángel; Vaquero, Juan J.; Gago, Federico CSIC ORCID; Alajarín, Ramón; Jimenez-Ruiz, Antonioartículo
openAccessaccesoRestringido.pdf.jpg2019Pyrrolopyrimidine vs imidazole-phenyl-thiazole scaffolds in nonpeptidic dimerization inhibitors of leishmania infantum trypanothione reductaseRevuelto, Alejandro CSIC ORCID; Ruiz-Santaquiteria, Marta CSIC ORCID; Lucio, Héctor de; Gamo, Ana; Carriles, Alejandra A. CSIC ORCID; Gutiérrez, Kilian Jesús; Sánchez-Murcia, Pedro A. CSIC ORCID; Gago, Federico CSIC ORCID; Camarasa Rius, María José CSIC ORCID; Jiménez-Ruiz, Antonio; Velázquez, Sonsoles CSIC ORCID CVNartículo
openAccessBioinformatica_OrgBiomolChem_1543.pdf.jpg3-nov-2011Rationale for the opposite stereochemistry of the major monoadducts and interstrand crosslinks formed by mitomycin C and its decarbamoylated analogue at CpG steps in DNA and the effect of cytosine modification on reactivityBueren-Calabuig, Juan A.; Negri, Ana; Morreale, Antonio; Gago, Federico CSIC ORCIDartículo
closedAccessaccesoRestringido.pdf.jpg2019Reaction mechanism of nucleoside 2′-deoxyribosyltransferases: Free-energy landscape supports an oxocarbenium ion as the reaction intermediateDel Arco, J.; Perona, Almudena CSIC ORCID CVN; González, L.; Fernández-Lucas, J.; Gago, Federico CSIC ORCID; Sánchez-Murcia, Pedro A. CSIC ORCIDartículo
closedAccess2012Recent Advances in Thymidine Kinase 2 (TK2) Inhibitors and New Perspectives for Potential ApplicationsPriego, Eva María CSIC ORCID; Karlsson, Anna; Gago, Federico CSIC ORCID; Camarasa Rius, María José CSIC ORCID; Balzarini, Jan; Peréz-Pérez, María-Jesús CSIC ORCID artículo
openAccessSanjuan_PlantPhysiology 2020_Author copy.pdf.jpg2020Recognition and activation of the plant AKT1 potassium channel by the kinase CIPK23Sánchez-Barrena, María José CSIC ORCID; Chaves Sanjuán, Antonio CSIC ORCID; Raddatz, Natalia CSIC ORCID; Mendoza, Imelda CSIC ORCID; Cortés, Álvaro; Gago, Federico CSIC ORCID; González-Rubio, Juana M. CSIC; Benavente, Juan Luis CSIC ORCID; Quintero, Francisco J. CSIC ORCID ; Pardo, José M. CSIC ORCID ; Albert, Armando CSIC ORCIDartículo
closedAccessaccesoRestringido.pdf.jpg18-dic-2015Restoration of microtubule interaction and cytotoxicity in D-seco taxanes upon incorporation of 20-hydroxymethyl-4-allyloxy groupsWang, Shao-Rong; Yang, Chun-Gang; Sánchez-Murcia, Pedro A. CSIC ORCID; Snyder, James P.; Yan, Ning; Sáez-Calvo, Gonzalo CSIC; Díaz, José Fernando CSIC ORCID ; Gago, Federico CSIC ORCID; Fang, Wei-Shuoartículo
openAccessASF9 REVISED jm-2019-01737d.pdf.jpgene-2020Scaffold Simplification Strategy Leads to a Novel Generation of Dual Human Immunodeficiency Virus and Enterovirus-A71 Entry InhibitorsMartínez-Gualda, Belén CSIC; Sun, Liang; Martí-Marí, Olaia CSIC ORCID; Abdelnabi, Rana; Noppen, Sam; Bator, Carol M.; Quesada, Ernesto CSIC ORCID ; Delang, Leen; Mirabelli, Carmen; Lee, Hyunwook; Schols, Dominique; Neyts, Johan; Hafenstein, Susan; Camarasa Rius, María José CSIC ORCID; Gago, Federico CSIC ORCID; San-Félix, Ana CSIC ORCID artículo
openAccesspharmaceuticals-14-00689-v2-1.pdf.jpg17-jul-2021Small Molecule–Peptide Conjugates as Dimerization Inhibitors of Leishmania infantum Trypanothione Disulfide ReductaseRevuelto, Alejandro CSIC ORCID; López-Martín, Isabel; Lucio, Héctor de; García-Soriano, Juan Carlos; Zanda, Nicola; Castro, Sonia de CSIC ORCID; Gago, Federico CSIC ORCID; Jiménez-Ruiz, Antonio; Velázquez, Sonsoles CSIC ORCID CVN; Camarasa Rius, María José CSIC ORCIDartículo